SV2002000624A - SILDENAFIL MALEATE - Google Patents
SILDENAFIL MALEATEInfo
- Publication number
- SV2002000624A SV2002000624A SV2001000624A SV2001000624A SV2002000624A SV 2002000624 A SV2002000624 A SV 2002000624A SV 2001000624 A SV2001000624 A SV 2001000624A SV 2001000624 A SV2001000624 A SV 2001000624A SV 2002000624 A SV2002000624 A SV 2002000624A
- Authority
- SV
- El Salvador
- Prior art keywords
- maleate
- treatment
- sexual dysfunction
- pharmaceutical compound
- sildenafil maleate
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Gynecology & Obstetrics (AREA)
- Cardiology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención se refiere tanto a un compuesto farmacéutico para el tratamiento de la disfunción sexual masculina como a el procedimiento para su preparación. La invención consiste en un compuesto farmacéutico 5-[2-etoxi-5-(4-metilpiperazina-1-isulfonil) penil]-1-metil-3-n-propil-1,6-dihidro-7H-pirazolo[4,3-d]pirimida-7ona MALEATE, que se utiliza en el tratamiento de la disfunción sexual, asi como procedimiento de elaboración.The present invention relates both to a pharmaceutical compound for the treatment of male sexual dysfunction and to the process for its preparation. The invention consists of a pharmaceutical compound 5- [2-ethoxy-5- (4-methylpiperazine-1-isulfonyl) penyl] -1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo [4, 3-d] pyrimide-7ona MALEATE, which is used in the treatment of sexual dysfunction, as well as elaboration procedure.
Priority Applications (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SV2001000624A SV2002000624A (en) | 2001-09-05 | 2001-09-05 | SILDENAFIL MALEATE |
PCT/EC2002/000003 WO2003020720A1 (en) | 2001-09-05 | 2002-07-16 | Sildenafil maleate |
MXPA04002149A MXPA04002149A (en) | 2001-09-05 | 2002-07-16 | Sildenafil maleate. |
KR10-2004-7003315A KR20040071117A (en) | 2001-09-05 | 2002-07-16 | Sildenafil maleate |
PA20028553601A PA8553601A1 (en) | 2001-09-05 | 2002-08-22 | SILDENAFIL MALEATE |
UY27426A UY27426A1 (en) | 2001-09-05 | 2002-08-29 | SILDENAFIL MALEATE |
GT200200177A GT200200177A (en) | 2001-09-05 | 2002-09-03 | SILDENAFIL MALEATE |
ARP020103342A AR037811A1 (en) | 2001-09-05 | 2002-09-04 | SILDENAFIL MALEATE FOR THE TREATMENT OF MALE SEXUAL DYSFUNCTION, PREPARATION PROCEDURE AND THE PHARMACEUTICAL COMPOSITION THAT INCLUDES IT |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SV2001000624A SV2002000624A (en) | 2001-09-05 | 2001-09-05 | SILDENAFIL MALEATE |
Publications (1)
Publication Number | Publication Date |
---|---|
SV2002000624A true SV2002000624A (en) | 2002-09-12 |
Family
ID=40091701
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SV2001000624A SV2002000624A (en) | 2001-09-05 | 2001-09-05 | SILDENAFIL MALEATE |
Country Status (8)
Country | Link |
---|---|
KR (1) | KR20040071117A (en) |
AR (1) | AR037811A1 (en) |
GT (1) | GT200200177A (en) |
MX (1) | MXPA04002149A (en) |
PA (1) | PA8553601A1 (en) |
SV (1) | SV2002000624A (en) |
UY (1) | UY27426A1 (en) |
WO (1) | WO2003020720A1 (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX2017016930A (en) * | 2017-12-19 | 2019-06-20 | Malesil Research & Tech Llc | Method of treatment of diabetic foot ulcers. |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2000000199A1 (en) * | 1998-06-26 | 2000-01-06 | Nastech Pharmaceutical Company, Inc. | Nasal delivery of sildenafil citrate |
IL130968A (en) * | 1999-07-15 | 2002-12-01 | Shmuel Simon | Pharmaceutical composition comprising sildenafil or its analogs, useful for the treatment of tinnitus and hearing loss |
AU1888800A (en) * | 1999-09-13 | 2001-04-17 | Cipla Limited | A novel process for the synthesis of sildenafil citrate |
-
2001
- 2001-09-05 SV SV2001000624A patent/SV2002000624A/en active IP Right Grant
-
2002
- 2002-07-16 KR KR10-2004-7003315A patent/KR20040071117A/en not_active Application Discontinuation
- 2002-07-16 MX MXPA04002149A patent/MXPA04002149A/en active IP Right Grant
- 2002-07-16 WO PCT/EC2002/000003 patent/WO2003020720A1/en not_active Application Discontinuation
- 2002-08-22 PA PA20028553601A patent/PA8553601A1/en unknown
- 2002-08-29 UY UY27426A patent/UY27426A1/en not_active Application Discontinuation
- 2002-09-03 GT GT200200177A patent/GT200200177A/en unknown
- 2002-09-04 AR ARP020103342A patent/AR037811A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
UY27426A1 (en) | 2003-04-30 |
AR037811A1 (en) | 2004-12-09 |
GT200200177A (en) | 2003-06-05 |
PA8553601A1 (en) | 2003-05-14 |
WO2003020720A1 (en) | 2003-03-13 |
MXPA04002149A (en) | 2005-03-07 |
KR20040071117A (en) | 2004-08-11 |
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SV2002000624A (en) | SILDENAFIL MALEATE |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant |