SU166326A1 - YULUCHENIE N-FENIL-N, N'-DIMETHYLMOLOCHEVINA - Google Patents

YULUCHENIE N-FENIL-N, N'-DIMETHYLMOLOCHEVINA

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Publication number
SU166326A1
SU166326A1 SU883452A SU883452A SU166326A1 SU 166326 A1 SU166326 A1 SU 166326A1 SU 883452 A SU883452 A SU 883452A SU 883452 A SU883452 A SU 883452A SU 166326 A1 SU166326 A1 SU 166326A1
Authority
SU
USSR - Soviet Union
Prior art keywords
yuluchenie
dimethylmolochevina
fenil
phenyl
dimethylamine
Prior art date
Application number
SU883452A
Other languages
Russian (ru)
Inventor
Н. М. Харитонова Г. Ф. Конева Н. А. Айкина СОЮ Н. Ф. Алексеев
Original Assignee
Кемеровский научно исследовательский институтм
химической промышленности
Publication of SU166326A1 publication Critical patent/SU166326A1/en

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Description

Известен способ получени  Ы-фенил-Ы, Nдкметилмочевнны , используемой в качестве гербицида (фенурон), взаимодействием фенилизоцианата с диметиламином. Дл  получени  исходного финнлизоцианата используют фосген -  довитый агрессивный реагент.A known method of producing N-phenyl-N, N-methyl urea, used as a herbicide (phenuron), by the interaction of phenyl isocyanate with dimethylamine. Phosgene, a poisonous aggressive reagent, is used to prepare the initial finisocyanate.

Предложено взаимодействию с диметилфталатом подвергать бутил-Ы-фенилкарбамат.It was proposed to subject the interaction with dimethyl phthalate to butyl-L-phenylcarbamate.

Реакцию провод т в сосуде, соединенном с пр мым холодильником. Нелетучий целевой продукт накапливают в реакторе, а сннрт и избыток амина отгон ют. Спирт и амин иснользуют повторно.The reaction is carried out in a vessel connected to a direct cooler. The non-volatile target product is accumulated in the reactor, and the snort and excess amine are distilled off. Alcohol and amine are reused.

Пример. Дл  синтеза М-фенил-М, N-диметилмочевины (фенурон) используют 97 г (0,5 моль) бутил-К-фенилкарбамата (т. ил. 82°С).Example. For the synthesis of M-phenyl-M, N-dimethylurea (phenuron), 97 g (0.5 mol) of butyl-K-phenylcarbamate (T. Il. 82 ° C) are used.

Карбамат расплавл етс  и быстро нагреваетс  до 180°С. После этого в течение 2,5 час свод т 56,25 г диметиламина (1,25 моль).The carbamate melts and heats quickly to 180 ° C. Then, over 2.5 hours, 56.25 g of dimethylamine (1.25 mol) are reduced.

Температура реакции держитс  в пределах 175-185°С.The reaction temperature is kept in the range of 175-185 ° C.

Получают реакцнонной N-фeнил-N , N-диметилмочевины 90 г; реакционного бутанола- 63 мл (насыщен диметиламином). Реакционный продукт имеет т. нл. . 5 г нррдукта измельчают и промывают 15 мл бензола. Не растворимого в бензоле остатка (очищенный фенурон) получают 4,6 г. Т. нл. очищенного продукта 123°С; продукт идентичен с образцом X. ч. Ы-фенил-М, N-диметнлмочевины (добавка дает повыщение температуры плавлени  до 123,5°С).Receive reactionary N-phenyl-N, N-dimethylurea 90 g; reaction butanol - 63 ml (saturated with dimethylamine). The reaction product is so nl. . 5 g of the mineral powder are crushed and washed with 15 ml of benzene. The residue not soluble in benzene (purified phenuron) is 4.6 g. T. nl. purified product 123 ° C; the product is identical with sample X. h. N-phenyl-M, N-dimethyl urea (the additive raises the melting point to 123.5 ° C).

Предмет изобретени Subject invention

Способ получени  -фенил-Ы, N-днметилмочевпны на основе диметиламина, отличающийс  тем, что, с целью уирощени  и обеспечени  безопасностн нроцесса, диметиламин подвергают взаимодействию с расплавленным бутил-N-фенилкарбаматом.The method for the preparation of α-phenyl-L, N-dimethyl urea based on dimethylamine, characterized in that, in order to alleviate and ensure the safety of the process, dimethylamine is reacted with molten butyl-N-phenylcarbamate.

SU883452A YULUCHENIE N-FENIL-N, N'-DIMETHYLMOLOCHEVINA SU166326A1 (en)

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SU166326A1 true SU166326A1 (en)

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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1981002156A1 (en) * 1980-01-25 1981-08-06 Reanal Finomvegyszergyar Process for the preparation of n-aryl-n'-(mono-or disubstiuted)-urea derivatives
US5283362A (en) * 1991-08-16 1994-02-01 Chemie Linz Gesellschaft M.B.H. Process for the preparation of pure N,N'-asymmetrically substituted phenylureas

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1981002156A1 (en) * 1980-01-25 1981-08-06 Reanal Finomvegyszergyar Process for the preparation of n-aryl-n'-(mono-or disubstiuted)-urea derivatives
US5283362A (en) * 1991-08-16 1994-02-01 Chemie Linz Gesellschaft M.B.H. Process for the preparation of pure N,N'-asymmetrically substituted phenylureas

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