SU1563187A1 - 1-(2-ethoxyethyl)-4-hydroxypiperidine as an intermediate compound for synthesis of 1-(2-ethoxyethyl)-4-acylhydroxypiperidine hydrochlorides showing local anesthetic activity - Google Patents

1-(2-ethoxyethyl)-4-hydroxypiperidine as an intermediate compound for synthesis of 1-(2-ethoxyethyl)-4-acylhydroxypiperidine hydrochlorides showing local anesthetic activity

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Publication number
SU1563187A1
SU1563187A1 SU4445654/04A SU4445654A SU1563187A1 SU 1563187 A1 SU1563187 A1 SU 1563187A1 SU 4445654/04 A SU4445654/04 A SU 4445654/04A SU 4445654 A SU4445654 A SU 4445654A SU 1563187 A1 SU1563187 A1 SU 1563187A1
Authority
SU
USSR - Soviet Union
Prior art keywords
ethoxyethyl
synthesis
hydroxypiperidine
local anesthetic
acylhydroxypiperidine
Prior art date
Application number
SU4445654/04A
Other languages
Russian (ru)
Inventor
К.Д. Пралиев
В.К. Ю
С.А. Тараков
С.Н. Шин
Д.М. Кадырова
И.А. Козбагарова
Original Assignee
Институт химических наук АН КазССР
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Институт химических наук АН КазССР filed Critical Институт химических наук АН КазССР
Priority to SU4445654/04A priority Critical patent/SU1563187A1/en
Application granted granted Critical
Publication of SU1563187A1 publication Critical patent/SU1563187A1/en

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Abstract

FIELD: organic chemistry, heterocyclic compounds. SUBSTANCE: product: 1-(2-ethoxyethyl)-4-hydroxypiperidine. Synthesis of new compound is carried out by reaction of 1-(2-ethoxyethyl)-4-ketopiperidine with sodium borohydride in isopropanol. Yield is 99.9%, $$$ = 0.18; empirical formula is $$$. Substances synthesized on the base of new compound show local anesthetic activity comparable with that of novocaine. EFFECT: synthesis of new compound indicated above.
SU4445654/04A 1988-06-22 1988-06-22 1-(2-ethoxyethyl)-4-hydroxypiperidine as an intermediate compound for synthesis of 1-(2-ethoxyethyl)-4-acylhydroxypiperidine hydrochlorides showing local anesthetic activity SU1563187A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
SU4445654/04A SU1563187A1 (en) 1988-06-22 1988-06-22 1-(2-ethoxyethyl)-4-hydroxypiperidine as an intermediate compound for synthesis of 1-(2-ethoxyethyl)-4-acylhydroxypiperidine hydrochlorides showing local anesthetic activity

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SU4445654/04A SU1563187A1 (en) 1988-06-22 1988-06-22 1-(2-ethoxyethyl)-4-hydroxypiperidine as an intermediate compound for synthesis of 1-(2-ethoxyethyl)-4-acylhydroxypiperidine hydrochlorides showing local anesthetic activity

Publications (1)

Publication Number Publication Date
SU1563187A1 true SU1563187A1 (en) 1996-11-20

Family

ID=60527416

Family Applications (1)

Application Number Title Priority Date Filing Date
SU4445654/04A SU1563187A1 (en) 1988-06-22 1988-06-22 1-(2-ethoxyethyl)-4-hydroxypiperidine as an intermediate compound for synthesis of 1-(2-ethoxyethyl)-4-acylhydroxypiperidine hydrochlorides showing local anesthetic activity

Country Status (1)

Country Link
SU (1) SU1563187A1 (en)

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