SK10298A3 - Phenyl acetic acid derivatives, process and intermediate products for their production and their use as parasiticides and fungicides - Google Patents

Abstract

Phenyl acetic acid derivatives of formula (I) in which: X is NOCH3, CHOCH3 and CHCH3; Y is NMR and O; R, R<1> are hydrogen and C1-4 alkyl; R<2> is hydrogen, C1-C6 alkyl, C1-C4 alkyl halide and C3-C6 cycloalkyl; R<3> is C4-C6 alkyl, substituted C1-C6 alkyl, possibly substituted C2-C6 alkinyl or possibly substituted C2-C6 alkenyl; R<4> is hydrogen, possibly substituted C1-C10 alkenyl, C2-C10 alkinyl, C1-10 alkyl carbonyl, C2-C10 alkenyl carbonyl, C3-C10 alkinyl carbonyl or C1-C10 alkyl sulphonyl, aryl, aryl carbonyl, aryl sulphonyl, hetaryl, hetaryl carbonyl or hetaryl sulphonyl; and their salts, a process and intermediate products for their production and their use.

Description

(57) Annotation: i

Phenylacetic acid derivatives of general formula (I) are described in which the individual substituents and indices have the following meanings: X represents NOCH ₃ , CHOCH ₃ and CHCH ₃ ; Y is NR and O; R 1, R ¹ is hydrogen or C 1 -C 4 -alkyl; R ² is H, -C ₆ alkyl, C _r C ₄ haloalkyl, and Q-Cg-cycloalkyl; R ³ is C 4 -C 6 -cycloalkyl, C 2 -C 6 alkyl, substituted C 4 -alkyl, optionally substituted C 2 -C 6 -alkynyl or optionally substituted C 2 -C 6 -alkenyl; R ⁴ is hydrogen, optionally substituted C 1 -C 10 -alkyl, C 3 -C ₆ -cycloalkyl, C ₂ -C 10 -alkynyl, C 1 -C ₁₀ -alkylcarbonyl, C ₂ -C ₁₀ -alkenylcarbonyl, C ₃ -C ₁₀ -alkinylkarbonyl or C _r C | _O- alkylsulfonyl, aryl, arylcarbonyl, arylsulfonyl, hetaryl, hetarylcarbonyl or hetarylsulfonyl, as well as their salts, processes and intermediates for their preparation and their use.

R "ON-C (R ^d) -C (R ^a}» NOCH _s r,

O-C-Y-F (I)

Phenylacetic acid derivatives, process and intermediates for their preparation and their use as a pest and fungicide preparation

Technical field

The present invention relates to phenylacetic acid derivatives, processes for their preparation, intermediates for their preparation and their use as pests and as fungicides.

SUMMARY OF THE INVENTION

The present invention relates to phenylacetic acid derivatives of the general formula I

O = CYR ¹ in which the substituents and the index have the following meanings:

X NOCH ₃ , CHOCH ₃ and CHCH ₃ ;

Y NR and oxygen;

R 1, R ^{1 is} hydrogen or C ₁ -C ₄ -alkyl;

R ^{2 is} hydrogen, C 1 -C 6 -alkyl, C ₁ -C ₄ -haloalkyl and C ₃ -C 8 -cycloalkyl;

R ³ -C ₄ -C 8 -cycloalkyl, C ₂ -C 8 -alkyl or C ₁ -C 8 -alkyl which is partially or fully halogenated and / or carries one to three of the following: cyano, nitro, hydroxy, mercapto, amino, carboxyl , aminocarbonyl, aminothiocarbonyl, halogen, C1-C6-alkylaminocarbonyl, di-C1-C6-alkylaminocarbonyl, C1-C6-alkylaminothiocarbonyl, di-C1-C6-alkylaminothiocarbonyl, C1-C6-alkylsulfonyl, C1-C6-alkylsulfoxyl , (^ -C alkoxy, C ₁ -C haloalkoxy, C ^ -C alkoxycarbonyl, C - ^ - Cg alkylthio, C ^^ - Cg-alkylamino, di-C ^ -C-alkyl amino, C ₂ - cg-alkenyloxy, C ₃ -C -cycloalkyl, C ₃ -C cycloalkoxy, heterocyclyl, heterocyclyloxy, aryl, aryloxy, aryl-C ₁ -C ₄ -alkoxy, arylthio, aryl-C? -C? -alkylthio, hetaryl, hetaryloxy, hetaryl-C ₁ -C ₄ -alkoxy, hetarylthio, hetaryl-C ₁ -C ₄ alkylthio, wherein the cyclic radicals to be partially or fully halogenated and / or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, C 1 -C 6 g-alkyl, C ^ -C haloalkyl, C - ^ - C alkylsulfonyl, C -C alkylsulfonyl-oxy, C ₃ -C cycloalkyl, C -C alkoxy, C ^^ - Cg-haloalkoxy, C -C -alkoxycarbonyl, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylamino, di-C 1 -C 8 -alkylamino, C 1 -C 8 -alkylaminocarbonyl, di-C 1 -C 8 -alkylaminocarbonyl, C 1 -C 8 -alkylaminothiocarbonyl, di- C 1 -C 8 -alkylaminothiocarbonyl, C ₂ -C 8 -alkenyl, C ₂ -C 8 -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarythio and C (= NOR ^a ) -A _n -R 6;

C ₂ -C 8 -alkynyl or C ₂ -C 8 -alkenyl, which may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C- C1-C6-alkylaminocarbonyl, di-C1-C6-alkylaminocarbonyl, C1-C6-alkylaminothiocarbonyl, di-C1-C6-alkylaminothiocarbonyl, C1-C6-alkylsulfonyl, C1-C6-alkylsulfoxyl, C1-C6 -alkoxy, C ^ -C-haloalkoxy, C ^ -C alkoxycarbonyl, C ^ -C alkylthio, C -C alkylamino, di-Cl-Cg-alkylamino, _C2 ~ Cg-alkenyloxy, C -C cycloalkyl , C -C cycloalkyloxy, heterocyclyl, heterocyclyloxy, aryl, aryloxy, aryl-C ₁ -C ₄ -alkoxy, arylthio, _{aryl-C1-C4-alkylthio,} hetaryl, hetaryloxy, hetaryl-C? -C? -alkoxy , hetarylthio, hetaryl-aryl-C ₁ -C ₄ -alkylthio, wherein the cyclic moieties may be partially or fully halogenated and / or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl C 1 -C 8 -alkyl, C 1 -C 8 -alkyl -C -haloalkyl, C ₁ -C -alkylsulfonyl, C ^^ - Cg-alkylsulfoxyl, C ₃ -C cycloalkyl, C -C ^ alkoxy, C ^ -C-haloalkoxy, C ^ -C alkoxycarbonyl, C -C -alkylthio, C ₁ -C 8 -alkylamino, di-C 1 -C 8 -alkylamino, C 1 -C 8 -alkylaminocarbonyl, di-C 1 -C 8 -alkylaminocarbonyl, C 1 -C 8 -alkylaminothiocarbonyl, di-C 1 -C 8 -alkylaminothiocarbonyl, C ₂ -C-alkenyl, ^C2-C6 ~

-alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarythio and C (= NOR ^a ) -A _n -R ^b ;

R ⁴ hydrogen,

C ^ -Cio-alkyl, C ₃ -C -cycloalkyl, C ₂ -C ₁₀ -alkenyl, C ₂ -C ₁₀ -alkynyl, C ₂ -C ₁₀ ~ alkylcarbonyl, ^C 2 -C ₁₀ -alkenylkarbonyl, C ₃ -C _10- alkynylcarbonyl or C 1 -C 4 -alkylsulfonyl, which radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1-6 alkyl; C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl, C ₁ -C 8 -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C 1 -C 8 -alkoxycarbonyl, C 1 -C 8 -alkoxy -C8-alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, C1-C6-alkylaminocarbonyl, di-C1-C6-alkylaminocarbonyl, C1-C6-alkylaminothiocarbonyl, di-C1-C6-alkylamino -C -alkylaminothiocarbonyl, C ₂ -C alkenyl, C ₂ -C alkenyloxy, C ₃ -C -cycloalkyl, C ₃ -C cycloalkoxy, heterocyclyl, heterocyclyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy wherein the cyclic radicals may be partially or fully halogenated or carry one to three of the following of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkylsulfonyl, C1-C6-alkylsulfoxyl , C ₃ -C 8 -cycloalkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C ₃ -C 8 -alkoxy

-alkoxycarbonyl, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylamino, di-C 1 -C 8 -alkylamine ⁰ , C 1 -C 8 -alkylaminocarbonyl, di-C 1 -C 8 -alkylaminocarbonyl, C 1 -C 8 -alkylaminothiocarbonyl, di- C 1 -C 8 -alkylaminothiocarbonyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarythio or C (= NOR ^a ) -An-R 6 ⁾ ;

aryl, arylcarbonyl, arylsulfonyl, hetaryl, hetarylcarbonyl wherein these radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carbonyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1 -C 6 alkyl, C -C haloalkyl, C ^ -C alkylsulfonyl, C ^ -C-alkylsulfoxyl, C ₃ -C cycloalkyl, C ^ -C alkoxy, C - ^ - Cg-haloalkoxy, C ^ -CG- alkoxycarbonyl, C1-C6-alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, C1-C6-alkylaminocarbonyl, di-C1-C6-alkylaminocarbonyl, C1-C6-alkylaminothiocarbonyl, di-C1 C 1 -C 8 -alkylaminothiocarbonyl, C ₂ -C 8 -alkenyl, C ₂ -C 8 -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, hetaryl, hetaryloxy, or C (= NOR ^a ) -A _n -R ^b ;

where

A represents oxygen, sulfur or nitrogen, the nitrogen bearing hydrogen or C1-C6-alkyl;

n is 0 or 1;

R ^a is hydrogen or C 1 -C 8 -alkyl and

R ^b is hydrogen or C ₁ -C 8 -alkyl, and salts thereof, with the exception of compounds in which R ¹ and R ² are methyl, R ³ ethyl, R ⁴ methyl or ethyl, X NOCH ₃ and Y NH or O, as well as with the exception of compounds of formula I wherein R ³ is tert-butyl.

In addition, the invention relates to processes and intermediates in the preparation of these compounds, as well as compositions containing them for use against animal pests and harmful fungi.

Phenylacetic acid derivatives for use against animal pests are known from the literature [EP-A 422 597, EP-A 463 488, EP-A 370 629, EP-A 460575, EP-A 472 300, WO-A 90 / 07,493, WO -A 92 / 13,830, WO-A 92 / 18,487, WO-A 95 / 18,789, WO-A 95 / 21,153, WO-A 95 / 21,154].

The present invention has been developed in accordance with the specification of compounds having improved activity.

Initially, the phenylacetic acid derivatives of the general formula (I) were initially defined. In addition, processes and intermediates for their production, as well as preparations containing them on animal pests and harmful fungi, have been found and used in this sense.

The compounds of formula I are obtained by various methods according to literature procedures.

In principle, not in the synthesis of compounds of formula I, material, or by first forming a group -CÍXjCOYR ¹ or -CH ₂ ON = C ^(R2) -C ^(R3) = NOR ^fourth

The formation of the group -CfXjCOYR ¹ is known, for example, from the literature cited in the introduction and from the following literature: EP-A 222 070, EP-A 254 426, EP-A 370 629, EP-A 413 580, EP-A 656 352, PCT / EP 95/02013, EP-A 398,692.

1. For the formation of the group -CH ₂ ON = C (R ² ) -C (R ³ ) = NOR ⁴ , the benzyl derivative of the general formula

II reacts. with a hydroxyimine of formula III.

R ⁴ -ON = C ^(R3) -C ^(R2) = NOH (III)

R ⁴ -OH-C ^(R3) -C ^(R2) = NOCH,

c = x

C ^ CYR ¹

L ¹ in formula II is a nucleophilically exchangeable leaving group, for example halogen or sulfonate groups, preferably chlorine, bromine, iodine, mesylate, tosylate or triflate.

The reaction is carried out in a manner known per se in an inert organic solvent in the presence of a base such as sodium hydride, potassium hydroxide, potassium carbonate and triethylamine according to the methods described in Houben-Weyl, Vol. E 14b, p. 370 et seq. and Houben-Weyl, Vol. 10/1, p. 1189 et seq.

The necessary carbonic acid hydrazide is obtained, for example, by reacting the corresponding dihydroxyimine of formula IV with a nucleophilically substituted reagent of formula VI

HON = C (R ³ ) -C (R ² ) = NOH (IV) (VI) -> R ⁴ -ON = C (R ³ ) -C (R ² ) = NOH (III)

L ² in formula VI is a nucleophilically exchangeable leaving group, for example halogen or sulfonate groups, preferably chlorine, bromine, iodine, mesylate, tosylate or triflate.

The reaction is carried out in a known manner in an inert organic solvent in the presence of a base such as potassium carbonate, potassium hydroxide, sodium hydride, pyridine and triethylamine according to the methods described in Houben-Weyl, Vol. E 14b, p. 307 et seq., P. 370 et seq. and p. 385 et seq .; Houben-Weyl, Vol. 10/4, p. 55 et seq., P. 180 et seq. and p. 217 et seq .; Houben-Weyl, Vol. E5, p. 780 et seq.

1.1. Alternatively, the compounds of formula I can also be obtained by first reacting a benzyl derivative of formula II with a dihydroxyimine derivative of formula IV to the corresponding benzyloxime of formula V, followed by reacting the compound V with a nucleophilically substituted reagent of formula VI to give a compound of formula I.

HON = C ^(R3) -C ^(R2) = NOH (IV)

->

HON = C (R ³ ) -C (R ² ) = NO-CH (V) r ⁴ -1 ¹² (VI) r ⁴ -on = c (R ³ ) -c (r ² ) = no ₂ (I)

c = x (II)

O = CYR ¹

c = x

C ^ ¹ CYR

The reaction is carried out in a known manner in an inert organic solvent in the presence of a base such as potassium carbonate, potassium hydroxide, sodium hydride, pyridine and triethylamine according to the methods described in Houben-Weyl, Vol. E 14b, p. 307 et seq., P. 370 et seq. and p. 385 et seq .; Houben-Weyl, Vol. 10/4, p. 55 et seq., P. 180 et seq. and p. 217 et seq .; Houben-Weyl, Vol. E5, p. 780 et seq.

1.2. Analogously, the required hydroxyimine of formula III can also be prepared from a carbonylhydroxyimine of formula VII by reaction with a hydroxylamine of formula IXa or its salts of formula IXb.

+ O = C (R ³ ) -C (R ² ) = NOH -> R ⁴ -ON = C (R ³ ) -C (R ² ) = NOH (VII) (III)

Q in formula IXb is an anion of an acid, preferably an inorganic acid, for example a halide such as chloride.

The reaction is carried out in a known manner in an inert organic solvent according to the methods described in EP-A 513 580; Houben-Weyl, Vol. 10/4, p. 73 et seq .; Houben-Weyl, Vol. E 14b, p. 369 and p. 385 et seq.

Carbonylhydroxyimines of formula VII are known either from the literature (for example, Chem. Ber. 46, (1913) 1864; J. Chem. Soc. Perkin Trans. 2 (1994) 3, 415-420; Gazz. Chim. Ital. 63. 1933) 917 et seq., J. Indian, Chem. Soc. 35, (1958) 898) or may be prepared according to analogous procedures.

1.3 Alternatively, the compounds of formula I may be prepared by first reacting a benzyl derivative of formula II with a carbonylhydroxyimine of formula VII to give the corresponding benzyloxyimine of formula VIII, followed by reacting the compound of formula VIII with hydroxylamine of formula IXa, respectively. a salt of formula IXb to a compound of formula I.

O = C (R ³ ) -C (R ² ) = NOH (VII)

(Ii) c = x

OC-1'-R ¹

IXa / IXb

(VIII) c = x

C ^ CYR ¹

(I) c = x

O = C — YR ¹ (VI)

The reaction is carried out in a manner known per se in an inert organic solvent according to the methods described in Houben-Weyl, Vol. E 14b, p. 369 et seq .; Houben-Weyl, Vol. 10/1, p. 1189 et seq. and Houben-Weyl, Vol. 10/4, p. 73 et seq. or EP-A 13 580.

1.4. Another possibility for the preparation of the compounds of the formula I is the reaction of the benzyl II derivative with N-hydroxyphthalimide and subsequent hydrazinolysis to the benzylhydroxylamine IIa and the further reaction of the compound of the formula IIa with the carbonyl compound of the formula X.

N-OCH;

R ⁴ -ON = C (R ³⁾ -C (R ²⁾ = 0 (X)

C = X

O = CY — R ¹ h ₂ nnh ₂

->

(Ha)

> (I)

The reaction is carried out in a known manner in an inert solvent according to the methods described in EP-A 463 488, DE 42 42 867-3.

The required carbonyl compound X is obtained for example by reaction of a corresponding compound of formula Villa hydroxyiminokarbonylu a nucleophilically substituted reagent VI R ⁴ -L ^2-ON = C (R ³⁾ -C (R ²⁾ = a -> r = c ^{4-one (3} R ) -c (r ² ) = o (VI) (VIIa) (x) or by reacting the corresponding dicarbonyl compound of formula XI with hydroxylamine IXa or a salt thereof of formula IXb / r ⁴ -onh _{2 '} (IXa)

Example - + 0 = C (R ³ ) -C (R ² ) = O -> R ⁴ -ON = C (R ³ ) -C (R ² ) = O (XI) (X) r ⁴ -onh ₃ ®

V (IXb) /

The reaction is carried out in a known manner in a solvent according to the methods described by Houben-Weyl, Vol. 10/4, p. 55 et seq., P. 180 et seq. and p. 217 et seq .; Houben-Weyl, 307 et seq. and p. 369 et seq .; Houben-Weyl, et al.

inert organic in EP-A 513 580, et seq. , p. Vol. E 14 / b, p. Vol. E5, p. 780

1.5. The compounds may also be obtained by first reacting a benzylhydroxylamine derivative of formula IIa with a hydroxylimine derivative of formula VIIa to give the corresponding benzyloxyimine of formula V, followed by reacting the compound of formula V with a nucleophilically substituted reagent of formula VI as described above I.

HON = C (R ³ ) -C (R ² ) = NOH (Villa)

(Ha)

C ^ CYR ¹

(I) c = x

OC-YR ¹

1.6. Analogously, compounds of formula I can also be obtained by first reacting a benzylhydroxylamine of formula IIa with a dicarbonyl derivative of formula XI to the corresponding benzyloxyimine derivative of formula VIII and subsequently reacting the compound of formula VIII with IXa or a salt of formula IXb to compound of formula I.

with a hydroxylamine of the formula as described above,

O = C — Y — R ³ (XI) (Ha)

IXa / IXb

->

(VI)

R ⁴ ON = C (R ³ ) -C (R ² ) = NO-CH

(I) c = x

C ^ CYR ¹

1.7. Compounds of formula VIII wherein R ³ optionally represents substituted alkenyl may also be prepared; from a compound of formula VIIa.

Here, the double bond C = C moiety is formed by reaction of alkenyl compound of formula VIIIa with a carbonyl compound of the formula VIIIb in a known manner under aldol reaction (for example Organikum, 15th edition, pp. 565 ff.), Wherein the radicals R ³ ', R ^3' * and R ³ '''enter through the rest of R ³ :

(VIIIa) of 11-O == C (R ^J (VIIIb)

OC-YR ¹

(VIII)

IXa / IXb

Compounds of formula VIII may be reacted as described above to give compounds of formula I.

1.8. In addition, compounds of formula I in which R ³ is optionally substituted alkenyl can be synthesized from halogen compounds of formula VIIIc according to the following reaction scheme. For the sake of clarity, the group -C (= X) -COYR ^{1 is} abbreviated as # in this scheme.

(VIIIc)

principle principle ψ

Ψ

Here, the C = C double bond of the alkenyl moiety is formed by the Wittig-Horner reaction (according to the schematic representation; see Houben-Weyl, Vol. VIb, 4th edition, p. 383 et seq.) Or correspondingly via the Wittig-Horner reaction. The group CR ^{2 3} '= CR ³ ''R ³ '' ¹ corresponds to the alkenyl radical R ³ .

2. Compounds of formula I wherein Y is oxygen are most preferably prepared by converting compounds of formula X according to the methods described in EP-A 493 711, a lactone of formula XII, first to the corresponding benzoic acid of formula XIII and XIII via the corresponding halides to cyanocarboxylic acid of formula XIV, which is converted by the Pinner reaction (Angew. Chem. 94, 1 (1982)) to the alpha-keto ester of formula XV and subsequently to derivatives of formula I (see EP-A 348 766, DE-A 37 05 389 EP-A 178 826, DE-A 36 23 921).

R ⁵ -ON = C (R ⁴ ) -C (R ³ ) = NOH (X)

->

O (XII)

every ₂ h (XIII) ->

(Hal = halogen)

(XIII.)

-ΐ>

CN

R ⁴ -ON = C ^(R3) -C ^(R2) = NO-CH

C = 0 (R = H)

(Xv)

R ⁴ -ON = C (R ³⁾ -C (R ²⁾ = NOCH

(I) which R ₂ ^j

Compounds of formula I wherein R ¹ is hydrogen are prepared according to this procedure by saponification of an ester of formula XV and subsequent reaction to compounds of formula I.

3. Compounds of formula I wherein Y is NR are most preferably prepared by converting a compound of formula X according to the methods described in EP-A 493 711 with a lactone of formula XII first to the corresponding benzoic acid of formula XIII and the compound of formula XIII via the corresponding halides are converted to cyanocarboxylic acid of formula XIV, which is converted to the alpha-ketoester by a Pinel reaction (Angew. Chem. 94, 1 (1982)). The desired carbonic acid amides of formula XVI are prepared from the derivatives of formula XV by amidation and subsequently converted to compounds of formula I.

(X)

(XII)

R ⁴ -ON = C (R 3) .C (F _{{2) = NO. CH2} .

(ΧΗΙ)

co ₂ h

-j5 **

R <ON = C {R 3) -C (R 2> _{N-CH 2} O - γ (Hal Halog _S n) (Xllt.a) COHal

R ⁴ ON = C (R 3) -C (R 2) = NO-CH ₂ (XIV)

c = o

- £ >>

(R * H) XVI

R ⁴ -ON = C (R 3) -C (R 2) = HO-CH ₂

c = o

OC-NRR ¹

(I)

R ⁴ ON = C (R 3) -C (R 2) = NOCH.

c = x

H = CNRR1

4th

 cyanates followed by hydrolysis of a compound of formula XVI in which R is hydrogen (EP-A 547 825).

R ¹ -NC = S =>

5. In another variation, compounds of formula XVI are obtained by converting an ortho-halogen compound after metallization with oxalyl chloride to the corresponding keto acid chloride, which is subsequently reacted with an amine to give the corresponding amide of formula XVI (see J. Org. Chem. 46, 212 and et al. (1981) DE-A

42 280; Houben-Weyl, Vol. E5, p. 972 et seq.).

R <ON = C (R ³ ) -C (R ² ) = NO-CH 2 (Hal = Haogen)

sludge

6. In another variation, compounds of formula I in which Y is NR are obtained on the basis of ketoesters of formula XV by first derivatizing ketofunction and converting the derivatives thus obtained into the amide (Houben-Weyl, vol. E5, p. 941 et seq.).

R 4 -ON = C (R ³ ) -C (R ² ) = NO-CH ₂ γ

C = O (XV) i (R * H) CO ₂ R

R4ON = C (R ³ ) -C (R ² ) = NO-CH ₂ ·

c = x co ₂ y

O = C-NRR *

The compounds of formula II are known (EP-A 513 580, EP-A 477 631, EP-A 463 488, EP-A 585 751, EP-A 400 417, EP-A 251 082) or can be prepared by processes which are described in the above sources.

The compounds of the formula I can be prepared as isomeric E / Z mixtures in the preparation by virtue of their double bonds C = C and C = N, which, for example, can be separated into the individual compounds by crystallization or chromatography.

If isomeric mixtures are formed in the synthesis, separation is usually not absolutely necessary, since the individual isomers may be partially converted to one another during treatment for use or in use (for example under the influence of light, acids or bases). Conversion may also occur when used, for example, in the treatment of plants in the treated plant itself or in the treated harmful fungus or animal pest.

Due to the C = X double bond, isomers E are preferred over compounds of formula I for efficiency (configuration relative to -CH ₃ or -CH ₃ relative to (C = C) YR ¹ ).

Due to the double bond of -C (R ² ) -NOCH ₂ -, cis isomers are preferred over compounds of formula I (configuration based on the remainder of the -OCH ₂ group) for efficiency.

In the definitions of the compounds of formula I given in the introduction, collective terms have been used, which generally represent the following groups in general:

Halogen: fluorine, chlorine, bromine, iodine;

Alkyl: linear or branched alkyl groups having 1 to 4, 6 or 10 carbon atoms, for example C 1 -C 6 -alkyl such as methyl, ethyl, propyl, 1-methylethyl, butyl, 1-methylpropyl, 2-methylpropyl,

1,1-dimethylethyl, pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl, 1-ethylpropyl, hexyl, 1,1-dimethylpropyl, 1,2-dimethylpropyl, 1-methylpentyl, 2- methylpentyl, 3-methylpentyl, 4-methylpentyl, 1,1-dimethylbutyl, 1,2-dimethylbutyl, 1,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1,1,2-trimethylpropyl, 1,2,2-trimethylpropyl, 1-ethyl-1-methylpropyl, 1-ethyl-2-methylpropyl;

Alkylamino: an amino group which bears a linear or branched alkyl group having 1 to 6 carbon atoms as described above;

Dialkylamino: an amino group which carries two independent, linear or branched alkyl groups having from 1 to 6 carbon atoms, as mentioned above;

Alkylcarbonyl: linear or branched alkyl groups having 1 to 10 carbon atoms, which are bonded to the structure via a carbonyl group (-CO-);

Alkylsulfonyl: linear or branched alkyl groups having 1 to 6 or 10 carbon atoms, which are bonded to the structure via a sulfonyl group (-SO ₂ -);

Alkylsulfoxyl: linear or branched alkyl groups having 1 to 6 carbon atoms, which are bonded to the structure via a sulfoxyl group (-S (= O) -);

Alkylaminocarbonyl: (C 1 -C 6) alkylamino groups as described above which are bonded to the structure via a carbonyl group (-CO-);

Dialkylaminocarbonyl: dialkylamino groups having 1 to 6 carbon atoms per alkyl radical as mentioned above, which are bonded to the structure via a carbonyl group (-CO-);

Alkylaminothiocarbonyl: (C 1 -C 6) alkylamino groups as described above, which are bonded to the structure via a thiocarbonyl (-CS-) group;

Dialkylaminothiocarbonyl: dialkylamino groups having 1 to 6 carbon atoms per alkyl moiety as described above, which are bonded to the structure via a thiocarbonyl (-CS-) group;

Haloalkyl: straight-chain or branched alkyl group having 1 to 6 carbon atoms, which groups may be partially or fully hydrogen replaced by halogen atoms as mentioned above, for example C ₁ -C ₂ -haloalkyl, such as chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2- difluoroethyl,

2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl and pentafluoroethyl;

Alkoxy: linear or branched alkyl groups having 1 to 4 or 6 carbon atoms as mentioned above which are bonded to the structure via an oxygen atom (-O-), for example C 1 -C 8 -alkoxy such as methyloxy, ethyloxy, propyloxy, -methyletyloxy, butyloxy, 1-methylpropyloxy, 2-methylpropyloxy, 1,1-dimethyletyloxy, pentyloxy, 1-methylbutyloxy, 2-methylbutyloxy, 3-methylbutyloxy, 2,2-dimethylpropyloxy, 1-ethylpropyloxy, hexyloxy,

1,1-dimethylpropyloxy, 1,2-dimethylpropyloxy, 1-methylpentyloxy,

2-methylpentyloxy, 3-methylpentyloxy, 4-methylpentyloxy,

1,1-dimethylbutyloxy, 1,2-dimethylbutyloxy, 1,3-dimethylbutyloxy,

2,2-dimethylbutyloxy, 2,3-dimethylbutyloxy, 3,3-dimethylbutyloxy,

1-ethylbutyloxy, 2-ethylbutyloxy, 1,1,2-trimethylpropyloxy,

1,2.2-trimethylpropyloxy, 1-ethyl-1-methylpropyloxy and 1-ethyl-2-methylpropyloxy;

Alkoxycarbonyl: linear or branched alkyl groups having 1 to 6 carbon atoms which are bonded to the structure via an oxycarbonyl group (-CO (= O) -);

Haloalkoxy: linear or branched alkyl groups having 1 to 6 carbon atoms, in which groups the hydrogen atoms may be partially or totally replaced by halogen atoms as mentioned above, and which groups are bonded to the structure via an oxygen atom;

Alkylthio: linear or branched alkyl groups having 1 to 4 or 6 carbon atoms as described above, which are bonded to the structure via a sulfur atom (-S-), for example C 1 -C 8 -alkylthio such as methylthio, ethylthio, propylthio -methylethylthio, butylthio, 1-methylpropylthio, 2-methylpropylthio, 1,1-dimethylethylthio, pentylthio, 1-methylbutylthio, 2-methylbutylthio, 3-methylbutylthio, 2,2-dimethylpropylthio, 1-ethylpropylthio, hexylthio,

1,1-dimethylpropylthio, 1,2-dimethylpropylthio, 1-methylpentylthio,

2-methylpentylthio, 3-methylpentylthio, 4-methylpentylthio, 1,1-dimethylbutylthio, 1,2-dimethylbutylthio, 1,3-dimethylbutylthio,

2,2-dimethylbutylthio, 2,3-dimethylbutylthio, 3,3-dimethylbutylthio,

1-ethylbutylthio, 2-ethylbutylthio, 1,1,2-trimethylpropylthio,

1,2.2-trimethylpropylthio, 1-ethyl-1-methylpropylthio and 1-ethyl-228

-metylpropyltio;

Alkenyl: linear or branched alkenyl groups having 2 to 6 or 10 carbon atoms and a double bond at any position, for example C ₂ -C 8 -alkenyl such as ethenyl, 1-propenyl,

2-propenyl, 1-methyletenyl, 1-butenyl, 2-butenyl, 3-butenyl,

1-Methyl-1-propenyl, 2-methyl-1-propenyl, 1-methyl-2-propenyl,

2-Methyl-2-propenyl, 1-pentenyl, 2-pentenyl, 3-pentenyl,

4-pentenyl, 1-methyl-1-butenyl, 2-methyl-1-butenyl,

-butenyl, -butenyl, 1-methyl-2-butenyl, 1-methyl-3-butenyl,

3-methyl-13-methyl-23-methyl-32-methyl-2-butenyl, 2-methyl-3-butenyl,

-butenyl, 1,1-dimethyl-2-propenyl, 1,2-dimethyl-1-propenyl, 1,2-dimethyl-2-propenyl, 1-ethyl-1-propenyl, 1-ethyl-2-propenyl, 1 -hexenyl, 2-hexenyl, 3-hexenyl, 4-hexenyl, 5-hexenyl, 1-methyl-1-pentenyl, 2-methyl-1-pentenyl, 3-methyl-1-pentenyl, 4-methyl-1-pentenyl , 1-methyl-2-pentenyl, 2-methyl-2-pentenyl, 3-methyl-2-pentenyl, 4-methyl-2-pentenyl, 1-methyl-3-pentenyl, and 2-methyl-3-pentenyl, 3 -methyl-3-pentenyl, 4-methyl-3-pentenyl, 1-methyl-4-pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl, 4-methyl-4-pentenyl, 1,1 -dimethyl-2-butenyl, 1,1-dimethyl-3-butenyl,

1,2-dimethyl-1-butenyl, 1,2-dimethyl-2-butenyl, 1,2-dimethyl-3-butenyl, 1,3-dimethyl-1-butenyl, 1,3-dimethyl-2-butenyl, 1,3-dimethyl-3-butenyl, 2,2-dimethyl-3-butenyl, 2,3-dimethyl-1-butenyl, 2,3-dimethyl-2-butenyl, 2,3-dimethyl-3-butenyl, 3,3-dimethyl-1-butenyl, 3,3-dimethyl-2-butenyl, 1-ethyl-1-butenyl, 1-ethyl-2-butenyl, 1-ethyl-3-butenyl, 2-ethyl-1- butenyl, 2-ethyl-2-butenyl, 2-ethyl-3-butenyl, 1,1,2-trimethyl-2-propenyl, 1-ethyl-1-methyl-2-propenyl, 1-ethyl-2-methyl- 1-propenyl and 1-ethyl-2-methyl-2-propenyl;

Alkenyloxy: linear or branched alkenyl groups having 2 to 6 carbon atoms and a double bond at any position, which are bonded to the structure via an oxygen atom (-O-);

Alkenylthio: linear or branched alkenyl groups having 2 to 6 carbon atoms and a double bond at any position, which are bonded to the structure via an oxygen atom;

Alkenylamino: an amino group which carries a linear or branched alkenyl group having 2 to 6 carbon atoms, as described above;

Alkenylcarbonyl: linear or branched alkenyl groups having 2 to 10 carbon atoms and a double bond at any position, which are bonded to the structure via a carbonyl group (-CO-);

alkynyl; linear or branched alkynyl groups having 2 to 10 carbon atoms and a triple bond in any desired position, for example C ₂ -C ₆ -alkynyl, such as ethynyl, 2-propynyl, 2-btinyl,

3-butynyl, 1-methyl-2-propynyl, 2-pentynyl, 3-pentynyl,

4-pentynyl, 1-methyl-2-butynyl, 1-methyl-3-butynyl, 2-methyl-3-butynyl, 1,1-dimethyl-2-propynyl, 1-ethyl-2-propynyl, 2-hexynyl,

3-hexinyl, 4-hexinyl, 5-hexinyl, 1-methyl-2-pentynyl, 1-methyl-3-pentynyl, 1-methyl-4-pentynyl, 2-methyl-3-pentynyl, 2-methyl-4- pentynyl, 3-methyl-4-pentynyl, 4-methyl-2-pentynyl, 1,1-dimethyl-2-butynyl, 1,1-dimethyl-3-butynyl, 1,2-dimethyl-3-butynyl,

2,2-dimethyl-3-butynyl, 1-ethyl-2-butynyl, 1-ethyl-3-butynyl,

2-ethyl-3-butynyl and 1-ethyl-1-methyl-2-propynyl;

Alkinyloxy: linear or branched alkynyl groups having 2 to 6 carbon atoms and a triple bond at any position attached to the structure via an oxygen atom (-O-);

Alkynylthio: linear or branched alkynyl groups having 2 to 6 carbon atoms and a triple bond at any position attached to the structure via a sulfur atom (-S-);

Alkynylamino: an amino group bearing linear or branched alkynyl groups having 2 to 6 carbon atoms as described above;

Alkynylcarbonyl: linear or branched alkynyl groups having 3 to 10 carbon atoms and a triple bond at any position, which are bonded to the structure via a carbonyl group (-CO-);

Cycloalkyl: monocyclic alkyl groups having 3 to 6 cyclic carbon members, for example cyclopropyl, cyclobutyl, cyclopentyl or cyclohexyl;

Cycloalkoxy: monocyclic alkyl groups having 3 to 6 cyclic carbon members as mentioned above, which are attached to the structure via an oxygen atom (-O-);

Cycloalkylthio: monocyclic alkyl groups having 3 to 6 cyclic carbon members as mentioned above, which are attached to the structure via a sulfur atom (-S-);

Cycloalkylamino: an amino group which carries a monocyclic alkyl group having 3 to 6 cyclic carbon members as mentioned above;

Cycloalkenyl: monocyclic alkenyl groups having 5 to 8 cyclic carbon members such as cyclopentenyl, cyclohexenyl, cycloheptenyl and cyclooctenyl;

Cycloalkenyloxy: monocyclic alkenyl groups having 5 to 8 cyclic carbon members as mentioned above, which are attached to the structure via an oxygen atom (-O-);

Cycloalkenylthio: monocyclic alkenyl groups having 5 to 8 cyclic carbon members as mentioned above, which are attached to the structure via a sulfur atom (—S-);

Cycloalkenylamino: an amino group that carries monocyclic alkyl groups of 5 to 8 cyclic carbon members as described above;

Heterocyclyl, optionally heterocyclyloxy, heterocyclylthio and heterocyclylamino: 3- to 6-membered, saturated or partially unsaturated mono- or polycyclic heterocycles containing one to three heteroatoms selected from the group consisting of oxygen, nitrogen and sulfur, and which are bonded directly to the structures, optionally via an oxygen atom (heterocyclyloxy) or a sulfur atom (heterocyclythio) or a nitrogen atom (heterocyclylamino) such as 2-tetrahydrofuranyl, oxiranyl, 3-tetrahydrofuranyl, 2-tetrahydrothienyl, 3-tetrahydrothienyl, 2-pyrrolidinyl,

3-pyrrolidinyl, 3-isoxazolidinyl, 4-isoxazolidinyl, 5-isoxazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl, 5-isothiazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl,

2-oxazolidinyl, 4-oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl,

4-thiazolidinyl, 5-thiazolidinyl, 2-imidazolidinyl, 4-imidazolidinyl, 1,2,4-oxadiazolidin-3-yl, 1,2,4-oxadiazolidin-5-yl, 1,2,4-thiadiazolidin-3- yl, 1,2,4-thiadiazolidin-5-yl, 1,2,4-thiazolidin-3-yl, 1,3,4-oxadiazolidin-2-yl, 1,3,4-thiadiazolidin-2-yl, 1,3,4-triazolidin-2-yl, 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,3-dihydrofur-4-yl, 2,3-dihydrofur-5- yl,

2,5-dihydrofur-2-yl, 2,5-dihydrofur-3-yl, 2,3-dihydrothien-2-yl,

2,3-dihydrothien-3-yl, 2,3-dihydrothien-4-yl, 2,3-dihydrothien-5-yl, 2,5-dihydrothien-2-yl, 2,5-dihydrothien-3-yl, 2, 3-dihydropyrrol-2-yl, 2,3-dihydropyrrol-3-yl, 2,3-dihydropyrrol-4-yl,

2,3-dihydropyrrol-5-yl, 2,5-dihydropyrrol-2-yl, 2,5-dihydropyrrol-3-yl, 2,3-dihydroisoxazol-3-yl, 2,3-dihydroisoxazol-4-yl, 2, 3-dihydroisoxazol-5-yl, 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl, 4,5-dihydroisoxazol-5-yl, 2,5-dihydroisothiazol-3-yl, 2, 5-dihydroisothiazol-4-yl, 2,5-dihydroisothiazol-5-yl,

2,3-dihydroisopyrazol-3-yl, 2,3-dihydroisopyrazol-4-yl, 2,3-dihydroisopyrazol-5-yl, 4,5-dihydroisopyrazol-3-yl, 4,5-dihydroisopyrazol-4-yl, 4, 5-dihydroisopyrazol-5-yl, 2,5-dihydroisopyrazol-3-yl, 2,5-dihydroisopyrazol-4-yl, 2,5-dihydroisopyrazol-5-yl, 2,3-dihydrooxazol-3-yl, 2, 3-dihydro-oxazol-4-yl,

2,3-dihydrooxazol-5-yl, 4,5-dihydrooxazol-3-yl, 4,5-dihydrooxazol-4-yl, 4,5-dihydrooxazol-5-yl, 2,5-dihydrooxazol-3-yl,

2,5-dihydrooxazol-4-yl, 2,5-dihydrooxazol-5-yl, 2,3-dihydrothiazol-2-yl, 2,3-dihydrothiazol-4-yl, 2,3-dihydrothiazol-5-yl,

4,5-dihydrothiazol-2-yl, 4,5-dihydrothiazol-4-yl, 4,5-dihydrothiazol-5-yl, 2,5-dihydrothiazol-2-yl, 2,5-dihydrothiazol-4-yl,

2,5-dihydrothiazol-5-yl, 2,3-dihydroimidazol-2-yl, 2,3-dihydroimidazol-4-yl, 2,3-dihydroimidazol-5-yl, 4,5-dihydroimidazol-2-yl, 4, 5-dihydroimidazol-4-yl, 4,5-dihydroimidazol-5-yl,

2,5-dihydroimidazol-2-yl, 2,5-dihydroimidazol-4-yl, 2,5-dihydroimidazol-5-yl, 2-morpholinyl, 3-morpholinyl, 2-piperidinyl,

3-piperidinyl, 4-piperidinyl, 3-tetrahydropyridazinyl, 4-tetra-32 hydropyridazinyl, 2-tetrahydropyrimidinyl, 4-tetrahydropyrimidinyl, 5-tetrahydropyrimidinyl, 2-tetrahydropyrazinyl, 1,3,5-tetrahydrotriazin-2-yl, 1,2,4 —Tetrahydrotriazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, 2-tetrahydropyranyl, 1,3-dioxolan-2-yl, 3,4,5,6-tetrahydropyridin-2 -yl, 4H-1,3-thiazin-2-yl, 4H-1,3-benzothiazin-2-yl, 1,1-dioxo-2,3,4,5-tetrahydrothien-2-yl, 2H-1 4-benzothiazin-3-yl, 2H-1,4-benzooxazin-3-yl,

1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl;

Aryl, optionally aryloxy, arythio, arylamino, arylcarbonyl and arylsulfonyl: aromatic mono- or polycyclic hydrocarbon radicals which are bonded to the structure directly, optionally via an oxygen atom (-O-) (aryloxy) or sulfur atom (-S-) (arylthio) ), via a nitrogen atom (arylamino) or via a carbonyl group (-CO-) (alkylcarbonyl) or via a sulfonyl group (-SO ₂ -) (arylsulfonyl), for example phenyl, naphthyl and phenanthrenyl, optionally phenyloxy, naphthyloxy and phenanthrenyloxy and the corresponding carbonyl groups and sulfonyl residues;

Hetaryl, optionally hetaryloxy, hetarythio, hetarylamino, hetarylcarbonyl and hetarylsulfonyl: aromatic mono- or polycyclic radicals which may contain, in addition to the cyclic carbon members. furthermore, one to four nitrogen atoms or one to three nitrogen atoms and one oxygen atom or one sulfur atom, which are attached to the structure directly, optionally via an oxygen atom (-O-) (hetaryloxy) or a sulfur atom (-S-) (hetarylthio), via a nitrogen atom (hetarylamino) or via a carbonyl group (-CO-) (hetalkylcarbonyl) or via a sulfonyl group (-SO ₂ -) (hetarylsulfonyl), for example

5-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one oxygen or one sulfur atom: a 5-membered heterocycle which, in addition to carbon atoms, may contain: one to three nitrogen atoms or one to three nitrogen atoms, and one sulfur or oxygen atom or one oxygen or sulfur atom as ring members, for example

2-furyl, 3-furyl, 2-thienyl, 3-thienyl, 2-pyrrolyl, 3-pyrrolyl,

3-isoxazolyl, 4-isoxazolyl, 5-isoxazolyl, 3-isothiazolyl,

4-isothiazolyl, 5-isothiazolyl, 3-pyrazolyl, 4-pyrazolyl, 5-pyrazolyl, 2-oxazolyl, 4-oxazolyl, 5-oxazolyl, 2-thiazolyl, 4-thiazolyl, 5-thiazolyl, 2-imidazolyl, 4- imidazolyl, 1,2,4-oxadiazol-3-yl, 1,2,4-oxadiazol-5-yl, 1,2,4-thiadiazol-3-yl, 1,2,4-thiadiazol-5-yl, 1,2,4-triazol-3-yl, 1,3,4-oxadiazol-2-yl, 1,3,4-thiadiazol-2-yl, 1,3,4-triazol-2-yl;

benzocondensed 5-membered heteroaryl containing one to three nitrogen atoms or one to two nitrogen atoms and / or one oxygen atom or one sulfur atom: a 5-membered heterocycle containing, in addition to carbon atoms, one to three nitrogen atoms or one to two atoms and one sulfur atom or one oxygen atom or one oxygen atom or sulfur atom as ring members and in which two adjacent cyclic carbon members or one cyclic nitrogen member and one adjacent cyclic carbon member may be linked by a buta-1,3-diene-1 group , 4-diyl;

a nitrogen-bonded 5-membered heteroaryl containing one to four nitrogen atoms, or a nitrogen-bonded benzocondensed

5-membered heteroaryl containing one to three nitrogen atoms:

A 5-membered heterocycle and a benzo-fused 5-membered heterocycle as described above, wherein the two adjacent cyclic carbon members or one cyclic nitrogen member and one adjacent cyclic carbon member may be bridged by buta-1,3-diene-1,4- diyl, wherein the cycles may be attached to the structure through one of the cyclic nitrogen members;

6-membered heteroaryl containing one to three or one to four nitrogen atoms: a 6-membered heterocycle which, in addition to the carbon atoms, may contain one to three or one to four nitrogen atoms as ring members, for example 2-pyridinyl,

3-pyridinyl, 4-pyridinyl, 3-pyridazinyl, 4-pyridazinyl, 2-pyrimidinyl, 4-pyrimidinyl, 5-pyrimidinyl, 2-pyrazinyl, 1,3,5-triazin-2-yl, 1,2,4- triazin-3-yl and 1,2,4,5-tetrazin-3-yl;

benzocondensed 6-membered heteroaryl containing one to four nitrogen atoms: a 6-membered heterocycle in which two adjacent ring members may be linked by a buta-1,3-diene-1,434 group

diyl, for example quinoline, isoquinoline, quinazoline and quinoxaline, optionally with the given oxy, thio, amine, carbonyl or sulfonyl groups.

Partially or totally halogenated is intended to indicate that in the groups so characterized, the hydrogen atoms may be partially or totally replaced by the same or different halogen atoms as mentioned above.

In view of their biological activity, compounds of the formula I are preferably used in which Y is oxygen and r is 1. means methyl.

In addition, compounds of formula I are preferably used in which X is NOCH ₃ and Y is NR or oxygen.

Also preferred are compounds of formula I wherein X is NOCH ₃ and Y is NR and R is hydrogen or methyl.

Equally, preferred compounds I, wherein X is NOCH ₃ and Y is NR, and R ¹ is hydrogen or methyl.

Further preferred are compounds of formula I wherein X is NOCH ₃ and Y is NR and R and R ^{1 are} both hydrogen or methyl.

Further preferred are compounds of formula I wherein X is NOCH ₃ and Y is NR and R is hydrogen and R ¹ is methyl.

Except in which X is meant compounds noch ₃ and Y is 0.

of formula I,

In addition, in which X stands for CHOCH ₃ and Y stands for O,

Furthermore, preferred compounds I, wherein X is CHCH ₃ and Y is 0th

Furthermore, preferred compounds of the formula I in which R ² is hydrogen.

Furthermore, preferred compounds I, wherein R ² is methyl.

In addition, compounds of formula I, o

wherein R is ethyl.

Furthermore, preferred compounds I, wherein R ² is n-propyl or isopropyl.

Furthermore, preferred compounds I, wherein R ² is trifluoromethyl.

Other preferred compounds of formula I in which R ² is cyclopropyl.

Other preferred compounds of formula I, wherein R ³ is C ₂ -C alkyl.

In addition, compounds of the formula I are used in which the radical R ³ shows no branching or only one.

Furthermore, preferred compounds I, wherein R ³ is ethyl.

Furthermore, preferred compounds I, wherein R ³ is isopropyl.

Also used are compounds of formula I wherein R is n-propyl.

Furthermore, preferred compounds I, wherein R ³ is isobutyl or n-butyl.

Furthermore, preferred compounds I are those where R ³ is C ₅ or C ~ alkyl.

Preference is furthermore given to compounds of the formula I in which R ³ represents C ₄ -C 8 -cycloalkyl.

Furthermore, preferred compounds I, wherein R ³ is C ₂ -C ₆ -alkenyl.

Also used are compounds of formula I wherein R ³ is vinyl, allyl, prop-1-enyl, 2-methylprop-1-enyl or isopropenyl.

Equally, preferred compounds I, wherein R ³ is C ₂ -C alkynyl.

Equally, preferred compounds I, wherein R ³ is ethynyl, propargyl, l-butyn-3-yl, l-butyn-4-yl, 2-butyn-4-yl, in particular ethynyl and propargyl.

Furthermore, preferred compounds I, wherein R ³ is C -C alkyl.

Furthermore, preferred compounds I, wherein R ³ is substituted or unsubstituted C ₂ -C alkenyl.

Furthermore, preferred compounds I, wherein R ³ is substituted or unsubstituted C ₂ -C ₆ -alkynyl.

Also preferred are compounds of formula I wherein R ³ is substituted C 1 -C 6 -alkyl, wherein the alkyl moiety is partially or fully halogenated and / or carries one to three of the following substituents: nitro, hydroxy, amino, cyano, C ^ -C alkylsulfonyl, C ₁ -C alkoxy, C - ^ - Cg-haloalkoxy, C ^ -C alkylthio, C ^ -C-alkyl amino, di ^"C l ^-C 6 ^alk y ⁿ ° ^phenylamino, C ₃ -C ₆ -cycloalkyl, heterocyclyl, aryl, aryloxy, hetaryl, hetaryloxy, wherein the cyclic radicals may be. partially or fully halogenated and / or carry one to three of the following groups: cyano, nitro, amino, aminocarbonyl, aminothiocarbonyl, C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl, C 1 -C 8 -alkylsulfonyl, C C1-C6-alkylsulfoxyl, C1-C6-alkoxy, C1-C6-haloalkoxy, C1-C6-alkyloxycarbonyl, C1-C6-alkylthio, C1-C6-alkylamino, C1-C6-alkylaminocarbonyl, di- C ₁ -C 8 -alkylaminocarbonyl, C ₂ -C 8 -alkenyloxy, aryl and aryloxy.

Equally, preferred compounds I, wherein R ³ is substituted C - ^ - Cg alkyl, the alkyl radical being partially or fully halogenated and / or carries one to three of the following substituents: cyano, C ₁ -C ₃ ~ alkoxy, phenyl, phenoxy, hetaryl, hetaryloxy, wherein the (hetero) aromatic may carry one to three of the following groups: halogen, C? -C - ^ - alkyl, _C-L-C3 haloalkyl, C ₃ -C _L alkoxy, cyano, phenyl, C ₁ -C ₃ -alkylamino, di-C ₁ -C ₃ -alkylamino and C 1 -C 8 -haloalkyl.

Furthermore, preferred compounds I, wherein R ³ is C? -C? Alkyl, the alkyl moiety is substituted by phenyl or phenoxy, and the aromatic radical bears one to three of the following substituents: halogen, C ₁ -C ₃ ~ alkyl, C 1 -C 3 -alkoxy, cyano, CF ₃ and phenyl, especially halogen, C ₁ -C ₃ -alkyl, C ₁ -C ₃ -alkoxy.

Furthermore, preferred compounds I, wherein R ³ is a C-C-alkyl, where the alkyl radical is partially or fully halogenated and / or carries a cyano and / or C ₁ -C ₃ -alkoxy.

Also preferred are compounds of formula I wherein R ³ is C ₁ -C ₄ -alkyl, wherein the alkyl moiety is substituted with hetaryl or hetaryloxyl and the heteroaromate bears one to three of the following groups: halogen, C 1 -C 6 -alkyl, C 1 -C 8 -alkoxy, cyano, CF 3 and phenyl, especially halogen, C 1 -C 8 -alkyl, C 1 -C 8 -alkoxy.

Other preferred compounds of formula I, wherein R ³ is substituted or unsubstituted C ₂ -C ₄ alkenyl, wherein the alkenyl radical is partially or fully halogenated and / or carries one to three of the following radicals: cyano, C ^ -CG- alkoxy ,.

Other preferred compounds of formula I, wherein R ³ is substituted or unsubstituted C ₂ -C ₄ alkenyl, wherein the alkenyl radical may carry one to three halogen atoms.

Further preferred are compounds of the formula I in which R @ 1³ is also substituted C₂-C₅-alkenyl, wherein the alkenyl radical is substituted by a phenol or hetaryl group which may carry one to three of the following substituents: halogen, C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl,^Cand^-C3 -alkoxy, cyano, C1-C6-alkylamino and di-C1-C6-alkylamino, in particular halogen, C1-C6-alkyl and C1-C6-alkoxy.

Other preferred compounds of formula I, wherein R ³ is substituted or unsubstituted C ₂ -C ₆ -alkenyl, wherein the alkenyl radical may be substituted by phenyl.

Other preferred compounds of formula I, wherein R ³ is substituted or unsubstituted C ₂ -C alkenyl, wherein the alkenyl radical may be substituted by a hetaryl radical, which may carry one to three of the following substituents: halogen, C -C alkyl, and C ^ -C alkoxy.

Other preferred compounds of formula I, wherein R ³ is substituted or unsubstituted Cg-Cg alkenyl, wherein the alkenyl radical may be substituted by a hetaryl radical.

Other preferred compounds of formula I, wherein R ³ is substituted or unsubstituted C ₂ -C alkenyl, wherein the alkenyl radical may carry one to three of the following groups: halogen, hydroxy, amino, C ^ -C j-alkoxy, CJ C 1-6 alkylthio, C ₁ -C ₃ -alkylamino, di-C ₁ -C ₃ -alkylamino and phenyl, preferably halogen and alkoxy.

Other preferred compounds of formula I, wherein R ³ is substituted or unsubstituted C ₂ -C-alkynyl wherein the alkynyl radical may be substituted by a phenyl radical, in particular phenylethynyl.

Furthermore, preferred compounds I, wherein R ³ is substituted or unsubstituted C ₁ -C -alkyl, Cj.-Cg-alkenyl, C - ^ - Cg-alkynyl, arylalkyl, hetarylalkyl, aryloxyalkyl, hetaryloxyalkyl, aryl or hetaryl .

Preference is also given to compounds of the formula I in which R ⁴ is hydrogen.

Except for this is preferably use general compounds of formula I, v of which R ⁴ is C by lower alkyl. Except for this is preferably use general compounds of formula I, v of which R ⁴ is methyl or ethyl. Except for this is preferably use general compounds of formula I, v of which R ⁴ is aryl or hetarylalkyl. Except for this is preferably use general compounds

of formula I wherein R ⁴ is aryloxyalkyl or hetaryloxyalkyl.

In addition, compounds of formula I in which R ⁴ is aryl or hetaryl are preferably used.

In addition, compounds of formula I are preferably used in which R ⁴ is optionally substituted C 1 -C 10 -alkyl.

In addition, compounds of formula I are preferably used in which R ⁴ is optionally substituted C ₂ -C 8 -alkenyl.

In addition, compounds of the formula I are preferably used in which R ⁴ is optionally substituted C ₂ -C ₆ -alkynyl.

Furthermore, preferred compounds I, wherein R ⁴ represents C by lower alkyl, wherein the alkyl radical may be partially or fully halogenated and / or carries one to three of the following substituents: cyano, hydroxyl, amino, C C1-C6-alkoxy, C1-C6-haloalkoxy, C1-C6-alkoxycarbonyl, C1-C6-alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, aminocarbonyl, C1-C6-alkylaminocarbonyl , di-C 1 -C 8 -alkylaminocarbonyl, alkenyloxy, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ -cycloalkyloxy, wherein the cyclic radicals may be completely or partially halogenated and / or carry one to three C ₁ -C ₆ -cyclic radicals -alkyl or C ₁ -C ₃ -alkoxy.

Further preferred are compounds of formula I wherein R ⁴ is C ₂ -C 8 -alkenyl, wherein the alkenyl radical may be partially or fully halogenated or bears one to three of the following substituents: cyano, hydroxy, amino, C 1 -C 8 -alkoxy, C1-C6-haloalkoxy, C1-C6-alkoxycarbonyl, C1-C6-alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, aminocarbonyl, C1-C6-alkylaminocarbonyl, di-C ₁ -C 8 -alkylaminocarbonyl, alkenyloxy, C ₃ -C 8 -cycloalkyl, C ₃ -C 8 -cycloalkyloxy, wherein the cyclic groups may be partially or fully halogenated or carry one to three C ₁ -C ₃ -alkyl or C- -C j ^ alkoxy.

Further preferred are compounds of formula I wherein R ⁴ is C ₂ -C 8 -alkynyl, wherein the alkynyl moiety may be partially or fully halogenated and / or carries one to three of the following substituents: cyano, hydroxy, amino, C 1-4 alkyl. C1-C6-alkoxy, C1-C6-haloalkoxy, C1-C6-alkoxycarbonyl, C1-C6-alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, amino41 carbonyl, C1-C6-alkylaminocarbonyl, di -C 1-6 -C 8 -alkylaminocarbonyl, alkenyloxy, C ₃ -C 8 -cycloalkyl, C 1 -C 8 -cycloalkyloxy, wherein the cyclic groups may be partially or fully halogenated or carry one to three C ₁ -C ₃ -alkyl or C ₁ - _C3-alkoxy.

Furthermore, preferred compounds I, wherein R ⁴ is C ₂ -C-alkynyl wherein the alkynyl radical may carry one to three of the following substituents: halogen, cyano and C-Cg-alkoxy, in particular halogen.

Furthermore, preferred compounds I, wherein R ⁴ is C ₂ -C alkenyl, wherein the alkenyl radical may carry one to three of the following substituents: halogen, cyano and C - ^ - Cg alkoxy, in particular halogen.

Furthermore, preferred compounds I, wherein R ⁴ is C ₂ -C-alkyl, wherein the alkyl radical may be partially or fully halogenated and / or carry one to three of the following radicals: C - ^ - Cg-alkoxy, and cyano.

Further preferred are compounds of formula I wherein R ⁴ is C ₂ -C 8 -alkenyl.

Other preferred compounds of formula I, wherein R ⁴ is C ₂ -C-alkynyl, especially propargyl.

Further preferred are compounds of formula I wherein R ⁴ is propargyl.

Furthermore, preferred compounds of the formula I in which ^R4 is trans-3-chloro-prop-2-enyl.

In addition, compounds of the formula I in which R @ ⁴ is 2-methoxyethyl are preferably used.

In addition, compounds of formula I in which R ⁴ is allyl are preferably used.

Further preferred are compounds of formula I in which the substituents are selected from a combination of the above-mentioned preferably used substituents.

Particularly with respect to use, the compounds of formulas 1.1 to 1.4 listed in the following tables are preferably used.

R ⁴ ON

co ₂ ch ₃ (1.1)

co ₂ ch ₃

R ⁴ ON

R ^z

(1.3) co ₂ ch ₃

o = cnhch ₃

Table 1 q

Compounds of the formula 1.1 in which R ^J is ethyl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line in the Table A.

Table 2

The compounds of formula 1.2 wherein ^R3 is ethyl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line in the Table A.

Table 3

Compounds of formula 1.3 wherein R ³ is ethyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 4;

Compounds of the formula 1.4 in which R ^J is ethyl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line in the Table A.

Table 5

Compounds of formula 1.1 wherein R ³ is n-propyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 6

Compounds of formula 1.2 wherein R ³ is n-propyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 7

Compounds of formula 1.3 wherein R ³ is n-propyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 8

Compounds of formula 1.4 wherein R ³ is n-propyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 9

Compounds of formula 1.1, n

pollen and combinations of R substituents in one row in Table A.

Table 10

Compounds of general formula 1.2, pollen and combinations of substituents R ^{2 in} one row in Table A.

Table 11

Compounds of formula 1.3, pollen and combinations of substituents R ^{2 in} one row in Table A.

Table 12

Compounds of general formula 1.4, pollen and combinations of substituents R ^{2 in} one row in Table A.

wherein R ³ isopro and R ⁴ for the compound corresponds to q wherein R ^J isopro and R ⁴ for the compound corresponds to _x wherein R ^J isopro and R ⁴ for the compound corresponds wherein R ³ is isopro and R ⁴ for the compound corresponds to

Table 13

Compounds of formula 1.1 wherein R ³ is n-butyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 14

Compounds of formula 1.2 wherein R ³ is n-butyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 15

ABOUT

Compounds of formula 1.3 in which R is n-butyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 16

Compounds of formula (1.4) in which R @ 1 is n-butyl and the combination of substituents R @ ² and R @ ⁴ for the compound corresponds to one row in Table A.

Table 17

Compounds of formula 1.1 wherein R ³ is isobutyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 18

Compounds of formula 1.2 wherein R ³ is isobutyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 19

Compounds of formula 1.3 wherein R ³ is isobutyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 20

Compounds of formula 1.4 wherein R ³ is isobutyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 21

Compounds of formula 1.1 wherein R ³ is sec-butyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 22

Compounds of formula 1.2 wherein R ³ is sec-butyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 23

Compounds of formula 1.3 wherein R ³ is sec-butyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 24

Compounds of formula 1.4 wherein R ³ is sec-butyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 25

Compounds of formula 1.1 wherein R ³ is cyclobutyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 26.

Compounds of formula 1.2 wherein R ³ is cyclobutyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 27

Compounds of formula 1.3 wherein R ³ is cyclobutyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 28

Compounds of formula 1.4 wherein R ³ is cyclobutyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 29

Compounds of formula 1.1 wherein R ³ is n-pentyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 30

Compounds of formula 1.2 wherein R ³ is n-pentyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 31

Compounds of formula 1.3 wherein R ³ is n-pentyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 32

Compounds of formula 1.4 wherein R ³ is n-pentyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 33

Compounds of formula 1.1 wherein R ³ is cyclopentyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 34

Compounds of formula 1.2 wherein R ³ is cyclopentyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 35

Compounds of formula 1.3 wherein R ³ is cyclopentyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 36

Compounds of formula 1.4 wherein R ³ is cyclopentyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 37

Compounds of the formula 1.1 in which R ^J is n-hexyl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line in the Table A.

Table 38

Compounds of formula 1.2 wherein R ³ is n-hexyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 39

Compounds of formula 1.3 wherein R ³ is n-hexyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 40

Compounds of formula 1.4 wherein R ³ is n-hexyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 41

Compounds of formula 1.1 wherein R ³ is cyclohexyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 42

Compounds of formula 1.2 wherein R ³ is cyclohexyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 43

Compounds of formula 1.3 wherein R ³ is cyclohexyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 44

Compounds of formula 1.4 wherein R ³ is cyclohexyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 45

The compounds of formula 1.1 wherein ^R3 is ethenyl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line of Table A.

Table 46

Compounds of formula 1.2 wherein R ³ is ethenyl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 47

Compounds of formula 1.3 wherein R ³ is ethenyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 48

The compounds of formula 1.4 wherein ^R3 is ethenyl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line of Table A.

propene means the compound of the invention

Table 49

Compounds of general formula 1.1 in which R @ 1

2-yl and the combination of the substituents R ² and R ⁴ to criticism to one line of table A.

Table 50

Compounds of formula (1.2) in which R-2-yl and the combination of substituents R ² and R ⁴ pro give one line in Table A.

Table 51

Compounds of formula (1.3) in which R -2-yl and the combination of substituents R ² and R ⁴ pro give one line in Table A.

Table 52

Compounds of formula (1.4) in which R-2-yl and the combination of substituents R ² and R ⁴ pro have one line in Table A.

Table 53

Compounds of general formula 1.1 in which R 1 -1-yl and the combination of substituents R ² and R ⁴ pro give one line in Table A.

Table 54

Compounds of formula (1.2) in which R @ 1 -

1-yl and the combination of the substituents R ² and R ⁴ to criticism to one line of table A.

means propene compound zodpo means propene compound zodpo means propene compound zodpo means propene compound zodpo means propene compound zodpo

Table 55 * 5

Compounds of formula 1.3 in which R is propen-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 56

Compounds of formula 1.4 wherein R ³ is propen-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 57

Compounds of formula 1.1 wherein R ³ is isobuten-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 58

Compounds of formula 1.2 wherein R ³ is isobuten-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 59

Compounds of formula 1.3 wherein R ³ is isobuten-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 60

Compounds of formula 1.4 wherein R ³ is isobuten-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 61

Compounds of formula 1.1 wherein R ³ is propen-3-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 62

Compounds of formula 1.2 wherein R ³ is propen-3-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 63

Compounds of formula 1.3 wherein R ³ is propen-3-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 64 o

The compounds of formula 1.4, wherein R is propen-3-yl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line in the Table A.

Table 65

Compounds of formula 1.1 wherein R ³ is isobuten-3-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 66

Compounds of formula 1.2 wherein R ³ is isobuten-3-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 67

ABOUT

Compounds of formula 1.3 wherein R is isobuten-3-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 68

Compounds of formula 1.4 wherein R ³ is isobuten-3-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 69

Compounds of formula 1.1 wherein R ³ is but-2-en-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 70>> X

Compounds of formula 1.2 in which R is but-2-en-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 71

Compounds of formula 1.3 wherein R ³ is but-2-en-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 72

Compounds of formula 1.4 wherein R ³ is but-2-en-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 73

ABOUT

The compounds of formula 1.1, wherein R is but-3-en-l-yl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line in the Table A.

Table 74

Compounds of formula 1.2 wherein R ³ is but-3-en-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 75

Compounds of formula 1.3 wherein R ³ is but-3-en-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 76

Compounds of formula 1.4 wherein R ³ is but-3-en-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 77

Compounds of formula 1.1 wherein R ³ is ethynyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 78

Compounds of formula 1.2 wherein R ³ is ethynyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 79

Compounds of formula 1.3 wherein R ³ is ethynyl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 80

ABOUT

The compounds of formula 1.4, wherein R is ethynyl and the combination of the substituents R ² and R ⁴ for a compound corresponds to one line of Table A.

Table 81

Compounds of formula 1.1 wherein R ³ is prop-1-yn-3-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 82

Compounds of formula 1.2 wherein R ³ is prop-1-yn-3-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 83

Compounds of formula 1.3 wherein R ³ is prop-1-yn-3-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 84

Compounds of formula X.4 wherein R ³ is prop-1-yn-3-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 85

Compounds of formula 1.1 wherein R ³ is but-1-yn-3-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 86

Compounds of formula 1.2 wherein R ³ is but-1-yn-3-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 87

Compounds of formula 1.3 wherein R ³ is but-1-yn-3-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 88

Compounds of formula 1.4 wherein R ³ is but-1-yn-3-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 89

Compounds of formula 1.1 wherein R ³ is but-2-yn-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Tabuika 90

Compounds of formula 1.2 wherein R ³ is but-2-yn-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 91

Compounds of formula 1.3 wherein R ³ is but-2-yn-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 92

Compounds of formula 1.4 wherein R ³ is but-2-yn-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 93

Compounds of formula 1.1 wherein R ³ is but-3-yn-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 94

Compounds of formula 1.2 wherein R ³ is but-3-yn-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 95

Compounds of formula 1.3 wherein R ³ is but-3-yn-1-yl and the combination of substituents R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 96

Compounds of formula 1.4 wherein R ³ is but-3-yn-1-yl and the combination of R ² and R ⁴ for the compound corresponds to one row in Table A.

Table 97 * 2>

Compounds of formula 1.1 wherein R is methyl and R ^{4 is} hydrogen and R ³ for the compound corresponds to one row in Table B.

Table 98

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} hydrogen and the substituent R ³ for the compound corresponds to one row in Table B.

Table 99

Compounds of formula (1.3) wherein R is methyl and R ^{4 is} hydrogen and R ³ for the compound corresponds to one row in Table B.

Table 100

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} hydrogen and the substituent R ³ for the compound corresponds to one row in Table B.

Table 101

The compounds of formula 1.1, wherein R ² is methyl and R ⁴ is methyl and R ³ for a compound corresponds to one line in Table B.

Table 102

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ methyl and R ³ for the compound corresponds to one row in Table B.

Table 103

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ is methyl and R ³ for a compound corresponds to one line in Table B.

Table 104

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ methyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 105

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ ethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 106

The compounds of formula 1.2, wherein R ² is methyl and R ⁴ ethyl and R ³ for a compound corresponds to one line in Table B.

Table 107

The compounds of formula 1.3, wherein R ² is methyl

and R ^{4 is} ethyl and the row substituent in Table B. R ³ for the compound responsible one Table 108 Compounds of general formula 1.4 about R stands for methyl and R ^{4 is} ethyl and substituent R ³ for the compound responsible one

row in Table B.

Table 109 # 9>

Compounds of formula 1.1 in which R is methyl and R ^{4 is} n-propyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 110

The compounds of formula 1.2, wherein R ² is methyl and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 111

ABOUT

Compounds of formula (1.3) wherein R is methyl and R ^{4 is} n-propyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 112

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} n-propyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 113

The compounds of formula 1.1, wherein R ² is methyl and isopropyl, and R ^J R for a compound corresponds to one line in Table B.

Table 114

Compounds of formula 1.2 wherein R ² is methyl and R isopropyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 115

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 116

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 117

The compounds of formula 1.1, wherein R ² is methyl and R ⁴ n-butyl and R ³ for a compound corresponds to one line in Table B.

Table 118

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} n-butyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 119

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ n-butyl and R ³ for a compound corresponds to one line in Table B.

Table 120

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} n-butyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 121 n

Compounds of formula 1.1 in which R is methyl and R ⁴ sec-butyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 122

Compounds of formula (1.2) wherein R ² is methyl and R ⁴ sec-butyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 123

ABOUT

Compounds of formula 1.3 wherein R is methyl and R ⁴ sec-butyl and R ³ for the compound correspond to one row in Table B.

Table 124

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ sec-butyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 125

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ isobutyl and R ³ for the compound corresponds to one row in Table B.

Table 126

The compounds of formula 1.2, wherein R ² is methyl

Λ * 3 and R isobutyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 127

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ isobutyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 128

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ isobutyl and R ³ for the compound corresponds to one row in Table B.

Table 129

Compounds of general formula 1.1, v of which R ^z is methyl and R ⁴ t-butyl and the substituent R ³ for the mu row in Table B. the compound corresponds jedné- Table 130 Compounds of general formula 1.2, v wherein R ² is methyl and R ⁴ t-butyl and the substituent R ³ for the mu row in Table B. the compound corresponds jedné- Table 131 Compounds of general formula 1.3, v wherein R ² is methyl

and R t-butyl and R for the compound corresponds to one row in Table B.

Table 132

Compounds of formula 1.4 wherein R ² is methyl 4 and R t-butyl and the substituent R ^j for the compound corresponds to one row in Table B.

Table 133

The compounds of formula 1.1, wherein R ² is methyl and R @ ^4, n-pentyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 134

The compounds of formula 1.2, wherein R ² is methyl and R @ ^4, n-pentyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 135

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} n-pentyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 136

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} n-pentyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 137

The compounds of formula 1.1, wherein R ² is methyl and R and R isopentyl ^J for a compound corresponds to one line in Table B.

Table 138

Compounds of formula 1.2 wherein R ² is methyl and R isopentyl and the R substituent for the compound corresponds to one row in Table B.

Table 139

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ isopentyl and R ³ for the compound corresponds to one row in Table B.

Table 140

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ isopentyl and R ³ for the compound corresponds to one row in Table B.

Table 141 _# o

The compounds of formula 1.1, wherein R is methyl and R ⁴ neopentyl, and R ³ for a compound corresponds to one line in Table B.

Table 142 _> 9

Compounds of formula 1.2 wherein R is methyl and R ^{4 is} neopentyl and R ³ for the compound corresponds to one row in Table B.

Table 143

I

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} neopentyl and R ³ for the compound corresponds to one row in Table B.

Table 144

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} neopentyl and R ³ for the compound corresponds to one row in Table B.

Table 145

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-methylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 146

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-methylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 147

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 2-methylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 148

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-methylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 149

Compounds of formula (1.1) wherein R ² is methyl and R ^{4 is} 1-methylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 150

The compounds of formula 1.2, wherein R ² is methyl

A * 5 and R 1-methylbutyl and the R substituent for the compound corresponds to one row in Table B.

Table 151

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 1-methylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 152

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 1-methylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 153

ABOUT

Compounds of formula 1.1 in which R is methyl and R ^{4 is} pentan-3-yl and R ³ for the compound corresponds to one row in Table B.

Table 154 '9

Compounds of formula (1.2) wherein R is methyl and R ⁴ pentan-3-yl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 155

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ pentan-3-yl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 156

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ pentan-3-yl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 157

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3-methylbutan-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 158

ABOUT

Compounds of formula (1.2) in which R is methyl and R ^{4 is} 3-methylbutan-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 159

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 3-methylbutan-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 160

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3-methylbutan-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 161

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-methylbutan-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 162

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-methylbutan-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 163 p

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 2-methylbutan-2-yl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 164

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-methylbutan-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 165

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ hexyl and R ³ for the compound corresponds to one row in Table B.

Table 166

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ hexyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 167

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ hexyl and R ³ for a compound corresponds to one line in Table B.

Table 168

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ hexyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 169

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3,3-dimethylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 170

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3,3-dimethylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 171

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 3,3-dimethylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 172

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3,3-dimethylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 173

Compounds of formula (1.1) wherein R ² is methyl o

and R 2 -ethylbutyl and R for the compound corresponds to one row in Table B.

Table 174

Compounds of formula 1.2 wherein R ² is methyl and R 2 -ethylbutyl and the substituent R for the compound corresponds to one row in Table B.

Table 175

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-ethylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 176

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-ethylbutyl and R ³ for the compound corresponds to one row in Table B.

Table 177

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 4-methylpentyl and R ³ for the compound corresponds to one row in Table B.

Table 178

Compounds of formula X.2 wherein R ² is methyl and R ^{4 is} 4-methylpentyl and R ³ for the compound corresponds to one row in Table B.

Table 179

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 4-methylpentyl and R ³ for the compound corresponds to one row in Table B.

Table 180

Compounds of formula 1.4 wherein R ² is methyl * 3 and R 4 -methylpentyl and the substituent R for the compound corresponds to one row in Table B.

Table 181

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ cyclopropylmethyl and R ³ for the compound corresponds to one row in Table B.

Table 182

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} cyclopropylmethyl and R ³ for the compound corresponds to one row in Table B.

Table 183

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ cyclopropylmethyl and R ³ for the compound corresponds to one row in Table B.

Table 184

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} cyclopropylmethyl and R ³ for the compound corresponds to one row in Table B.

Table 185

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-cyclopropylet-1-yl and R ³ for the compound corresponds to one row in Table B.

Table 186

The compounds of formula 1.2, wherein R ² is methyl

Λ * 5 and R '2-cyclopropylet-1-yl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 187

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-cyclopropylet-1-yl and R ³ for the compound corresponds to one row in Table B.

Tabuika 188

The compounds of formula 1.4, wherein R ² is methyl and R ⁴ 2-cyclopropylene-l-yl and the substituent ^R3 for a compound corresponds to one line in Table B.

Tabuika 189

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ cyclohexylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 190

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ cyclohexylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 191

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ cyclohexylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 192

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ cyclohexylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 193

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-cyclohexylet-1-yl and R ³ for the compound corresponds to one row in Table B.

Table 194

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-cyclohexylet-1-yl and R ³ for the compound corresponds to one row in Table B.

Table 195

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-cyclohexylet-1-yl and R ³ for the compound corresponds to one row in Table B.

Table 196

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-cyclohexylet-1-yl and R ³ for the compound corresponds to one row in Table B.

Table 197

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} cyclopropyl and R ³ for the compound corresponds to one row in Table B.

Table 198

The compounds of formula 1.2, wherein R ² is methyl

4. o and R cyclopropyl and the substituent R for the compound corresponds to one row in Table B.

Table 199

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} cyclopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 200

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} cyclopropyl and R ³ for the compound corresponds to one row in Table B.

Table 201

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ cyclopentyl and R ³ for the compound corresponds to one row in Table B.

Table 202

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ cyclopentyl and R ³ for the compound corresponds to one row in Table B.

Table 203

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} cyclopentyl and R ³ for the compound corresponds to one row in Table B.

Table 204

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} cyclopentyl and R ³ for the compound corresponds to one row in Table B.

- 79 Table 205

Compounds of formula 1.1, in and R ⁴ cyclohexyl and R ^{3 in} one row in Table B.

whose R ² is methyl for the compound corresponds to

Table 206

Compounds of general formula 1.2, and in R ⁴ cyclohexyl and R ^{3 in} one row in Table B.

whose R ² is methyl for the compound corresponds to

Table 207

Compounds of formula 1.3, in and R ⁴ cyclohexyl and R ^{3 in} one row in Table B.

whose R ² is methyl for the compound corresponds to

Table 208

Compounds of formula 1.4, in and R ⁴ cyclohexyl and R ^{3 in} one row in Table B.

wherein R is methyl for the compound corresponds

Table 209

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} difluoromethyl and R ³ for the compound corresponds to one row in Table B.

Table 210

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} difluoromethyl and R ³ for the compound corresponds to one row in Table B.

Table 211

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} difluoromethyl and R ³ for the compound corresponds to one row in Table B.

Table 212

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} difluoromethyl and R ³ for the compound corresponds to one row in Table B.

Table 213

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-fluoroethyl and R ³ for the compound corresponds to one row in Table B.

Table 214

The compounds of formula 1.2, wherein R ² is methyl and R 2-fluoroethyl and R ^J for a compound corresponds to one line in Table B.

Table 215

The compounds of formula 1.3, wherein R ² is methyl

2 and R 2 -fluoroethyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 216

The compounds of formula 1.4, wherein R ² is methyl *

and R 2-fluoroethyl and R ^J for a compound corresponds to one line in Table B.

Table 217

The compounds of formula 1.1, wherein R ² is methyl and R ⁴ 3-fluoropropyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 218

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-fluoropropyl and R ³ for the compound corresponds to one row in Table B.

Table 219

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 3-fluoropropyl and R ³ for the compound corresponds to one row in Table B.

Table 220

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3-fluoropropyl and R ³ for the compound corresponds to one row in Table B.

Table 221

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2,2-difluoroethyl and R ³ for the compound corresponds to one row in Table B.

Table 222

The compounds of formula 1.2, wherein R ² is methyl

9 and R 2,2-difluoroethyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 223

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ 2,2-difluoroethyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 224

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2,2-difluoroethyl and R ³ for the compound corresponds to one row in Table B.

Table 225

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ 2,2,2-trifluoroethyl and R ³ for the compound corresponds to one row in Table B.

Table 226

The compounds of formula 1.2, wherein R ² is methyl and R ⁴ 2,2,2-trifluoroethyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 227

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ 2,2,2-trifluoroethyl and R ³ for the compound corresponds to one row in Table B.

Table 228

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ 2,2,2-trifluoroethyl and R ³ for the compound corresponds to one row in Table B.

Table 229

Compounds of formula 1.1 in which R @ ⁶ is methyl and R @ ^{4 is} 2-bromomethyl and R @ ³ for the compound corresponds to one row in Table B.

Table 230 p

Compounds of formula (1.2) wherein R is methyl and R ^{4 is} 2-bromomethyl and R ³ for the compound corresponds to one row in Table B.

Table 231 * 2>

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 2-bromomethyl and R ³ for the compound corresponds to one row in Table B.

Table 232

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-bromomethyl and R ³ for the compound corresponds to one row in Table B.

Table 233

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3-bromopropyl and R ³ for the compound corresponds to one row in Table B.

Table 234

Compounds of formula (1.2) in which R ² is methyl 4 and R 3 -bromopropyl and the substituent R for the compound corresponds to one row in Table B.

Table 235

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 3-bromopropyl and R ³ for the compound corresponds to one row in Table B.

Table 236

Compounds of formula (1.4) in which R ⁶ is methyl and R ^{4 is} 3-bromopropyl and R ³ for the compound corresponds to one row in Table B.

Table 237

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 4-bromobutyl and R ³ for the compound corresponds to one row in Table B.

Table 238

Compounds of formula 1.2 wherein R is methyl and R ^{4 is} 4-bromobutyl and R ³ for the compound corresponds to one row in Table B.

Table 239

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 4-bromobutyl and R ³ for the compound corresponds to one row in Table B.

Table 240

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 4-bromobutyl and R ³ for the compound corresponds to one row in Table B.

Table 241

Compounds of formula 1.1 wherein R is methyl and R ^{4 is} 2-iodoethyl and R ³ for the compound corresponds to one row in Table B.

Table 242

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-iodoethyl and R ³ for the compound corresponds to one row in Table B.

Table 243 * 9

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 2-iodoethyl and R ³ for the compound corresponds to one row in Table B.

Table 244 n

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 2-iodoethyl and R ³ for the compound corresponds to one row in Table B.

Table 245

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-chloroethyl and R ³ for the compound corresponds to one row in Table B.

Table 246

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-chloroethyl and R ³ for the compound corresponds to one row in Table B.

Table 247

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-chloroethyl and R ³ for the compound corresponds to one row in Table B.

Table 248 _x

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 2-chloroethyl and R ³ for the compound corresponds to one row in Table B.

Table 249

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3-chloropropyl and R ³ for the compound corresponds to one row in Table B.

Table 250

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-chloropropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 251

The compounds of formula 1.3, wherein R ² is methyl and R 3-chloropropyl and R for a compound corresponds to one line in Table B.

Table 252

The compounds of formula 1.4, wherein R ² is methyl and R 3-chloropropyl and R ^J for a compound corresponds to one line in Table B.

Tabuika 253

The compounds of formula 1.1, wherein R ² is methyl and R ⁴ 4-chlorobutyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Tabuika 254

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 4-chlorobutyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 255

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ 4-chlorobutyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Tabuika 256

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 4-chlorobutyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 257

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ cyanomethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 258

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ cyanomethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 259

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ cyanomethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 260

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} cyanomethyl and R ³ for the compound corresponds to one row in Table B.

Table 261

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-cyanoethyl and R ³ for the compound corresponds to one row in Table B.

Table 262

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-cyanoethyl and R ³ for the compound corresponds to one row in Table B.

Table 263

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ 2-cyanoethyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 264

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-cyanoethyl and R ³ for the compound corresponds to one row in Table B.

Table 271 _Λ o

Compounds of formula (1.3) wherein R is methyl and R ^{4 is} 4-cyanobutyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 272

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ 4-cyanobutyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 273

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ 6-cyanohexyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 274

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ 6-cyanohexyl and R ³ for the compound corresponds to one row in Table B.

Table 275

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ 6-cyanohexyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 276

The compounds of formula 1.4, wherein R ² is methyl the

and R * 6-cyanohexyl ^J and R for a compound corresponds to one line in Table B.

Table 277

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 278

Compounds of formula 1.2 wherein R is methyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 279

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 280 "f

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 281

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-ethoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 282

Compounds of formula 1.2 wherein R ² is methyl λ 9 and R 2 -ethoxyethyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 277

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 278

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 279 _of p

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 280

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 281

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-ethoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 282

The compounds of formula 1.2, wherein R ² is methyl

T and R 2 -ethoxyethyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 283

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-ethoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 284

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-ethoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 285

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-isopropoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 286

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-isopropoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 287

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-isopropoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 288

The compounds of formula 1.4, wherein R ² is methyl and R 3 * 2-isopropoxy-ethyl, and R ^J for a compound corresponds to one line in Table B.

Table 289

Compounds of formula 1.1 in which R is methyl and R ^{4 is} 3-methoxypropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 290

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-methoxypropyl and R ³ for the compound corresponds to one row in Table B.

Table 291> 2

Compounds of formula 1.3 in which R is methyl and R ^{4 is} 3-methoxypropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 292

Compounds of formula 1.4 in which R is methyl and R ^{4 is} 3-methoxypropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 293

The compounds of formula 1.1, wherein R ² is methyl and R ⁴ 3-ethoxypropyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 294

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-ethoxypropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 295

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ 3-ethoxypropyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 296

The compounds of formula 1.4, wherein R is methyl and R ⁴ 3-ethoxypropyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 297

The compounds of formula 1.1, wherein R ² is methyl and R ⁴ 3-isopropoxypropyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 298

The compounds of formula 1.2, wherein R ² is methyl and R ⁴ 3-isopropoxypropyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 299

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ 3-isopropoxypropyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 300

Compounds of formula 1.4 wherein R ² is methyl and R 3 -isopropoxypropyl and R ^J for the compound corresponds to one row in Table B.

Table 301 p

Compounds of formula 1.1 wherein R * is methyl and R ^{4 is} 4-methoxybutyl and R ³ for the compound corresponds to one row in Table B.

Table 302

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 4-methoxybutyl and R ³ for the compound corresponds to one row in Table B.

Table 303

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 4-methoxybutyl and R ³ for the compound corresponds to one row in Table B.

Table 304

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 4-methoxybutyl and R ³ for the compound corresponds to one row in Table B.

Table 305

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ 4-ethoxybutyl and R ³ for the compound corresponds to one row in Table B.

Table 306

The compounds of formula 1.2, wherein R ² is methyl

4. * 3 and R '4-ethoxybutyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 307

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 4-ethoxybutyl and R ³ for the compound corresponds to one row in Table B.

Table 308 n

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 4-ethoxybutyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 309

The compounds of formula 1.1, wherein R ² is methyl and R ⁴ 4-izopropoxybutyl and R ³ for a compound corresponds to one line in Table B.

Table 310

The compounds of formula 1.2, wherein R ² is methyl and R ⁴ 4-izopropoxybutyl and R ³ for a compound corresponds to one line in Table B.

Table 311

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ 4-izopropoxybutyl and R ³ for a compound corresponds to one line in Table B.

Table 312

Compounds of formula 1.4 wherein R ² is methyl and R 14 -isopropoxybutyl and the substituent R for the compound corresponds to one row in Table B.

Tabuika 313

Compounds of formula 1.1 in which R is methyl and R ^{4 is} prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 314 * 9 *

Compounds of formula 1.2 wherein R is methyl and R ^{4 is} prop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Tabuika 315

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 316 o

Compounds of formula 1.4 wherein R is methyl and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 317

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} cis-but-2-enyl and R ³ for the compound corresponds to one row in Table B.

Tabuika 318

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} cis-but-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 319

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} cis-but-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 320 o

Compounds of formula 1.4 wherein R ⁶ is methyl and R ^{4 is} cis-but-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 321

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ trans -but-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 322 o

Compounds of formula 1.2 wherein R * ⁵ is methyl and R ⁴ trans -but-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 323

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ trans -but-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 324

The compounds of formula 1.4, wherein R ² is methyl

4. q and R trans -but-2-enyl and the R substituent for the compound corresponds to one row in Table B.

Table 325

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3-methylbut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 326

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-methylbut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 327

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 3-methylbut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 328

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 3-methylbut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 329

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-methylprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 330

The compounds of formula 1.2, wherein R ² is methyl

AO and R 2 -methylprop-2-enyl and the substituent R ^J for the compound corresponds to one row in Table B.

100

Table 331

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-methylprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 332

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 2-methylprop-2-enyl and R ³ for the compound corresponds to one row in the table

Table 333

Compounds of formula and R ⁴ but-3-enyl and the substituent on the row of Table B.

Table 334

Compounds of formula and R ⁴ but-3-enyl and the substituent on the row in Table B.

Table 335

Compounds of formula and R ⁴ but-3-enyl and the substituent on the row in Table B.

Table 336

Compounds of formula and R ⁴ but-3-enyl and the substituent on the row in Table B.

B.

1.1, V wherein R ² is methyl R ³ for the compound corresponds jedné- 1.2, v whose R stands for methyl R ³ for the compound corresponds jedné- 1.3, v of which R is methyl R ³ for the compound corresponds jedné- 1.4, h whose R stands for methyl R ³ for the compound corresponds jedné-

101

Table 337

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} cis-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 338

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} cis-3-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 339

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} cis-3-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 340

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} cis-3-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 341

Compounds of formula 1.1 wherein R ² is methyl

A, O and R trans-3-chloroprop-2-enyl and the R substituent for the compound corresponds to one row in Table B.

Table 342

The compounds of formula 1.2, wherein R ² is methyl and R-trans 3-chloro-prop-2-enyl and R ^J for a compound corresponds to one line in Table B.

102

Table 343

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ trans-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 344 _of o

Compounds of formula 1.4 wherein R is methyl and R ⁴ trans-3-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 345

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 346

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 347

Compounds of formula 1.3 wherein R ² is methyl and R 2 -chloroprop-2-enyl and the substituent R for the compound corresponds to one row in Table B.

Table 348

The compounds of formula 1.4, wherein R ² is methyl Q

and R @ 2-chloro-prop-2-enyl and R ^J for a compound corresponds to one line in Table B.

103

Table 349

Compounds of formula 1.1 in which R is methyl and R ^{4 is} 3,3-dichloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 350

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 351>> 9

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 3,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 352

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 353

The compounds of formula 1.1, wherein R ² is methyl and R @ 2,3,3-trichloroprop-2-enyl and R ^J for a compound corresponds to one line in Table B.

Table 354

The compounds of formula 1.2, wherein R ² is methyl

R 9 and 2,3,3-trichloroprop-2-enyl and R ^J for a compound corresponds to one line in Table B.

104

Table 355

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ 2,3,3-trichloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 356

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ 2,3,3-trichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 357

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} cis-2,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 358

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} cis-2,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one line in Table B.

Table 359

The compounds of formula 1.3, wherein R ² is methyl and R CXS-2,3-dichloropropene-2-enyl and R ^J for a compound corresponds to one line in Table B.

Table 360

The compounds of formula 1.4, wherein R ² is methyl and R @ cis-2,3-dichloropropene-2-enyl and R ^J for a compound corresponds to one line in Table B.

105

Table 361

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ trans-2,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 362

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ trans-2,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 363 * 9

Compounds of formula 1.3 wherein R is methyl and R ⁴ trans-2,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 364

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ trans-2,3-dichloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 365

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} cis-3-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 366

The compounds of formula 1.2, wherein R ² is methyl and R @ cis-3-bromoprop-2-enyl and R ^J for a compound corresponds to one line in Table B.

106

Table 367

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} cis-3-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 368

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} cis-3-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 369

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ trans-3-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 370

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ trans-3-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 371

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ trans-3-bromoprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 372

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ trans-3-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

107

Table 373

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 374 *

Compounds of formula (1.2) wherein R is methyl and R ^{4 is} 2-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 375

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-bromoprop-2-enyl and R ³ for the compound corresponds to one line in Table B.

Table 376

Compounds of formula 1.4 wherein R * ¹ is methyl and R ^{4 is} 2-bromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 377

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 378

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

108

Table 379 * 9

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 3,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 380

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 381

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ 2,3,3-tribromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 382

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ 2,3,3-tribromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 383

The compounds of formula 1.3, wherein R ² is methyl and R tribromprop-2,3,3-2-enyl and R ^J for a compound corresponds to one line in Table B.

Table 384

The compounds of formula 1.4, wherein R ² is methyl and R tribromprop-2,3,3-2-enyl and R ^J for a compound corresponds to one line in Table B.

109

Table 385, J

Compounds of formula 1.1 wherein R is methyl and R ^{4 is} cis-2,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 386

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} cis-2,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 387

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ cis-2,3-dibromoprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 388

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} cis-2,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 389

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ trans-2,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 390

The compounds of formula 1.2, wherein R ² is methyl

Λ O and R trans-2,3-dibromoprop-2-enyl and the substituent R ^J for the compound corresponds to one row in Table B.

110

Table 391

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ trans-2,3-dibromoprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 392

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ trans-2,3-dibromoprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 393

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ trans-2-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 394

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ trans-2-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 395

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ trans-2-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 396

The compounds of formula 1.4, wherein R ² is methyl and R 5 * trans-2-chloro-but-2-enyl and R ^J for a compound corresponds to one line in Table B.

111

Table 397 n _x

Compounds of formula 1.1 wherein R is methyl and R ^{4 is} cis-2-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 398

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} cis-2-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 399

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} cis-2-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 400

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} cis-2-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 401

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ trans-3-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 402

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ trans-3-chlorobut-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

112

Table 403

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ trans-3-chlorobut-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 404

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ trans-3-chlorobut-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 405

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} cis-3-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 406

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} cis-3-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 407

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} cis-3-chlorobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 408

The compounds of formula 1.4, wherein R ² is methyl and R @ cis-3-chloro-2-enyl and R ^J for a compound corresponds to one line in Table B.

113

Table 409> 2

Compounds of formula 1.1 in which R is methyl and R ⁴ trans-2-bromobut-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 410

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ trans-2-bromobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 411

Compounds of formula 1.3 wherein R is methyl and R ⁴ trans-2-bromobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 412

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ trans-2-bromobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 413

Compounds of formula 1.1 wherein R ² is methyl

A, O and R cis-2-bromobut-2-enyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 414

The compounds of formula 1.2, wherein R ² is methyl and R @ cis-2-bromo-but-2-enyl and R ^J for a compound corresponds to one line in Table B.

114

Table 415

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} cis-2-bromobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 416

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} cis-2-bromobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 417

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} cis-3-bromobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 418

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} cis-3-bromobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 419

Compounds of formula 1.3 wherein R ² is methyl and R cis-3-bromobut-2-enyl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 420

Compounds of formula 1.4 wherein R ² is methyl and R is cis-3-bromobut-2-enyl and the R substituent for the compound corresponds to one row in Table B.

115

Table 421

Compounds of formula 1.1 in which R ² is methyl and R ⁴ trans-3-bromobut-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 422

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ trans-3-bromobut-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 423 _of n

Compounds of formula (1.3) in which R @ ¹ is methyl and R @ ⁴ trans -3-bromobut-2-enyl and the substituent R @ ³ for the compound corresponds to one row in Table B.

Table 424

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ trans-3-bromobut-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 425

Compounds of formula 1.1 wherein R ² is methyl

AO and R prop-2-yl and the substituent R ^J for the compound corresponds to one row in Table B.

Table 426

Compounds of formula 1.2 wherein R ² is methyl and R prop-2-ynyl and the substituent R ^J for the compound corresponds to one row in Table B.

116

Tabuika 427

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ prop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Tabuika 428

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ prop-2-ynyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 429

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3-chloroprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 430 * 9

Compounds of formula (1.2) in which R ⁶ is methyl and R ^{4 is} 3-chloroprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Tabuika 431

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 3-chloroprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Tabuika 432

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3-chloroprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

117

Table 433 n

Compounds of formula 1.1 wherein R is methyl and R ^{4 is} 3-bromoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 434

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-bromoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 435

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 3-bromoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 436

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3-bromoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 437

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 438

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

118

Table 439

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 440

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 441

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ but-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 442

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ but-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 443

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ but-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 444

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ but-2-ynyl and R ³ for the compound corresponds to one row in Table B.

119

Table 445 n *

Compounds of formula 1.1 in which R is methyl and R ^{4 is} but-3-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 446

Compounds of formula (1.2) wherein R ² is methyl and R ⁴ but-3-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 447

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ but-3-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 448

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} but-3-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 449

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ but-3-yn-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 450

The compounds of formula 1.2, wherein R ² is methyl and R 4 but-3-yn-2-yl, and R ^J for a compound corresponds to one line in Table B.

120

Table 451

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ but-3-yn-2-yl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 452

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ but-3-yn-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 453

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ pent-4-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 454

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} pent-4-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 455

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} pent-4-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 456

The compounds of formula 1.4, wherein R ² is methyl d

and R pent-4-ynyl and R ^j for the compound corresponds to one row in Table B.

121

Table 457

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ pent-3-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 458

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ pent-3-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 459

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ pent-3-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 460

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} pent-3-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 461

Compounds of formula 1.1 wherein R ² is methyl

A o and R pent-3-m-2-yl and the R substituent for the compound corresponds to one row in Table B.

Table 462

Compounds of formula 1.2 wherein R ² is methyl and R pent-3-yn-2-yl and the substituent R ^j for the compound corresponds to one row in Table B.

122

Table 463

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ pent-3-yn-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 464

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ pent-3-yn-2-yl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 465

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ pent-4-yn-2-yl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 466

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ pent-4-yn-2-yl and R ³ for the compound corresponds to one row in Table B.

Table 467

The compounds of formula 1.3, wherein R ² is methyl and R @ pent-4-yn-2-yl, and R ^J for a compound corresponds to one line in Table B.

Table 468

Compounds of formula 1.4 wherein R ² is methyl * 3 and R 5 pent-4-yn-2-yl and the substituent R ^j for the compound corresponds to one row in Table B.

123

Table 469 '9

Compounds of formula 1.1 wherein R is methyl and R ^{4 is} 2-vinyloxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 470

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-vinyloxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 471

The compounds of formula 1.3, in which R ^o is methyl and R ⁴ 2-vinyloxyethyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 472> 9 *

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 2-vinyloxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 473

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-allyloxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 474

The compounds of formula 1.2, wherein R ² is methyl

9 and R 2 -allyloxyethyl and the R substituent for the compound corresponds to one row in Table B.

124

Table 475

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 2-allyloxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 476

The compounds of formula 1.4, wherein R ² is methyl and R ⁴ 2-allyloxyethyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 477>> 9

Compounds of formula 1.1 in which R is methyl and R ^{4 is} 2-trifluoromethoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 478

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-trifluoromethoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 479

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-trifluoromethoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 480

The compounds of formula 1.4, wherein R ² is methyl

Z and R 2 -trifluoromethoxyethyl and the substituent R ^J for the compound corresponds to one row in Table B.

125

Table 481, n

Compounds of formula 1.1 in which R is methyl and R ^{4 is} 3-trifluoromethoxypropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 482

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-trifluoromethoxypropyl and R ³ for the compound corresponds to one row in Table B.

Table 483, 2

Compounds of formula 1.3 in which R is methyl and R ^{4 is} 3-trifluoromethoxypropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 484

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 3-trifluoromethoxypropyl and R ³ for the compound corresponds to one row in Table B.

Table 485

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 4-trifluoromethoxybutyl and R ³ for the compound corresponds to one row in Table B.

Table 486

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 4-trifluoromethoxybutyl and R ³ for the compound corresponds to one row in Table B.

126

Table 487 "o

Compounds of formula (1.3) wherein R and R ⁴ 4-trifluoromethoxybutyl and R ³ correspond to one row in Table B.

Table 488

Compounds of formula 1.4 wherein R ² and R ⁴ 4-trifluoromethoxybutyl and R ³ correspond to one row in Table B.

Table 489

Compounds of formula 1.1 in which R and R ⁴ hydroxycarbonylmethyl and R ³ pro give one line in Table B.

Table 490

Compounds of formula (1.2) in which R ² and R ⁴ hydroxycarbonylmethyl and the substituent R ³ for give one line in Table B.

Table 491

The compounds of formula 1.3, wherein R ² and R and R hydroxycarbonylmethyl to say one line of Table B.

Table 492

Compounds of formula 1.4 wherein R ² and R ⁴ hydroxycarbonylmethyl and the substituent R ³ for give one line in Table B.

means methyl for a compound means methyl for a compound means methyl compound means methyl compound means methyl compound means methyl compound from127

Table 493, 2 *

Compounds of formula 1.1 in which R is and R ^{4 is} methoxycarbonylmethyl and the substituent R ³ for the compound leads to one row in Table B.

Table 494

The compounds of formula 1.2, wherein R ² is methoxycarbonylmethyl and R @ ⁴ and R ³ for the compound of criticism to one line of Table B.

Table 495, 2 Compounds of formula 1.3 in which R is and R ^{4 is} methoxycarbonylmethyl and the substituent R ³ for the compound leads to one row in Table B.

Table 496

Compounds of formula 1.4 wherein R ² is and R ⁴ methoxycarbonylmethyl and the substituent R ³ for the compound leads to one row in Table B.

Table 497

The compounds of formula 1.1, wherein R ² is and R and R ammokarbonylmetyl ^J criticism for the compound to one line of Table B.

Table 498

The compounds of formula 1.2, wherein R ² is and R ⁴ aminocarbonylmethyl and R ³ for the compound of criticism to one line of Table B.

Methyl odpovedometyl odpovedometyl odpovedometyl odpovedometyl zodpo128

Table 499

The compounds of formula 1.3, wherein R ² is methyl and R ⁴ aminocarbonylmethyl and R ³ for a compound corresponds to one line in Table B.

Table 500

The compounds of formula 1.4, wherein R ² is methyl and R ⁴ aminocarbonylmethyl and R ³ for a compound corresponds to one line in Table B.

Table 501

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ N-methylaminocarbonylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 502

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ N-methylaminocarbonylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 503

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} N-methylaminocarbonylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 504

The compounds of formula 1.4, wherein R ² is methyl

R 1 and R N -methylaminocarbonylmethyl and the substituent R ^J for the compound corresponds to one row in Table B.

129

Table 505, 9

Compounds of formula 1.1 in which R is methyl and R ^{4 is} Ν, Ν-dimethylaminocarbonylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 506

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ Ν, Ν-dimethylaminocarbonylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 507

Compounds of formula 1.3 wherein R ² is methyl and R ⁴ Ν, Ν-dimethylaminocarbonylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 508

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ Ν, Ν-dimethylaminocarbonylmethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 509

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-hydroxycarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 510

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-hydroxycarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

130

Table 511

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-hydroxycarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 512

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 2-hydroxycarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 513

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-methoxycarbonylethyl and R ³ for the compound corresponds to one row in Table B.

Table 514

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-methoxycarbonylethyl and R ³ for the compound corresponds to one row in Table B.

Table 515

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-methoxycarbonylethyl and R ³ for the compound corresponds to one row in Table B.

Table 516

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-methoxycarbonylethyl and R ³ for the compound corresponds to one row in Table B.

131

Table 517

Compounds of formula 1.1 wherein R is methyl and R ^{4 is} 2-aminocarbonylethyl and R ³ for the compound corresponds to one row in Table B.

Table 518

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-aminocarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 519 ^ 9

Compounds of formula 1.3 in which R is methyl and R ^{4 is} 2-aminocarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 520

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 2-aminocarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 521

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-N-methylaminocarbonylethyl and R ³ for the compound corresponds to one row in Table B.

Table 522

The compounds of formula 1.2, wherein R ² is methyl

9 and R @ 2 N-R metylaminokarbonyletyl and ^J for a compound corresponds to one line in Table B.

132

Table 523, n

Compounds of formula 1.3 in which R is methyl and R ^{4 is} 2-N-methylaminocarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 524

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-N-methylaminocarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 525

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-N, N-dimethylaminocarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 526 _of 9

Compounds of formula 1.2 wherein R is methyl and R ^{4 is} 2-N, N-dimethylaminocarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 527

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-N, N-dimethylaminocarbonylethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 528

The compounds of formula 1.4, wherein R ² is methyl the

and R 2-N, N-dimetylammokarbonyletyl ^J and R for a compound corresponds to one line in Table B.

133

Table 529

Compounds of formula 1.1 wherein R is methyl and R ^{4 is} 2-aminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 530

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-aminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 531, 2 Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 2-aminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 532

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-aminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 533

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-N-methylaminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 534

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-N-methylaminoethyl and R ³ for the compound corresponds to one row in Table B.

134

Table 535

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 2-N-methylaminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 536

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 2-N-methylaminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 537

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-N, N-dimethylaminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 538

Compounds of formula 1.2 wherein R is methyl and R ^{4 is} 2-N, N-dimethylaminoethyl and R ³ for the compound corresponds to one row in Table B.

Table 539

The compounds of formula 1.3, wherein R ² is methyl

and R ^{4 is} 2-N, N-dimethylaminoethyl and a substituent R ³ for the compound corresponds to one row in Table B. Table 540 Compounds of general formula 1.4 R ² means methyl and R ^{4 is} 2-N, N-dimethylaminoethyl and a substituent R ³ for the compound

corresponds to one row in Table B.

135

Table 541

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-aminopropyl and R ³ for the compound corresponds to one row in Table B.

Table 542

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 2-aminopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 543

Compounds of formula (1.3) wherein R is methyl and R ^{4 is} 2-aminopropyl and R ³ for the compound corresponds to one row in Table B.

Table 544

Compounds of formula 1.4 wherein R is methyl and R ^{4 is} 2-aminopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 545

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 2-N-methylaminopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 546

The compounds of formula 1.2, wherein R ² is methyl

9 and R @ 2 N-R metylammopropyl and ^J for a compound corresponds to one line in Table B.

136

Table 547 '·)

Compounds of formula (1.3) in which R and R ⁴ 2-N-methylaminopropyl and the substituent R ³ for one line in Table B.

Table 548

Compounds of formula 1.4 wherein R ² and R ^{4 of} 2-N-methylaminopropyl and the substituent R ³ for one line in Table B.

Table 549

Compounds of formula 1.1 in which R ² and R ⁴ 2 -N, N-dimethylaminopropyl and R ³ correspond to one row in Table B.

Table 550

The compounds of formula 1.2, wherein R ² and R 2 ^4-N, N-dimethylaminopropyl, and R ³ corresponds to one line in Table B.

Table 551

Compounds of formula (1.3) wherein R ²

4- 2 and R 2 -N, N-dimethylaminopropyl and the substituent R corresponds to one row in Table B.

Table 552

Compounds of formula (1.4) wherein R ²

2 and R 2 -N, N-dimethylaminopropyl and R ^J corresponds to one row in Table B.

means methyl compound means methyl compound means methyl for compound means methyl for compound means methyl for compound means methyl for compound

137

Tabuika 553

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3-aminopropyl and R ³ for the compound corresponds to one row in Table B.

Table 554

Compounds of formula 1.2 in which R is methyl and R ^{4 is} 3-aminopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 555

Compounds of formula 1.3 wherein R ² is methyl and R ^{4 is} 3-aminopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 556

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3-aminopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 557

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 3-N-methylaminopropyl and R ³ for the compound corresponds to one row in Table B.

Tabuika 558

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-N-methylaminopropyl and R ³ for the compound corresponds to one row in Table B.

138

Table 559

The compounds of formula 1.3, wherein R ^a is methyl and R ⁴ 3-N-dimethylaminopropyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 560

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 3-N-methylaminopropyl and R ³ for the compound corresponds to one row in Table B.

Table 561 _x o

Compounds of formula 1.1 in which R is methyl and R ^{4 is} 3-N, N-dimethylaminopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 562

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 3-N, N-dimethylaminopropyl and R ³ for the compound corresponds to one row in Table B.

Table 563

The compounds of formula 1.3, wherein R ² is methyl

7 and R 3 -N, N-dimethylammopropyl and the R substituent for the compound corresponds to one row in Table B.

Table 564

The compounds of formula 1.4, wherein R ² is methyl

7 and R 3 -N, N-dimethylaminopropyl and the R substituent for the compound corresponds to one row in Table B.

139

Table 565

Compounds of formula 1.1 wherein R ² is methyl and R ^{4 is} 4-aminobutyl and R ³ for the compound corresponds to one row in Table B.

Table 566

Compounds of formula 1.2 wherein R ² is methyl and R ^{4 is} 4-aminobutyl and R ³ for the compound corresponds to one row in Table B.

Table 567

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 4-aminobutyl and R ³ for the compound corresponds to one row in Table B.

Table 568

Compounds of formula 1.4 wherein R ² is methyl and R ^{4 is} 4-aminobutyl and R ³ for the compound corresponds to one row in Table B.

Table 569

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ 4-N-methylaminobutyl and R ³ for the compound corresponds to one row in Table B.

Table 570

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ 4-N-methylaminobutyl and R ³ for the compound corresponds to one row in Table B.

140

Table 571, J

Compounds of formula 1.3 wherein R is methyl and R ^{4 is} 4-N-methylaminobutyl and R ³ for the compound corresponds to one row in Table B.

Table 572

Compounds of formula 1.4 wherein R ² is methyl and R ⁴ 4-N-methylaminobutyl and R ³ for the compound corresponds to one row in Table B.

Table 573

Compounds of formula 1.1 wherein R ² is methyl and R ⁴ 4-N, N-dimethylaminobutyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 574

Compounds of formula 1.2 wherein R ² is methyl and R ⁴ 4-N, N-dimethylaminobutyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 575

The compounds of formula 1.3, wherein R ² is methyl. 3 and R 4-N, N-dimethylammobutyl and the R substituent for the compound corresponds to one row in Table B.

Table 576

The compounds of formula 1.4, wherein R ² is methyl

2 and R 11 ^is 4-N, N-dimethylammobutyl and the R substituent for the compound corresponds to one row in Table B.

141

Table 577

The compounds of formula 1.1, wherein R ² is hydrogen and R ⁴ is hydrogen and R ³ for a compound corresponds to one line in Table B.

Table 578

Compounds of formula 1.2 wherein R ² is hydrogen and R ⁴ hydrogen and the substituent R ³ for the compound corresponds to one row in Table B.

Table 579

The compounds of formula 1.3, wherein R ² is hydrogen and R ⁴ is hydrogen and R ³ for a compound corresponds to one line in Table B.

Table 580

Compounds of formula 1.4 wherein R ² is hydrogen and R ⁴ hydrogen and the substituent R ³ for the compound corresponds to one row in Table B.

Table 581

The compounds of formula 1.1, wherein R ² is hydrogen and R is methyl and R ^J for a compound corresponds to one line in Table B.

Table 582

Compounds of formula 1.2 wherein R ² is hydrogen and R ⁴ methyl and R ³ for the compound corresponds to one row in Table B.

142

Table 583

Compounds of formula 1.3 wherein R ² is hydrogen and R ⁴ methyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 584

Compounds of formula 1.4 wherein R ² is hydrogen and R ⁴ methyl and R ³ for the compound corresponds to one row in Table B.

Table 585 'n

The compounds of formula 1.1, wherein R is hydrogen and R ⁴ ethyl and R ³ for a compound corresponds to one line in Table B.

Table 586

The compounds of formula 1.2, wherein R ² is hydrogen and R ⁴ ethyl and R ³ for a compound corresponds to one line in Table B.

Table 587

The compounds of formula 1.3, wherein R ² is hydrogen

and R ^{4 is} ethyl and the row substituent in Table B. R ³ for the compound corresponds to one Table 588 Compounds of general formula 1.4 R ² is hydrogen and R ^{4 is} ethyl and substituent R ³ for the compound corresponds to one

row in Table B.

143

Table 589 _x o

The compounds of formula 1.1, wherein R is hydrogen and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 590

The compounds of formula 1.2, wherein R ² is hydrogen and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 591

The compounds of formula 1.3, wherein R ² is hydrogen and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 592

The compounds of formula 1.4, wherein R ² is hydrogen and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 593

Compounds of formula 1.1 wherein R ² is hydrogen and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 594

The compounds of formula 1.2, wherein R ² is hydrogen and R isopropyl, and R ^J for a compound corresponds to one line in Table B.

144

Table 595

Compounds of formula 1.3 wherein R ² is hydrogen and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 596

Compounds of formula 1.4 wherein R ² is hydrogen and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 597

Compounds of formula 1.1 wherein R ² is hydrogen and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 598

Compounds of formula X.2 wherein R ² is hydrogen and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 599

Compounds of formula 1.3 wherein R ² is hydrogen and R 2 -methoxyethyl and the substituent R 6 'for the compound corresponds to one row in Table B.

Table 600

The compounds of formula 1.4, wherein R ² is hydrogen and R 2-methoxyethyl and R ^J for a compound corresponds to one line in Table B.

145

Table 601

Compounds of formula 1.1 wherein R ² is hydrogen and R ⁴ prop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 602

Compounds of formula 1.2 wherein R ² is hydrogen and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 603

Compounds of formula 1.3 wherein R ² is hydrogen and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 604

Compounds of formula 1.4 wherein R ² is hydrogen and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 605

Compounds of formula 1.1 wherein R ² is hydrogen and R ⁴ trans-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 606

Compounds of formula 1.2 wherein R ² is hydrogen and R ⁴ trans-3-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

146

Table 607

Compounds of formula 1.3 wherein R ² is hydrogen and R ⁴ trans-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 608

Compounds of formula 1.4 wherein R ² is hydrogen and R ⁴ trans-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 609

Compounds of formula 1.1 wherein R ² is hydrogen and R ⁴ prop-2-ynyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 610

The compounds of formula 1.2, wherein R ² is hydrogen and R ⁴ prop-2-ynyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 611

Compounds of formula 1.3 wherein R ² is hydrogen and R ⁴ prop-2-ynyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 612

Compounds of formula 1.4 wherein R ² is hydrogen and R prop-2-ynyl and the substituent R ^j for the compound corresponds to one row in Table B.

147

Table 613

Compounds of formula 1.1 wherein R is hydrogen and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 614 _Λ 2

Compounds of formula 1.2 wherein R is hydrogen and R ^{3 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 615

Compounds of formula 1.3 wherein R ² is hydrogen and R ^{4 is} 3-iodoprop-2-ynyl and the substituent R ³ for the compound corresponds to one row in Table B. Table 616

Compounds of formula 1.4 wherein R ² is hydrogen and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 617

Compounds of formula a R ⁴ hydrogen and the substituent R ^{3 of the} row in Table B.

I.1, wherein R ² is ethyl for the compound corresponds to one

Table 618

1.2 wherein R ² is ethyl for the compound corresponds to one

Compounds of formula a R ⁴ hydrogen and the substituent R ^{3 of the} row in Table B.

148

Table 619

Compounds of formula and R ⁴ hydrogen and substituent R ^{3 of the} row in Table B.

Table 620

Compounds of formula a R ⁴ hydrogen and the substituent R ^{3 of the} row in Table B.

Table 621

Compounds of formula and R ⁴ methyl and substituent R ^{3 of the} row in Table B.

Table 622

Compounds of formula and R ⁴ methyl and substituent R ^{3 of the} row in Table B.

Table 623

Compounds of formula and R ⁴ methyl and substituent R ^{3 of the} row in Table B.

Table 624

Compounds of formula and R ⁴ methyl and substituent R ^{3 of the} row in Table B.

1.3, wherein R ² represents ethyl for the compound corresponds to one

1.4 wherein R ² represents ethyl for the compound corresponds to one

I.1, wherein R is ethyl for the compound corresponds to one

1.2 wherein R ² is ethyl for the compound corresponds to one

1.3, wherein R ² represents ethyl for the compound corresponds to one

1.4 wherein R ² represents ethyl for the compound corresponds to one

149

Table 625

Compounds of formula and R ⁴ ethyl and substituent R ^{3 of the} row in Table B.

I.1, wherein R ² is ethyl for the compound corresponds to one

Table 626

Compounds of formula and R ⁴ ethyl and substituent R ^{3 of the} row in Table B.

1.2 wherein R ² is ethyl for the compound corresponds to one

Table 627

Compounds of formula and R ⁴ ethyl and substituent R ^{3 of the} row in Table B.

1.3, wherein R ² represents ethyl for the compound corresponds to one

Table 628

Compounds of formula and R ⁴ ethyl and substituent R ^{3 of the} row in Table B.

1.4 wherein R ² represents ethyl for the compound corresponds to one

Table 629

The compounds of formula 1.1, wherein R ² is ethyl fourth * 3 and R n -propyl and the R substituent for the compound corresponds to one row in Table B.

Table 630

The compounds of formula 1.2, wherein R ² is ethyl and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

150

Table 631

The compounds of formula 1.3, wherein R ² is ethyl and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 632

Compounds of formula 1.4 wherein R ² is ethyl and R ^{4 is} n-propyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 633

Compounds of formula 1.1 wherein R ² is ethyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 634

Compounds of formula 1.2 wherein R ² is ethyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 635

Compounds of formula 1.3 wherein R ² is ethyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 636

Compounds of formula 1.4 wherein R ² is ethyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

151

Table 637

Compounds of formula 1.1 wherein R ² is ethyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 638.

Compounds of formula 1.2 wherein R ² is ethyl and R ^{4 is} 2-methoxyethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 639 n

Compounds of formula 1.3 wherein R is ethyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 640

Compounds of formula 1.4 wherein R * ¹ is ethyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 641

Compounds of formula 1.1, in and R ⁴ prop-2-enyl and R ^{3 in} one row in Table B.

whose R ² represents ethyl for the compound corresponds to

Table 642 wherein R ² is ethyl for the compound corresponds

Compounds of general formula 1.2, v

9 and R is prop-2-enyl and R is substituted in one row in Table B.

152

Compounds of formula 1.3, in and R ⁴ prop-2-enyl and R ^{3 in} one row in Table B.

Table 643 wherein R ⁶ represents ethyl for the compound corresponds

Table 644

Compounds of formula 1.4, v and R ⁴ prop-2-enyl and substituent R ^{3 in} one row in Table B.

whose R ² represents ethyl for the compound corresponds to

Table 645

Compounds of formula 1.1 wherein R ² is ethyl and R ⁴ trans-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 646 _x 2 Compounds of formula (1.2) in which R ⁶ is ethyl and R ⁴ trans-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 647

Compounds of formula 1.3 wherein R ² is ethyl and R trans-3-chloroprop-2-enyl and the R substituent for the compound corresponds to one row in Table B.

Table 648

Compounds of formula 1.4 wherein R ² is ethyl and R trans-3-chloroprop-2-enyl and the R substituent for the compound corresponds to one row in Table B.

153

Table 649

Compounds of formula 1.1, in and R ⁴ prop-2-ynyl and R ^{3 in} one row in Table B.

whose R is ethyl for the compound corresponds

Table 650

Compounds of general formula 1.2, and in R ⁴ prop-2-ynyl and substituent R ^{3 in} one row in Table B.

whose R ² represents ethyl for the compound corresponds to

Table 651

Compounds of formula 1.3, in and R ⁴ prop-2-ynyl and substituent R ^{3 in} one row in Table B.

> 9 whose R is ethyl for the compound corresponds

Table 652

Compounds of general formula 1.4, in and R ⁴ prop-2-ynyl and substituent R ^{3 in} one row in Table B.

Wherein R is ethyl for the compound

Table 653

Compounds of formula 1.1 wherein R ² is ethyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 654

The compounds of formula 1.2, wherein R ² is ethyl and R @ 3-iodo-2-ynyl and R ^J for a compound corresponds to one line in Table B.

154

Table 655

Compounds of formula 1.3 wherein R ² is ethyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 656

Compounds of formula 1.4 wherein R ² is ethyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 657

Compounds of formula 1.1 wherein R ² is trifluoromethyl and R ^{4 is} hydrogen and R ³ for the compound corresponds to one row in Table B.

Table 658

Compounds of formula (1.2) wherein R is trifluoromethyl and R ^{4 is} hydrogen and R ³ for the compound corresponds to one row in Table B.

Table 659

Compounds of formula 1.3 wherein R ² is trifluoromethyl and R ^{4 is} hydrogen and R ³ for the compound corresponds to one row in Table B.

Table 660

Compounds of formula 1.4 wherein R ² is trifluoromethyl and R ^{4 is} hydrogen and R ³ for the compound corresponds to one row in Table B.

155

Tabuika 661

The compounds of formula 1.1, wherein R is trifluoromethyl and R ⁴ is methyl and R ³ for a compound corresponds to one line in Table B.

Tabuika 662

Compounds of formula 1.2 wherein R ² is trifluoromethyl and R ⁴ methyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 663

Compounds of formula 1.3 wherein R ² is trifluoromethyl and R ⁴ methyl and R ³ for the compound corresponds to one row in Table B.

Table 664

Compounds of formula 1.4 wherein R ² is trifluoromethyl and R ⁴ methyl and R ³ for the compound corresponds to one row in Table B.

Tabuika 665

Compounds of formula 1.1 wherein R ² is trifluoromethyl and R ⁴ ethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Tabuika 666

Compounds of formula 1.2 wherein R ² is trifluoromethyl and R ⁴ ethyl and the substituent R ³ for the compound corresponds to one row in Table B.

156

Table 667

Compounds of formula 1.3 wherein R ² is trifluoromethyl and R ⁴ ethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 668

Compounds of formula 1.4 wherein R ² is trifluoromethyl and R ⁴ ethyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 669

The compounds of formula 1.1, wherein R ² is trifluoromethyl and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 670

The compounds of formula 1.2, wherein R ² is trifluoromethyl and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 671

The compounds of formula 1.3, wherein R ² is trifluoromethyl and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 672

The compounds of formula 1.4, wherein R ² is trifluoromethyl and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

157

Table 673

Compounds of formula 1.1 wherein R ² is trifluoromethyl and R ⁴ isopropyl and R ³ for the compound corresponds to one row in Table B.

Table 674

Compounds of formula 1.2 wherein R ² is trifluoromethyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 675

Compounds of formula 1.3 wherein R ² is trifluoromethyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 676 n

Compounds of formula 1.4 wherein R is trifluoromethyl and R ⁴ isopropyl and R ³ for the compound corresponds to one row in Table B.

Table 677

Compounds of formula 1.1 wherein R ² is trifluoromethyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 678

Compounds of formula 1.2 wherein R ² is trifluoromethyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

158

Table 679

Compounds of formula 1.3 wherein R ² is trifluoromethyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 680

Compounds of formula 1.4 wherein R ² is trifluoromethyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 681

Compounds of formula 1.1 wherein R ² is trifluoromethyl and R ⁴ prop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 682

Compounds of formula 1.2 wherein R ² is trifluoromethyl and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 683

Compounds of formula 1.3 wherein R ² is trifluoromethyl and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 684

Compounds of formula 1.4 wherein R ² is trifluoromethyl and R ⁴ prop-2-enyl and R ³ for the compound corresponds to one row in Table B.

159

Table 685

Compounds of formula 1.1 wherein R ² is trifluoromethyl and R ⁴ trans -3-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 686

Compounds of formula 1.2 wherein R ² is trifluoromethyl and R ⁴ trans -3-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 687

Compounds of formula (1.3) wherein R is trifluoromethyl and R ⁴ trans-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 688

Compounds of formula 1.4 wherein R ² is trifluoromethyl-1 and R ⁴ trans-3-chloroprop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 689

Compounds of formula 1.1 wherein R ² is trifluoromethyl and R ⁴ prop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 690

Compounds of formula 1.2 wherein R ² is trifluoromethyl and R ⁴ prop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

160

Table 691, 9

Compounds of formula 1.3 wherein R is trifluoromethyl and R ^{4 is} prop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 692

The compounds of formula X.4, wherein R ² is trifluoromethyl and R @ ⁴ prop-2-ynyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 693

Compounds of formula 1.1 wherein R ² is trifluoromethyl and R ⁴ 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 694

Compounds of formula 1.2 wherein R ² is trifluoromethyl and R ⁴ 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 695

Compounds of formula 1.3 wherein R ² is trifluoromethyl and R ⁴ 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 696

Compounds of formula 1.4 wherein R ² is trifluoromethyl and R ⁴ 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

161

Table 697

Compounds of formula 1.1 wherein R ² is cyclopropyl and R ^{4 is} hydrogen and the substituent R ³ for the compound corresponds to one row in Table B.

Table 698

Compounds of formula 1.2 wherein R ² is cyclopropyl and R ^{4 is} hydrogen and R ³ for the compound corresponds to one row in Table B.

Table 699

Compounds of formula 1.3 wherein R ² is cyclopropyl and R ^{4 is} hydrogen and the substituent R ³ for the compound corresponds to one row in Table B.

Table 700

Compounds of formula 1.4 wherein R ⁶ is cyclopropyl and R ^{4 is} hydrogen and R ³ for the compound corresponds to one row in Table B.

Table 701

Compounds of formula 1.1 wherein R ² is cyclopropyl and R ⁴ methyl and R ³ for the compound corresponds to one row in Table B.

Table 702

Compounds of formula 1.2 wherein R ² is cyclopropyl and R ⁴ methyl and R ³ for the compound corresponds to one row in Table B.

162

Table 703

Compounds of formula 1.3 wherein R ² is cyclopropyl and R ⁴ methyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 704

Compounds of formula 1.4 wherein R ² is cyclopropyl and R ⁴ methyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 705

Compounds of formula 1.1 wherein R ² is cyclopropyl and R ⁴ ethyl and R ³ for the compound corresponds to one row in Table B.

Table 706

Compounds of formula 1.2 wherein R ² is cyclopropyl and R ⁴ ethyl and R ³ for the compound corresponds to one row in Table B.

Table 707

The compounds of formula 1.3, wherein R ² is cyclopropyl and R ⁴ ethyl and R ³ for a compound corresponds to one line in Table B.

Table 708

Compounds of formula 1.4 wherein R ² is cyclopropyl and R ethyl and the substituent R ^J for the compound corresponds to one row in Table B.

163

Table 709

The compounds of formula 1.1, wherein R ² is cyclopropyl and R ⁴ of n-propyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 710

Compounds of formula 1.2 wherein R ² is cyclopropyl and R ^{4 is} n-propyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 711

Compounds of formula 1.3 wherein R is cyclopropyl and R ^{4 is} n-propyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 712

Compounds of formula 1.4 wherein R is cyclopropyl and R ^{4 is} n-propyl and R ³ for the compound corresponds to one row in Table B.

Table 713

Compounds of formula 1.1 wherein R ² is cyclopropyl and R ⁴ isopropyl and R ³ for the compound corresponds to one row in Table B.

Table 714

Compounds of formula 1.2 wherein R ² is cyclopropyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

164

Table 715

Compounds of formula 1.3 wherein R ² is cyclopropyl and R ⁴ isopropyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 716

Compounds of formula 1.4 wherein R ² is cyclopropyl and R ⁴ isopropyl and R ³ for the compound corresponds to one row in Table B.

Table 717, o

Compounds of formula 1.1 in which R @ 1 is cyclopropyl and R @ ^{4 is} 2-methoxyethyl and R @ ³ for the compound corresponds to one row in Table B.

Table 718

Compounds of formula 1.2 wherein R ² is cyclopropyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 719

Compounds of formula 1.3 wherein R ² is cyclopropyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

Table 720

Compounds of formula 1.4 wherein R ² is cyclopropyl and R ^{4 is} 2-methoxyethyl and R ³ for the compound corresponds to one row in Table B.

165

Table 721 of

The compounds of formula 1.1, wherein R ^£ is cyclopropyl and R @ ⁴ prop-2-enyl and the substituent ^R3 for a compound corresponds to one line in Table B.

Table 722

Compounds of formula 1.2 wherein R ² is cyclopropyl and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 723

Compounds of formula 1.3 wherein R is cyclopropyl and R ⁴ prop-2-enyl and R ³ for the compound corresponds to one row in Table B.

Table 724 of 9 of

Compounds of formula 1.4 wherein R is cyclopropyl and R ⁴ prop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 725

Compounds of formula 1.1 wherein R ² is cyclopropyl and R ⁴ trans-3-chloroprop-2-enyl and the substituent R ³ for the compound corresponds to one row in Table B.

Table 726

Compounds of formula 1.2 wherein R ² is cyclopropyl and R trans-3-chloroprop-2-enyl and the R substituent for the compound corresponds to one row in Table B.

166 cycloR ³ for

Table 727

Compounds of formula 1.3 wherein R ² is propyl and R ⁴ trans-3-chloroprop-2-enyl and the substituent compound corresponds to one row in Table B.

Table 728

Compounds of formula 1.4 wherein R ² is propyl and R ⁴ trans-3-chloroprop-2-enyl and the substituent compound corresponds to one row in Table B.

Table 729

Compounds of formula 1.1 wherein R ² is propyl and R ^{4 is} prop-2-ynyl and the substituent R ³ for the compound leads to one row in Table B.

Table 730

Compounds of formula 1.2 wherein R ² is propyl and R ^{4 is} prop-2-ynyl and R ³ for the compound leads to one row in Table B.

Table 731

Compounds of formula 1.3 wherein R ² is propyl and R ^{4 is} prop-2-ynyl and R ³ for the compound leads to one row in Table B.

Table 732

Compounds of formula 1.4 wherein R ² is propyl and R ^{4 is} prop-2-ynyl and R ³ for the compound leads to one row in Table B.

CycloR ³ for cyclicconsultingconsultingconsumingconsumingtoor167

Table 733

Compounds of formula 1.1 wherein R ² is cyclopropyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 734

Compounds of formula 1.2 wherein R ² is cyclopropyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 735 _x 2

Compounds of formula 1.3 wherein R is cyclopropyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table 736

Compounds of formula 1.4 wherein R ² is cyclopropyl and R ^{4 is} 3-iodoprop-2-ynyl and R ³ for the compound corresponds to one row in Table B.

Table A

Nr. R 2 R ⁴ | A. 1 ch ₃ h 1 A. 2 ch ₃ ch ₃ 1 A. 3 ch ₃ c ₂ h ₅ A.4 ch ₃ nC ₃ H7 1 A.5 ch ₃ 1-C ₃ H7 A.6 ch ₃ Cyclopropyl 1 A.7 ch ₃ n-C 1 H 8 A.8 ch ₃ S'C ₄ phi I A.9 ch ₃ t-c ₄ h ₉ 1 A.10 ch ₃ tC ₄ Hg | A.11 ch ₃ n CsHii A.12 ch ₃ I-C5HU A.13 ch ₃ neo-CsHn I A.14 ch ₃ Cyclopentyl 1 A.15 ch ₃ nC ₆ H ₁₃ A.16 ch ₃ Cyfclohexyl A.17 ch ₃ n-C 6 H 17 J A.18 ch ₃ CH ₂ CH ₂ C1 j A.19 ch ₃ (CH _{2) 4} C 1 J A.20 ch ₃ ch ₂ cn j A.21 ch ₃ ch ₂ ch ₂ cn J A.22 ch ₃ (CH ₂ ) ₃ CN J A.23 ch ₃ (ch ₂ ) ₄ cn 1 A.24 ch ₃ (CH ₂ ) s CN 1 A.25 ch ₃ Cyclohexylmethyl 1 A.26 ch ₃ 2-Cyferlohexyleth-1-yl A.27 ch ₃ Cyclopropylmethyl I A.28 ch ₃ 2-Cyclopropyl-ethyl-1-yl | A.29 ch ₃ 2-Methoxyeth-1-yl 1 A.30 ch ₃ 2-Ethoxyeth-1-yl A.31 ch ₃ 2-Isopropoxyeth-1-yl A.32 ch ₃ 3-Methoxyprop-1-yl A.33 ch ₃ 3-Ethoxyprop-1-yl | A.34 3H ₃ 3-Isopropoxyprop-1-yl 1 A.35 HH ₃ 4methoxybut-1-yl A.36 3H ₃ 4-Isopropoxy-but-1-yl 1 A.37 3H ₃ Propen-3-yl A.38 ( : h ₃ I 3ut-2-en-1-yl |

 - // / <-

Nr. R ² R ⁴ A.39 ch ₃ 3-methyl-but-2-en-l-yl A.40 ch ₃ 2-Vinyloxyeth-1-yl A.41 ch ₃ Allyloxyeth-1-yl A.42 ch ₃ 2-Trifluormethoxyeth-yl A.43 ch ₃ Trifluormethoxyprop 3-yl A.44 ch ₃ Difluormethoxybut 4-yl A.45 ch ₃ Hydroxycarbonylmethyl A.46 ch ₃ Methoxycarbonylmethyl A.47 ch ₃ Aminocarbonylmethyl A. 48 ch ₃ N-Methylaminocarbonylmethyl A.49 ch ₃ Ν, Ν-Dimethylaminocarbonyl-methyl A.50 ch ₃ 2-Hydroxycarbonyleth-1-yl A.51 ch ₃ 2-Methoxycarbonyleth-1-yl A.52 ch ₃ 2-Aminocarbonyleth-yl A. 53 ch ₃ 2-N-Methylaminocarbonyleth-1-yl A. 54 ch ₃ 2-Dimethylaminocarbonyleth-1-yl A.55 ch ₃ 2-aminoethyl-1-yl A. 56 ch ₃ 2-Aminoprop-1-yl A. 57 ch ₃ 4-amino-but-1-yl A.58 ch ₃ 3-dimethylaminopropyl-l-yl A. 59 ch ₃ 4-Aminothiocarbonylbut-1-yl A.60 ch ₃ 2-oxo-propyl A.61 ch ₃ cyclohexyl .62 ch ₃ cyclopropyl .63 ch ₃ cyclopentyl A.64 ch ₃ 2-Methoxyiminoprop-1-yl A.65 ch ₃ 2-Methoxyiminoeth-1-yl A.66 ch ₃ 6-Aminocarbonylhex-1-yl A.67 ch ₃ 3-Aminothiocarbonylprop-1-yl A.68 ch ₃ 2-Aminothiocarbonyleth-1-yl A.69 ch ₃ Aminothiocarbonylmethyl A.70 ch ₃ 4- (N, N-dimethylamino) but-l-yl A. 71 ch ₃ 2- (Methylthio) eth-l-yl A.72 ch ₃ 2- (methylsulfonyl) eth-l-yl A. 73 ch ₃ 4- (Methylthio) prop-l-yl A. 74 ch ₃ 4- (methylsulfonyl) prop-1-yl A.75 ch ₃ benzyl A.76 2H ₃ 2-FC ₆ H ₄ -CH ₂ A. 77 : h ₃ ifc ₆ h ₄ -ch ₂

Y -

Nr. R 2 R ⁴ A.78 ch ₃ 4-FC ₆ H ₄ -CH ₂ A.79 ch ₃ 2,3-F ₂ -CfiHa-CH ₂ A. 80 ch ₃ 2,4-F ₂ -C ₆ H 3 -CH ₂ A. 81 ch ₃ 2,5-F ₂ -C ₆ H ₃ -CH ₂ A.82 ch ₃ 2,6-F ₂ -C ₆ H 3 -CH ₂ A. 83 ch ₃ 3,4-F ₂ -C ₆ H ₃ -CH ₂ A.84 ch ₃ . 3,5-F ₂ -C ₆ H ₃ -CH ₂ A.85 ch ₃ 2-C 1 -C ₆ H ₄ -CH ₂ A. 86 ch ₃ 3-Cl-C ₅ H ₄ -CH ₂ A.87 ch ₃ 4-C1-C ₆ H ₄ CH ₂ A.88 ch ₃ 2,3-Cl ₂ -C ₆ H ₃ -CH ₂ A.89 ch ₃ 2,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.90 ch ₃ 2,5-Cl ₂ -C ₆ H 3 -CH 2 A.91 ch ₃ 2,6-Cl ₂ -C ₆ H ₃ -CH ₂ A.92 ch ₃ 3,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.93 ch ₃ 3,5-Cl ₂ -C ₆ H ₃ -CH ₂ A.94 ch ₃ 2,3,4 -Cl ₃ -C ₆ H ₂ -CH ₂ A.95 ch ₃ 2,3,5-C 1 -C ₃ -C ₆ H ₂ -CH ₂ A.96 ch ₃ 2,3,6-Cl ₃ -C ₆ H ₂ -CH ₂ A.97 ch ₃ 2,4,5 -Cl ₃ -C ₆ H ₂ -CH ₂ A.98 ch ₃ 2,4,6-Cl ₃ -C 1 H ₂ -CH ₂ A.99 ch ₃ 3,4,5 -Cl ₃ -C ₆ H ₂ -CH ₂ A.100 ch ₃ 2-Br-C ₆ H ₄ CH ₂ A.101 ch ₃ 3 -Br, -C ₆ H ₄ -CH ₂ A.102 ch ₃ 4 -Br-C ₆ H ₄ CH ₂ A.103 ch ₃ 2,3-Br ₂ -C ₆ H ₃ -CH ₂ A.104 ch ₃ 2,4-Br ₂ -C ₆ H ₃ -CH ₂ A.105 ch ₃ 2,5-Br ₂ -C ₆ H ₃ -CH ₂ A, 106 ch ₃ 2,6 -Br ₂ -C ₆ H ₃ -CH ₂ A.107 ch ₃ 3,4-Br ₂ -C ₆ H ₃ -CH ₂ A.108 ch ₃ 3,5-Br ₂ -C ₆ H ₃ -CH ₂ A.109 ch ₃ 2-F, 3-C 1-C ₆ H ₃ CH ₂ A.110 ch ₃ 2-F, 4-C 1 -C ₅ H ₃ -CH ₂ A.111 ch ₃ 2-F, 5-C 1-C ₆ H ₃ CH ₂ A.112 SRŠ 2-F, 3-Br-C ₆ H ₃ CH ₂ A.113 HH ₃ 2-F, 4-Br-C ₆ H ₃ CH ₂ A.114 : h ₃ 2-F, 5-Br-C ₆ H ₃ CH ₂ A.115 : h ₃ 2-C1, 3-Br-C ₆ H ₃ CH ₂ MSC.116 : h ₃ 2-C1, 4-Br-C ₆ H ₃ CH ₂

[

Nr. R ² R ⁴ A.117 ch ₃ 2-C1, 5-Br-C ₆ H ₃ CH ₂ A.118 ch ₃ 3-F, 4-C1-C ₆ H ₃ CH ₂ A.119 ch ₃ 3-F, 5-C 1-C ₆ H ₃ CH ₂ A.120 ch ₃ 3-F, 6-Cl-C ₆ H ₃ CH ₂ A.121 ch ₃ 3-F, 4-Br-C ₆ H ₃ CH ₂ A.122 ch ₃ 3-F, 5-Br-C ₆ H ₃ CH ₂ A. 123 ch ₃ 3-F, 6-Br-C ₆ H ₃ CH ₂ A.124 ch ₃ 3-C1, 4-Br-C ₆ H ₃ CH ₂ A.125 ch ₃ 3-C1, 5-Br-C ₆ H ₃ CH ₂ A.126 ch ₃ 3-C1, 6-Br-C ₆ H ₃ CH ₂ A.127 ch ₃ 4-F, 5-C 1-C ₆ H ₃ CH ₂ A.128 ch ₃ 4-F, 6-C1-C ₆ H ₃ CH ₂ A.129 ch ₃ 4-F, 5-Br-C ₆ H ₃ CH ₂ A.130 ch ₃ 4-F, 6-Br-C ₆ H ₃ CH ₂ A.131 ch ₃ 4-C1, 5-Br-C ₆ H ₃ CH ₂ A.132 ch ₃ 5-F, 6-C1-C ₆ H ₃ CH ₂ A.133 ch ₃ 5-F, 6-Br-C ₆ H ₃ CH ₂ A.134 ch ₃ 5-C1, 6-Br-C ₆ H ₃ CH ₂ A.135 ch ₃ 3-Br, 4-C1, 5-Br-C ₆ H ₂ CH ₂ A.136 ch ₃ 2 -CN-C ₆ H ₄ -CH ₂ A.137 ch ₃ 3 -CN -C ₆ H ₄ -CH ₂ A.138 ch ₃ 4 -CN-C ₆ H ₄ -CH ₂ A.139 ch ₃ 2-NO ₂ -C ₆ H ₄ -CH ₂ A.140 ch ₃ 3-NO ₂ -C ₆ H ₄ -CH ₂ A.141 ch ₃ 4-NO ₂ -C ₆ H ₄ -CH ₂ A.142 ch ₃ 2-CH ₃ -C ₆ H ₄ -CH ₂ A.143 ch ₃ 3-CH ₃ -C ₆ H ₄ -CH ₂ A.144 ch ₃ 4-CH ₃ -C ₆ H ₄ -CH ₂ A.145 ch ₃ 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.146 ch ₃ 2,4- (CH ₃ ) ₂ -C ₈ H ₃ -CH ₂ A.147 ch ₃ 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.148 ch ₃ 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.149 ch ₃ 3,4- (CH ₃ ) ₂ -C ₆ H 3 -CH ₂ A.150 ch ₃ 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.151 ch ₃ 2-C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.152 ch ₃ 3-C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.153 ch ₃ ic ₂ h ₅ -c ₆ h ₄ -ch ₂ A.154 ch ₃ 2- i -C ₃ H ₇ -C ₆ H ₄ -CH ₂ A.155 ch ₃ i -i -c ₃ h ₇ -c ₆ h ₄ -ch ₂

// ť • T ŕ-

Nr. R ² R ⁴ A. 156 ch ₃ 4-C ₃ H ₇ -C ₆ H ₄ -CH ₂ A.157 ch _{3 2-Cyclohexyl-C6H4-CH2} A.158 ch ₃ 3-Cyclohexyl-C6H4-CH2 A. 159 ch ₃ 4-Cyclohexyl-C6H4-CH2 A.160 ch ₃ 2-Vinyl -C ₆ H ₄ -CH ₂ A.161 ch ₃ 3-vinyl-C ₆ H ₄ CH ₂ A. 162 ch ₃ 4-vinyl-CH2-C6ÍÍ4 A. 163 ch ₃ 2-Allyl-C ₆ H ₄ -CH ₂ A. 164 ch ₃ 3-Allyl-C ₆ H ₄ CH ₂ A. 165 ch ₃ 4-Allyl-C ₆ H ₄ CH ₂ A.166 ch ₃ 2-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.167 ch ₃ 3-C ₆ H ₅ -C ₆ H 4 -CH ₂ A.168 ch ₃ 4-C ₆ H ₅ -C ₆ H 4 -CH ₂ A. 169 ch ₃ 3-CH ₃ , 5 -1-C 4 H 9 -C ₆ H ₃ -CH ₂ A. 170 ch ₃ 2-OH-C ₆ H 4 -CH ₂ A.171 ch ₃ 3-OH-C ₆ H 4 -CH ₂ A. 172 ch ₃ 4-OH-C ₆ H 4 -CH ₂ A. 173 ch ₃ 2-OCH ₃ -C ₆ H 4 -CH ₂ A.174 ch ₃ 3-OCH ₃ -C ₆ H ₄ -CH ₂ A. 175 ch ₃ 4-OCH ₃ -C ₆ H 4 -CH ₂ A. 176 ch ₃ 2,3- (OCH ₃ , ₂ -C ₆ H ₃ -CH ₂₎ A. 177 ch ₃ 2,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.178 ch ₃ 2,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A. 179 ch ₃ 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.180 ch ₃ 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A. 181 ch ₃ 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH ₂ A. 182 ch ₃ 2-OC 2 H 5 -C ₆ H ₄ -CH ₂ A.183 ch ₃ 3 -OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.184 ch ₃ 4 -OC ₂ H _S -C ₆ H ₄ -CH ₂ A.185 ch ₃ 2-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.186 ch ₃ 3-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.187 ch ₃ 4-O- (nC ₃ H ₇ ) -C ₆ H 4 -CH ₂ A.188 ch ₃ 2-O- (iC ₃ H ₇ ) -C ₆ H 4 -CH ₂ A.189 ch ₃ 3-O- (iC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.190 CH ₃ 4-O- (iC ₃ H ₇ ) -C ₆ H 4 -CH ₂ A.191 zh ₃ 4-O- (nC ₄ H ₉ ) -C ₆ H 4 -CH ₂ A.192 ľh ₃ 3-O- (t C ₄ H ₉ ) -C ₆ H ₄ -CH ₂ A.193 HH ₃ 1-O- (nC ₆ H ₁₃ ) -C ₆ H ₄ -CH ₂ A.194 : h ₃ 2-Ο-Allyl-C ₆ H ₄ -CH ₂

-m-

Nr. R ² R ⁴ A.195 ch ₃ 3-O-allyl-C ₆ H ₄ CH ₂ A.196 ch ₃ 4-O-allyl-C ₆ H ₄ CH ₂ A.197 ch ₃ 2-CF ₃ -C ₆ H ₄ -CH ₂ A.198 ch ₃ 3-CF ₃ -C ₆ H ₄ -CH ₂ A.199 ch ₃ 4-CF ₃ -C ₆ H ₄ -CH ₂ A.200 ch ₃ 2 - Ace tulle - CgH ₄ - (¾ A.201 ch ₃ 3-Acetyl-C ₆ H ₄ CH ₂ A.202 ch ₃ 4 - acetyl - ₄ CGH - _CH2 A.203 ch ₃ 2-Methoxycarbonyl-C 8 H ₄ -CH ₂ A.204 ch ₃ 3-Methoxycarbonyl-C 8 H ₄ -CH ₂ A.205 ch ₃ Methoxycarbonyl-4-C ₆ H ₄ CH ₂ A.206 ch ₃ 2-Aminocarbonyl-C 8 H ₄ -CH ₂ A.207 ch ₃ 3-aminocarbonyl-C ₆ H ₄ CH ₂ A.208 ch _{3 4-aminocarbonyl-4 -CH2} CGH A.209 ch ₃ 2-Dimethylaminocarbonyl-C 8 H ₄ -CH ₂ A.210 ch ₃ 3-DimethylaminocarbonylCgH ₄ -CH ₂ A.211 ch ₃ 4 - CGH _{Dimethylaminocarbonyl-4-CH 2} A.212 ch ₃ 2- (N-Methylaminocarbonyl) -C ₆ H ₄ -CH ₂ A.213 ch ₃ 3- (N-Methylaminocarbonyl) -C ₈ H ₄ -CH ₂ A.214 ch ₃ 4- (N-Methylaminocarbonyl) -C ₈ H ₄ -CH ₂ A.215 ch ₃ 2-H ₂ N-C 8 H ₄ -CH ₂ A.216 ch ₃ 3-H ₂ NC ₆ H ₄ -CH ₂ A.217 ch ₃ 4-H ₂ NC ₆ H ₄ -CH ₂ A.218 ch ₃ 2-Amino thiocarbonyl -C ₈ H ₄ -CH ₂ A.219 ch ₃ 3-Aminothiocarbonyl -C ₈ H ₄ -CH ₂ A.220 ch ₃ 4-Aminothiocarbonyl -C ₈ H ₄ -CH ₂ A.221 ch ₃ 2-C 6 H ₄ -Methoxyiminomethyl _CH2 A.222 ch _{3 3-methoxyimino-methyl-4-CH 2} CGH A.223 ch _{3 4-methoxyimino-methyl-4-CH 2} CGH A.224 ch ₃ 2 - Forms 1 - C 8 H ₄ - CH ₂ A.225 ch ₃ 3 - _{formyl-4 -CH2} CGH A.226 ch ₃ 4 - Forms 1 - Cg H ₄ - CH ₂ A.227 ch ₃ 2- (1'-Methoxyiminoeth-1'-yl) -C ₈ H ₄ -CH ₂ A.228 ch ₃ 3 - (1 '-Methoxyiminoe th -1' - yl) - ₄ CGH - _CH2 A.229 ch ₃ 4- (1'-Methoxyiminoeth-1'-yl) -C ₈ H ₄ -CH ₂ A.230 ch ₃ 2-SCH ₃ -C ₆ H ₄ -CH ₂ A.231 2H ₃ 3-SCH ₃ -C ₆ H ₄ -CH ₂ A.232 HH ₃ 4-SCH ₃ -C ₈ H ₄ -CH ₂ A.233 : h ₃ 2-SO ₂ CH ₃ -C ₈ H ₄ -CH ₂

'rťt-

Nr. R ² R4 A. 234 ch ₃ 3-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ A.235 ch ₃ 4 · SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ A. 236 ch ₃ 2-OCF ₃ -C ₆ H ₄ -CH ₂ A.237 ch ₃ 3-OCF ₃ -C ₆ H ₄ -CH ₂ A.238 ch ₃ 4-OCF ₃ -C ₆ H ₄ -CH ₂ A.239 ch ₃ 2-OCHF ₂ -C ₆ H ₄ -CH ₂ A.240 ch ₃ 3-OCHF ₂ -C ₆ H ₄ -CH ₂ A. 241 ch ₃ 4OCHF ₂ -C ₆ H ₄ -CH ₂ A. 242 ch ₃ 3-CF ₃ , 4-OCF ₃ -C ₆ H ₃ -CH ₂ A. 243 ch _{3 1-Naphthyl-CH2} A. 244 ch _{3 2-Naphthyl-CH2} A.245 ch ₃ 2-Phenoxy-th-1-yl A.246 ch ₃ 2- (2 * -Chlorphenoxy) eth-l-yl A.247 ch ₃ 2- (3'-Chlorphenoxy) eth-l-yl A.248 ch ₃ 2- (4'-Chlorphenoxy) eth-1-yl A.249 ch ₃ 2- (3 ', 5'-Dichlorphenoxy) eth-1-yl A.250 ch ₃ 2- (2'-Cyanophenoxy) eth-1-yl A.251 ch ₃ 2- (3'-Cyanophenoxy) eth-l-yl A.252 ch ₃ 2- (4'-Cyanophenoxy) eth-1-yl A.253 ch ₃ 2- (2'-methylphenoxy) eth-1-yl A.254 ch ₃ 2- (3'-methylphenoxy) eth-l-yl A.255 ch ₃ 2- (4'-methylphenoxy) eth-l-yl A.256 ch ₃ 2- (3'-t-Butylphenoxy) eth-l-yl A.257 ch ₃ 2- (4'-t-Butylphenoxy) eth-1-yl A.258 ch ₃ 2- (2'-Nitrophenoxy) eth-1-yl A.259 ch ₃ 2- (3'-Nitrophenoxy) eth-1-yl A.260 ch ₃ 2- (4'-Nitrophenoxy) eth-l-yl A.261 ch ₃ 2- (2-methoxyphenoxy) eth-1-yl A.262 ch ₃ 2- (3'-methoxyphenoxy) eth-l-yl A.263 ch ₃ 2- (4'-methoxyphenoxy) eth-l-yl A.264 ch ₃ 2- (2 ' Trifluormethylphenoxy) eth-l-yl A.265 ch ₃ 2- (3'-Trifluoromethylphenoxy) eth-1-yl A. 266 ch ₃ 2- (4'-Trifluoromethylphenoxy) eth-1-yl A.267 ch ₃ 2- (2'-Acetylphenoxy) eth-l-yl A.268 CH ₃ 2- (3'-Acetylphenoxy) eth-1-yl A.269 HH ₃ 2- (4'-Acetylphenoxy) eth-1-yl A.270 HH ₃ 2- (2'-methoxycarbonyl) eth-l-yl A.271 : h ₃ 2- (3'-methoxycarbonyl) eth-l-yl A.272 : h ₃ 2- (4'-methoxycarbonyl) eth-l-yl

W-

Nr. R 2 R ⁴ A.273 ch ₃ 2- (2'-Dimethylaminocarbonyl) eth-1-yl A.274 ch ₃ 2- (3'-Dimethylaminocarbonyl) eth-1-yl A.275 ch ₃ 2- (4'-Dimethylaminocarbonyl) eth-1-yl A.276 ch ₃ 2- (2-Aminothiocarbonyl) eth-l-yl A.277 ch ₃ 2- (3'-Aminothiocarbonyl) eth-1-yl A.278 ch ₃ 2- (4'-Aminothiocarbonyl) eth-1-yl A.279 ch ₃ 2- (2'-Methylsulfonyl) eth-1-yl A.280 ch ₃ 2- (3'-Methylsulfonyl) eth-1-yl A.281 ch ₃ 2- (4'-Methylsulfonyl) eth-1-yl; A.282 ch ₃ 3-Phenoxyprop-1-yl A.283 ch ₃ 3- (2'-Chloro-phenoxy) -prop-1-yl A.284 ch ₃ 3- (3'-Chloro-phenoxy) -prop-1-yl A.285 ch ₃ 3- (4'-Chlorphenoxy) prop-1-yl A.286 ch ₃ 3- (3 ', 5', Dichlorphenoxy) prop-1-yl A.287 ch ₃ 3- (2'-Cyanophenoxy) prop-1-yl A.288 ch ₃ 3- (3'-Cyanophenoxy) prop-1-yl A.289 ch ₃ 3- (4'-Cyanophenoxy) prop-1-yl A.290 ch ₃ 3- (2'-Methylphenoxy) prop-1-yl A.291 ch ₃ 3- (3'-Methylphenoxy) prop-1-yl; A.292 ch ₃ 3- (4'-Methylphenoxy) prop-1-yl A.293 ch ₃ 3- (2'-Methoxyphenoxy) prop-1-yl A.294 ch ₃ 3- (3'-Methoxyphenoxy) prop-1-yl A.295 ch ₃ 3- (4'-Methoxyphenoxy) prop-1-yl A.296 ch ₃ 3- (2-Trifluormethylphenoxy) prop-1-yl A.297 ch ₃ 3- (3'-Trifluoromethylphenoxy) prop-1-yl; A.298 ch ₃ 3- (4'-Trifluoromethylphenoxy) prop-1-yl A.299 ch ₃ 4-Phenoxybut-1-yl A.300 ch ₃ 2-Phenyleth-1-yl i A.301 ch ₃ 2- (2'-Chlorophenyl) eth-1-yl A.302 ch ₃ 2- {3'-Chlorphenyl) eth-l-yl A.303 ch ₃ 2- (4'-Chlorphenyl) eth-1-yl A.304 ch ₃ 2- (3 ', 5'-Dichlorophenyl) eth-1-yl' A.305 ch ₃ 2- (2'-cyanophenyl) eth-1-yl A.306 2H ₃ 2- (3'-cyanophenyl) eth-l-yl A.307 2H ₃ 2- (4'-Cyanophenyl) eth-1-yl A.308 2H ₃ 2- (2'-Methylphenyl) eth-l-yl A.309 : h ₃ 2- (3'-Methylphenyl) eth-l-yl A.310 < : h ₃ 2- (4'-Methylphenyl) eth-1-yl A.311 ( : h ₃ 2- (2'-Methoxyphenyl) eth-1-yl

ΊΊ-i-

Nr. R ² R ⁴ A.312 ch ₃ 2- (3'-Methoxyphenyl) eth-1-yl A.313 ch ₃ 2- (4'-Methoxyphenyl) eth-1-yl A.314 ch ₃ 2- (2'-Trifluoromethylphenyl) eth-1-yl A.315 ch ₃ 2- (3 ' Trifluormethylphenyl) eth-1-yl A.316 ch ₃ 2- (4'-Trifluormethylphenyl) eth-1-yl A.317 ch ₃ 3-Phenylprop-1-yl A.318 ch ₃ 3- (2'-Chlorophenyl-prop-1-yl) A.319 ch ₃ 3- (3'-Chlorophenyl-prop-1-yl) A.320 ch ₃ 3- (4'-Chlorophenyl-prop-1-yl) A.321 ch ₃ 3- (2'-Cyanophenyl) prop-1-yl A.322 ch ₃ 3- (3'-Cyanophenyl) prop-1-yl A.323 ch ₃ 3- (4'-Cyanophenyl) prop-1-yl A.324 ch ₃ 3- (2-Trifluormethylphenyl) prop-1-yl A.325 ch ₃ 4-Phenylbut-1-yl A.326 ch ₃ 4- (4'-Chlorphenyl) but-l-yl A.327 ch ₃ 6- (4'-Chlorphenyl) hex-1-yl A.328 ch ₃ 2 -Pyridylmethyl A.329 ch ₃ 3 -Pyridylmethyl A.330 ch ₃ 4-pyridylmethyl A.331 ch ₃ 4-Chloro-pyridin-2-ylmethyl A.332 ch ₃ 5-Chloro-pyridin-2-ylmethyl A.333 ch ₃ 6-Chloropyridin-2-ylmethyl A.334 ch ₃ 5-Chloropyridin-3-ylmethyl A.335 ch ₃ 6-Chloro-pyridin-3-ylmethyl A.336 ch ₃ 2-Chloropyridin-4-ylmethyl A.337 ch ₃ 2 -Pyrimidinylmethyl A.338 ch ₃ 4-Chloro-pyrimidin-2-ylmethyl A.339 ch ₃ 5-Chloro-pyrimidin-2-ylmethyl A.340 ch ₃ 2-Chloro-pyrimidin-4-ylmethyl A.341 ch ₃ 6-Chloro-pyrimidin-4-ylmethyl A.342 ch ₃ 2-Chloro-pyrimidin-5-ylmethyl A.343 ch ₃ 4-Pyridazinylmethyl A.344 ch ₃ 2 -Pyrazinylmethyl A.345 ch ₃ 5-Chloro-pyrazin-2-ylmethyl A.346 ch ₃ S-Chloro-pyrazin-2-ylmethyl A.347 ch ₃ 3-Pyridazinylmethyl A.348 ch ₃ 5-chloropyridazine-3-ylmethyl A.349 7H ₃ 1,3,5-Triazinylmethyl A.350 : h ₃ 2-furylmethyl

'Ή / -

Nr. R ² R ⁴ A.351 ch ₃ 3-furylmethyl A.352 ch ₃ 4-bromofuro-2-ylmethyl A.353 ch ₃ 5-Chlorofur-2-ylmethyl A.354 ch ₃ 2-thienylmethyl A.355 ch ₃ 3-thienylmethyl A.356 ch ₃ 5-methyl-thien-3-ylmethyl A.357 ch ₃ 5-Chlorothien-2-ylmethyl A.358 ch ₃ 2-Chlorothien-4-ylmethyl A.359 ch ₃ 2-pyrrolylmethyl A.360 ch ₃ 3-pyrrolylmethyl A.361 ch ₃ 2-oxazolylmethyl A.362 ch ₃ 4-Methyl-oxazol-2-ylmethyl A.363 ch ₃ 5-Methyl-oxazol-2-ylmethyl A.364 ch ₃ 4-Chlorooxazol-2-ylmethyl A.365 ch ₃ 5-chlorooxazole-2-ylmethyl A.366 ch ₃ 4-Oxazolylmethyl A.367 ch ₃ 2-Methyloxazol-4-ylmethyl A.368 ch ₃ 5-Methyl-oxazol-4-ylmethyl A.369 ch ₃ 2-Chlorooxazol-4-ylmethyl A.370 ch ₃ 5-Chlorooxazol-4-ylmethyl A.371 ch ₃ 5-Oxazolylmethyl A. 372 ch ₃ 2-Methyloxazol-5-ylmethyl A.373 ch ₃ 4-Methyl-oxazol-5-ylmethyl A.374 ch ₃ 2-chlorooxazole-5-ylmethyl A.375 ch ₃ 4-Chlorooxazol-5-ylmethyl A.376 ch ₃ 2-thiazolylmethyl A.377 ch ₃ 4-Methyl-thiazol-2-ylmethyl A.378 ch ₃ 5-Methylthiazol-2-ylmethyl A.379 ch ₃ 4-Chloro-thiazol-2-ylmethyl A.380 ch ₃ 5-Chlorothiazol-2-ylmethyl A.381 ch ₃ 4-thiazolylmethyl A.382 ch ₃ 2-Methylthiazol-4-ylmethyl A.383 ch ₃ 5-Methylthiazol-4-ylmethyl A.384 ch ₃ 2-Chlorothiazol-4-ylmethyl A.385 ch ₃ 5-Chloro-thiazol-4-ylmethyl A.386 ch ₃ 5thiazolylmethyl A.387 7H ₃ 2-Methyl-thiazol-5-ylmethyl A.388 2H ₃ 4-Methylthiazol-5-ylmethyl A.389 2H ₃ 2-Chlorothiazol-5-ylmethyl

r ‘Γ (Γ ')

Nr. R ² R ⁴ 1 A.390 ch ₃ 4-Chlorothiazol-5-ylmethyl | A.391 ch ₃ 3-Isoxazolylmethyl | A.392 ch ₃ 4-Methylisoxazol-3-ylmethyl J A.393 ch ₃ 5-Methylisoxazol-3-ylmethyl | A.394 ch ₃ 4-Chloroisoxazol-3-ylmethyl j A.395 ch ₃ 5-Chloroisoxazol-3-ylmethyl A.396 ch ₃ 4-Isoxazolylmethyl J A.397 ch ₃ 3-Methylisoxazol-4-ylmethyl 1 A.398 ch ₃ 5-Methylisoxazol-4-ylmethyl 1 A.399 ch ₃ 3-Chloroisoxazol-4-ylmethyl | A.400 ch ₃ 5-Chloroisoxazol-4-ylmethyl 1 A.401 ch ₃ 5-Isoxazolylmethyl 1 A.402 ch ₃ 3-Methylisoxazol-5-ylmethyl 1 A.403 ch ₃ 4-Methylisoxazol-5-ylmethyl 1 A.404 ch ₃ 3-Chloroisoxazol-5-ylmethyl 1 A.405 ch ₃ 4-Chloroisoxazol-5-ylmethyl 1 A.406 ch ₃ 3-Isothiazolylmethyl 1 A.407 ch ₃ 4-Methylisothiazol-3-ylmethyl 1 A.408 ch ₃ 5-Methylisothiazol-3-ylmethyl 1 A.409 ch ₃ 4-Chloroisothiazol-3-ylmethyl A.410 ch ₃ 5-Chlorisothiazol-3-ylmethyl A.411 ch ₃ 4-Isothiazolylmethyl 1 A.412 ch ₃ 3-Methylisothiazol-4-ylmethyl 1 A.413 ch ₃ 5-Methylisothiazol-4-ylmethyl 1 A.414 ch ₃ 3-Chloroisothiazol-4-ylmethyl A.415 ch ₃ 5-Chloroisothiazol-4-ylmethyl 1 A.416 ch ₃ 5 - Isothiazolylmethyl A.417 ch ₃ 3-Methylisothiazol-5-ylmethyl A.418 Cfí ₃ 4-Methylisothiazol-5-ylmethyl A.419 ch ₃ 3-Chlorisothiazol-5-ylmethyl A.420 ch ₃ 4-Chloroisothiazol-5-ylmethyl A.421 ch ₃ 4-Imidazolylmethyl 1 A.422 ch ₃ 1-Phenylpyrazol-3-ylmethyl A.423 ch ₃ 1-Methylimidazol-4-ylmethyl 1 A.424 ch ₃ 1-Phenyl-1,2,4-triazol-3-ylmethyl | A.425 ch ₃ 1,2,4-Oxadiazol-3-ylmethyl A.426 CH ₃ 3-chloro-1,2,4-oxadiazol-3-ylmethyl A.427 2H ₃ 5-Methyl-1,2,4-oxadiazol-3-ylmethyl A.428 HH ₃ j-Trifluoromethyl-1,2,4-oxadiazol-3-ylmethyl

Nr. R ² R ⁴ A.429 ch ₃ 1,3,4-oxadiazol-2-ylmethyl A.430 ch ₃ 5-chloro-1,3,4-oxadiazol-2-ylmethyl A.431 ch ₃ 5-Methyl-1,3,4-oxadiazol-2-ylmethyl A.432 ch ₃ 5-Methoxy-l, 3,4-oxadiazol-2-ylmethyl A. 433 ch ₃ 1,2,4-thiadiazol-3-ylmethyl A.434 čh ₃ 5-chloro-1,2,4-thiadiazol-3-ylmethyl A.435 ch ₃ 5-Methyl-1,2,4-thiadiazol-3-ylmethyl A.436 ch ₃ 1,3,4-thiadiazol-2-ylmethyl A.437 ch ₃ 5-chloro-1,3,4-thiadiazol-2-ylmethyl A.438 ch ₃ 5-methyl-1,3,4-thiadiazol-2-ylmethyl A.439 ch ₃ 5-Cyano-1,3,4-thiadiazol-2-ylmethyl A.440 ch ₃ 2- (2'-Pyridinyloxy) eth-1-yl A.441 ch ₃ 2- (3'-Pyridinyloxy) eth-1-yl A.442 ch ₃ 2- (4'-Pyridinyloxy) eth-1-yl A.443 ch ₃ 2- (2'-Pyrimidinyloxy) eth-1-yl A.444 ch ₃ 2- (4'-Pyrimidinyloxy) eth-1-yl A.445 ch ₃ 2- (5'-Pyrimidinyloxy) eth-1-yl A.446 ch ₃ 2- (2'-Pyrazinyloxy) eth-1-yl A.447 ch ₃ 2- (2'-Pyridazinyloxy) eth-1-yl A.448 ch ₃ 2- (3'-pyridazinyloxy) eth-1-yl A.449 ch ₃ 2- (1 ', 3', 5'-Triazinyloxy) eth-1-yl A.450 ch ₃ 2- (5'-Methylisoxazol-3'-yloxy) eth-1-yl A.451 ch ₃ 2- (5'-Chloroisoxazol-3'-yloxy) eth-1-yl A.452 ch ₃ 2- (2-methoxythiazole-4-yloxy) eth-1-yl A.453 ch ₃ 2- (4'-chlorooxazole-2-yloxy) eth-l-yl A.454 ch ₃ 2- (1'-Phenyl-1'H-1 ', 2' _of 4'-triazol-3'-yloxy) eth-1-yl A.455 ch ₃ 2- (1'-Phenylpyrazol-3'-yloxy) eth-1-yl A.456 ch ₃ C ₆ h ₅ A.457 ch ₃ 2-Cl-C ₆ H ₄ A.458 ch ₃ 3-Cl-C ₆ H ₄ A.459 ch ₃ 4-Cl-C ₆ H ₄ A.460 ch ₃ 2.3 -C 1 -C ₂ -C 6 H ₃ A.461 ch ₃ 2,4-Cl ₂ -C ₆ H ₃ A.462 ch ₃ 2,5-Cl ₂ -C ₆ H ₃ A. 463 ch ₃ 3,4-Cl ₂ -C ₆ H ₃ A. 464 ch ₃ 3,5-Cl ₂ -C ₆ H ₃ A. 465 ch ₃ and-CN-C ₆ H ₄ A.466 HH ₃ 2-NO ₂ -C ₆ H ₄

^ 0-

Nr. R ² R ⁴ 1 A.467 ch ₃ 3-NO 2 * C 8 H 4 J A.468 ch ₃ 4-no ₂ -c6h ₄ 1 A.469 ch ₃ 2,4- (NO ₂ ) 2 -C ₆ H 3 1 A.470 ch ₃ 2-CH ₃ -C ₆ H ₄ I A.471 ch ₃ 3-CH ₃ -C ₆ H ₄ A.472 ch ₃ 4-CH ₃ -C ₆ H ₄ 1 A.473 ch ₃ 2,3- (CH ₃ ) ₂ -C ₆ H ₃ I A.474 ch ₃ 2,4 - (CH ₃ ) 2 * C ₆ H ₃ 1 A.475 ch ₃ 2,5- (CH ₃ ) ₂ -C ₆ H ₃ 1 A.476 ch ₃ 2,6- (CH ₃ ) ₂ -C ₆ H ₃ J A.477 ch ₃ 2-C6H5-C6H4J A.478 ch ₃ 3-C ₆ H ₅ -C ₆ H ₄ j A.479 ch ₃ 4-C ₆ H ₅ -C ₆ H ₄ j A.480 ch ₃ 3-OCH ₃ -C ₆ H ₄ J A.481 ch ₃ 4-OCH ₃ -C ₆ H ₄ j A.482 ch ₃ 3-Acetyl-C ₆ H ₄ J A.483 ch ₃ 4-Acetyl-C 6 H ₄ S A.484 ch ₃ 3-methoxycarbonyl-1 C 6 H ₄ A.485 ch _{3 4-methoxycarbonyl-4} CEH J A.486 ch ₃ 3-CF ₃ -C ₆ H ₄ 1 A.487 ch ₃ 4-CF ₃ -C ₆ H ₄ 1 A.488 ch ₃ 2-Naphthyl | A.489 ch ₃ 6-Chloropyridazin-3-yl f A.490 ch ₃ 5-Chloro-pyrazin-2-yl A.491 ch ₃ Quinolin-2-yl A.492 ch ₃ 2,5-Dimethylpyrazin-3-yl 1 A.493 ch ₃ Pyrazin-2-yl 1 A.494 ch ₃ 3-chloropyrid-2-yl A.495 ch ₃ 6-Chloropyrid-2-yl | A.496 ch ₃ 4-Trifluoromethyl, 6-Chloropyrid-2-yl 1 A.497 ch ₃ 4-Trifluoromethylpyrid-2-yl 1 A.498 ch ₃ 6-trifluoromethylpyrid-2-yl A.499 ch ₃ 6-methoxypyridin-2-yl A. 500 ch ₃ 5-Chloropyrid-2-yl A.501 ch ₃ Pyrid-2-yl 1 A.502 2H ₃ 3-benzothiazol-2-yl A. 503 HH ₃ 7-Chloro-quinolin-4-yl A. 504 = h ₃ -Nitropyrid-2-yl 1 A.505 : h ₃ pyrrol-3-yl |

-1Ν-

Nr. R ² R ⁴ A.506 ch ₃ Pyrrol-2-yl A. 507 ch ₃ 2,6-Dioctylpyrid-4-yl A.508 ch ₃ 5-Ni-tropyrid-2-yl A. 509 ch ₃ Pyridin-4-yl A. 510 ch ₃ Pyridin-3-yl A.511 ch ₃ Pyrimidin-2-yl A.512 ch ₃ Pyrimidin-4-yl A.513 ch ₃ Quinazolin-4-yl A.514 ch ₃ 6-Chloro-pyrimidin-4-yl A.515 ch ₃ 6-Methoxy-pyrimidin-4-yl A.516 ch ₃ 2,5,6-Trichloro-4-yl A. 517 ch ₃ 2,6-dimethyl-pyrimidin-4-yl A.518 ch ₃ 2-Methyl, 6-chloropyrimidin-4-yl A.519 ch ₃ 2-Methyl, 6-Ethoxy-pyrimidin-4-yl A.520 ch ₃ 4,5,6-trichloro-2-yl A.521 ch ₃ 4,6-Dimethoxy-pyrimidin-2-yl A.522 ch ₃ 4,6-dimethyl-2-yl A.523 ch ₃ 4,6-dichloropyrimidine-2-yl A. 524 ch ₃ 4-Methyl, 6-methoxy-pyrimidin-2-yl A.525 ch ₃ 4-Chloro, 6-methoxypyrimidin-2-yl A.526 ch ₃ 6-Chloro-quinoxalin-2-yl A.527 ch ₃ 3,6-Dichloro-1,2,4-triazin-5-yl A. 528 ch ₃ 4-methoxy-1,3,5-triazin-2-yl A.529 ch ₃ 4-Ethoxy-1,3,5-triazin-2-yl A.530 ch ₃ 4,6-Dichloro-1,3,5-triazin-2-yl A.531 ch ₃ 4-Ethoxy, 6-Chloro-1,3,5-triazin-2-yl A.532 ch ₃ Isoxazol-3-yl A.533 čh ₃ Thien-2-yl A.534 ch ₃ Fur-2-yl A.535 ch ₃ Thiatriazol-5-yl A.536 ch ₃ E) -l-chloropropene-3-yl A.537 ch ₃ E) -4- (4'-Chlorophenyl) but-2-en-1-yl A.538 ch ₃ Propyn-3-yl A.539 ch ₃ Methylcarbonyl A.540 '' TJ wti3 Ethylcarbonyl A.541 2H ₃ n Propylcarbonyl A.542 3H ₃ i-Propylcarbonyl A.543 ( : h ₃ n Butylcarbony1 A.544 ( HH ₃ p-Butylcarbonyl

- 1? 2-

Nr. R ² R ⁴ A. 545 ch ₃ i -Butylcarbonyl | A. 546 ch ₃ t-Butylcarbonyl | A.547 ch ₃ n-Pentylcarbonyl. | A.548 ch ₃ i-Pentylcarbonyl | A.549 ch ₃ neo-Pentylcarbonyl | A. 550 ch ₃ n-Hexylcarbonyl | A.551 ch ₃ n-Octylcarbonyl 1 A.552 ch ₃ 1-Propenylcarbonyl 1 A.553 ch ₃ 2-Penten-1-yl-carbonyl A.554 ch ₃ 2,5-Heptadien-1-yl-carbonyl A.555 ch ₃ Benzoyl I A. 556 ch ₃ 2-Chlorobenzoyl A. 557 ch ₃ 3-Chlorobenzoyl A. 558 ch ₃ 4-Chlorobenzoyl A. 559 ch ₃ 2 -Cyanobenzyl 1 A. 560 ch ₃ 3-Cyanobenzoyl 1 A.561 ch ₃ 4-Cyanobenzoyl J. A. 562 ch ₃ 4-Methoxybenzoyl J. A. 563 ch ₃ 2-Pyridylcarbonyl J A. 564 ch ₃ 3 -Pyr idyll rbony1 1 A. 565 ch ₃ 4-Pyridylcarbonyl J A.566 ch ₃ 2-Pyrimidinylcarbonyl 1 A. 567 ch ₃ 2 Oxazolylcarbonyl 1 A. 568 ch ₃ 4-Methylisoxazol-5-ylcarbonyl 1 A. 569 ch ₃ Methylsulfonyl J A. 570 ch ₃ Ethylsulfonyl 1 A.571 ch ₃ n-Propylsulfonyl J A. 572 ch ₃ i-Propyl sulfones J A.573 ch ₃ n-Butylsulfonyl 1 A. 574 ch ₃ t-Butylsulfonyl; A.575 ch ₃ n-Pentylsulfonyl 1 A. 576 ch ₃ Neo-Pentylsulfonyl 1 A.577 ch ₃ n-Hexylsulfonyl 1 A.578 HH ₃ n-Octylsulfonyl 1 A.579 3H ₃ Phenylsulfonyl 1 A.580 HH ₃ 2-Chlorophenylsulfonyl J A. 581 : h ₃ 3-Chlorophenylsulfonyl J A.582 ( : h ₃ 4-Chlorophenylsulfonyl 1 A.583 ( : h ₃ 2-Cyanophenylsulfonyl 1

Ίϊ; <-

Nr. R ² R ⁴ A. 584 ch ₃ 3-Cyanophenylsulfonyl A. 585 ch ₃ 4-Cyanophenylsulfonyl A. 586 ch ₃ 2-Pyridylsulfonyl A.587 ch ₃ 3-Pyridylsulfonyl A.588 ch ₃ 4-Pyridylsulfonyl A. 589 ch ₃ 2-Pyrimidinylsulfonyl A. 590 ch ₃ 4-Oxazolylsulfonyl A.591 ch ₃ 5-Chloro-thiazol-2-ylsulfonyl A. 592 ch ₃ 2 -1-C ₄ H ₉ -C ₆ H ₄ -CH ₂ A. 593 ch ₃ 3 -1-C ₄ H ₉ -C ₆ H ₄ -CH ₂ A. 594 ch ₃ 4-C ₄ H ₉ -C ₆ H ₄ -CH ₂ A.595 ch ₃ 2- (4'-Chloro-thiazol-2'-yloxy) eth-1-yl A.596 ch ₃ 2- (1'-Methylpyrazol-4'-yloxy) eth-1-yl A.597 ch ₃ 4-Br-C ₆ H ₄ A.598 ch ₃ 3,5- (CH ₃ ) ₂ -C ₆ H ₃ A.599 ch ₃ 4-C2H5-C6H4 A.600 ch ₃ 3-Dimethylaminocarbonyl -C 6 H 4 A.601 ch ₃ 4-Dimethylaminocarbonyl-C6H4 A.602 ch ₃ 2-Hydroxyprop-1-yl A.603 ch ₃ 6-hydroxy-2-methylpyrimidin-4-ylmethyl A.604 ch ₃ [6-OH, 2-CH (CH ₃ ) 2 * pyrimidin-4-yl] -CH ₂ A.605 ch ₃ [6-OH, 2-CH (CH ₂ ) 2 -pyrimidin-4-yl] -CH ₂ A.606 ch ₃ 5- (2'-furan) pent-l-yl A.607 ch ₃ 5- (2'-N-Methyl-pyrrole) -pent-1-yl A.608 ch ₃ [2- (4-Cl-C ₆ H ₄₎ -oxazole-4-yl] _-CH2 A.609 ch ₃ 3-CF _3- pyridin-2-yl A.610 ch ₃ 5-CF ₃ -pyridin-2-yl A.611 ch ₃ 6- (2'-Thienyl) hex-1-yl A.612 ch ₃ <E) -3-chloro-but-2-en-l-yl A.613 ch ₃ CZ) -3-chloro-but-2-en-l-yl A.614 ch ₃ ΪΕ) -2-bromo-but-2-en-l-yl A.615 ch ₃ Z) -2-bromo-but-2-en-l-yl A.616 ch ₃ (E) -l-chloro-prop-l-en-3-yl A.617 ch ₃ 'Z) -l-chloro-prop-l-en-3-yl A.618 ch ₃ But-en-3-yl A.619 ch ₃ CH ₂ CH ₂ Br A.620 2H ₃ CH ₂ CH ₂ CH ₂ Br A.621 2H ₃ CH ₂ CH ₂ CH ₂ CH ₂ Br A.622 : h ₃ Methylprop-2-yl

-Ο

Nr. R ² R ⁴ A.623 ch ₃ 2-Ethoxyprop-1-yl | A.624 ch ₃ 2-Isopropoxyprop-1-yl | A.625 ch ₃ But-1-yn-S-yl | A.626 ch ₃ But-1-yn-4-yl | A.627 ch ₃ But-2-yn-4-yl i A.628 ch ₃ Pent-1-yn-4-yl A.629 ch ₃ Pent-2-yn-4-yl | A.630 ch ₃ Pent-1-yn-5-yl | A.631 ch ₃ Pent-2-yn-5-yl 1 A.632 ch ₃ E-2-Chlorobut-2-en-1-yl | A.633 ch ₃ Z-2-Chlorobut-2-en-1-yl | A.634 ch ₃ Z-1-Chlorprop-1-en-3-yl A.635 ch ₃ 2-Methylprop-1-en-3-yl 1 A.636 ch ₃ 2-Chloroprop-1-en-3-yl A.637 ch ₃ 2-Bromo-prop-1-en-3-yl 1 A. 638 ch ₃ But-2-en-l-yl A.639 ch ₃ But-3-en-1-yl A.640 ch ₃ 1-Iodoprop-1-yn-3-yl j A.641 ch ₃ E-3-Bromobut-2-en-1-yl | A.642 ch ₃ Z-3-Bromobut-2-en-1-yl A.643 C ₂ H ₅ h 1 A.644 C ₂ Hs ch ₃ I A.645 C ₂ Hs c ₂ h ₅ A.646 C ₂ H _p n.-C ₃ H ₇ J A.647 C ₂ H _p I-C3H7 A.648 C ₂ H _p Cyclopropyl 1 A.649 c ₂ h ₅ nC ₄ 19 A.650 C ₂ H ₅ S'C ₄ Hg J A.651 c ₂ h ₅ 1 * C ₄ Hg | A.652 c ₂ Hs tC ₄ H ₉ J A.653 c ₂ h ₅ n-CsHn J A.654 c ₂ h ₅ i C5H1I I A.655 c ₂ h ₅ neo-CsHn I A.656 c ₂ h ₅ cyclopentyl A.657 c ₂ h ₅ 1-C6H13 J A.658 c ₂ h ₅ cyclohexyl A.659 ^C 2 ^H 5 l-CgHIV | A.660 -2H5 3H ₂ CH ₂ Cl 1 A.661 3 ₂ Hs (ch ₂ ) ₄ or 1

../Ír siM

Nr. R ² R ⁴ A.662 c ₂ h ₅ ch ₂ cn A. 663 c ₂ h ₅ ch ₂ ch ₂ cn A.664 c ₂ h ₅ (CH ₂ ) ₃ CN A.665 c ₂ h ₅ (CH ₂ ) ₄ CN A.666 c ₂ h ₅ (ch ₂ ) ₆ cn A.667 c ₂ h ₅ Cyclohexylmethyl A.668 c ₂ h ₅ 2-Cyclohexyleth-1-yl A.669 c ₂ h ₅ cyclopropylmethyl A.670 c ₂ h ₅ 2-Cyclopropyleth-1-yl A.671 c ₂ h ₅ 2-methoxyethyl-1-yl A.672 C ₂ Hs 2-ethoxyethanol 1-y1 A.673 c ₂ h ₅ 2-1-propoxye th-1-yl A.674 c ₂ h ₅ 3-methoxypropyl-1-yl A.675 c ₂ h ₅ 3-Ethoxyprop-1-yl A.676 c ₂ h ₅ 3 -1sopropoxyprop-1-yl A.677 c ₂ h ₅ 4-methoxy-but yl A.678 c ₂ h ₅ Isopropoxybut 4-yl A.679 C2H5 Propen-3-yl A.680 c ₂ H ₅ But-2-en-l-yl A.681 C ₂ Hs 3-methyl-but-2-en-l-yl A. 682 c ₂ h ₅ 2-Vinyloxyeth-yl A.683 C ₂ H ₅ Allyloxyeth-1-yl A.684 C ₂ H ₅ 2-Trifluormethoxyeth-1-yl A.685 C ₂ H ₅ 3-Trifluormethoxyprop-1-yl A.686 c ₂ h ₅ Dífluormethoxybut 4-yl A.687 C ₂ H ₅ Hydroxycarbonylmethy1 A.688 C ₂ H _p Methoxycarbonylmethyl i A.689 c ₂ h ₅ Aminocarbonylmethyl A.690 C ₂ Hs N-Methylaminocarbonylmethyl A.691 c ₂ h ₅ Ν, Ν-methyl-Dimethylaminocarbonyl A.692 C ₂ Hs 2-Hydroxycarbonyleth-1-yl A.693 c ₂ h ₅ 2-Methoxycarbonyleth-1-yl j A.694 c ₂ h ₅ 2-Aminocarbonyleth-1-yl; A.695 C ₂ H _p 2-N-Methylaminocarbonyleth-1-yl i A.696 C ₂ H ₅ 2-Dimethylaminocarbonyleth-1-yl; A.697 c ₂ h ₅ 2-Aminoeth-1-yl i A.698 C ₂ H ₅ 2-Aminoprop-1-yl; 1 A.699 C ₂ Hs 4-Aminobut-1-yl i s 2 A.700 c ₂ h ₅ 3-Dimethylaminoprop-1-yl j

Nr. R ² R ⁴ A.701 c ₂ h ₅ Aminothiocarbonylbut 4-yl A.702 C ₂ Hs 2-oxo-propyl A.703 c ₂ h ₅ cyclohexyl A.704 c ₂ h ₅ cyclopropyl A.705 c ₂ h ₅ cyclopentyl A.706 C ₂ Hs 2-Methoxyiminoprop-yl A.707 c ₂ h ₅ 2-Methoxyiminoeth-1-yl A.708 C ₂ Hs 6-Aminocarbonylhex-1-yl A.709 C ₂ H ₅ Aminothiocarbonylprop 3-yl A.710 c ₂ h ₅ 2-Aminothiocarbonyleth-yl A.711 c ₂ h ₅ Aminothiocarbonylmethyl A.712 c ₂ h ₅ 4- (N, N-dimethylamino) but-l-yl A.713 C ₂ H ₅ 2- (Methylthio) eth-1-yl A.714 c ₂ h ₅ 2- (methylsulfonyl) eth-1-yl A.715 c ₂ h ₅ 4- (Methylthio) prop-1-yl A.716 C ₂ H _p 4- (Methylsulfonyl) prop-1-yl A.717 c ₂ h ₅ Benyzl A.718 c ₂ h ₅ 2-FC ₆ H ₄ -CH ₂ A. 719 c ₂ h ₅ 3-FC ₆ H ₄ -CH ₂ A. 720 C ₂ Hs 4-FC ₆ H ₄ -CH ₂ A.721 c ₂ h ₅ 2,3-F ₂ -C ₆ H ₃ -CH ₂ A.722 c ₂ h ₅ 2,4-F ₂ -C ₆ H ₃ -CH ₂ A.723 c ₂ h ₅ 2,5-F ₂ -C ₆ H ₃ -CH ₂ A.724 C ₂ Í 5 2,6-F ₂ -C ₆ H ₃ -CH ₂ A.725 C ₂ H5 3,4-F ₂ -C ₆ H ₃ -CH ₂ A.726 c ₂ h ₅ 3,5-F ₂ -C ₆ H ₃ -CH ₂ A.727 c ₂ h ₅ 2 -C 1 -C ₆ H ₄ -CH ₂ A.728 c ₂ h ₅ 3-Cl-C ₆ H ₄ CH ₂ A.729 c ₂ h ₅ 4-C1-C ₆ H ₄ CH ₂ A.730 c ₂ h _p 2,3-Cl ₂ -C ₆ H ₃ -CH ₂ A.731 C ₂ Hs 2,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.732 c ₂ h ₅ 2,5-Cl ₂ -C ₆ H ₃ -CH ₂ A.733 c ₂ h ₅ 2,6-Cl ₂ -C ₆ H ₃ -CH ₂ A.734 c ₂ h ₅ 3,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.735 C2H5 3,5-Cl ₂ -C ₆ H ₃ -CH ₂ A.736 c ₂ h ₅ 2,3,4-Cl ₃ -C ₆ H ₂ -CH ₂ A.737 3 ₂ H ₅ 2,3,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.738 -2H5 2,3,6-Cl ₃ -C ₆ H ₂ -CH ₂ A.739 -2H ₅ 2,4,5-Cl ₃ -C ₆ H ₂ -CH ₂

- m-

Nr. R ² R ⁴ I A.740 C ₂ Hs 2,4,6-Cl ₃ -C ₆ H ₂ -CH ₂ L A.741 C2H5 3,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.742 C2H5 2-Br-C ₆ H ₄ -CH ₂ j A.743 C2H5 3-Br-C ₆ H ₄ -CH ₂ 1 A.744 c ₂ h ₅ 4-Br-C ₆ H ₄ -CH ₂ J A.745 c ₂ h ₅ 2,3-Br ₂ -C ₆ H ₃ -CH ₂ | A.746 C2H5 2,4-Br ₂ -C ₆ H ₃ -CH ₂ A.747 C2H5 2,5-Br ₂ -C ₆ H ₃ -CH ₂ A.748 C2H5 2,6-Br _{2 C} 6 H ₃ -CH ₂ J A.749 C ₂ H ₅ 3,4-Br ₂ -C ₆ H ₃ -CH ₂ L A.750 C2H5 3,5-Br ₂ -C ₆ H ₃ -CH ₂ A.751 C2H5 2-F, 3-C 1 -C ₆ H ₃ -CH ₂ 1 A.752 C2H5 2-F, 4-C 1 -C ₆ H ₃ -CH ₂ 1 A.753 C2H5 2-F, 5-C 1 -C ₆ H ₃ -CH ₂ J A.754 C2H5 2-F, 3-Br-C ₆ H ₃ -CH ₂ 1 A.755 C2H5 2-F, 4-Br-C ₆ H ₃ -CH ₂ | A.756 C2H5 2-F, 5-Br-C ₆ H ₃ -CH ₂ | A.757 C2H5 2-Cl, 3-Br-C ₆ H ₃ -CH ₂ 1 A.758 C2H5 2-Cl, 4-Br-C ₆ H ₃ -CH ₂ j A.759 C2H5 2-C1, 5-Br-C ₆ H ₃ -CH ₂ | A.760 C2H5 3-F, 4-C 1 -C ₆ H ₃ -CH ₂ J A.761 C ₂ Hs 3-F, 5-C 1 -C ₆ H ₃ -CH ₂ J A.762 C2H5 3-F, 6-C 1 -C ₆ H ₃ -CH ₂ j A.763 C2H5 3-F, 4-Br-C ₆ H ₃ -CH ₂ J A.764 c ₂ h ₅ 3-F, 5-Br-C ₆ H ₃ -CH ₂ | A.765 c ₂ h ₅ 3-F, 6-Br-C ₆ H ₃ -CH ₂ f A.766 C2H5 3-Cl, 4-Br-C ₆ H ₃ -CH ₂ J A.767 C ₂ H ₅ 3-C1, 5-Br-C ₆ H ₃ -CH ₂ | A.768 c ₂ h _p 3-C1, 6-Br-C ₆ H ₃ CH ₂ A.769 C2H5 4-F, 5-C 1 -C ₆ H ₃ -CH ₂ j A.770 C2H5 4-F, 6-C 1 -C ₆ H ₃ -CH ₂ J A.771 c ₂ h ₅ 4-F, 5-Br-C ₆ H ₃ -CH ₂ | A.772 C2H5 4-F, 6-Br-C ₆ H ₃ -CH ₂ J A.773 C ₂ H _S 4-C1, 5-Br-C ₆ H ₃ -CH ₂ | A.774 C2H5 5-F, 6-C 1 -C ₆ H ₃ -CH ₂ J A.775 C ₂ H _S 5-F, 6-Br-C ₆ H ₃ -CH ₂ | A.776 C2H5 5-C1, 6-Br-C ₆ H ₃ -CH ₂ | A.777 -2H5 and-Br, 4-C1, 5-Br-C ₆ H ₂ -CH ₂ | A.778 2 ₂ H ₅ 2-CN-C ₆ H ₄ -CH ₂ J

Nr. R ² R ⁴ A.779 c ₂ h ₅ 3-CN-C ₆ H ₄ CH ₂ A.780 c ₂ h ₅ 4-CN-C ₆ H ₄ CH ₂ A.781 c ₂ h ₅ 2-NO ₂ -C ₆ H ₄ -CH ₂ I A.782 c ₂ h ₅ 3-NO ₂ -C ₆ H ₄ -CH ₂ 1 A.783 c ₂ h ₅ 4-NO ₂ -C ₆ H ₄ -CH ₂ 1 A.784 c ₂ h ₅ 2-CH ₃ -C ₆ H ₄ -CH ₂ L A.785 c ₂ h ₅ 3 -CH ₃ -C ₆ H ₄ -CH ₂ A.786 c ₂ h ₅ 4-CH ₃ -C ₆ H ₄ -CH ₂ L A.787 c ₂ h ₅ 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ I A.788 c ₂ h ₅ 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.789 c ₂ h ₅ 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ L A.790 c ₂ h ₅ 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ j A.791 c ₂ h ₅ 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ J A.792 c ₂ h ₅ 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ j A.793 c ₂ h ₅ 2-c ₂ h ₅ -c _s h ₄ -ch ₂ 1 A.794 c ₂ h ₅ 3-C ₂ H ₅ -C ₆ H ₄ -CH ₂ j A.795 c ₂ h ₅ 4-c ₂ h _with -c ₆ h ₄ -ch ₂ J A.796 c ₂ h ₅ 2-C ₃ H ₇ -C ₆ H ₄ -CH ₂ j A.797 c ₂ h ₅ 3-C ₃ H ₇ -C ₆ H ₄ -CH ₂ J A.798 C ₂ Hs 4-C ₃ H ₇ -C ₆ H ₄ -CH ₂ j A.799 C ₂ Hs 2-Cyclohexyl-C 6 H ₄ -CH ₂ L A.800 c ₂ h ₅ 3-Cyclohexyl-C 6 H ₄ -CH ₂ | A.801 c ₂ h ₅ 4-CGH -Cyclohexy1 ₄ - CH ₂ A.802 c ₂ h ₅ 2-Vinyl-C ₆ H ₄ -CH ₂ J A.803 c ₂ h ₅ 3-vinyl-C ₆ H ₄ -CH ₂ | A.804 c ₂ h ₅ 4-Vinyl-C ₆ H ₄ -CH ₂ | A.805 c ₂ h ₅ 2-allyl-C ₆ H ₄ -CH ₂ | A.806 C ₂ Hs 3-allyl-C ₆ H ₄ -CH ₂ | A.807 C ₂ Hs 4-allyl-C ₆ H ₄ -CH ₂ | A.808 c ₂ h ₅ 2-C ₆ H 5 -C ₆ H ₄ -CH ₂ j A.809 C ₂ Hs 3-c ₆ h ₅ -c ₆ h ₄ -ch ₂ 1 A. 810 C ₂ F 15 4-C ₆ H 5 -C ₆ H ₄ -CH 2 j A.811 c ₂ H ₅ 3-CH ₃ , 5 -1-C ₄ H ₉ -C ₆ H ₃ -CH ₂ L A.812 c ₂ h ₅ 2-OH-C ₆ H ₄ -CH ₂ j A.813 C ₂ Hs 3-oh-c ₆ h ₄ -ch ₂ J A. 814 c ₂ h ₅ 1-OH-C ₆ H ₄ -CH ₂ 1 A. 815 = ₂ Hs 2 -OCH ₃ -C ₆ H ₄ -CH ₂ L A. 816 3 ₂ H ₅ 3-OCH ₃ -C ₆ H ₄ -CH ₂ 1 A. 817 3 ₂ Hs 1-OCH ₃ -C ₆ H ₄ -CH ₂ 1

U'3-

Nr. R 2 R ⁴ A.818 C ₂ H ₅ 2,3- (OCH 3) ₂ -C ₆ H ₃ -CH ₂ A.819 c ₂ h ₅ 2,4- (OCH ₃ ) 2 -C ₆ H ₃ -CH ₂ A.820 c ₂ h ₅ 2,5 - (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.821 c ₂ h ₅ 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.822 C ₂ Hs 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ L A.823 C2H5 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH ₂ ! A.824 c ₂ H ₅ 2-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ t A.825 C2H5 3-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ j A.826 C ₂ Hs 4-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.827 C ₂ Hs 2-O- (nC ₃ H ₇ ) -c ₆ h ₄ -ch ₂ ; A.828 C2H5 3-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ ; A.829 C2H5 4-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.830 C2H5 2-O- (t-C ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.831 C ₂ H ₅ 3-O- (t-C ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A. 832 C2H5 4-o- (i-c ₃ h ₇ ) -c ₆ h ₄ -ch ₂ : A. 833 C2H5 4-O- (nC ₄ H ₉ ) -C ₆ H ₄ -CH ₂ A. 834 C2H5 3-O- (t C ₄ H ₉ ) -C ₆ H ₄ -CH ₂ A.835 C2H5 4-O- (nC ₆ H ₃ ) -C ₆ H ₄ -CH ₂ A. 836 C2H5 2-o-Alyl-c ₆ h ₄ -CH ₂ ; A. 837 c ₂ H ₅ 3-Allyl-O-C ₆ H ₄ CH ₂ A. 838 C2H5 4-O-allyl-C ₆ H ₄ CH ₂ A. 839 C ₂ H ₅ 2 -CP ₃ -C ₆ H ₄ -CH ₂ A. 840 c ₂ h ₅ 3-CP ₃ -C ₆ H ₄ -CH ₂ A. 841 C2H5 4-CP ₃ -C ₆ H ₄ -CH ₂ A. 842 C2H5 2-Acetyl-C ₆ H ₄ CH ₂ A. 843 C2H5 3-Acetyl-C ₆ H ₄ CH ₂ A. 844 c ₂ H ₅ 4-Acetyl-C ₆ H ₄ CH ₂ A. 845 c ₂ h ₅ 2-Methoxycarboethyl -C ₈ H ₄ -CH ₂ A. 846 C ₂ Hs 3-Methoxycarbonyl -C ₈ H ₄ -CH ₂ A. 847 c ₂ h ₅ 4-Methoxycarbonyl -C ₈ H ₄ -CH ₂ A. 848 c ₂ h ₅ 2 -Aminocarbonyl - CGH ₄ - CH ₂ A. 849 c ₂ h _{5 3-aminocarbonyl-4 -CH2} ΟβΗ A.850 C ₂ H ₅ 4 - aminocarbonyl - CGH ₄ - CH ₂ A. 851 c ₂ h _p 2-Dimethylaminocarbonyl -CeH ₄ -CH ₂ A. 852 c ₂ h ₅ 3-Dimethylaminocarbonyl -C ₈ H ₄ -CH ₂ A. 853 3 ₂ h ₅ 4-Dimethylaminocarbonyl -C ₈ H ₄ -CH ₂ A. 854 3 ₂ H ₅ 2- (N-Methylaminocarbonyl) _{4 -CH2} -C5H A.855 -2? 5 3- (N-Methylaminocarbonyl) -C ₆ H ₄ -CH ₂ A.856 - ₂ H ₅ 4- (N-Methylaminocarbonyl) -C 5 H ₄ -CH ₂

Nr. R ² R ⁴ J A. 857 c ₂ h ₅ 2-H ₂ NC ₆ H ₄ -CH ₂ 1 A.858 C ₂ H ₅ 3-H ₂ NC ₆ H ₄ -CH ₂ 1 A. 859 c ₂ h ₅ 4-H ₂ NC ₆ H ₄ -CH ₂ 1 A. 860 c ₂ h ₅ 2-Aminothiocarbonyl-C6H4-CH2 | A.861 c ₂ h ₅ 3-Aminothiocarbonyl-C 6 H ₄ -CH ₂ | A. 862 c ₂ h ₅ 4-Aminothiocarbonyl-C6H4-CH2 A. 863 c ₂ h _{5 2-methoxyimino-C6H4-CH2} | A.864 C ₂ H ₅ 3-methoxyimino-methyl-C 6 H ₄ CH ₂ I A.865 C ₂ H _{5 4-methoxyiminomethyl-C6H4-CH2} | A.866 c ₂ h ₅ 2-Formyl-C ₆ H ₄ -CH ₂ | A. 867 c ₂ h ₅ 3 - Forms 1 -C 6 H 4 -CH ₂ J A.868 C ₂ H _{5 4-formyl-C6H4-CH2} | A.869 C ₂ H ₅ 2- (1'-Methoxyiminoeth-1'-yl) -C 6 H 4 -CH 2 A.870 C ₂ H _p 3- (1'-Methoxyiminoeth-1'-yl) -C 6 H 4 -CH 2 J A.871 C ₂ H ₅ 4- (1'-Methoxyiminoeth-1'-yl) -C 6 H 4 -CH 2, A.872 C ₂ H ₅ 2-SCH ₃ -C ₆ H ₄ -CH ₂ 1 A.873 C ₂ H ₅ 3-SCH 3 -C ₆ H ₄ -CH ₂ | A.874 c ₂ h ₅ 4 -SCH 3 -C ₆ H ₄ -CH ₂ J A.875 c ₂ h ₅ 2 -so ₂ ch ₃ -c ₆ h ₄ -ch ₂ j A.876 C ₂ Hs 3-SO ₂ CH ₃ -C ₆ H 4 -CH ₂ f A.877 C ₂ Hs 4 -so ₂ ch ₃ -c ₆ h ₄ -ch ₂ J A.878 C ₂ Hs 2-OCF ₃ -C ₆ H 4 -CH ₂ j A.879 c ₂ h ₅ 3-OCF ₃ -C ₆ H ₄ -CH ₂ J A.880 c ₂ h ₅ 4-OCF 3 -C 6 H 4 -CH 2 J A.881 c ₂ h ₅ 2-OCHF ₂ -C ₆ H ₄ -CH ₂ j A.882 C ₂ Hs 3-OCHF 2 -C 6 H 4 -CH 2 i A.883 c ₂ h ₅ 4 -ochf ₂ -c ₆ h ₄ -ch ₂ J A. 884 c ₂ h ₅ 3-CF 3, 4-OCF 3 -C ₆ H ₃ -CH ₂ A.885 c ₂ h ₅ 1-Naphthyl-CH ₂ J A.886 c ₂ h ₅ 2-Naphthyl-CH ₂ J A.887 c ₂ h ₅ 2-Phenoxyethyl 1 A.888 c ₂ h ₅ 2- <2'-Chlorphenoxy) eth-l-yl A.889 c ₂ h ₅ 2- (3'-Chlorphenoxy) ethyl] J A.890 c ₂ h ₅ 2- (4'-Chlorphenoxy) eth-l-yl A.891 c ₂ h _p 2- (3 ', 5'-Dichlorophenoxy) eth-1-yl A.892 3 ₂ Hs 2- (2'-Cyanophenoxy) eth-1-yl 1 A.893 = ₂ h ₅ 2- (3'-Cyanophenoxy) eth-l-yl A.894 : ₃ h ₅ 2- (4'-Cyanophenoxy) eth-1-yl 1 A.895 : ₂ H ₅ 2- (2'-Methylphenoxy) eth-1-yl |

- ý / / / -

Nr. R ² R ⁴ A.896 c ₂ h ₅ 2- (3'-Methylphenoxy) eth-1-yl A.897 C ₂ H5 2- (4'-Methylphenoxy) eth-1-yl A.898 C ₂ H ₅ 2- (3'-t-Butylphenoxy) eth-1-yl A.899 C ₂ H ₅ 2- (4'-t-Butylphenoxy) eth-1-yl A.900 C2H5 2- (2'-Nitrophenoxy) eth-1-yl A.901 C2H5 2- (3'-Nitrophenoxy) eth-1-yl A.902 C2H5 2- (4'-Nitrophenoxy) eth-1-yl A.903 C2H5 2- (2'-Methoxyphenoxy) eth-1-yl A.904 C2H5 2- (3'-Methoxyphenoxy) eth-1-yl A.905 c ₂ h ₅ 2- (4'-Methoxyphenoxy) eth-1-yl A. 906 C ₂ H ₅ 2- (2'-Trifluoromethylphenoxy) eth-1-yl A.907 C2H5 2- (3'-Trifluoromethylphenoxy) eth-1-yl A. 908 C2H5 2- (4'-Trifluoromethylphenoxy) eth-1-yl A.909 C ₂ Hs 2- (2'-Acetylphenoxy) eth-1-yl A.910 C ₂ H ₅ 2- (3 &apos; -Acetylphenoxy) eth-1-yl A.911 C ₂ Hs 2- (4'-Acetylphenoxy) eth-1-yl A.912 C ₂ Hs 2- (2'-Methoxycarbonyl) eth-1-yl A.913 C2H5 2- (3'-Methoxycarbonyl) eth-1-yl A. 914 C2H5 2- (4'-Methoxycarbonyl) eth-1-yl A.915 C2H5 2- (2'-Dimethylaminocarbonyl) eth-1-yl A.916 C ₂ H _S 2- (3'-Dimethylaminocarbonyl) eth-1-yl A. 917 C2H5 2- (4'-Dimethylaminocarbonyl) eth-1-yl A.918 c ₂ H ₅ 2- (2'-Aminothiocarbonyl) eth-1-yl A.919 C2H5 2- (3'-Aminothiocarbonyl) eth-1-yl A.920 C ₂ H ₅ 2- (4'-Aminothiocarbonyl) eth-1-yl A.921 C ₂ Hs 2- (2'-Methylsulfonyl) eth-1-yl A.922 C ₂ H _p 2- (3'-methylsulfonyl) eth-1-yl A.923 c ₂ h _p 2- (4'-methylsulfonyl) eth-1-yl A.924 C ₂ Hs 3-Phenoxyprop-1-yl A.925 c ₂ h _p 3- (2'-Chlorophenoxy) prop-1-yl A.926 C ₂ Hs 3- (3'-Chlorphenoxy) prop-l-yl A.927 C2H5 3- (4'-Chlorophenoxy) prop-1-yl A.928 C ₂ H ₅ 3- (3 ', 5', Dichlorophenoxy) prop-1-yl A.929 C ₂ Hs 3- (2'-Cyanophenoxy) prop-1-yl A.930 c ₂ h ₅ 3- (3'-Cyanophenoxy) prop-1-yl A.931 C ₂ Hs 3- (4'-Cyanophenoxy) prop-1-yl A.932 C ₂ Hs 3- (2-methylphenoxy) prop-1-yl A.933 2 ₂ h ₅ 3- (3'-Methylphenoxy) prop-1-yl A.934 - ₂ h ₅ 3 '(4'-Methylphenoxy) prop-1-yl

Nr.

A.935

A.936

A.937

A.938

A.939

A.940

A.941

A.942

A.943

A.944

A.945

A.946

A.947

A.948

A.949

A.950

A.951

A.952

A.953

A.954

A.955

A.956

A.957

A.958

A.959

A.960

A.961

A.962

A.963

A.964

A.965

A.966

A.967

A.968

A.969

A.970.971, 972.973

C ₂ H ₅

C ₂ f ₅ c ₂ h ₅

C ₂ H ₅

C ₂ H _S c ₂ h ₅

C ₂ H ₅

C ₂ H ₅ c ₂ h ₅

C ₂ H ₅ c ₂ h ₅ c ₂ h ₅ c ₂ h ₅ c ₂ h ₅ c ₂ h ₅

C ₂ H ₅

C ₂ h ₅ c ₂ h ₅ c ₂ h ₅ c ₂ h ₅ c ₂ h ₅ c ₂ h ₅ c ₂ h ₅

C ₂ H ₅ c ₂ h ₅ c ₂ h ₅ c ₂ h ₅

C ₂ H _S c ₂ h ₅

C ₂ H _S

C ₂ H ₅ c ₂ h ₅

C ₂ H ₅

C ₂ Hs

C ₂ H ₅

C ₂ H _S c ₂ h ₅ c ₂ h ₅ c ₂ h ₅

R ²

R ⁴

3- (2'-Methoxyphenoxy) prop-yl

3- (3'-Methoxyphenoxy) prop-yl

3- (4'-Methoxyphenoxy) prop-yl

3- (2'-Trifluoromethylphenoxy) prop-yl

3- (3 ' Trifluormethylphenoxy) prop-l-yl

3- (4'-Trifluormethylphenoxy) prop-1-yl

-Phenoxybut-1-yl

2-Phenyleth-yl

2- (2-Chlorphenyl) eth-l-yl

2- (3'-Chlorphenyl) eth-l-yl

2- (4'-Chlorphenyl) eth-1-yl

2- (3 ', 5'-Dichlorophenyl) eth-1-yl

2- (2'-cyanophenyl) eth-l-yl

2- (3'-cyanophenyl) eth-l-yl

2- (4'-cyanophenyl) eth-l-yl

2- (2 * -Methylphenyl) eth-1-yl

2- (3'-methylphenyl) eth-1-yl

2- (4'-Methylphenyl) eth-l-yl

2- (2'-Methoxyphenyl) eth-1-yl

- (3'-Methoxyphenyl) eth-l-yl

- (4'-Methoxyphenyl) eth-l-yl

2- (2 ' Trifluormethylphenyl) eth-1-yl

- (3 ' Trifluormethylphenyl) eth-1-yl

- (4'-Trifluormethylphenyl) eth-1-yl

-Phenylprop-1-yl

- (2'-Chlorphenyl) prop-1-yl

- (3'-Chlorphenyl) prop-1-yl

- (4'-Chlorophenyl) prop-1-yl (2'-Cyanophenyl) prop-1-yl

- (3'-Cyanophenyl) prop-1-yl (4'-Cyanophenyl) prop-1-yl

- (2 ' Trifluormethylphenyl) prop-1-yl

-Phenylbut-1-yl

- (4'-Chlorphenyl) but-1-yl

- (4'-Chlorphenyl) hex-1-yl

-Pyridylmethyl

pyridylmethyl

-Pyridylmethyl

Chloropyridin-2-ylmethyl

- / ýj-

Nr. R ² r ⁴ A. 974 c ₂ h ₅ 5-Chloro-pyridin-2-ylmethyl A.975 c ₂ h ₅ 6-Chloro-pyridin-2-ylmethyl A. 976 c ₂ h ₅ 5-Chloro-pyridin-3-ylmethyl A.977 C ₂ Hs 6-Chloro-pyridin-3-ylmethyl A.978 C ₂ Hs 2-Chloropyridin-4-ylmethyl A. 979 c ₂ h ₅ 2-Pyrimidinylmethyl i A.980 c ₂ h ₅ 4-Chloropyrimidin-2-ylmethyl i A.981 c ₂ h ₅ 5-Chloropyrimidin-2-ylmethyl A.982 c ₂ h ₅ 2-Chloropyrimidin-4-ylmethyl | A.983 C ₂ Hs 6-Chloro-pyrimidin-4-ylmethyl A.984 c ₂ h ₅ 2-Chloropyrimidin-5-ylmethyl A.985 c ₂ h ₅ 4-Pyridazinylmethyl A.986 c ₂ h ₅ 2 -Pyr and zynyme thy1 A.987 c ₂ h ₅ 5-Chloro-pyrazin-2-ylmethyl A.988 C ₂ Hs 6-Chloro-pyrazin-2-ylmethyl A.989 c ₂ h ₅ 3-Pyridazinylmethyl A.990 c ₂ h ₅ 6-chloropyridazine-3-ylmethyl A.991 c ₂ h ₅ 1,3,5-Triazinylmethyl A.992 c ₂ h ₅ 2-furylmethyl A.993 C ₂ Hs 3-furylmethyl A.994 c ₂ h ₅ 4-bromofuro-2-ylmethyl A.995 C ₂ Hs 5-chloro-furo-2-ylmethyl A.996 C ₂ H _p 2-thienylmethyl A.997 c ₂ h ₅ 3-thienylmethyl A.998 c ₂ h ₅ 5-methyl-thien-3-ylmethyl A.999 C ₂ H _p 5-Chlorothien-2-ylmethyl A.1000 c ₂ h ₅ 2-Chlorothien-4-ylmethyl A.1001 c ₂ h ₅ 2-pyrrolylmethyl A.1002 c ₂ h ₅ 3-pyrrolylmethyl A.1003 C ₂ H ₅ 2-oxazolylmethyl A.1004 C ₂ Hs 4-Methyl-oxazol-2-ylmethyl A.1005 C ₂ Hs 5-Methyl-oxazol-2-ylmethyl A.1006 C ₂ Hs 4-chlorooxazole-2-ylmethyl A.1007 c ₂ h ₅ 5-chlorooxazole-2-ylmethyl A.1008 No. ₂ h ₅ 4-oxazolylmethyl A.1009 c ₂ h ₅ 2-Methyl-oxazol-4-ylmethyl A.1010 = ₂ Hs 5-Methyl-oxazol-4-ylmethyl A.1011 = ₂ h ₅ 2-chlorooxazole-4-ylmethyl A.1012 - ₂ Hs 5-chlorooxazole-4-ylmethyl

Nr. R ² R ⁴ A.1013 C ₂ H ₅ 5-Oxazolylmethyl | . A.1014 C ₂ Hs 2-Methyl-oxazol-5-ylmethyl J A.1015 C ₂ H _p 4-Methyl-oxazol-5-ylmethyl | A.1016 c ₂ h ₅ 2-Chlorooxazol-5-ylmethyl | A.1017 c ₂ h ₅ 4-Chlorooxazol-5-ylmethyl | A.1018 c ₂ h ₅ 2-Thiazolylmethyl | A.1019 c ₂ h ₅ 4-Methylthiazol-2-ylmethyl | A.1020 C ₂ H ₅ 5-Methylthiazol-2-ylmethyl | A.1021 c ₂ h _p 4-Chlorothiazol-2-ylmethyl A.1022 C ₂ H ₅ 5-Chlorothiazol-2-ylmethyl | A.1023 C ₂ Hs 4-Thiazolylmethyl J A.1024 c ₂ h ₅ 2-Methylthiazol-4-ylmethyl A.1025 C ₂ H ₅ 5-Methyl-thiazol-4-ylmethyl A.1026 C ₂ H ₅ 2-Chlorothiazol-4-ylmethyl A.1027 c ₂ h ₅ 5-Chloro-thiazol-4-ylmethyl A.1028 c ₂ h _p 5-Thiazolylmethyl 1 A.1029 c ₂ h ₅ 2-Methylthiazol-5-ylmethyl A.1030 c ₂ h ₅ 4-Methylthiazol-5-ylmethyl j A.1031 c ₂ h ₅ 2-Chlorothiazol-5-ylmethyl J A.1032 c ₂ h ₅ 4-Chlorothiazol-5-ylmethyl 1 A.1033 C ₂ H ₅ 3-Isoxazolylmethyl 1 A.1034 c ₂ h ₅ 4-Methylisoxazol-3-ylmethyl 1 A.1035 c ₂ h ₅ 5-Methylisoxazol-3-ylmethyl 1 A.1036 C ₂ Hs 4-Chloroisoxazol-3-ylmethyl J A.1037 c ₂ h ₅ 5-Chloroisoxazol-3-ylmethyl 1 A.1038 c ₂ h ₅ 4-Isoxazolylmethyl 1 A.1039 c ₂ h ₅ 3-Methylisoxazol-4-ylmethyl A.1040 c ₂ Hs 5-Methylisoxazol-4-ylmethyl A.1041 c ₂ h ₅ 3-Chloroisoxazol-4-ylmethyl 1 A.1042 c ₂ h ₅ 5-Chloroisoxazol-4-ylmethyl 1 A.1043 C ₂ Hs 5-Isoxazolylmethyl 1 A.1044 c ₂ h ₅ 3-Methylisoxazol-5-ylmethyl A.1045 c ₂ h ₅ 4-Methyl-isoxazol-5-ylmethyl A.1046 c ₂ h ₅ 3-Chloroisoxazol-5-ylmethyl 1 A.1047 c ₂ h ₅ 4-Chloroisoxazol-5-ylmethyl A.1048 C ₂ H _p 5-Isothiazolylmethyl 1 A.1049 3 ₂ H ₅ 1-Methylisothiazol-3-ylmethyl 1 A.1050 3 ₂ H ₅ j-Methylisothiazol-3-ylmethyl A.1051 - ₂ Hs 1-Chloroisothiazol-3-ylmethyl |

Nr. R ² R ⁴ A.1052 C ₂ H ₅ 5-Chlorisothiazol-3-ylmethyl A.1053 c ₂ h ₅ 4-Isothiazolylmethyl A.1054 c ₂ h ₅ 3-Methylisothiazol-4-ylmethyl A.1055 c ₂ h ₅ 5-methylisothiazol-4-ylmethyl A.1056 C ₂ H ₅ 3-Chlorisothiazol-4-ylmethyl A.1057 C ₂ H ₅ 5-Chlorisothiazol-4-ylmethyl A.1058 C ₂ H _S 5-Isothiazolylmethyl A.1059 c ₂ h _p 3-Methylisothiazol-5-ylmethyl A.1060 c ₂ h ₅ 4-Methylisothiazol-5-ylmethyl A. 10.61 C ₂ H ₅ 3-Chloroisothiazol-5-ylmethyl A.1062 C ₂ H ₅ 4-Chloroisothiazol-5-ylmethyl A.1063 c ₂ h ₅ 4-Imidazolylmethyl A.1064 c ₂ h ₅ 1-Phenylpyrazol-3-ylmethyl A.1065 c ₂ h ₅ 1-Methylimidazol-4-ylmethyl A.1066 c ₂ h ₅ 1-Phenyl-l, 2,4-triazol-3-ylmethyl A.1067 c ₂ h ₅ 1,2,4-oxadiazol-3-ylmethyl A. 1068 c ₂ h ₅ 5-chloro-1,2,4-oxadiazol-3-ylmethyl A.1069 C ₂ H ₅ 5-Methyl-1,2,4-oxadiazol-3-ylmethyl A.1070 C2H5 5-Trifluoromethyl-1,2,4-oxadiazol-3-ylmethyl A.1071 c ₂ H ₅ 1,3,4-oxadiazol-2-ylmethyl A.1072 c ₂ h ₅ 5-chloro-1,3,4-oxadiazol-2-ylmethyl A.1073 c ₂ h ₅ 5-Methyl-1,3,4-oxadiazol-2-ylmethyl A.1074 c ₂ h ₅ 5-Methoxy-l, 3,4-oxadiazol-2-ylmethyl A.1075 C ₂ Hs 1,2,4-thiadiazol-3-ylmethyl A.1076 C2H5 5-Chloro-1,2,4-thiadiazol-3-ylmethyl A.1077 C2H5 5-methyl-1,2,4-thiadiazol-3-ylmethyl A.1078 C2H5 1,3,4-Thiadiazol-2-ylmethyl A.1079 C ₂ H ₅ 5-Chloro-1,3,4-thiadiazol-2-ylmethyl A.1080 C2H5 5-methyl-1,3,4-thiadiazol-2-ylmethyl A.1081 C2H5 5-Cyano-1,3,4-thiadiazol-2-ylmethyl A. 1082 C ₂ H ₅ 2- (2'-Pyridinyloxy) eth-l-yl A.1083 C2H5 2- (3'-Pyridinyloxy) eth-1-yl A.1084 C2H5 2- (4'-Pyridinyloxy) eth-l-yl A.1085 C2H5 2- (2'-pyrimidinyloxy) eth-l-yl A.1086 C2H5 2- (4'-pyrimidinyloxy) eth-l-yl A.1087 C2H5 2- (5'-pyrimidinyloxy) eth-l-yl A.1088 c ₂ h ₅ 2- (2'-pyrazinyloxy) eth-l-yl A.1089 C2H5 2- (2'-pyridazinyloxy) eth-l-yl A.1090 -2H5 2- (3'-pyridazinyloxy) eth-l-yl

- Ί% -

Nr. R ² R ⁴ A.1091 c ₂ h ₅ 2- (1 ', 3', 5'-Triazinyloxy) eth-1-yl A.1092 C ₂ H ₅ 2- (5'-methylisoxazole-3'-yloxy) eth-1-yl A.1093 c ₂ h ₅ 2- (5 ' Chlorisoxazol-3'-yloxy) eth-l-yl A.1094 c ₂ h ₅ 2- (2-methoxythiazole-4-yloxy) eth-1-yl A.1095 C ₂ H ₅ 2- (4'-Chlorooxazol-2'-yloxy) eth-1-yl A.1096 c ₂ h ₅ 2- (1'-Phenyl-1'H-1 ', 2', 4'-triazol-3'-yl- oxy) eth-l-yl A.1097 c ₂ h ₅ 2- (L-Phenylpyrazol-3'-yloxy) eth-l-yl A.1098 C ₂ Hs c ₆ h _p A.1099 C ₂ Hs 2-Cl-C ₆ H ₄ A.1100 C ₂ H ₅ 3-Cl-C ₆ H ₄ A. 1101 c ₂ h ₅ 4-Cl-C ₆ H ₄ A.1102 c ₂ h ₅ 2,3-Cl ₂ -C _s H ₃ A. 1103 C ₂ H _p 2,4-Cl ₂ -C ₆ H ₃ A.1104 C ₂ H ₅ 2,5-Cl ₂ -C ₆ H ₃ A.1105 C ₂ Hs 3,4-Cl ₂ -C ₆ H ₃ A.1106 C ₂ Hs 3,5-Cl ₂ -C ₆ H ₃ A.1107 C ₂ Hs 4-CN-C ₆ H ₄ A.1108 c ₂ h ₅ 2-NO ₂ -C ₆ H ₄ A.1109 c ₂ h ₅ 3-NO ₂ -C ₆ H ₄ A.1110 C ₂ Hs 4-NO ₂ -C ₆ H ₄ A.1111 c ₂ h ₅ 2,4 - (NO ₂ ) ₂ -C ₆ H ₃ A.1112 c ₂ h ₅ 2-CH ₃ -C ₆ H ₄ A.1113 C ₂ H ₅ 3-CH ₃ -C ₆ H ₄ A.1114 c ₂ h ₅ 4-CH ₃ -C ₆ H ₄ A.1115 c ₂ h ₅ 2,3- (CH ₃ ) ₂ -C ₆ H ₃ A.1116 c ₂ h _p 2,4- (CH ₃ ) ₂ -C ₆ H ₃ A.1117 c ₂ h ₅ 2,5- (CH ₃ ) ₂ -C ₆ H ₃ A.1118 c ₂ h ₅ 2,6- (CH ₃ ) ₂ -C ₆ H ₃ A.1119 c ₂ h ₅ 2-C ₆ H ₅ -C ₆ H ₄ A.1120 c ₂ h ₅ 3-C ₆ H ₅ -C ₆ H ₄ A.1121 c ₂ h ₅ 4-C ₆ H _with -C ₆ H ₄ A.1122 C ₂ Hs 3-OCI ₃ -C ₆ H ₄ A.1123 C ₂ H _p 4-OCH ₃ -C ₆ H ₄ A.1124 C ₂ H ₅ 3-Acetyl-C 6 H ₄ A.1125 c ₂ h ₅ 4-Acetyl-C 6 H ₄ A.1126 = ₂ H ₅ 3-Methoxycarbonyl-ββ ₄ A.1127 = ₂ H _{5 4-methoxycarbonyl-4} CGH A.1128 7 ₂ H ₅ 3-CF ₃ -C ₆ H ₄

Nr. R ² R ⁴ A.1129 C ₂ H ₅ 4-CF ₃ -C _s H ₄ A.1130 C ₂ Hs 2-Naphthyl A.1131 c ₂ h ₅ 6-chloropyridazine-3-yl A.1132 c ₂ h ₅ 5-Chloro-pyrazin-2-yl A.1133 c ₂ h ₅ Quinolin-2-yl A.1134 c ₂ h ₅ 2,5-Dimethylpyrazin-3-yl A.1135 c ₂ h ₅ Pyrazin-2-y1 A.1136 c ₂ Hs 3-chloropyrid-2-yl A.1137 C ₂ Hs 6-chloropyrid-2-yl A.1138 c ₂ h ₅ 4-Trifluoromethyl, 6-chloropyrid-2-yl A.1139 c ₂ h _p 4-trifluoromethylpyrid-2-yl A.1140 C ₂ H ₅ 6-trifluoromethylpyrid-2-yl A.1141 c ₂ h ₅ 6-methoxypyridin-2-yl A.1142 c ₂ h ₅ 5-chloropyrid-2-yl A.1143 c ₂ h ₅ Pyridin-2-yl A.1144 c ₂ h ₅ Benzothiazol-2-yl A.1145 C ₂ Hs 7-Chloro-quinolin-4-yl A.1146 C ₂ Hs 3-nitro-pyridin-2-yl A. 1147 C ₂ Hs Pyrrole-3-yl A. 1148 c ₂ h ₅ Pyrrol-2-yl A. 1149 c ₂ h ₅ 2,6-Dioctylpyrid-4-yl A.1150 c ₂ h ₅ 5-nitro-pyridin-2-yl A.1151 C ₂ Hs Pyridin-4-yl A.1152 C ₂ Hs Pyridin-3-yl A.1153 c ₂ h ₅ Pyrimidin-2-yl A.1154 c ₂ h ₅ Pyrimidin-4-yl A. 1155 c ₂ Hs Quinazolin-4-yl A. 1156 C ₂ Hs 6-Chloropyrimidin-4-yl A.1157 c ₂ h ₅ 6-Methoxypyrimidin-4-yl A. 1158 c ₂ h ₅ 2,5,6-Trichloro-4-yl A. 1159 c ₂ h ₅ 2,6-dimethyl-pyrimidin-4-yl A.1160 C ₂ H ₅ 2-Methyl, 6-chloropyrimidin-4-yl A.1161 c ₂ h ₅ 2-Methyl, 6-Ethoxy-pyrimidin-4-yl A.1162 c ₂ h _p 4,5,6-trichloro-2-yl A.1163 C ₂ Hs 4,6-Dimethoxy-pyrimidin-2-yl A. 1164 3 ₂ H ₅ 1,6-dimethyl-pyrimidin-2-yl A.1165 = ₂ Hs 1,6-dichloropyrimidine-2-yl A.1166 -2H5 1-Methyl, 6-methoxy-pyrimidin-2-yl A.1167 : ₃ h ₅ 1-Chloro, 6-methoxypyrimidin-2-yl

'in'

Nr. R ² R ⁴ A.1168 C ₂ H ₅ 6-Chloro-quinoxalin-2-yl A.1169 c ₂ h ₅ 3,6-Dichloro-1,2,4-triazin-5-yl A.1170 C2H5 4-Methoxy-l, 3,5-triazin-2-yl A.1171 c ₂ h ₅ 4-Ethoxy-1,3,5-triazin-2-yl; A.1172 C ₂ Hs 4,6-Dichloro-1,3,5-1-triazin-2-yl A.1173 c ₂ h ₅ 4-Ethoxy, 6-Chloro-1,3,5-triazin-2-yl A.1174 c ₂ h ₅ Isoxazol-3-yl A.1175 c ₂ h ₅ Thien-2-yl A.1176 c ₂ h ₅ Fur-2-yl A.1177 C ₂ H ₅ Thiatriazole-5-yl A.1178 c ₂ h ₅ (E) -l-chloropropene-3-yl A.1179 c ₂ h ₅ (E) -4- (4'-Chlorophenyl) but-2-en-1-yl A.1180 C ₂ Hs Propyn-3-yl A.1181 C ₂ Hs Methylcarbonyl A.1182 c ₂ h ₅ Ethylcarbonyl A.1183 C2H5 n Propylcarbonyl A.1184 c ₂ h ₅ i-Propylcarbonyl A.1185 C ₂ Hs n-Butylcarbonyl A.1186 c ₂ Hs p-Butylcarbonyl A.1187 C ₂ Hs i-Butylcarbonyl A.1188 C ₂ Hs t-Butylcarbonyl A.1189 c ₂ Hs n Pentylcarbony1 A.1190 c ₂ h ₅ i -Pentylcarbonyl A.1191 c ₂ h ₅ neo-Pentylcarbonyl A.1192 C ₂ Hs n Hexylcarbony1 A.1193 c ₂ h ₅ n-Octylca rbony1 A.1194 c ₂ h ₅ 1-Propenylcarbonyl A.1195 c ₂ h ₅ 2-Penten-1-yl-carbonyl A.1196 C ₂ Hs 2,5-heptadiene-yl-carbonyl A.1197 c ₂ h ₅ benzoyl A.1198 C ₂ Hs 2-chlorobenzoyl A.1199 C ₂ Hs 3-chlorobenzoyl A.1200 c ₂ h ₅ 4 -Chlorobenzoyl A. 1201 c ₂ h ₅ 2-Cyanobenzoyl A.1202 C ₂ Hs 3-Cyanobenzoyl A.1203 - ₂ h ₅ 4-Cyanobenzoyl A.1204 = ₂ Hs 4-methoxybenzoyl A.1205 3 ₂ H ₅ 2-Pyridylcarbonyl A.1206 3 ₂ H5 3-Pyridylcarbonyl

79ý

Nr. R ² R ⁴ A.1207 c ₂ h ₅ 4-Pyridylcarbony1 A.1208 c ₂ h ₅ 2 -Pyrimidinylcarbonyl A.1209 c ₂ h ₅ 2-Oxazolylcarbonyl A.1210 c ₂ h ₅ 4-Methylisoxazol-5-ylcarbonyl j A.1211 C ₂ H ₅ Methylsulfonyl ’ A.1212 c ₂ h ₅ ethylsulfonyl A.1213 c ₂ h ₅ n-propylsulfonyl A.1214 c ₂ h ₅ i-Propylsulfonyl j A.1215 c ₂ h ₅ n-Butylsulfonyl; A.1216 C ₂ H ₅ t-Butylsulfonyl; A.1217 c ₂ h ₅ n-pentylsulfonyl A.1218 C ₂ H ₅ neo-pentylsulfonyl A.1219 c ₂ h ₅ n Hexy1su1fony1 A.1220 C ₂ H ₅ n-Octylsulfonyl A.1221 c ₂ h ₅ phenylsulfonyl A.1222 C ₂ H ₅ 2-Chlorphenylsulfonyl A.1223 C ₂ III 3-Chlorphenylsulfonyl A.1224 C2H5 4-Chlorphenylsulfonyl A.1225 c ₂ h ₅ 2-Cyanophenylsulfonyl A.1226 C ₂ H5 3-Cyanophenylsulfonyl A.1227 C ₂ Hs 4-Cyanophenylsulfonyl A.1228 C ₂ H ₅ 2-Pyridylsulfonyl A.1229 c ₂ h ₅ 3-Pyridylsulfonyl A.1230 c ₂ h ₅ 4-Pyridylsulfonyl A.1231 c ₂ h ₅ 2-Pyrimidinylsulfonyl A.1232 C ₂ Hs 4-Oxazolylsulfonyl A.1233 C ₂ H _p 5-Chlorothiazol-2-ylsulfonyl A.1234 C ₂ Hs 2 -1-C ₄ H ₉ -C ₆ H ₄ -CH ₂ A.1235 C ₂ H ₅ 3- t C ₄ H ₉ -C ₆ H ₄ -CH ₂ A.1236 c ₂ h ₅ 4-tC ₄ H ₉ -C ₆ H ₄ -CH ₂ A.1237 c ₂ h ₅ 2- (4'-Chloro-thiazol-2'-yloxy) eth-1-yl A.1238 C ₂ Hs 2- (1'-Methylpyrazol-4'-yloxy) eth-1-yl A.1239 c ₂ h ₅ 4-Br-Ce ₄ A.1240 C ₂ H _p 3,5- (CH ₃ ) ₂ -C ₆ H ₃ A.1241 c ₂ h ₅ 4-C ₂ H ₅ -C ₆ H ₄ A.1242 C ₂ Hs 3-Dimethylaminocarbonyl-C 5 H ₄ A.1243 3 ₂ Hs 4-Dimethylaminocarbonyl-C 6 H ₄ A.1244 7 ₂ h ₅ 2-Hydroxyprop-1-yl A.1245 -2H5 5-Hydroxy-2-methylpyrimidin-4-ylmethyl

Nr. R ² R ⁴ A.1246 C ₂ H ₅ [6 - OH, 2 - CH (CH ₃ ) ₂ - pyrimidin - 4 - yl] - CH ₂ A.1247 C ₂ Hs [6-OH, 2-CH (CH ₂ ) ₂ -pyrimidin-4-yl] -CH ₂ A.1248 c ₂ h ₅ 5- (2'-furan) pent-l-yl A.1249 c ₂ h ₅ 5- (2'-N-Methylpyrrol) pent-l-yl A.1250 c ₂ h ₅ [2- (4-Cl-C ₆ H ₄₎ -oxazole-4-yl] _-CH2 A.1251 c ₂ h ₅ 3-CF _3- pyridin-2-yl A.1252 c ₂ h ₅ 5-CF ₃ -pyridin-2-yl A.1253 c ₂ h ₅ 6- (2'-Thienyl) hex-1-yl A.1254 C ₂ Hs (E) -3-chloro-but-2-en-l-yl A.1255 c ₂ h ₅ (Z) -3-chloro-but-2-en-l-yl A.1256 c ₂ h ₅ (E) -2-bromo-but-2-en-l-yl A.1257 c ₂ h ₅ (Z) -2-bromo-but-2-en-l-yl A.1258 c ₂ h ₅ (E) -l-chloro-prop-l-en-3-yl A.1259 C ₂ H ₅ (Z) -l-chloro-prop-l-en-3-yl A.1260 c ₂ h ₅ But-en-3-yl A.1261 c ₂ h ₅ CH ₂ CH ₂ Br A.1262 c ₂ h ₅ CH ₂ CH ₂ CH ₂ Br A.1263 C ₂ Hs CH ₂ CH ₂ CH ₂ CH ₂ Br A.1264 c ₂ h ₅ Methylprop-2-yl A.1265 C ₂ Hs 2-E-thoxyprop-1-yl A.1266 C ₂ Hs 2-isopropoxypropanoic-yl A.1267 c ₂ h ₅ But-in-3-yl A.1268 c ₂ h ₅ But-in-4-yl A.1269 c ₂ h ₅ But-2-yn-4-yl A.1270 C ₂ H ₅ Pent-in-4-yl A.1271 c ₂ h _p Pent-2-yn-4-yl A.1272 c ₂ h ₅ Pent-in-5-yl A.1273 c ₂ h ₅ Pent-2-yn-5-yl A.1274 c ₂ h ₅ E-2-chloro-but-2-en-l-yl A.1275 C ₂ Hs Z-2-chloro-but-2-en-l-yl A.1276 c ₂ h ₅ Z-l-chloro-prop-l-en-3-yl A.1277 c ₂ h ₅ 2-methyl-prop-l-en-3-yl A.1278 = ₂ h ₅ 2-chloro-prop-l-en-3-yl A.1279 2 ₂ H ₅ 2-bromoprop-l-en-3-yl A.1280 - ₂ H5 But-2-en-l-yl A.1281 < 7 ₂ H ₅ But-3-en-l-yl A.1282 ( - ₂ Hs l-Iodprop-l-yn-3-yl A.1283 < - ₂ Hs E-3-bromo-but-2-en-l-yl A.1284 C : ₂ Hs S-3-bromo-but-2-en-l-yl

Nr. R ² R ⁴ A.1285 iC ₃ H ₇ H A.1286 I-C3H7 ch ₃ A.1287 iC ₃ H ₇ C2H5 A.1288 t-c ₃ h ₇ nC ₃ H ₇ A.1289 1-C ₃ H ₇ iC ₃ H ₇ A.1290 1-C ₃ H ₇ cyclopropyl A.1291 t-c ₃ h ₇ I1-C4H9 A.1292 1-C ₃ H ₇ S ”C4H9 A.1293 1-C ₃ H ₇ I-C4H9 A.1294 1-C ₃ H ₇ tC ₄ Hg A.1295 1-C ₃ H ₇ n CSHN A.1296 1-C ₃ H ₇ I-C5H11 A.1297 1-C ₃ H ₇ neo-CSHN A.1298 1-C ₃ H ₇ cyclopentyl A.1299 t-c ₃ h ₇ n-C ₆ H 13 A.1300 1-C ₃ H ₇ cyclohexyl A.1301 1-C ₃ H ₇ nC ₈ Hi ₇ A.1302 1-C ₃ H ₇ CH ₂ CH ₂ Cl A.1303 t-c ₃ h ₇ (CH ₂ ) ₄ Cl A.1304 1-C ₃ H ₇ ch ₂ cn A.1305 1-C ₃ H ₇ ch ₂ ch ₂ cn A.1306 1 ^- C ₃ H ₇ (ch ₂ ) ₃ cn A.1307 1-C ₃ H ₇ (CH ₂ ) ₄ CN A.1308 iC ₃ H ₇ (CH ₂ ) ₆ CN A.1309 1-C ₃ H ₇ Cyclohexylmethyl A.1310 1-C ₃ H ₇ 2-Cyclohexyleth-1-yl A.1311 1-C ₃ H ₇ Cyclopropylme thyl A.1312 ic ₃ h ₇ 2-Cyclopropyleth-1-yl A.1313 1-C ₃ H ₇ 2-methoxyethyl-1-yl A.1314 t-c ₃ h ₇ 2-ethoxyethanol-1-yl A.1315 t-c ₃ h ₇ 2-Isopropoxyeth-1-yl A.1316 1-C ₃ H ₇ 3-methoxypropyl-1-yl A.1317 1-C ₃ H ₇ 3-Ethoxyprop-1-yl A.1318 1-C ₃ H ₇ 3-isopropoxypropanoic-yl A.1319 t-c ₃ h ₇ 4methoxybut-1-yl A.1320 í ~ c ₃ h ₇ 4-Isopropoxybut-1-yl A.1321 _β -C ₃ H ₇ Propen-3-yl A.1322 1-C ₃ H ₇ But-2-en-1-yl A.1323 1-C ₃ H ₇ 3-methyl-but-2-en-1-yl

-2 ¢ 2-

Nr. R ² R ⁴ A.1324 iC ₃ H ₇ 2-Vinyloxyeth-1-yl A.1325 Í ~ C ₃ H ₇ Allyloxyeth-1-yl A.1326 ° C ₃ H ₇ 2-Trifluoromethoxyeth-1-yl A.1327 Ϊ — C ₃ H ₇ 3-Trifluoromethoxyprop-1-yl A.1328 i — C ₃ H ₇ 4-Difluoromethoxybut-1-yl A.1329 iC ₃ H ₇ Hydroxycarbonylmethyl A. 1330 iC ₃ H ₇ Methoxycarbonylmethyl A.1331 iC ₃ H ₇ Aminocarbonyme methyl A.1332 iC ₃ H ₇ N-Methylaminocarbonylmethyl A.1333 1-C ₃ H ₇ Ν, Ν-methyl-Dimethylaminocarbonyl A.1334 1-C ₃ H ₇ 2-Hydroxycarbonyleth-1-yl A.1335 1-C ₃ H ₇ 2-Methoxycarbonyleth-1-yl A. 1336 1-C ₃ H ₇ 2-Aminocarbonyleth-yl A.1337 1-C ₃ H ₇ 2 -N-Methylaminocarbonyleth-1-yl A.1338 t-c ₃ h ₇ 2-Dimethylaminocarbonyleth-1-yl A.1339 1-C ₃ H ₇ 2-aminoethyl-1-yl A.1340 1-C ₃ H ₇ 2-amino-prop-1-yl A.1341 I-C3H7 4-Aminobut-1-yl A.1342 iC ₃ H ₇ 3-Dimethylaminoprop-1-yl A.1343 CI-C ₃ H ₇ 4-Aminothiocarbonylbut-1-yl A.1344 iC ₃ H ₇ 2-oxo-propyl A.1345 iC ₃ H ₇ cyclohexyl A. 1346 t-c ₃ h ₇ cyclopropyl A.1347 1-C3H7 cyclopentyl A.1348 iC ₃ H ₇ 2-Methoxyiminoprop-1-yl A.1349 iC ₃ H ₇ 2-Methoxyiminoeth-1-yl A.1350 iC ₃ H ₇ 6-Aminocarbonylhex-1-yl A.1351 CI-C ₃ H ₇ 3-Aminothiocarbonylprop-1-yl A.1352 iC ₃ H ₇ 2-Aminothiocarbonyleth-1-yl · A.1353 1-C3H7 Aminothiocarbonylmethyl A.1354 I-C3H7 4- (N, N-Dimethylamino) but-1-yl A.1355 iC ₃ H ₇ 2- (Methylthio) eth-1-yl A. 1356 1-C ₃ H ₇ 2- (Methylsulfonyl) eth-1-yl A.1357 1-C ₃ H ₇ 4- (Methylthio) prop-1-yl A.1358 1-C ₃ H ₇ 4- (methylsulfonyl) prop-l-yl A.1359 1-C ₃ H ₇ Benyz1 A.1360 I-C3H7 2-FC ₆ H ₄ -CH ₂ A.1361 1-C ₃ H ₇ 3-FC ₆ H ₄ -CH ₂ A.1362 ~ c ₃ h ₇ t-fc ₆ h ₄ -ch ₂

Nr. R 2 R ⁴ A.1363 I-C3H7 2,3-F ₂ -C ₆ H ₃ -CH ₂ A.1364 I-C3H7 2,4-F ₂ -C ₆ H ₃ -CH ₂ A.1365 I-C3H7 2,5-F ₂ -C ₆ H ₃ -CH ₂ A.1366 I-C3H7 2,6-F ₂ -C ₆ H ₃ -CH ₂ A.1367 I-C3H7 3,4-F ₂ -C ₆ H ₃ -CH ₂ A.1368 1-C3H7 3,5-F ₂ -C ₆ H ₃ -CH 2 A.1369 I-C3H7 2-C 1 -C ₆ H ₄ -CH ₂ A.1370 I-C3H7 3-Cl-C ₆ H ₄ CH ₂ A.1371 I-C3H7 4-C 1 -C ₆ H ₄ -CH ₂ A.1372 I-C3H7 2,3-Cl ₂ -C ₆ H ₃ -CH ₂ A.1373 1-C3H7 2,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.1374 I-C3H7 2,5-Cl ₂ -C ₆ H ₃ -CH ₂ A.1375 I-C3H7 2,6-Cl ₂ -C ₆ H ₃ -CH ₂ A.1376 iC ₃ H ₇ 3,4-Cl ₂ -C ₆ H ₃ -CH ₂ A. 1377 I-C3H7 3.5-Cl ₂ -C ₆ H ₃ -CH ₂ A.1378 I-C3H7 2,3,4-Cl ₃ -C ₆ H ₂ -CH ₂ A.1379 I-C3H7 2,3,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.1380 I-C3H7 2,3,6-Cl ₃ -C ₆ H ₂ -CH ₂ A.1381 iC ₃ H ₇ 2,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.1382 I-C3H7 2,4,6-Cl ₃ -C ₆ H ₂ -CH ₂ A.1383 I-C3H7 3,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.1384 I-C3H7 2 -Br-C ₆ H ₄ -CH ₂ A.1385 I-C3H7 3-Br-C ₆ H ₄ CH ₂ A.1386 I-C3H7 4 -Br-C ₆ H ₄ CH ₂ A.1387 ic ₃ H ₆ 2,3-Br ₂ -C ₆ H ₃ -CH ₂ A.1388 t-c ₃ h ₇ 2,4-Br ₂ -C ₆ H ₃ -CH ₂ A.1389 ic ₃ h ₇ 2,5-Br ₂ -C ₆ H ₃ -CH ₂ A.1390 1-C ₃ H ₇ 2,6-Br 2 -C ₆ H ₃ -CH 2 A.1391 t-c ₃ h ₇ 3,4-Br ₂ -C ₆ H ₃ -CH ₂ A.1392 t-c ₃ h ₇ 3,5-Br ₂ -C ₆ H ₃ -CH 2 A.1393 CI-C ₃ H ₇ 2-F, 3-Cl-C ₆ H ₃ CH ₂ A.1394 t-c ₃ h ₇ 2-F, 4-C1-C ₆ H ₃ CH ₂ A.1395 t-c ₃ h ₇ 2-F, 5-Cl-C ₆ H ₃ CH ₂ A.1396 t-c ₃ h ₇ 2-F, 3-Br-C ₆ H ₃ CH ₂ A.1397 t-c ₃ h ₇ 2-F, 4-Br-C ₆ H ₃ CH ₂ A.1398 1-C ₃ H ₇ 2-F, 5-Br-C ₆ H ₃ CH ₂ A.1399 1-C ₃ H ₇ 2-C1, 3-Br-C ₆ H ₃ CH ₂ A.1400 iC ₃ H ₇ 2-C1, 4-Br-C ₆ H ₃ CH ₂ A.1401 t-c ₃ h ₇ 2-C1, 5-Br-C ₆ H ₃ -CH ₂ - -----

- -

Nr. R ² R ⁴ A.1402 iC ₃ H ₇ 3-F, 4-Cl-C ₆ H ₃ CH ₂ A.1403 t-c ₃ h ₇ 3-F, 5-C 1 -C ₆ H ₃ -CH ₂ A.1404 1-C ₃ H ₇ 3-F, 6-C 1 -C ₆ H ₃ -CH ₂ A.1405 t-c ₃ h ₇ 3-F, 4-Br-C ₆ H ₃ CH ₂ A. 1406 1-C ₃ H ₇ 3-F, 5-Br-C ₆ H ₃ CH ₂ A.1407 1-C ₃ H ₇ 3-F, 6-Br-C ₆ H ₃ CH ₂ A.1408 t-c ₃ h ₇ 3-C1, 4-Br-C ₆ H ₃ CH ₂ A.1409 1-C ₃ H ₇ 3-Cl, 5-Br-C ₆ H ₃ -CK ₂ A.1410 1-C ₃ H ₇ 3-C1, 6-Br-C ₆ H ₃ CH ₂ A.1411 1-C ₃ H ₇ 4-F, 5-C 1-C ₆ H ₃ CH ₂ A.1412 1-C ₃ H ₇ 4-F, 6-Cl-C ₆ H ₃ CH ₂ A.1413 1-C ₃ H ₇ 4-F, 5-Br-C ₆ H ₃ CH ₂ A.1414 1-C ₃ H ₇ 4-F, 6-Br-C ₆ H ₃ CH ₂ A.1415 1-C ₃ H ₇ 4-C1, 5-Br-C ₆ H ₃ CH ₂ A.1416 1-C ₃ H ₇ 5-F, 6-Cl-C ₆ H ₃ CH ₂ A.1417 1-C ₃ H ₇ 5-F, 6-Br-C ₆ H ₃ CH ₂ A.1418 1-C ₃ H ₇ 5-C1, 6-Br-C ₆ H ₃ CH ₂ A.1419 1-C ₃ H ₇ 3-Br, 4-C1, 5-Br-C ₆ H ₂ CH ₂ A.1420 1-C ₃ H ₇ 2 -CN-C ₆ H ₄ -CH ₂ A.1421 1-C ₃ H ₇ 3 -CN-C 6 H 4 -CH ₂ A.1422 1-C ₃ H ₇ 4 -CN-C ₆ H ₄ -CH ₂ A.1423 t-c ₃ h ₇ 2-NO ₂ -C ₆ H ₄ -CH ₂ A.1424 1-C ₃ H ₇ 3-NO ₂ -C ₆ H ₄ -CH ₂ A.1425 1-C ₃ H ₇ 4-NO ₂ -C ₆ H ₄ -CH ₂ A.1426 1-C ₃ H ₇ 2-CH ₃ -C ₆ H ₄ -CH ₂ A.1427 t-c ₃ h ₇ 3-CH ₃ -C ₆ H ₄ -CH ₂ A.1428 1-C ₃ H ₇ 4-CH ₃ -C ₆ H ₄ -CH ₂ A.1429 t-c ₃ h ₇ 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1430 xc ₃ h ₇ 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1431 1-C ₃ H ₇ 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1432 ic ₃ h ₇ 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1433 iC ₃ H ₇ 3.4; (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1434 1-C ₃ H ₇ 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1435 1-C ₃ H ₇ 2-C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.1436 1-C ₃ H ₇ 3-C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.1437 iC ₃ H ₇ 4-C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.1438 t-c ₃ h ₇ 2-C ₃ H ₇ -C ₆ H 4 -CH ₂ A.1439 t-c ₃ h ₇ i - ic ₃ h _{7 -} c ₆ h _{4 -} ch ₂ A.1440 CI-C ₃ H ₇ i-i-c ₃ h _7- c ₆ h ₄ -ch ₂

- Ζο5 ~ -

Nr. R ² R ⁴ A.1441 I-C3H7 2-Cyclohexyl-C 6 H 4 -CH 2 A.1442 I-C3H7 _{3-Cyclohexyl-C6H4-CH2} A.1443 I-C3H7 4 - _{Cyclohexyl-C6H4-CH2} A.1444 I-C3H7 2-Vinyl -C ₆ H ₄ -CH ₂ A.1445 I-C3H7 3-vinyl-C ₆ H ₄ CH ₂ A.1446 I-C3H7 4-Vinyl -C ₆ H ₄ -CH ₂ A.1447 I-C3H7 2-Allyl-C ₆ H ₄ -CH ₂ A.1448 I-C3H7 3-Allyl-C ₆ H ₄ CH ₂ A.1449 I-C3H7 4-Allyl-C ₆ H ₄ CH ₂ A.1450 I-C3H7 2-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.1451 I-C3H7 3-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.1452 I-C3H7 4-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.1453 I-C3H7 3-CH3, 5-1-C ₄ H _9, -C _p H ₃ CH ₂ A.1454 I-C3H7 2-OH-C ₆ H ₄ CH ₂ A.1455 xC ₃ H ₇ 3-OH-C ₆ H ₄ CH ₂ A.1456 I-C3H7 4-OH-C ₆ H ₄ CH ₂ A.1457 I-C3H7 2-OCH 3 -C ₆ 14 -CH ₂ A.1458 I-C3H7 3-OCH ₃ -C ₆ H ₄ -CH 2 A.1459 I-C3H7 4-OCH 3 -C ₆ H ₄ -CH ₂ A.1460 I-C3H7 2,3- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1461 X-C3H7 2,4- (OCH ₃ ) ₂ -C ₆ H 3 -CH ₂ A.1462 I-C3H7 2,5 - (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1463 X-C3H7 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1464 X-C3H7 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.1465 C3H7 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH ₂ A.1466 xC ₃ H ₇ 2-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.1467 I-C3H7 3-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.1468 xC ₃ H ₇ 4-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.1469 I-C3H7 2-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.1470 X-C3H7 3-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.1471 ic ₃ H ₆ 4-O- (nC ₃ H ₇ ) -C _G H ₄ -CH ₂ A.1472 X-C3H7 2-O- (iC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A. 1473 X-C3H7 3-O- (iC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.1474 I-C3H7 4-O- (iC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.1475 X-C3H7 4-O- (nC ₄ Hg) -C ₆ H ₄ -CH ₂ A.1476 X-C3H7 3-O- (t C ₄ H ₉ ) -C ₆ H ₄ -CH ₂ A. 1477 C3H7 4-O- (nC ₆ H ₁₃ ) -C ₆ H ₄ -CH ₂ A.1478 I-C3H7 2-Ο-Allyl-C ₆ H ₄ -CH ₂ A.1479 I-C3H7 3-Ο-Allyl-C ₆ H ₄ -CH ₂

~ 7 >έ> -

Nr. R ² R ⁴ A.1480 iC ₃ H ₇ 4-O-allyl-C ₆ H ₄ -CH ₂ | A.1481 iC ₃ H ₇ 2-CF ₃ -C ₆ H ₄ -CH ₂ I A.1482 iC ₃ H ₇ 3-CF ₃ -C ₆ H ₄ -CH ₂ L A.1483 t-c ₃ h ₇ 4-CF ₃ -C ₆ H ₄ -CH ₂ L A.1484 1-C ₃ H ₇ 2-Acetyl-C 6 H ₄ -CH ₂ | A.1485 iC ₃ H ₇ 3-Acetyl-C ₁ H ₄ -CH ₂ A.1486 t-c ₃ h ₇ 4-Acetyl-C ₆ H ₄ -CH ₂ | A.1487 t-c ₃ h _{7 2-methoxycarbonyl-4} CGH _-CH2 | A.1488 1-C ₃ H _{7 3-methoxycarbonyl-4} CGH _-CH2 | A.1489 1-C ₃ H ₇ Methoxycarbonyl-4-C 6 H ₄ -CH ₂ | A.1490 1-C ₃ H ₇ 2-Aminocarbonyl-C 8 H ₄ -CH ₂ L A.1491 1-C ₃ H ₇ 3-Aminocarbonyl-C 8 H ₄ -CH ₂ J A.1492 iC ₃ H ₇ 4-Aminocarbonyl-C 8 H ₄ -CH ₂ j A.1493 t-c ₃ h ₇ 2-Dimethylaminocarbonyl-C 6 H ₄ -CH ₂ I A.1494 1-C ₃ H ₇ 3-Dimethylaminocarbonyl-C 6 H ₄ -CH ₂ J A.1495 1-C ₃ H ₇ 4-Dimethylaminocarbonyl -C ₆ H ₄ -CH ₂ I A.1496 t-c ₃ h ₇ 2- (N-Methylaminocarbonyl) -C ₆ H ₄ -CH ₂ L A.1497 1-C ₃ H ₇ 3- (N-Methylaminocarbonyl) -C 6 H ₄ -CH ₂ | A.1498 I-C3H7 4- (N-Methylaminocarbonyl) -C ₆ H ₄ -CH ₂ J A.1499 ic ₃ H ₆ 2 -h ₂ nc ₆ h ₄ -ch ₂ j A.1500 1-C ₃ H ₇ 3 -H ₂ NC ₆ H ₄ -CH ₂ J A.1501 1-C ₃ H ₇ 4-H ₂ NC ₆ H ₄ -CH ₂ J A.1502 1-C ₃ H ₇ 2-Aminothiocarbonyl-C 6 H ₄ -CH ₂ J A.1503 1-C ₃ H ₇ 3-Aminothiocarbonyl-C 6 H ₄ -CH ₂ S A.1504 iC ₃ H ₇ 4-Aminothiocarbonyl-C 6 H ₄ -CH ₂ S A.1505 1-C ₃ H ₇ 2-methoxyimino-methyl-C ₆ H ₄ CH ₂ S A.1506 t-c ₃ h ₇ 3-methoxyimino-methyl-C 6 H ₄ -CH ₂ S A.1507 iC ₃ H ₇ 4-methoxyimino-methyl-C 6 H ₄ CH ₂ 1 A.1508 iC ₃ H ₇ 2-Formyl-C 6 H ₄ -CH ₂ L A.1509 iC ₃ H ₇ 3-Formyl-C 8 H ₄ -CH ₂ I A.1510 CI-C ₃ H ₇ 4-Formyl-C 6 H ₄ -CH ₂ J A.1511 ic ₃ h ₇ 2- (1'-Methoxyiminoeth-1'-yl) -C ₆ H ₄ -CH ₂ I A.1512 1-C ₃ H ₇ 3- (1'-Methoxyiminoeth-1'-yl) -C ₆ H ₄ -CH ₂ J A.1513 1-C ₃ H ₇ 4- (1'-Methoxyiminoeth-1'-yl) -CeH ₄ -CH ₂ A.1514 1-C ₃ H ₇ 2-SCH ₃ -C ₆ H ₄ -CH ₂ J A.1515 iC ₃ H ₇ 3-sch ₃ -c ₆ h ₄ -ch ₂ J A.1516 1-C ₃ H ₇ 4 -SCH ₃ -C ₆ H ₄ -CH ₂ j A.1517 t-c ₃ h ₇ 2-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ J A.1518 i ~ C ₃ phi ₇ 3-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ J

'Ζη-

Nr. R ² R ⁴ A.1519 I-C3H7 4-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ A.1520 t-c ₃ h ₇ 2-OCF ₃ -C ₆ H ₄ -CH ₂ A.1521 t-c ₃ h ₇ 3-OCF ₃ -C ₆ H ₄ -CH ₂ A.1522 1-C ₃ H ₇ 4-OCF ₃ -C ₆ H ₄ -CH ₂ A.1523 iC ₃ H ₇ 2-OCHF ₂ -C ₆ H ₄ -CH ₂ A.1524 1-C ₃ H ₇ 3-OCHF ₂ -C ₆ H ₄ -CH ₂ A.1525 iC ₃ H ₇ 4 -OCHF ₂ -C _S H ₄ CH ₂ A.1526 iC ₃ H ₇ 3-CF ₃ , 4-OCF ₃ -C ₆ H ₃ -CH ₂ A.1527 t-c ₃ h _{7 1-Naphthyl-CH2} A.1528 t-c ₃ h ₇ 2 -Naphthyl-CH ₂ A.1529 1-C ₃ H ₇ 2-Phenoxyeth-1-yl A.1530 1-C ₃ H ₇ 2- (2-Chlorphenoxy) eth-1-yl A.1531 1-C ₃ H ₇ 2- (3'-Chlorphenoxy) eth-1-yl A.1532 1-C ₃ H ₇ 2- (4'-Chlorphenoxy) eth-1-yl A.1533 1-C ₃ H ₇ 2- (3 ', 5'-Dichlorophenoxy) eth-1-yl A.1534 1-C ₃ H ₇ 2- (2'-Cyanophenoxy) eth-l-yl A.1535 1-C ₃ H ₇ 2- (3'-Cyanophenoxy) eth-l-yl A.1536 1-C ₃ H ₇ 2- (4'-Cyanophenoxy) eth-1-yl A.1537 1-C ₃ H ₇ 2- (2'-Methylphenoxy) eth-1-yl A.1538 1-C ₃ H ₇ 2- (3'-methylphenoxy) eth-1-yl A.1539 t-c ₃ h ₇ 2- (4'-methylphenoxy) eth-1-yl A.1540 t-c ₃ h ₇ 2- (3 ' 1-Butylphenoxy) eth-l-yl A.1541 CI-C ₃ H ₇ 2- (4'-t-Butylphenoxy) eth-l-yl A.1542 CI-C ₃ H ₇ 2- (2'-Nitrophenoxy) eth-1-yl A.1543 1-C ₃ H ₇ 2- (3'-Nitrophenoxy) eth-l-yl A.1544 t-c ₃ h ₇ 2- (4'-Nitrophenoxy) eth-l-yl A.1545 t-c ₃ h ₇ 2- (2-methoxyphenoxy) eth-l-yl A.1546 t-c ₃ h ₇ 2- (3'-methoxyphenoxy) eth-1-yl A.1547 1-C ₃ H ₇ 2- (4'-methoxyphenoxy) eth-l-yl A.1548 1-C ₃ H ₇ 2- (2 ' Trifluormethylphenoxy) eth-1-yl A.1549 t-c ₃ h ₇ 2- (3 ' Trifluormethylphenoxy) eth-l-yl A.1550 t-c ₃ h ₇ 2- (4'-Trifluormethylphenoxy) eth-1-yl A.1551 1-C ₃ H ₇ 2- (2'-Acetylphenoxy) eth-1-yl A.1552 iC ₃ H ₇ 2- (3'-Acetylphenoxy) eth-l-yl A.1553 t-c ₃ h ₇ 2- {4'-Acetylphenoxy) eth-l-yl A.1554 1-C ₃ H ₇ 2- (2'-methoxycarbonyl) eth-1-yl A.1555 t-c ₃ h ₇ 2- (3'-methoxycarbonyl) eth-1-y1 A. 1556 t-c ₃ h ₇ 2- (4'-methoxycarbonyl) eth-1-yl A. 1557 t-c ₃ h ₇ 2- (2'-Dimethylaminocarbonyl) eth-1-yl

Nr. R ² R ⁴ A.1558 I-C3H7 2- (3'-Dimethylaminocarbonyl) eth-1-yl A.1559 I-C3H7 2- (4'-Dimethylaminocarbonyl) eth-1-yl A.1560 I-C3H7 2- (2'-Aminothiocarbonyl) eth-1-yl A.1561 I-C3H7 2- (3'-Aminothiocarbonyl) eth-1-yl A.1562 I-C3H7 2- (4'-Aminothiocarbonyl) eth-1-yl A.1563 I-C3H7 2- (2 * methylsulfonylbenzoic) eth-1-yl A.1564 I-C3H7 2- (3'-Methylsulfonyl) eth-1-yl A.1565 iC ₃ H ₇ 2- (4'-methylsulfonyl) eth-1-yl A. 1566 iC ₃ H ₇ 3-Phenoxyprop-1-yl A.1567 I-C3H7 3- (2'-Chloro-phenoxy) -prop-1-yl A.1568 iC ₃ H ₇ 3- (3'-Chlorophenoxy) prop-1-yl A.1569 I-C3H7 3- (4'-Chlorphenoxy) prop-1-yl A.1570 I-C3H7 3- (3 ', 5', Dichlorophenoxy) prop-1-yl A. 1571 I-C3H7 3- (2'-Cyanophenoxy) prop-1-yl A.1572 iC ₃ H ₇ 3- (3'-Cyanophenoxy) prop-1-yl A.1573 1-C ₃ H ₇ 3- (4'-Cyanophenoxy) prop-1-yl A.1574 1-C ₃ H ₇ 3- (2'-Methylphenoxy) prop-1-yl A.1575 I-C3H7 3- (3'-Methylphenoxy) prop-1-yl A.1576 iC ₃ H ₇ 3- (4'-Methylphenoxy) prop-1-yl A. 1577 1-C ₃ H ₇ 3- (2'-Methoxyphenoxy) prop-1-yl A.1578 t-c ₃ h ₇ 3- (3'-Methoxyphenoxy) prop-1-yl A.1579 1-C ₃ H ₇ 3- (4'-Methoxyphenoxy) prop-1-yl A.1580 t-c ₃ h ₇ 3- (2'-Trifluoromethylphenoxy, prop-1-yl) A.1581 1-C ₃ H ₇ 3- (3'-Trifluoromethylphenoxy) prop-1-yl A.1582 t-c ₃ h ₇ 3- (4'-Trifluoromethylphenoxy) prop-1-yl A.1583 1-C ₃ H ₇ 4-Phenoxy-but-1-yl A.1584 iC ₃ H ₇ 2-Phenyleth-1-yl A.1585 t-c ₃ h ₇ 2- (2'-Chlorophenyl) eth-1-yl A.1586 t-c ₃ h ₇ 2- (3'-Chlorophenyl) eth-1-yl A.1587 1-C ₃ H ₇ 2- (4'-Chlorophenyl) eth-1-yl A.1588 1-C ₃ H ₇ 2- (3 ', 5'-Dichlorophenyl) eth-1-yl A.1589 t-c ₃ h ₇ 2- (2'-Cyanophenyl) eth-1-yl A.1590 1-C ₃ H ₇ 2- (3'-Cyanophenyl) eth-1-yl A.1591 t-c ₃ h ₇ 2- (4'-Cyanophenyl) eth-1-yl A.1592 1-C ₃ H ₇ 2- (2'-Methylphenyl) eth-1-yl A.1593 1-C ₃ H ₇ 2- (3'-Methylphenyl) eth-1-yl A. 1594 1-C ₃ H ₇ 2- (4'-Methylphenyl) eth-1-yl A.1595 t-c ₃ h ₇ 2- (2'-Methoxyphenyl) eth-1-yl A.1596 t-c ₃ h ₇ 2- (3'-Methoxyphenyl) eth-1-yl

Nr. R ² R ⁴ A.1597 I-C3H7 2- (4'-Methoxyphenyl) eth-1-yl A.1598 iC ₃ H ₇ 2- (2'-Trifluoromethylphenyl) eth-1-yl A.1599 1-C ₃ H ₇ 2- (3 ' Trifluormethylphenyl) eth-1-yl A.1600 t-c ₃ h ₇ 2- (4'-Trifluoromethylphenyl) eth-1-yl A.1601 t-c ₃ h ₇ 3-Phenylprop-1-yl A.1602 1-C ₃ H ₇ 3- (2'-Chloro-phenyl) -prop-1-yl A.1603 1-C ₃ H ₇ 3- (3'-Chlorophenyl) prop-1-yl A.1604 t-c ₃ h ₇ 3- (4'-Chloro-phenyl) -prop-1-yl A.1605 1-C ₃ H ₇ 3- (2'-Cyanophenyl) prop-1-yl A.1606 t-c ₃ h ₇ 3- (3'-Cyanophenyl) prop-1-yl A.1607 1-C ₃ H ₇ 3- (4'-Cyanophenyl) prop-1-yl A.1608 I-C3H7 3- (2'-Trifluoromethylphenyl) prop-1-yl A.1609 iC ₃ H ₇ 4-Phenylbut-1-yl A.1610 t-c ₃ h ₇ 4- (4'-Chloro-phenyl) -but-1-yl A.1611 ° C ₃ h ₇ 6 · (4'-Chlorphenyl) hex-1-y1 A.1612 1-C ₃ H ₇ 2 -Pyridylmethyl A.1613 1-C ₃ H ₇ 3-pyridylmethyl A.1614 1-C ₃ H ₇ 4-Pyridylmethyl A.1615 1-C ₃ H ₇ 4-Chloro-pyridin-2-ylmethyl A.1616 1-C ₃ H ₇ 5-Chloropyridin-2-ylmethyl A.1617 1-C ₃ H ₇ 6-Chloro-pyridin-2-ylmethyl A.1618 1-C ₃ H ₇ 5-Chloro-pyridin-3-ylmethyl A.1619 t-c ₃ h ₇ 6-Chloropyridin-3-ylmethyl A.1620 1-C ₃ H ₇ 2-Chloro-pyridin-4-ylmethyl A.1621 1-C ₃ H ₇ 2-pyrimidinylmethyl A.1622 1-C3H7 4-Chloropyrimidin-2-ylmethyl A.1623 iC ₃ H ₇ 5-Chloropyrimidin-2-ylmethyl A.1624 1-C ₃ H ₇ 2-Chloropyrimidin-4-ylmethyl A.1625 t-c ₃ h ₇ 6-Chloro-pyrimidin-4-ylmethyl A.1626 ic ₃ h ₇ 2-Chloropyrimidin-5-ylmethyl A.1627 1-C ₃ H ₇ 4-Pyridazinylmethyl A.1628 1-C ₃ H ₇ 2-pyrazinylmethyl A.1629 iC ₃ H ₇ 5-Chloro-pyrazin-2-ylmethyl A.1630 t-c ₃ h ₇ 6-Chloro-pyrazin-2-ylmethyl A.1631 i — c ₃ h ₇ 3-Pyridazinylmethyl A.1632 1-C ₃ H ₇ 6-chloropyridazine-3-ylmethyl A.1633 IC ₃ H ₇ 1,3,5-Triazinylmethyl A.1634 1-C ₃ H ₇ 2-furylmethyl A.1635 1-C ₃ H ₇ 3-furylmethyl

Λ- ίν -

Nr. R ² R ⁴ A.1636 iC ₃ H ₇ 4-Bromofur-2-ylmethyl A.1637 I-C3H7 5-chloro-furo-2-ylmethyl A.1638 I-C3H7 2-thienylmethyl A.1639 I-C3H7 3-thienylmethyl A.1640 I-C3H7 5-methyl-thien-3-ylmethyl A.1641 I-C3H7 5-Chlorothien-2-ylmethyl A.1642 I-C3H7 2-Chlorothien-4-ylmethyl A.1643 I-C3H7 2-pyrrolylmethyl A.1644 I-C3H7 3-Pyrylmethyl1 A.1645 I-C3H7 2-oxazolylmethyl A.1646 I-C3H7 4-Methyl-oxazol-2-ylmethyl A.1647 I-C3H7 5-Methyl-oxazol-2-ylmethyl A.1648 I-C3H7 4-chlorooxazole-2-ylmethyl A.1649 1-C3H7 5-chlorooxazole-2-ylmethyl A.1650 ic ₃ H ₆ 4-oxazolylmethyl A.1651 I-C3H7 2-Methyloxazol-4-ylmethyl A.1652 I-C3H7 5-Methyl-oxazol-4-ylmethyl A.1653 I-C3H7 2-chlorooxazole-4-ylmethyl A.1654 I-C3H7 5-chlorooxazole-4-ylmethyl A.1655 I-C3H7 5-Oxazolylmethyl A.1656 X-C3H7 2-Methyl-oxazol-5-ylmethyl A.1657 I-C3H7 4-Methyl-oxazol-5-ylmethyl A.1658 I-C3H7 2-Chlorooxazol-5-ylmethyl A.1659 I-C3H7 4-chlorooxazole-5-ylmethyl A.1660 I-C3H7 2-thiazolylmethyl A.1661 I-C3H7 4-Methyl-thiazol-2-ylmethyl A.1662 I-C3H7 5-Methylthiazol-2-ylmethyl A.1663 I-C3H7 4-Chlorothiazol-2-ylmethyl A.1664 I-C3H7 5-Chloro-thiazol-2-ylmethyl A.1665 I-C3H7 4-thiazolylmethyl A.1666 I-C3H7 2-Methylthiazol-4-ylmethyl A.1667 I-C3H7 5-Methylthiazol-4-ylmethyl A.1668 I-C3H7 2-Chloro-thiazol-4-ylmethyl A.1669 I-C3H7 5-Chlorothiazol-4-ylmethyl A.1670 I-C3H7 5thiazolylmethyl A.1671 - ^- C3H ₇ 2-Methylthiazol-5-ylmethyl A.1672 L-C3H7 1-Methylthiazol-5-ylmethyl A.1673 L-C3H7 2-Chlorothiazol-5-ylmethyl A.1674 .-C3H7 l-Chloro-thiazol-5-ylmethyl

- /// Nr.

A.1675

A.1676

A.1677

A.1678

A.1679

A.1680

A.1681

A.1682

A.1683

A.1684

A.1685

A.1686

R ²

I-C3H7

I-C3H7

I-C3H7

I-C3H7

C ₃ H ₇ Cl ₃ H ₇

H-C ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ i C ₃ H ₇

I-C3H7

A.1687 iC ₃ H ₇

A.1688

A.1689

A.1690

A.1691

A.1692

A.1693

A.1694

A.1695

A.1696

A.1697

A.1698

A.1699

A.1700

A.1701

A.1702

A.1703

A.1704

A.1705

A.1706

A.1707

A.1708

A.1709 .1710 .1711 .1712

1713

1-C3H7 iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇

I-C3H7 iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇

I-C3H7

I-C3H7

I-C3H7 iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇

I-C3H7 iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇ iC ₃ H ₇

3-isoxazolylmethyl

R ⁴

-Methylisoxazol-3-ylmethyl

5-Methyl-isoxazol-3-ylmethyl

4-Chlorisoxazol-3-ylmethyl

5-Chlorisoxazol-3-ylmethyl

-Isoxazolylmethyl

-Methylisoxazol-4-ylmethyl

-Methylisoxazol-4-ylmethyl

3-Chlorisoxazol-4-ylmethyl

-Chloroisoxazol-4-ylmethyl

-Isoxazolylmethyl

3-Methylisoxazol-5-ylmethyl

4-Methylisoxazol-5-ylmethyl

3-Chloroisoxazol-5-ylmethyl

-Chloroisoxazol-5-ylmethyl

-Isothiazolylmethyl

4-isothiazolin-3-ylmethyl

5-Methylisothiazol-3-ylmethyl

4-Chlorisothiazol-3-ylmethyl

5-Chlorisothiazol-3-ylmethyl

4-Isothiazolylmethyl

3-methylisothiazol-4-ylmethyl

5-Methylisothiazol-4-ylmethyl

3-Chlorisothiazol-4-ylmethyl

5-Chlorisothiazol-4-ylmethyl

5-Isothiazolylmethyl

3-methylisothiazol-5-ylmethyl

-Methylisothiazol-5-ylmethyl

3-Chloroisothiazol-5-ylmethyl

-Chloroisothiazol-5-ylmethyl Imidazolylmethyl

Phenylpyrazol-3-ylmethyl

Methylimidazol-4-ylmethyl 1 'phenyl 1,2,4-triazol-3-ylmethyl

1,2,4-oxadiazol-3-ylmethyl

5-chloro-1,2,4-oxadiazol-3-ylmethyl

5-methyl-l, 2,4-oxadiazol-3-ylmethyl

- Trifluoromethyl-1,2,4-oxadiazol-3-ylmethyl

1,3,4-oxadiazol-2-ylmethyl

- L '

Nr. R ² R ⁴ A.1714 iC ₃ H ₇ 5-chloro-1,3,4-oxadiazol-2-ylmethyl A.1715 XC ₃ H ₇ 5-Methyl-1,3,4-oxadiazol-2-ylmethyl A.1716 i — C ₃ H ₇ 5-Methoxy-l, 3,4-oxadiazol-2-ylmethyl A.1717 I-C3H7 1,2,4-thiadiazol-3-ylmethyl A.1718 iC ₃ H ₇ 5-Chloro-1,2,4-thiadiazol-3-ylmethyl A.1719 iC ₃ H ₇ 5-methyl-1,2,4-thiadiazol-3-ylmethyl A.1720 1-C ₃ H ₇ 1,3,4-Thiadiazol-2-ylmethyl A.1721 1-C ₃ H ₇ 5-Chloro-1,3,4-thiadiazol-2-ylmethyl A.1722 1-C ₃ H ₇ 5-methyl-1,3,4-thiadiazol-2-ylmethyl A.1723 I-C3H7 5-Cyano-1,3,4-thiadiazol-2-ylmethyl A.1724 1-C3H7 2- (2'-Pyridinyloxy) eth-1-yl A.1725 I-C3H7 2- (3'-Pyridinyloxy) eth-l-yl A.1726 I-C3H7 2- (4'-Pyridinyloxy) eth-l-yl A.1727 I-C3H7 2- (2'-pyrimidinyloxy) eth-l-yl A.1728 t-c ₃ h ₇ 2- (4'-pyrimidinyloxy) eth-l-yl A.1729 t-c ₃ h ₇ 2- (5'-pyrimidinyloxy) eth-l-yl A.1730 iC ₃ H ₇ 2- (2'-pyrazinyloxy) eth-l-yl A.1731 I-C3H7 2- (2'-pyridazinyloxy) eth-l-yl A.1732 ic ₃ H ₆ 2- (3'-pyridazinyloxy) eth-l-yl A.1733 t-c ₃ h ₇ 2 (I ', 3', 5'-Triazinyloxy) eth-l-yl A.1734 t-c ₃ h ₇ 2- (5'-methylisoxazole-3'-yloxy) eth-1-yl A.1735 t-c ₃ h ₇ 2- (5 ' Chlorisoxazol-3'-yloxy) eth-l-yl A.1736 t-c ₃ h ₇ 2- (2-methoxythiazole-4-yloxy) eth-l-yl A.1737 ic ₃ H ₆ 2- (4'-chlorooxazole-2-yloxy) eth-l-yl A.1738 1-C ₃ H ₇ 2- (1'-Phenyl-1'H-1 ', 2', 4'-triazol-3'-yloxy) eth-1-yl A.1739 1-C ₃ H ₇ 2- (1'-Phenylpyrazol-3'-yloxy) eth-1-yl A.1740 1-C ₃ H ₇ c ₆ h ₅ A.1741 t-c ₃ h ₇ 2-Cl-C ₆ H ₄ A.1742 t-c ₃ h ₇ 3-Cl-C ₆ H ₄ A.1743 1-C ₃ H ₇ 4-Cl-C ₆ H ₄ A.1744 1-C ₃ H ₇ 2,3-Cl ₂ -C ₆ H ₃ A.1745 t-c ₃ h ₇ 2,4-Cl ₂ -C ₆ H ₃ A.1746 t-c ₃ h ₇ 2,5-Cl ₂ -C ₆ H ₃ A.1747 1-C ₃ H ₇ 3,4-Cl ₂ -C ₆ H ₃ A.1748 1-C ₃ H ₇ 3,5-Cl ₂ -C ₆ H ₃ A.1749 1-C ₃ H ₇ 4-CN-C ₆ H ₄ A.1750 1-C ₃ H ₇ 2-NO ₂ -C ₆ H ₄ A.1751 1-C ₃ H ₇ 3-NO ₂ -C ₆ H ₄

i m

Nr. R ² R ⁴ A. 1752 I-C3H7 4-NO ₂ -C ₆ H ₄ A.1753 I-C3H7 2,4- (NO ₂ ) ₂ -C ₆ H 3 A. 1754 I-C3H7 2-CH ₃ -C ₆ H ₄ A.1755 I-C3H7 3-CH ₃ -C ₆ H ₄ A. 1756 I-C3H7 4-CH ₃ -C ₆ H ₄ A.1757 I-C3H7 2,3- (CH ₃ ) ₂ -C ₆ H ₃ A. 1758 I-C3H7 2,4 - (CH ₃ ) ₂ -C ₆ H ₃ A.1759 I-C3H7 2,5 - _{(CH3) 2} C H _{3 e} A.1760 I-C3H7 2,6- (CH ₃ ) ₂ -C ₆ H ₃ A.1761 I-C3H7 2-C ₆ H ₅ -C ₆ H ₄ A.1762 I-C3H7 3-C ₆ H ₅ -C ₆ H ₄ A.1763 I-C3H7 4-C ₆ H ₅ -C ₆ H ₄ A.1764 I-C3H7 3-OCH ₃ -C ₆ H ₄ A.1765 I-C3H7 4-OCH ₃ -C ₆ H ₄ A.1766 I-C3H7 3-Acetyl-C ₆ H ₄ A.1767 I-C3H7 4-Acetyl-C 6 H ₄ A.1768 I-C3H7 3-methoxycarbonyl-C6H4 A.1769 I-C3H7 4-methoxycarbonyl-C6H4 A.1770 I-C3H7 3-CF ₃ -C ₆ H ₄ A.1771 I-C3H7 4-CF ₃ -C ₆ H ₄ A.1772 I-C3H7 2-Naphthyl A.1773 I-C3H7 6-chloropyridazine-3-yl A.1774 I-C3H7 5-Chloro-pyrazin-2-yl A.1775 I-C3H7 Quinolin-2-yl A.1776 I-C3H7 2,5-Dimethylpyrazin-3-yl A.1777 iC ₃ H ₇ Pyrazin-2-y1 A.1778 I-C3H7 3-chloropyrid-2-yl A.1779 I-C3H7 6-chloropyrid-2-yl A.1780 I-C3H7 4-Trifluoromethyl, 6-chloropyrid-2-yl A.1781 I-C3H7 4-Trifluoromethylpyrid-2-yl A.1782 I-C3H7 6-Trifluoromethylpyrid-2-yl A.1783 i-C3H7 6-Methoxypyrid-2-yl A.1784 I-C3H7 5-chloropyrid-2-yl A.1785 1-C3H7 Pyridin-2-yl A.1786 I-C3H7 Benzothiazol-2-yl A.1787 I-C3H7 7-Chloroquinolin-4-yl A. 1788 I-C3H7 J-nitro-pyridin-2-yl A. 1789 I-C3H7 ? Yrrol-3-yl A.1790 I-C3H7 ? Yrrol-2-yl

Nr. R ² R ⁴ A.1791 iC ₃ H ₇ 2,6-Dioctylpyrid-4-yl A.1792 t-c ₃ h ₇ 5-nitro-pyridin-2-yl A.1793 1-C ₃ H ₇ Pyrid-4-yl A.1794 1-C ₃ H ₇ Pyridin-3-yl A.1795 t-c ₃ h ₇ Pyrimidin-2-yl A.1796 t-c ₃ h ₇ Pyrimidin-4-yl A.1797 ic ₃ H ₆ Quinazolin-4-yl A.1798 1-C ₃ H ₇ 6-Chloro-pyrimidin-4-yl A.1799 iC ₃ H ₇ 6-Methoxy-pyrimidin-4-yl A.1800 iC ₃ H ₇ 2,5,6-Trichloro-4-yl A.1801 iC ₃ H ₇ 2,6-dimethyl-pyrimidin-4-yl A.1802 iC ₃ H ₇ 2-Methyl, 6-chloropyrimidin-4-yl A.1803 CI-C ₃ H ₇ 2-Methyl, 6-Ethoxy-pyrimidin-4-yl A.1804 iC ₃ H ₇ 4,5,6-trichloro-2-yl A.1805 1-C ₃ H ₇ 4,6-Dimethoxypyrimidin-2-yl A.1806 1-C ₃ H ₇ 4,6-dimethyl-2-yl A.1807 iC ₃ H ₇ 4,6-dichloropyrimidine-2-yl A.1808 t-c ₃ h ₇ 4-Methyl, 6-methoxy-pyrimidin-2-yl A.1809 ic ₃ H ₆ 4-Chloro, 6-methoxypyrimidin-2-yl A.1810 t-c ₃ h ₇ 6-Chloro-quinoxalin-2-yl A.1811 1-C ₃ H ₇ 3,6-Dichloro-1,2,4-triazin-5-yl A.1812 1-C ₃ H ₇ 4-Methoxy-l, 3,5-triazin-2-yl A.1813 t-c ₃ h ₇ 4-Ethoxy-l, 3,5-triazin-2-yl A. 1814 1-C ₃ H ₇ 4,6-Dichloro-1,3,5-triazin-2-yl A.1815 t-c ₃ h ₇ 4-Ethoxy, 6-Chloro-1,3,5-triazin-2-yl A. 1816 t-c ₃ h ₇ Isoxazol-3-yl A.1817 1-C ₃ H ₇ Thien-2-yl A.1818 1-C ₃ H ₇ Fur-2-yl A. 1819 t-c ₃ h ₇ Thiatriazol-5-yl A.1820 1-C ₃ H ₇ (E) -1-chloropropene-3-yl A.1821 t-c ₃ h ₇ (E) -4- (4'-Chlorophenyl-but-2-en-1-yl) A.1822 1-C ₃ H ₇ Propyn-3-yl A.1823 t-c ₃ h ₇ Methylcarbonyl A.1824 1-C ₃ H ₇ Ethylcarbonyl A.1825 1-C ₃ H ₇ n Propylcarbonyl A.1826 1-C ₃ H ₇ . -Propylcarbonyl A.1827 t-c ₃ h ₇ i-Butylcarbonyl A.1828 1 ~ C ₃ H ₇ 3-Butylcarbonyl A.1829 t-c ₃ h ₇ L-Butylcarbonyl

Nr. R ² R ⁴ A.1830 I-C3H7 t-Butylcarbonyl A.1831 I-C3H7 n Pentylcarbonyl A.1832 I-C3H7 i -Pentylcarbonyl A.1833 1-C3H7 neo-Pentylcarbonyl A.1834 I-C3H7 n Hexylcarbonyl A.1835 I "C3ÍÍ7 n Octylcarbonyl A.1836 I-C3H7 1-Propenylcarbonyl A.1837 I-C3H7 2-Pentene-1-carbonyl A.1838 I-C3H7 2,5-heptadiene-1-yl-carbonyl A.1839 I-C3H7 benzoyl A.1840 I-C3H7 2-chlorobenzoyl A.1841 I-C3H7 3 - Chlorobenz o1 A.1842 I-C3H7 4 -Chlorobenzoyl A.1843 X-C3H7 2-Cyanobenzoyl A.1844 I-C3H7 3-Cyanobenzoyl A.1845 I-C3H7 4-Cyanobenzoyl A.1846 I-C3H7 4-methoxybenzoyl A.1847 I-C3H7 2-Pyridylcarbonyl A.1848 I-C3H7 3 -Pyridylcarbonyl A.1849 I-C3H7 4-Pyridylcarbonyl A.1850 I-C3H7 2-Pyrimidinylcarbonyl A.1851 I-C3H7 2-Oxazolylcarbonyl A.1852 I-C3H7 4-Methyl-isoxazol-5-ylcarbonyl A.1853 I-C3H7 methylsulfonyl A.1854 I-C3H7 ethylsulfonyl A.1855 I-C3H7 n-propylsulfonyl A.1856 I-C3H7 i-propylsulfonyl A.1857 I-C3H7 n-Bu tylsulfonyl A.1858 I-C3H7 t-Bu tylsu1f onyl A.1859 I-C3H7 n-pentylsulfonyl A.1860 I-C3H7 neo-pentylsulfonyl A.1861 I-C3H7 n-Hexylsulfonyl A.1862 I-C3H7 n-Octylsulfonyl A.1863 I-C3H7 phenylsulfonyl A.1864 I-C3H7 2-Chlorphenylsulfonyl A.1865 I-C3H7 3-Chlorphenylsulfonyl A.1866 L-C3H7 4-Chlorophenylsulfonyl A.1867 L-C3H7 2-Cyanophenylsulfonyl A.1868 L-C3H7 3-Cyanophenylsulfonyl

Nr. R ² R ⁴ A.1869 IC ₃ H ₇ 4-Cyanophenylsulfonyl A.1870 t-c ₃ h ₇ 2 -Pyridylsulfonyl A.1871 ic ₃ H ₆ 3-Pyridylsulfonyl A.1872 1-C ₃ H ₇ 4 -Pyridylsulfonyl A.1873 1-C ₃ H ₇ 2-Pyrimidinylsulfonyl A.1874 1-C ₃ H ₇ 4-Oxazolylsulfonyl A.1875 t-c ₃ h ₇ 5-Chloro-thiazol-2-ylsulfonyl A.1876 1-C ₃ H ₇ 2-C ₄ H ₉ -C ₆ H ₄ -CH ₂ A.1877 t-c ₃ h ₇ 3 1-C ₄ H ₉ C _s H ₄ CH ₂ A.1878 1-C ₃ H ₇ 4-tC ₄ H ₉ -C ₆ H ₄ -CH ₂ A.1879 1-C ₃ H ₇ 2- (4'-Chloro-thiazol-2'-yloxy) eth-1-yl A.1880 1-C ₃ H ₇ 2- (L-methyl-pyrazol-4-yloxy) eth-1-yl A.1881 1-C ₃ H ₇ 4-Br-C ₆ H ₄ A.1882 1-C ₃ H ₇ 3,5- (CH ₃ ) ₂ -C ₆ H ₃ A.1883 1-C ₃ H ₇ 4-C ₂ H ₅ -C ₆ H ₄ A.1884 1-C ₃ H ₇ 3-Dimethylaminocarbonyl-C ₆ H ₄ A.1885 t-c ₃ h ₇ 4-Dimethylaminocarbonyl-C 6 H ₄ A.1886 t-c ₃ h ₇ 2-Hydroxyprop-1-yl A.1887 1-C ₃ H ₇ 6-hydroxy-2-methyl-4-ylmethyl A.1888 t-c ₃ h ₇ 16 - OH, 2 - CH (CH _{3) 2} - pyr imi din - 4 - yl 1] - _CH2 A.1889 t-c ₃ h ₇ [6-OH, 2-CH (CH ₂ ) ₂ -pyrimidin-4-yl] -CH ₂ A.1890 1-C ₃ H ₇ 5- (2'-Furan) -pent-1-yl A.1891 t-c ₃ h ₇ 5- (2'-N-Methylpyrrol) pent-l-yl A.1892 t-c ₃ h ₇ [2- (4-Cl-C ₆ H ₄₎ -oxazole-4-yl] _-CH2 A.1893 t-c ₃ h ₇ 3-CF ₃ -pyridin-2-yl A.1894 t-c ₃ h ₇ 5-CF ₃ -pyridin-2-yl A.1895 t-c ₃ h ₇ 6- (2'-Thienyl) hex-l-yl A.1896 1-C ₃ H ₇ (E) -3-chloro-but-2-en-l-yl A.1897 ic ₃ H ₆ (Z) -3-chloro-but-2-en-l-yl A.1898 iC ₃ H ₇ (E) -2-bromo-but-2-en-l-yl A.1899 t-c ₃ h ₇ (Z) -2-Bromobut-2-en-yl A.1900 1-C ₃ H ₇ (E) -1-Chlorprop-l'-3-yl A.1901 1-C ₃ H ₇ (Z) -l-chloro-prop-l-en-3-yl A.1902 1-C ₃ H ₇ But-en-3-yl A.1903 ic ₃ h ₇ CH ₂ CH ₂ Br A.1904 IC ₃ H ₇ ¹ 1 H ₂ CH ₂ CH ₂ Br A.1905 iC ₃ H ₇ 3H ₂ CH ₂ CH ₂ CH ₂ Br A.1906 1-C ₃ H ₇ 2-methylprop-1-y1 A.1907 LC ₃ H ₇ 2-Ethoxyprop-1-yl

Nr. R ² R ⁴ A.1908 1-C3H7 2-isopropoxypropanoic-yl A.1909 I-C3H7 But-in-3-yl A.1910 I-C3H7 But-in-4-yl A.1911 I-C3H7 But-2-yn-4-yl A.1912 I-C3H7 Pent-in-4-yl A.1913 I-C3H7 Pent-2-yn-4-yl A.1914 I-C3H7 Pent-in-5-yl A.1915 I-C3H7 Pent-2-yn-5-yl A.1916 I-C3H7 E-2-chloro-but-2-en-l-yl A.1917 I-C3H7 Z-2-chloro-but-2-en-l-yl A.1918 I-C3H7 Z-l-chloro-prop-l-en-3-yl A.1919 I-C3H7 2-methyl-prop-1-en-3-y1 A.1920 I-C3H7 2-chloro-prop-l-en-3-yl A.1921 I-C3H7 2-bromoprop-l-en-3-yl A.1922 I-C3H7 But-2-en-l-yl A.1923 I-C3H7 But-3-en-l-yl A.1924 i — C ₃ H ₇ l-Iodprop-l-yn-3-yl A.1925 t-c ₃ h ₇ E-3-bromo-but-2-en-l-yl A.1926 I-C3H7 Z-3-bromo-but-2-en-l-yl A.1927 cyclopropyl H A.1928 cyclopropyl CH ₃ A.1929 cyclopropyl C2H5 A.1930 cyclopropyl nC ₃ H ₇ A.1931 cyclopropyl I-C3H7 A.1932 cyclopropyl cyclopropyl A.1933 cyclopropyl nC ₄ Hg A.1934 cyclopropyl S · c ₄ h ₉ A.1935 cyclopropyl iC ₄ H9 A.1936 cyclopropyl tC ₄ H ₉ A.1937 cyclopropyl n CSHN A.1938 cyclopropyl I-C5H11 A.1939 cyclopropyl neo-CSHN A.1940 cyclopropyl cyclopentyl A.1941 cyclopropyl n-C6Hi3 A.1942 cyclopropyl cyclohexyl A.1943 cyclopropyl n CeHi7 A.1944 cyclopropyl CH ₂ CH ₂ Cl A.1945 cyclopropyl (CH ₂₎ j C 1 -C ₄ A.1946 cyclopropyl ch ₂ cn j

~ / IR

Nr. R ² R ⁴ A.1947 cyclopropyl ch ₂ ch ₂ cn A.1948 cyclopropyl (CH ₂ ) ₃ CN A.1949 cyclopropyl (ch ₂ ) ₄ cn A.1950 cyclopropyl (ch ₂ ) ₆ cn A.1951 cyclopropyl Cyclohexylmethyl A.1952 cyclopropyl 2-Cyclohexyleth-1-yl A.1953 cyclopropyl Cyclopropyme 1 A.1954 cyclopropyl 2-Cyclopropyleth-1-yl A.1955 cyclopropyl 2-methoxyethyl-yl A.1956 cyclopropyl 2-ethoxyethanol-1-yl A.1957 cyclopropyl 2-Isopropoxyeth-1-yl A.1958 cyclopropyl 3-methoxypropyl-1-yl A.1959 cyclopropyl 3-ethoxypropyl-1-yl A.1960 cyclopropyl 3-1sopropoxyp rop-1-y1 A.1961 cyclopropyl 4-Methoxybut-1-yl A. 1962 cyclopropyl 4-Isopropoxybut-1-yl

'21 ^ -

Nr. R ² R ⁴ A.1963 cyclopropyl Propen-3-yl A.1964 cyclopropyl But-2-en-l-yl A.1965 cyclopropyl 3-methyl-but-2-en-1-yl A.1966 cyclopropyl 2-Vinyloxyeth-1-yl A.1967 cyclopropyl Allyloxy-th-1-yl A.1968 cyclopropyl 2-Trifluormethoxyeth-1-yl A.1969 cyclopropyl 3-Trifluormethoxyprop-1-yl A. 1970 cyclopropyl 4-Difluormethoxybut-1-yl A.1971 cyclopropyl Hydroxycarbonylmethyl A.1972 cyclopropyl Methoxycarbonylmethyl A.1973 cyclopropyl Aminocarbonylmethyl A.1974 cyclopropyl N-Methylaminocarbonylmethyl A.1975 cyclopropyl Ν, Ν-methyl-Dimethylaminocarbonyl A.1976 cyclopropyl 2-Hydroxycarbonyleth-1-yl A.1977 cyclopropyl 2-Methoxycarbonyleth-1-yl A.1978 cyclopropyl 2-Aminocarbonyleth-1-yl A.1979 cyclopropyl 2-N-Methylaminocarbonyleth-1-yl A.1980 cyclopropyl 2-Dimethylaminocarbonyleth-1-yl A.1981 cyclopropyl 2-aminoethyl-l-yl A.1982 cyclopropyl 2-amino-prop-1-yl A.1983 cyclopropyl 4-amino-but-l-yl A.1984 cyclopropyl 3-Dimethylamino-l-yl A.1985 cyclopropyl 4-Aminothiocarbonylbut-1-yl A.1986 cyclopropyl 2-oxo-propyl A.1987 cyclopropyl cyclohexyl A.1988 cyclopropyl cyclopropyl A.1989 cyclopropyl cyclopentyl A.1990 cyclopropyl 2-Methoxyiminoprop-1-yl A.1991 cyclopropyl 2--Methoxyiminoeth-1-yl A.1992 cyclopropyl 6-Aminocarbonylhex-1-yl A.1993 cyclopropyl 3-Aminothiocarbonylprop-1-yl A.1994 cyclopropyl 2-Aminothiocarbonyleth-1-yl A.1995 cyclopropyl Aminothiocarbonylmethyl A.1996 cyclopropyl 4- (N, N-dimethylamino) but-l-yl A.1997 cyclopropyl 2- (Methylthio) eth-l-yl A.1998 cyclopropyl 2- (methylsulfonyl) eth-1-yl A.1999 cyclopropyl 4- (Methylthio) prop-1-yl A.2000 cyclopropyl 4- (methylsulfonyl) prop-l-yl A.2001 cyclopropyl benzyl

Nr. R ² R ⁴ A.2002 cyclopropyl 2-FC ₆ H ₄ -CH ₂ A.2003 cyclopropyl 3-FC ₆ H ₄ -CH ₂ A.2004 cyclopropyl 4-FC ₆ H ₄ -CH ₂ A.2005 cyclopropyl 2,3-F ₂ -C ₆ H ₃ -CH ₂ A.2006 cyclopropyl 2,4-F ₂ -C ₆ H ₃ -CH ₂ A.2007 cyclopropyl 2,5-F ₂ -C ₆ H ₃ -CH ₂ A.2008 cyclopropyl 2,6-F ₂ -C ₆ H ₃ -CH ₂ A.2009 cyclopropyl 3,4-F ₂ -C ₆ H ₃ -CH ₂ A.2010 cyclopropyl 3,5-F ₂ -C ₆ H ₃ -CH ₂ A.2011 cyclopropyl 2-C 1 -C ₆ H ₄ -CH ₂ A.2012 cyclopropyl 3-Cl-C ₆ H ₄ CH ₂ A.2013 cyclopropyl 4 -C 1 -C ₆ H ₄ -CH ₂ A.2014 cyclopropyl 2,3-Cl ₂ -C ₆ H ₃ -CH ₂ A.2015 cyclopropyl 2,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.2016 cyclopropyl 2,5-Cl ₂ -C ₆ H ₃ -CH ₂ A.2017 cyclopropyl 2,6-Cl ₂ -C ₆ H ₃ -CH ₂ A.2018 cyclopropyl 3,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.2019 cyclopropyl 3,5-Cl ₂ -C ₆ H ₃ -CH ₂ A.2020 cyclopropyl 2,3,4-Cl ₃ -C ₆ H ₂ -CH ₂ A.2021 cyclopropyl 2,3,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.2022 cyclopropyl 2,3,6-C 1 -C ₃ -C ₆ H ₂ -CH ₂ A.2023 cyclopropyl 2,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.2024 cyclopropyl 2,4,6-C 1 -C ₃ -C ₆ H ₂ -CH ₂ A.2025 cyclopropyl 3,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.2026 cyclopropyl 2 -Br-C ₆ H ₄ -CH ₂ A. 2027 cyclopropyl 3-Br-C ₆ H ₄ CH ₂ A.2028 cyclopropyl 4-Br-C ₆ H ₄ CH ₂ A.2029 cyclopropyl 2,3-Br ₂ -C ₆ H ₃ -CH ₂ A.2030 cyclopropyl 2,4-Br ₂ -C ₆ H ₃ -CH ₂ A.2031 cyclopropyl 2,5-Br ₂ -C ₆ H ₃ -CH ₂ A.2032 cyclopropyl 2,6-Br ₂ -C ₆ H ₃ -CH ₂ A.2033 cyclopropyl 3,4-Br ₂ -C ₆ H ₃ -CH ₂ A.2034 cyclopropyl 3,5-Br ₂ -C ₆ H ₃ -CH ₂ A.2035 cyclopropyl 2-F, 3-Cl-C ₆ H ₃ CH ₂ A.2036 cyclopropyl 2-F, 4-C1-C ₆ H ₃ CH ₂ A.2037 cyclopropyl 2-F, 5-Cl-C ₆ H ₃ CH ₂ A.2038 cyclopropyl 2-F, 3-Br-C ₆ H ₃ CH ₂ A.2039 cyclopropyl 2-F, 4-Br-C ₆ H ₃ CH ₂ A.2040 cyclopropyl 2-F, 5-Br-C ₆ H ₃ CH ₂

Nr. R ² R ⁴ A.2041 cyclopropyl 2-C1, 3-Br-C ₆ H ₃ CH ₂ A.2042 cyclopropyl 2-C1, 4-Br-C ₆ H ₃ CH ₂ A.2043 cyclopropyl 2-C1, 5-Br-C ₆ H ₃ CH ₂ A.2044 cyclopropyl 3-F, 4-C1-C ₆ H ₃ CH ₂ A.2045 cyclopropyl 3-F, 5-Cl-C ₆ H ₃ CH ₂ A.2046 cyclopropyl 3-F, 6-Cl-C ₆ H ₃ CH ₂ A.2047 cyclopropyl 3-F, 4-Br-C ₆ H ₃ CH ₂ A.2048 cyclopropyl 3-F, 5-Br-C ₆ H ₃ CH ₂ A.2049 cyclopropyl 3-F, 6-Br-C ₆ H ₃ CH ₂ A.2050 cyclopropyl 3-C1, 4-Br-C ₆ H ₃ CH ₂ A.2051 cyclopropyl 3-C1, 5-Br-C ₆ H ₃ CH ₂ A.2052 cyclopropyl 3-C1, 6-Br-C ₆ H ₃ CH ₂ A.2053 cyclopropyl 4-F, 5-C 1-C ₆ H ₃ CH ₂ A.2054 cyclopropyl 4-F, 6-C1-C ₆ H ₃ CH ₂ A.2055 cyclopropyl 4-F, 5-Br-C ₆ H ₃ CH ₂ A.2056 cyclopropyl 4-F, 6-Br-C ₆ H ₃ CH ₂ A.2057 cyclopropyl 4-C1, 5-Br-C ₆ H 3 -CH ₂ A.2058 cyclopropyl 5-F, 6'C 1 -C ₆ H ₃ -CH ₂ A.2059 cyclopropyl 5-F, 6-Br-C ₆ H ₃ CH ₂ A.2060 cyclopropyl 5-C1, _6-Br-3 CEH -CH ₂ A.2061 cyclopropyl 3-Br, 4-Cl ,. 5-Br-C ₆ H ₂ CH ₂ A.2062 cyclopropyl 2-CN-C ₆ H ₄ CH ₂ A.2063 cyclopropyl 3-CN-C ₆ H ₄ CH ₂ A.2064 cyclopropyl 4 -CN-C ₆ H ₄ -CH ₂ A.2065 cyclopropyl 2-NO ₂ -C ₆ H ₄ -CH ₂ A.2066 cyclopropyl 3-NO ₂ -C ₆ H ₄ -CH ₂ A.2067 cyclopropyl 4-NO ₂ -C ₆ H ₄ -CH ₂ A.2068 cyclopropyl 2-CH ₃ -C ₆ H ₄ -CH ₂ A.2069 cyclopropyl 3 -CH ₃ -C ₆ H ₄ -CH ₂ A.2070 cyclopropyl 4-CH ₃ -C ₆ H ₄ -CH ₂ A.2071 cyclopropyl 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A. 2072 cyclopropyl 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2073 cyclopropyl 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2074 cyclopropyl 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2075 cyclopropyl 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2076 ľyclopropyl 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2077 ľyclopropyl 2-C ₂ H _with -C ₆ H ₄ -CH ₂ A.2078 ľyclopropyl 3-C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2079 ľyclopropyl 4-C ₂ H ₅ -C ₆ H ₄ -CH ₂

Nr. R ² R ⁴ A.2080 cyclopropyl 2 - i-C3H7-C ₆ H ₄ CH ₂ A.2081 cyclopropyl 3 - i-C3H7-C ₆ H ₄ CH ₂ A.2082 cyclopropyl 4 - i-C3H7-C ₆ H ₄ CH ₂ A.2083 cyclopropyl 2 - Cyclohexy1 - CGH ₄ - CH ₂ A.2084 cyclopropyl 3 - Cyc lohexy1 - CGH ₄ - CH ₂ A.2085 cyclopropyl 4 - Cyc lohexy 1 - C 8 H ₄ - CH ₂ A.2086 cyclopropyl 2-Vinyl -C ₆ H ₄ -CH ₂ A.2087 cyclopropyl 3-Vinyl -C ₆ H ₄ -CH ₂ A.2088 cyclopropyl 4-Vinyl-C 6 H ₄ - CH ₂ A.2089 cyclopropyl 2-allyl-C ₆ H ₄ CH ₂ A.2090 cyclopropyl 3-Allyl-C ₆ H ₄ CH ₂ A. 2091 cyclopropyl 4-allyl-C ₆ H ₄ CH ₂ A.2092 cyclopropyl 2-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.2093 cyclopropyl 3-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.2094 cyclopropyl 4-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.2095 cyclopropyl 3-CH3, 5-t C ₄ H9-C ₆ H ₃ CH ₂ A.2096 cyclopropyl 2-OH-C ₆ H ₄ CH ₂ A.2097 cyclopropyl 3-OH-C ₆ H ₄ CH ₂ A.2098 cyclopropyl 4-OH-C ₆ H ₄ CH ₂ A.2099 cyclopropyl 2-OCH 3 -C ₆ H ₄ -CH ₂ A.2100 cyclopropyl 3-OCH ₃ -C ₆ H ₄ -CH ₂ A. 2101 cyclopropyl 4-OCH 3 -C ₆ H ₄ -CH ₂ A.2102 cyclopropyl 2,3- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2103 cyclopropyl 2,4- (OCH ₃ ) 2 -C ₆ H 3 -CH ₂ A.2104 cyclopropyl 2,5- (OCH 3) ₂ -C ₆ H ₃ -CH ₂ A.2105 cyclopropyl 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2106 cyclopropyl 3,5- (OCH ₃ ) ₂ -C ₆ H 3 -CH ₂ A.2107 cyclopropyl 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH ₂ A.2108 cyclopropyl 2-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2109 cyclopropyl 3 -OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2110 cyclopropyl 4-OC ₂ H _S -C ₆ H ₄ -CH ₂ A.2111 cyclopropyl 2-0; (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.2112 cyclopropyl 3-O- (11-C ₃ H 7) -C ₆ H ₄ -CH ₂ A.2113 cyclopropyl 4-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.2114 cyclopropyl 2-O- (iC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.2115 ľyclopropyl 3-O- (1-C ₃ H 7) -C ₆ H ₄ -CH ₂ A.2116 ľyclopropyl 4-O- (1-C ₃ H 7) -C ₆ H ₄ -CH ₂ A.2117 ( ľyclopropyl 4-O- (nC ₄ H ₉ ) -C ₆ H ₄ -CH ₂ A.2118 ( Zyclopropyl ϊ-O- (t C ₄ H ₉ ) -C ₅ H ₄ -CH ₂

2ΖΖ-

Nr. R ² rl A.2119 cyclopropyl 4-O- (nc ₆ H ₁₃ ) -c ₆ h ₄ -ch ₂ A. 2120 cyclopropyl 2-O-allyl-C ₆ H ₄ CH ₂ A.2121 cyclopropyl 3-O-allyl-C ₆ H ₄ CH ₂ A.2122 cyclopropyl 4-O-allyl-C ₆ H ₄ CH ₂ A.2123 cyclopropyl 2-CF ₃ -C ₆ H ₄ -CH ₂ A.2124 cyclopropyl 3-CF ₃ -C ₆ H ₄ -CH ₂ L A.2125 cyclopropyl 4-CF ₃ -C ₆ H ₄ -CH ₂ j A.2126 cyclopropyl _2-Acetyl-4 CGH CH ₂ L A.2127 cyclopropyl 3-Acetyl-C ₆ H ₄ CH _2? A.2128 cyclopropyl 4-Acetyl - ₄ CGH - _CH2 A.2129 cyclopropyl 2-methoxycarbonyl-C 6 H ₄ -CH ₂ A.2130 cyclopropyl 3-methoxycarbonyl-C 6 H ₄ -CH ₂ A.2131 cyclopropyl Methoxycarbonyl-4-C 6 H ₄ CH _2, A.2132 cyclopropyl 2 -Aminocarbonyl -CeH ₄ -CH ₂ A.2133 cyclopropyl 3-aminocarbonyl-C 6 H ₄ -CH ₂ A.2134 cyclopropyl 4-Aminocarbonyl -C ₆ H ₄ -CH ₂ A.2135 cyclopropyl 2-Dimethylaminocarbonyl-C 6 H ₄ -CH ₂ A.2136 cyclopropyl 3 - Dimethylaminocarbonyl -C 6 H ₄ - CH ₂ A.2137 cyclopropyl 4 - Dimethylaminocarbonyl-C 6 H ₄ -CH ₂ A.2138 cyclopropyl 2- (N-Methylaminocarbonyl) -C ₆ H ₄ -CH ₂ A.2139 cyclopropyl 3- (N-Methylaminocarbonyl) -C ₈ H ₄ -CH ₂ A.2140 cyclopropyl 4- (N-Methylaminocarbonyl) -C ₆ H ₄ -CH ₂ A.2141 cyclopropyl 2 -H ₂ NC ₆ H ₄ -CH ₂ A.2142 cyclopropyl 3-H ₂ NC ₆ H ₄ -CH ₂ A.2143 cyclopropyl 4-H ₂ NC ₆ H ₄ -CH ₂ A.2144 cyclopropyl 2-Aminothiocarbonyl-C ₆ H ₄ CH ₂ A.2145 cyclopropyl 3-Aminothiocarbonyl-C 8 H ₄ -CH ₂ A.2146 cyclopropyl 4-Aminothiocarbonyl-C 6 H ₄ -CH ₂ A.2147 cyclopropyl 2-methoxyimino-methyl-C 6 H ₄ -CH _2; A.2148 cyclopropyl 3-Methoxyiminomethyl -C ₈ H ₄ -CH ₂ A.2149 cyclopropyl 4-methoxyimino-methyl-C 6 H ₄ -CH ₂ A.2150 cyclopropyl 2-Formyl-C6H ₄ -CH ₂ ( A.2151 cyclopropyl -Formy1 3 -C ₆ H ₄ -CH _2; A.2152 cyclopropyl 4-Formyl-C 8 H ₄ -CH ₂ A.2153 cyclopropyl 2- (1'-Methoxyiminoeth-1'-yl) -C ₆ H ₄ -CH ₂ A.2154 cyclopropyl 3- (1'-Methoxyiminoeth-1'-yl) -C ₆ H ₄ -CH ₂ A.2155 cyclopropyl 4- (1'-Methoxyiminoeth-1'-yl) -C ₆ H ₄ -CH ₂ A.2156 cyclopropyl 2-SCH ₃ -C ₆ H ₄ -CH ₂ A.2157 cyclopropyl 3-SCH ₃ -C ₆ H ₄ -CH ₂

. Nr. R ² R ⁴ A.2158 cyclopropyl 4-SCH ₃ -C ₆ H ₄ -CH ₂ A.2159 cyclopropyl 2-SO2CH3-C6H4-CH2 A.2160 cyclopropyl 3-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ A.2161 cyclopropyl 4-SO2CH3-C6H4-CH2 A.2162 cyclopropyl 2-OCF ₃ -C ₆ H ₄ -CH ₂ A.2163 cyclopropyl 3-OCF ₃ -C ₆ H ₄ -CH ₂ A.2164 cyclopropyl 4 -OCF ₃ -C ₆ H ₄ -CH ₂ A.2165 cyclopropyl 2-OCHF ₂ -C ₆ H ₄ -CH ₂ A.2166 cyclopropyl 3-OCHF ₂ -C ₆ H ₄ -CH ₂ A.2167 cyclopropyl 4-OCHF ₂ -C ₆ H ₄ -CH ₂ A.2168 cyclopropyl 3-CF ₃ , 4-OCF 3 -C ₆ H ₃ -CH ₂ A.2169 cyclopropyl _{1-Naphthyl-CH2} A.2170 cyclopropyl _{2-Naphthyl-CH2} A.2171 cyclopropyl 2-Phenoxyeth-1-yl A.2172 cyclopropyl 2- (2'-Chlorophenoxy) eth-1-yl A. 2173 cyclopropyl 2- (3'-Chlorophenoxy) eth-1-yl A.2174 cyclopropyl 2- (4'-Chlorphenoxy) eth-l-yl A.2175 cyclopropyl 2- (3 ', 5'-Dichlorophenoxy) eth-1-yl A.2176 cyclopropyl 2- (2'-Cyanophenoxy) eth-1-yl A.2177 cyclopropyl 2- (3'-Cyanophenoxy) eth-l-yl A.2178 cyclopropyl 2- (4'-Cyanophenoxy) eth-l-yl A.2179 cyclopropyl 2- (2'-Methylphenoxy) eth-1-yl A.2180 cyclopropyl 2- (3'-methylphenoxy) eth-l-yl A.2181 cyclopropyl 2- (4'-Methylphenoxy) eth-1-yl A.2182 cyclopropyl 2- (3'-t-Butylphenoxy) eth-l-yl A.2183 cyclopropyl 2- (4'-t-Butylphenoxy) eth-l-yl A.2184 cyclopropyl 2- (2'-Nitrophenoxy) eth-1-yl A.2185 cyclopropyl 2- (3'-Nitrophenoxy) eth-l-yl A.2186 cyclopropyl 2- (4'-Nitrophenoxy) eth-1-yl A.2187 cyclopropyl 2- (2-methoxyphenoxy) eth-l-yl A.2188 cyclopropyl 2- (3'-Methoxyphenoxy) eth-1-yl A.2189 cyclopropyl 2- (4'-Methoxyphenoxy) eth-1-yl A.2190 cyclopropyl 2- (2'-Trifluoromethylphenoxy) eth-1-yl A.2191 cyclopropyl 2- (3 ' Trifluormethylphenoxy) eth-1-yl A.2192 cyclopropyl 2- (4'-Trifluoromethylphenoxy) eth-1-yl A.2193 cyclopropyl 2- (2'-Acetylphenoxy) eth-l-yl A.2194 cyclopropyl 2- (3'-Acetylphenoxy) eth-l-yl A.2195 cyclopropyl 2- (4'-Acetylphenoxy) eth-l-yl A.2196 < ľyclopropyl 2- (2'-Methoxycarbonyl) eth-1-yl

- £ / <-

Nr. R ² R ⁴ A.2197 cyclopropyl 2- (3'-methoxycarbonyl) eth-1-yl A.2198 cyclopropyl 2- (4'-Methoxycarbonyl) eth-1-yl A.2199 cyclopropyl 2- (2'-Dimethylaminocarbonyl) eth-1-yl A.2200 cyclopropyl 2- (3'-Dimethylaminocarbonyl) eth-1-yl A.2201 cyclopropyl 2- (4'-Dimethylaminocarbonyl) eth-1-yl A.2202 cyclopropyl 2- (2'-Aminothiocarbonyl) eth-1-yl A.2203 cyclopropyl 2- (3'-Aminothiocarbonyl) eth-1-yl A.2204 cyclopropyl 2- (4'-Aminothiocarbonyl) eth-1-yl j A.2205 cyclopropyl 2- (2'-Methylsulfonyl) eth-1-yl ¹ A.2206 cyclopropyl 2- (3'-methylsulfonyl) eth-l-yl A.2207 cyclopropyl 2- (4'-Methylsulfonyl) eth-1-yl A.2208 cyclopropyl 3-Phenoxyprop-1-yl A.2209 cyclopropyl 3- (2'-Chloro-phenoxy) -prop-1-yl A.2210 cyclopropyl 3- (3'-Chlorphenoxy) prop-yl A.2211 cyclopropyl 3- (4'-Chlorophenoxy) prop-1-yl A.2212 cyclopropyl 3- (3 ', 5', Dichlorophenoxy) prop-1-yl A.2213 cyclopropyl 3- (2'-Cyanophenoxy) prop-1-yl A.2214 cyclopropyl 3- (3'-Cyanophenoxy) prop-1-yl j A.2215 cyclopropyl 3- (4'-Cyanophenoxy) prop-1-yl i A.2216 cyclopropyl 3- (2'-Methylphenoxy) prop-1-yl { A.2217 cyclopropyl 3- (3'-Methylphenoxy) prop-1-yl and 1 A.2218 cyclopropyl 3- (4'-methylphenoxy) prop-1-yl A.2219 cyclopropyl 3- (2'-Methoxyphenoxy) prop-1-yl A.2220 cyclopropyl 3- (3'-Methoxyphenoxy) prop-1-yl s A.2221 cyclopropyl 3- (4'-Methoxyphenoxy) prop-1-yl A.2222 cyclopropyl 3- (2'-Trifluoromethylphenoxy) prop-1-yl A.2223 cyclopropyl 3- (3'-Trifluoromethylphenoxy) prop-1-yl A.2224 cyclopropyl 3- (4'-Trifluoromethylphenoxy) prop-yl A.2225 cyclopropyl 4-Phenoxybut-1-yl A.2226 cyclopropyl 2-Phenyleth-1-yl A.2227 cyclopropyl 2- (2'-Chlorophenyl) eth-1-yl A.2228 cyclopropyl 2- (3'-Chlorphenyl) eth-1-yl A.2229 cyclopropyl 2- (4'-Chlorophenyl) eth-1-yl A.2230 cyclopropyl 2- (3 ', 5'-Dichlorophenyl) eth-1-yl A.2231 cyclopropyl 2- (2'-Cyanophenyl) eth-1-yl A.2232 cyclopropyl 2- (3'-Cyanophenyl) eth-1-yl A.2233 cyclopropyl 2- (4'-Cyanophenyl) eth-1-yl A.2234 ( Cyclopropyl i 2- (2'-Methylphenyl) eth-1-yl; A.2235 ( Cyclopropyl i 2- (3'-Methylphenyl) eth-l-yl

-22i-

Nr. R ² R ⁴ A.2236 cyclopropyl 2- (4'-Methylphenyl) eth-l-yl A.2237 cyclopropyl 2- (2'-Methoxyphenyl) eth-l-yl A.2238 cyclopropyl 2- (3'-Methoxyphenyl) eth-l-yl A.2239 cyclopropyl 2- (4'-Methoxyphenyl) eth-l-yl A.2240 cyclopropyl 2- (2'-Trifluoromethylphenyl) eth-1-yl A.2241 cyclopropyl 2- (3'-Trifluoromethylphenyl) eth-1-yl A.2242 cyclopropyl 2- (4'-Trifluoromethylphenyl) eth-1-yl A.2243 cyclopropyl 3-Phenylprop-1-yl A.2244 cyclopropyl 3- (2-Chlorphenyl) prop-1-yl A.2245 cyclopropyl 3- (3'-Chlorphenyl) prop-l-yl A.2246 cyclopropyl 3- (4'-Chlorophenyl) prop-1-yl A.2247 cyclopropyl 3- (2'-Cyanophenyl) prop-1-yl A.2248 cyclopropyl 3- (3'-Cyanophenyl) prop-1-yl A.2249 cyclopropyl 3- (4'-cyanophenyl) prop-1-yl A.2250 cyclopropyl 3- (2'-Trifluoromethylphenyl) prop-1-yl A.2251 cyclopropyl 4-Phenylbut-1-yl A.2252 cyclopropyl 4- (4'-Chlorophenyl) but-1-yl A.2253 cyclopropyl 6- (4'-Chlorophenyl) hex-1-yl A.2254 cyclopropyl 2-pyridylmethyl A.2255 cyclopropyl 3-pyridylmethyl A.2256 cyclopropyl 4-pyridylmethyl A.2257 cyclopropyl 4-Chloro-pyridin-2-ylmethyl A.2258 cyclopropyl 5-Chloro-pyridin-2-ylmethyl A.2259 cyclopropyl 6-Chloro-pyridin-2-ylmethyl A. 2260 cyclopropyl 5-Chloro-pyridin-3-ylmethyl A.2261 cyclopropyl 6-Chloro-pyridin-3-ylmethyl A.2262 cyclopropyl 2-Chloro-pyridin-4-ylmethyl A.2263 cyclopropyl 2-pyrimidinylmethyl A.2264 cyclopropyl 4-chloro-pyrimidin-2-ylmethyl A.2265 cyclopropyl 5-chloro-pyrimidin-2-ylmethyl A.2266 cyclopropyl 2-Chloro-pyrimidin-4-ylmethyl A.2267 cyclopropyl 6-Chloro-pyrimidin-4-ylmethyl A.2268 cyclopropyl 2-chloro-pyrimidin-5-ylmethyl A.2269 cyclopropyl 4-Pyridazinylmethyl A.2270 cyclopropyl 2-pyrazinylmethyl A.2271 cyclopropyl 5-Chloro-pyrazin-2-ylmethyl A.2272 cyclopropyl 5-Chloro-pyrazin-2-ylmethyl A.2273 cyclopropyl Ϊ-Pyridazinylmethyl A.2274 cyclopropyl 5-chloropyridazine-3-ylmethyl

Nr. R ² R ⁴ A.2275 cyclopropyl 1,3,5-Triazinylmethyl A.2276 cyclopropyl 2-furylmethyl A.2277 cyclopropyl 3-furylmethyl A.2278 cyclopropyl 4-bromofuro-2-ylmethyl A.2279 cyclopropyl 5-Chlorofur-2-ylmethyl A.2280 cyclopropyl 2-thienylmethyl A.2281 cyclopropyl 3-thienylmethyl A.2282 cyclopropyl 5-methyl-thien-3-ylmethyl A.2283 cyclopropyl 5-Chlorothien-2-ylmethyl A.2284 cyclopropyl 2-Chlorothien-4-ylmethyl A.2285 cyclopropyl 2 -Pyrrolylmethyl A.2286 cyclopropyl 3-pyrrolylmethyl A.2287 cyclopropyl 2-oxazolylmethyl A.2288 cyclopropyl 4-Methyl-oxazol-2-ylmethyl A.2289 cyclopropyl 5-Methyl-oxazol-2-ylmethyl A.2290 cyclopropyl 4-chlorooxazole-2-ylmethyl A.2291 cyclopropyl 5-chlorooxazole-2-ylmethyl A.2292 cyclopropyl 4-oxazolylmethyl A.2293 cyclopropyl 2-Methyl-oxazol-4-ylmethyl A.2294 cyclopropyl 5-Methyl-oxazol-4-ylmethyl A.2295 cyclopropyl 2-chlorooxazole-4-ylmethyl A.2296 cyclopropyl 5-chlorooxazole-4-ylmethyl A.2297 cyclopropyl 5-oxazolylmethyl A.2298 cyclopropyl 2-Methyl-oxazol-5-ylmethyl A.2299 cyclopropyl 4-Methyl-oxazol-5-ylmethyl A.2300 cyclopropyl 2-chlorooxazole-5-ylmethyl A.2301 cyclopropyl 4-Chlorooxazol-5-ylmethyl A.2302 cyclopropyl 2-Thiazolylmethyl ' A.2303 cyclopropyl 4-Methylthiazol-2-ylmethyl i A.2304 cyclopropyl 5-Methylthiazol-2-ylmethyl; A.2305 cyclopropyl 4-Chlorothiazol-2-ylmethyl A.2306 cyclopropyl 5-Chlorothiazol-2-ylmethyl j A.2307 cyclopropyl 4-Thiazolylmethyl j A.2308 cyclopropyl 2-Methylthiazol-4-ylmethyl | A.2309 cyclopropyl 5-Methylthiazol-4-ylmethyl j A.2310 cyclopropyl 2-Chlorothiazol-4-ylmethyl | A.2311 cyclopropyl 5-Chloro-thiazol-4-ylmethyl A.2312 cyclopropyl 5thiazolylmethyl A.2313 cyclopropyl 2-Methylthiazol-5-ylmethyl

- Uf -

Nr. R ² R ⁴ A.2314 cyclopropyl 4-Methylthiazol-5-ylmethyl A.2315 cyclopropyl 2-Chlorothiazol-5-ylmethyl A.2316 cyclopropyl 4-Chlorothiazol-5-ylmethyl A.2317 cyclopropyl 3-isoxazolylmethyl A.2318 cyclopropyl 4-Methyl-isoxazol-3-ylmethyl A.2319 cyclopropyl 5-Methyl-isoxazol-3-ylmethyl A.2320 cyclopropyl 4-Chloroisoxazol-3-ylmethyl A.2321 cyclopropyl 5-Chloroisoxazol-3-ylmethyl A.2322 cyclopropyl 4-Isoxazolylmethyl A.2323 cyclopropyl 3-Methylisoxazol-4-ylmethyl A.2324 cyclopropyl 5-Methyl-isoxazol-4-ylmethyl A.2325 cyclopropyl 3-Chloroisoxazol-4-ylmethyl A.2326 cyclopropyl 5-Chloroisoxazol-4-ylmethyl A.2327 cyclopropyl 5-Isoxazolylmethyl A.2328 cyclopropyl 3-Methylisoxazol-5-ylmethyl A.2329 cyclopropyl 4-Methyl-isoxazol-5-ylmethyl A.2330 cyclopropyl 3-Chloroisoxazol-5-ylmethyl A.2331 cyclopropyl 4-Chloroisoxazol-5-ylmethyl A.2332 cyclopropyl 3-Isothiazolylmethyl A. 2333 cyclopropyl 4-isothiazolin-3-ylmethyl A.2334 cyclopropyl 5-isothiazolin-3-ylmethyl A.2335 cyclopropyl 4-Chloroisothiazol-3-ylmethyl A.2336 cyclopropyl 5-Chlorisothiazol-3-ylmethyl A.2337 cyclopropyl 4-Isothiazolylmethyl A.2338 cyclopropyl 3-methylisothiazol-4-ylmethyl A.2339 cyclopropyl 5-methylisothiazol-4-ylmethyl A.2340 cyclopropyl 3-Chloroisothiazol-4-ylmethyl A.2341 cyclopropyl 5-Chloroisothiazol-4-ylmethyl A.2342 cyclopropyl 5-Isothiazolylmethyl A.2343 cyclopropyl 3-Methylisothiazol-5-ylmethyl A.2344 cyclopropyl 4-methylisothiazol-5-ylmethyl A.2345 cyclopropyl 3-Chlorisothiazol-5-ylmethyl A.2346 cyclopropyl 4-Chloroisothiazol-5-ylmethyl A.2347 cyclopropyl 4-Imidazolylmethyl A.2348 cyclopropyl 1-Phenylpyrazol-3-ylmethyl A.2349 cyclopropyl 1-methyl-4-ylmethyl A.2350 cyclopropyl 1-Phenyl-1,2,4-triazol-3-ylmethyl A.2351 cyclopropyl 1,2,4-oxadiazol-3-ylmethyl A.2352 cyclopropyl 5-Chloro-l, 2,4-oxadiazol-3-ylmethyl

- tzo-

Nr. R ² R ⁴ A. 2353 cyclopropyl 5-Methyl-1,2,4-oxadiazol-3-ylmethyl A. 2354 cyclopropyl 5-Trifluoromethyl-1,2,4-oxadiazol-3-ylmethyl A. 2355 cyclopropyl 1,3,4-oxadiazol-2-ylmethyl A. 2356 cyclopropyl 5-Chloro-1,3,4-oxadiazol-2-ylmethyl A. 2357 cyclopropyl 5-Methyl-1,3,4-oxadiazol-2-ylmethyl A.2358 cyclopropyl 5-methoxy-1,3,4-oxadiazol-2-ylmethyl A.2359 cyclopropyl 1,2,4-thiadiazol-3-ylmethyl A.2360 cyclopropyl 5-Chloro-1,2,4-thiadiazol-3-ylmethyl A.2361 cyclopropyl 5-Methyl-1,2,4-thiadiazol-3-ylmethyl A.2362 cyclopropyl 1,3,4-thiadiazol-2-ylmethyl A. 2363 cyclopropyl 5-Chloro-1,3,4-thiadiazol-2-ylmethyl A.2364 cyclopropyl 5-methyl-1,3,4-thiadiazol-2-ylmethyl A.2365 cyclopropyl 5-Cyano-1,3,4-thiadiazol-2-ylmethyl A.2366 cyclopropyl 2- (2'-Pyridinyloxy) eth-1-yl A.2367 cyclopropyl 2- (3'-Pyridinyloxy) eth-1-yl A.2368 cyclopropyl 2- (4'-Pyridinyloxy) eth-1-yl A.2369 cyclopropyl 2- (2'-Pyrimidinyloxy) eth-1-yl A.2370 cyclopropyl 2- (4'-Pyrimidinyloxy) eth-1-yl A.2371 cyclopropyl 2- (5'-Pyrimidinyloxy) eth-1-yl j A.2372 cyclopropyl 2- (2'-Pyrazinyloxy) eth-1-yl A.2373 cyclopropyl 2- (2'-Pyridazinyloxy) eth-1-yl A.2374 cyclopropyl 2- (3'-Pyridazinyloxy) eth-1-yl A.2375 cyclopropyl 2- (1 ', 3', 5'-Triazinyloxy) eth-1-yl A.2376 cyclopropyl 2- (5'-Methylisoxazol-3'-yloxy) eth-1-yl A.2377 cyclopropyl 2- (5'-Chloroisoxazol-3'-yloxy) eth-1-yl A.2378 cyclopropyl 2- (2'-Methoxythiazol-4'-yloxy) eth-1-yl A.2379 cyclopropyl 2- (4'-Chlorooxazol-2'-yloxy) eth-1-yl A.2380 cyclopropyl 2- (1'-Phenyl-1'H-1 ', 2', 4'-triazol-3'-yloxy) eth-1-yl A.2381 cyclopropyl 2- (1'-Phenylpyrazol-3'-yloxy) eth-1-yl A.2382 cyclopropyl c ₆ h ₅ A.2383 cyclopropyl 2-Cl-C ₆ H ₄ A.2384 cyclopropyl 3-Cl-C ₆ H ₄ f A.2385 cyclopropyl 4-Cl-C ₆ H ₄ ! A.2386 cyclopropyl 2,3-Cl ₂ -C ₆ H ₃ i A.2387 cyclopropyl 2,4-Cl ₂ -c ₆ h ₃ ; A.2388 cyclopropyl 2,5-Cl ₂ -C ₆ H ₃ ; A.2389 cyclopropyl 3,4-c ₂ -c ₆ h ₃ ; A.2390 cyclopropyl 1,5-Cl ₂ -C ₆ H ₃

Nr. R ² R ⁴ A.2391 cyclopropyl 4-CN-C ₆ H ₄ A.2392 cyclopropyl 2-NO ₂ -C ₆ H ₄ A.2393 cyclopropyl 3-NO ₂ -C ₆ H ₄ . A.2394 cyclopropyl 4-NO ₂ -C ₆ H ₄ A.2395 cyclopropyl 2,4- (NO ₂ ) ₂ -C ₆ H ₃ A.2396 cyclopropyl 2-CH ₃ -C ₆ H ₄ A. 2397 cyclopropyl 3-CH ₃ -C ₆ H ₄ A.2398 cyclopropyl 4-CH ₃ -C ₆ H ₄ A.2399 cyclopropyl _{{2,3-CH3) 2-C} H _{3 e} A.2400 cyclopropyl 2,4- (CH ₃ ) ₂ -C ₆ H ₃ A.2401 cyclopropyl 2,5- (CH ₃ ) ₂ -C ₆ H ₃ A.2402 cyclopropyl 2,6- (CH ₃ ) ₂ -C ₆ H ₃ A.2403 cyclopropyl 2-C ₆ H ₅ -C ₆ H ₄ A.2404 cyclopropyl 3-C ₆ H ₅ -C ₆ H ₄ A.2405 cyclopropyl 4-C ₆ H ₅ -C ₆ H ₄ A.2406 cyclopropyl 3-OCH ₃ -C ₆ H ₄ A.2407 cyclopropyl 4-OCH ₃ -C ₆ H ₄ A.2408 cyclopropyl 3 -AcetyľC6H ₄ A.2409 cyclopropyl 4 -AcetylCgH ₄ A.2410 cyclopropyl _{3-methoxycarbonyl-4} CEH A.2411 cyclopropyl Methoxycarbonyl-4-C 6 H ₄ A.2412 cyclopropyl 3-CF ₃ -C ₆ H ₄ A.2413 cyclopropyl 4-CF ₃ -C ₆ H ₄ A.2414 cyclopropyl 2-Naphthyl A.2415 cyclopropyl 6-chloropyridazine-3-yl A.2416 cyclopropyl 5-Chloro-pyrazin-2-yl A.2417 cyclopropyl Quinolin-2-yl A.2418 cyclopropyl 2,5-Dimethylpyrazin-3-yl A.2419 cyclopropyl Pyrazin-2-yl A.2420 cyclopropyl 3-chloropyrid-2-yl A.2421 cyclopropyl 6-chloropyrid-2-yl A.2422 cyclopropyl 4-Trifluoromethyl, 6-chloropyrid-2-yl A.2423 cyclopropyl 4-trifluoromethylpyrid-2-y1 A.2424 cyclopropyl 6-trifluoromethylpyrid-2-yl A.2425 cyclopropyl 6-methoxypyridin-2-y1 A.2426 cyclopropyl 5-Chloropyridin-2-yl A.2427 cyclopropyl Pyridin-2-yl A.2428 cyclopropyl Senzothiazol-2-yl A.2429 cyclopropyl 7-Chloro-quinolin-4-yl

-Ζ3Ί-

Nr. R ² R ⁴ A.2430 cyclopropyl 3-nitro-pyridin-2-yl A.2431 cyclopropyl Pyrrole-3-yl A.2432 cyclopropyl Pyrrol-2-yl A.2433 cyclopropyl 2,6-Dioctylpyrid-4-yl. A.2434 cyclopropyl 5-nitro-pyridin-2-yl A.2435 cyclopropyl Pyridin-4-yl A.2436 cyclopropyl Pyridin-3-yl A.2437 cyclopropyl Pyrimidin-2-yl A.2438 cyclopropyl Pyrimidin-4-yl A.2439 cyclopropyl Quinazolin-4-yl A.2440 cyclopropyl 6-Chloro-pyrimidin-4-yl A.2441 cyclopropyl 6-Methoxypyrimidin-4-yl A.2442 cyclopropyl 2,5,6-Trichloro-4-yl A.2443 cyclopropyl 2,6-dimethyl-pyrimidin-4-yl A.2444 cyclopropyl 2-Methyl, 6-chloropyrimidin-4-yl A.2445 cyclopropyl 2-Methyl, 6-Ethoxy-pyrimidin-4-yl A.2446 cyclopropyl 4,5,6-trichloro-2-yl A.2447 cyclopropyl 4,6-dimethoxypyrimidin-2-yl A.2448 cyclopropyl 4,6-Dimethylpyrimidin-2-yl A.2449 cyclopropyl 4,6-dichloropyrimidine-2-yl A.2450 cyclopropyl 4-Methyl, 6-methoxy-pyrimidin-2-yl A.2451 cyclopropyl 4-Chloro, 6-methoxypyrimidin-2-yl A.2452 cyclopropyl 6-Chloro-quinoxalin-2-yl A.2453 cyclopropyl 3,6-dichloro-l, 2,4-triazin-5-yl A.2454 cyclopropyl 4-Methoxy-1,3,5-triazin-2-yl; A.2455 cyclopropyl 4-Ethoxy-l, 3,5-triazin-2-yl A.2456 cyclopropyl 4,6-dichloro-l, 3,5-triazin-2-yl A.2457 cyclopropyl 4-Ethoxy, 6-Chloro-1,3,5-triazin-2-yl A.2458 cyclopropyl Isoxazol-3-yl A.2459 cyclopropyl Thien-2-yl A.2460 cyclopropyl Fur-2-yl A.2461 cyclopropyl Thiatriazole-5-yl A.2462 cyclopropyl E) -l-chloropropene-3-yl A.2463 cyclopropyl E) -4- (4'-Chlorophenyl) but-2-en-1-yl A.2464 cyclopropyl Propyn-3-yl A.2465 cyclopropyl Methylcarbonyl A.2466 cyclopropyl Ethylcarbonyl A.2467 ( cyclopropyl i-Propylcarbonyl A.2468 ( cyclopropyl i-Propylcarbonyl

'Z íl-

Nr. R ² R ⁴ A.2469 cyclopropyl n-Butylcarbonyl A.2470 cyclopropyl p-Butylcarbonyl A.2471 cyclopropyl i-Butylcarbonyl A.2472 cyclopropyl t-Butylcarbonyl A.2473 cyclopropyl n Pentylcarbonyl A.2474 cyclopropyl i-Pentylcarbonyl A.2475 cyclopropyl neo-Pentylcarbonyl A.2476 cyclopropyl n Hexylcarbonyl A.2477 cyclopropyl n Octylcarbonyl A.2478 cyclopropyl 1-Propenylcarbonyl A.2479 cyclopropyl 2-Penten-1-yl-carbonyl A.2480 cyclopropyl 2,5-heptadiene-yl-carbonyl A.2481 cyclopropyl benzoyl A.2482 cyclopropyl 2-chlorobenzoyl A.2483 cyclopropyl 3-chlorobenzoyl A.2484 cyclopropyl 4-chlorobenzoyl A.2485 cyclopropyl 2-Cyanobenzoyl A.2486 cyclopropyl 3 -Cyanobenzoyl A.2487 cyclopropyl 4-Cyanobenzoyl A.2488 cyclopropyl 4-methoxybenzoyl A.2489 cyclopropyl 2 -Pyridylcarbonyl A.2490 cyclopropyl 3 -Pyridylcarbonyl A.2491 cyclopropyl 4-Pyridylcarbonyl A.2492 cyclopropyl 2-Pyrimidinylcarbonyl A.2493 cyclopropyl 2-Oxazolylcarbonyl A.2494 cyclopropyl 4-Methyl-isoxazol-5-ylcarbonyl A.2495 cyclopropyl methylsulfonyl A.2496 cyclopropyl ethylsulfonyl A.2497 cyclopropyl n Propylsulfony1 A.2498 cyclopropyl i-propylsulfonyl A.2499 cyclopropyl n-butylsulfonyl A.2500 cyclopropyl t-butylsulfonyl A.2501 cyclopropyl n-pentylsulfonyl A.2502 cyclopropyl neo-pentylsulfonyl A.2503 cyclopropyl n-Hexylsulfonyl A.2504 cyclopropyl i-Octylsulfonyl A.2505 cyclopropyl ? henylsulfonyl A.2506 cyclopropyl 2-Chlorphenylsulfonyl A.2507 cyclopropyl 5-Chlorphenylsulfonyl

- 2i3-

Nr. R ² R ⁴ A.2508 cyclopropyl 4-Chlorophenylsulfonyl A.2509 cyclopropyl 2 -Cyanophenylsulfonyl A.2510 cyclopropyl 3 - Cyanophenyl sulphonyl A.2511 cyclopropyl 4 -Cyanophenylsulfonyl A.2512 cyclopropyl 2-Pyridylsulfonyl A.2513 cyclopropyl 3 -Pyridylsulfonyl A.2514 cyclopropyl 4-Pyridylsulfonyl A.2515 cyclopropyl 2-Pyrimidinylsulfonyl A.2516 cyclopropyl 4-0xazolylsulfonyl A.2517 cyclopropyl 5-Chloro-thiazol-2-ylsulfonyl A.2518 cyclopropyl 2-C ₄ H ₉ -C ₆ H ₄ -CH ₂ A.2519 cyclopropyl 3-C ₄ H ₉ -C ₆ H ₄ -CH ₂ j A.2520 cyclopropyl 4-C ₄ H ₉ -C ₆ H ₄ -CH ₂ j A.2521 cyclopropyl 2- (4'-Chlorothiazol-2'-yloxy) -eth-1-yl J A.2522 cyclopropyl 2- (1'-Methylpyrazol-4'-yloxy) eth-1-yl ( A.2523 cyclopropyl 4-Br-C ₆ H ₄ A.2524 cyclopropyl 3,5- (CH ₃ ) ₂ -C ₆ H ₃ I A.2525 cyclopropyl 4-C2H5-C6H4 A.2526 cyclopropyl 3-Dimethylaminocarbonyl-C6H4; A.2527 cyclopropyl 4-Dimethylaminocarbonyl-ββ4! A.2528 cyclopropyl 2-Hydroxyprop-1-yl A.2529 cyclopropyl 6-hydroxy-2-methylpyrimidin-4-ylmethyl A.2530 cyclopropyl [6-OH, 2-CH (CH ₃ ) ₂ -pyrimidin-4-yl] -CH 2 A.2531 cyclopropyl [6-OH, 2-CH (CH ₂ ) ₂ -pyrimidin-4-yl] -CH ₂ A.2532 cyclopropyl 5- (2'-Furan) -pent-1-yl A.2533 cyclopropyl 5- (2'-N-Methylpyrrol) pent-l-yl A.2534 cyclopropyl [2- (4-Cl-C ₆ H ₄₎ -oxazole-4-yl] _-CH2 A.2535 cyclopropyl 3 -CF ₃ -pyridin-2-yl A.2536 cyclopropyl 5-CF ₃ -pyridin-2-yl A. 2537 cyclopropyl 6- (2'-Thienyl) hex-1-yl; A.2538 cyclopropyl E) -3-Chlorobut-2-en-1-yl A.2539 cyclopropyl Z) -3-chloro-but-2-en-l-yl A.2540 cyclopropyl \ E) -2-bromo-but-2-en-l-yl A. 2541 cyclopropyl Z) -2-Bromobut-2-en-1-yl A.2542 cyclopropyl (E) -1-Chloroprop-1-en-3-yl A. 2543 cyclopropyl I'z) -l-chloro-prop-l-en-3-yl A.2544 cyclopropyl But-en-3-yl A.2545 cyclopropyl CH ₂ CH ₂ Br A.2546 Cyclopropyl CH ₂ CH ₂ CH ₂ Br

Nr. R ² R ⁴ A.2547 cyclopropyl CH ₂ CH ₂ CH ₂ CH ₂ Br A.2548 cyclopropyl Methylprop-2-yl A.2549 cyclopropyl Ethoxypropyl-2-yl A.2550 cyclopropyl 2-1sopropoxyprop-1-yl A.2551 cyclopropyl But-in-3-yl A.2552 cyclopropyl But-in-4-yl A.2553 cyclopropyl But-2-yn-4-yl A.2554 cyclopropyl Pent-in-4-yl A.2555 cyclopropyl Pent-2-yn-4-yl A.2556 cyclopropyl Pent-in-5-yl A.2557 cyclopropyl Pent-2-yn-5-yl A.2558 cyclopropyl E-2-chloro-but-2-en-l-yl A.2559 cyclopropyl Z-2-chloro-but-2-en-l-yl A.2560 cyclopropyl Z-l-chloro-prop-l-en-3-yl A.2561 cyclopropyl 2-methyl-prop-l-en-3-yl A.2562 cyclopropyl 2-chloro-prop-l-en-3-yl A.2563 cyclopropyl 2-bromoprop-l-en-3-yl A.2564 cyclopropyl But-2-en-l-yl A.2565 cyclopropyl But-3-en-l-yl A.2566 cyclopropyl l-Iodprop-l-yn-3-yl Oh. 2567 cyclopropyl E-3-bromo-but-2-en-l-yl A.2568 cyclopropyl Z-3-bromo-but-2-en-l-yl A.2569 11-C3H7 H A.2570 nC ₃ H ₇ ch ₃ A.2571 n-C3H7 c ₂ h ₅ A.2572 n-C3H7 nC3H7 A.2573 11-C3H7 I-C3H7 A.2574 nC ₃ H ₇ cyclopropyl A.2575 1V-C3H7 11-C4H9 A.2576 nC ₃ H ₇ SC ₄ Hg A.2577 nC ₃ H ₇ -C ₄ H9 A.2578 nC ₃ 17 t-č ₄ Hg A.2579 n-C3H7 n CSHN A.2580 nC ₃ H ₇ i-CsHu A.2581 n-C 3 H ₇ neo-CsHii A.2582 C1-C3H7 ľyclopentyl A.2583 1-C3H7 1-C6H13 A.2584 1-C3H7 Zyclohexyl A.2585 i I-C3H7 1 l-CgHi7

- from 3 r-

Nr. R ² R ⁴ A.2586 nC ₃ H ₇ CH ₂ CH ₂ Cl A.2587 nC ₃ H ₇ (ch ₂ ) ₄ ci A.2588 nC ₃ H ₇ ch ₂ cn A.2589 nC ₃ H ₇ ch ₂ ch ₂ cn A.2590 nC ₃ H ₇ (CH ₂ ) ₃ CN A.2591 nC ₃ H ₇ (CH ₂ ) ₄ CN A.2592 nC ₃ H ₇ (ch ₂ ) ₆ cn A. 2593 nC ₃ H ₇ Cyclohexylmethyl A.2594 nC ₃ H ₇ 2-Cyclohexyleth-1-yl A.2595 nC ₃ H ₇ cyclopropylmethyl A.2596 nC ₃ H ₇ 2-Cyclopropyleth-yl A.2597 nC ₃ H ₇ 2-methoxyethyl-yl A.2598 nC ₃ H ₇ 2-Ethoxyeth-1-yl A.2599 nC ₃ H ₇ 2-lsopropoxyeth-1-yl A.2600 nC ₃ H ₇ 3-methoxypropyl-1-yl A.2601 nC ₃ H ₇ 3-ethoxypropyl-1-yl A.2602 nC ₃ H ₇ 3-Isopropoxyprop-yl A.2603 nC ₃ H ₇ 4-Me thoxybut-1-yl A.2604 nC ₃ H ₇ 4-Isopropoxy-but-1-yl A.2605 nC ₃ H ₇ Propen-3-yl A.2606 nC ₃ H ₇ But-2-en-l-yl A.2607 nC ₃ H ₇ 3-methyl-but-2-en-1-yl A.2608 nC ₃ H ₇ 2-Vinyloxyeth-1-yl A.2609 nC ₃ H ₇ Allyloxyeth-1-yl A.2610 nC ₃ H ₇ 2-Trifluoromethoxyeth-1-yl A.2611 nC ₃ H ₇ -Trifluormethoxyprop-1-yl A.2612 nC ₃ H ₇ 4-Difluoromethoxybutyl A.2613 nC ₃ H ₇ Hydroxycarbonylmethyl A.2614 nC ₃ H ₇ Methoxycarbonylmethyl j A.2615 nC ₃ H ₇ Aminocarbonylmethyl j 1 A.2616 nC ₃ H ₇ N-Methylaminocarbonylmethyl A.2617 nC ₃ H ₇ N, N-Dimethylaminocarbonylmethyl i A.2618 nC ₃ H ₇ 2-Hydroxycarbonyleth-1-yl | A.2619 QC ₃ H ₇ 2-Methoxycarbonyleth-1-yl; A.2620 nC ₃ H ₇ 2-Aminocarbonyleth-1-yl; A.2621 iC ₃ H ₇ 2-N-Methylaminocarbonyleth-1-yl A.2622 iC ₃ H ₇ 2-Dimethylaminocarbonyleth-1-yl A.2623 i IC ₃ H ₇ 2-aminoethyl-l-yl A.2624 i iC ₃ H ₇ 2-amino-prop-1-yl

- 726-

Nr. R ² R ⁴ A.2625 nC ₃ H ₇ 4-Aminobut-1-yl A.2626 nC ₃ H ₇ 3-Dimethylaminoprop-1-yl A.2627 nC ₃ H ₇ 4-Aminothiocarbonylbut-1-yl A.2628 nC ₃ H ₇ 2-oxo-propyl A.2629 nC ₃ H ₇ cyclohexyl A.2630 nC ₃ H ₇ cyclopropyl A.2631 nC ₃ H ₇ cyclopentyl A.2632 nC ₃ H ₇ 2-Methoxyiminoprop-yl A.2633 nC ₃ H ₇ 2--Methoxyiminoeth-yl A.2634 nC ₃ H ₇ 6-Aminocarbonylhex-1-yl A.2635 nC ₃ H ₇ Aminothiocarbonylprop 3-yl A.2636 nC ₃ H ₇ 2-Aminothiocarbonyleth-yl A.2637 nC ₃ H ₇ Aminothiocarbonylmethyl A.2638 nC ₃ H ₇ 4- (N, N-dimethylamino) but-l-yl A.2639 nC ₃ H ₇ 2- (Methylthio) eth-1-yl A.2640 nC ₃ H ₇ 2- (methylsulfonyl) eth-1-yl A.2641 nC ₃ H ₇ 4- (Methylthio) prop-1-yl A.2642 nC ₃ H ₇ 4- (methylsulfonyl) prop-1-yl A.2643 nC ₃ H ₇ benzyl A.2644 nC ₃ H ₇ 2-FC ₆ H ₄ -CH ₂ A.2645 nC ₃ H ₇ 3 “FC ₆ H ₄ -CH ₂ A.2646 nC ₃ H ₇ 4-FC ₆ H ₄ -CH ₂ A.2647 nC ₃ H ₇ 2,3-F ₂ -C ₆ H ₃ -CH ₂ A.2648 nC ₃ H ₇ 2,4-F ₂ -C ₆ H ₃ -CH ₂ A.2649 nC ₃ H ₇ 2,5-F ₂ -C ₆ H ₃ -CH ₂ A.2650 nC ₃ H ₇ 2,6-P ₂ C ₆ H ₃ CH ₂ A.2651 nC ₃ H ₇ 3,4-F ₂ -C ₆ H ₃ -CH ₂ A.2652 nC ₃ H ₇ 3,5-F ₂ -C ₆ H ₃ -CH ₂ A.2653 nC ₃ H ₇ 2 -C 1 -C ₆ H ₄ -CH ₂ A.2654 nC ₃ H ₇ 3 -C 1 -C ₆ H ₄ -CH ₂ A.2655 nC ₃ H ₇ 4 -Cl -C ₆ H ₄ -CH ₂ A.2656 nC ₃ H ₇ 2,3-Cl ₂ -C ₆ H ₃ -CH ₂ A.2657 nC ₃ H ₇ 2,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.2658 nC ₃ H ₇ 2,5-Cl ₂ -C ₆ H ₃ -CH ₂ A.2659 n — C ₃ H ₇ 2,6-Cl ₂ -C ₆ H ₃ -CH ₂ A.2660 nC ₃ H ₇ 3,4-Cl ₂ -C ₆ H ₃ -CH ₂ A.2661 tl-C ₃ H ₇ 3,5-Cl ₂ -C ₆ H ₃ -CH ₂ A.2662 iC ₃ H ₇ 2,3,4-Cl ₃ -C ₆ H ₂ -CH ₂ A.2663 1-C ₃ H ₇ 2,3,5-Cl ₃ -C ₆ H ₂ -CH ₂

23Ί -

Nr. R ² R ⁴ A.2664 nC ₃ H ₇ 2,3,6-Cl ₃ -C ₆ H ₂ -CH ₂ A.2665 nC ₃ H ₇ 2,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ A.2666 nC ₃ H ₇ 2,4,6-Cl ₃ -C ₆ H ₂ -CH ₂ A.2667 nC ₃ H ₇ 3,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ A. 2668 nC ₃ H ₇ 2-Br-C ₆ H ₄ CH ₂ A.2669 nC ₃ H ₇ 3-Br-C ₆ H ₄ CH ₂ A.2670 nC ₃ H ₇ 4 -Br-C ₆ H ₄ CH ₂ A.2671 nC ₃ H ₇ 2,3-Br ₂ -C ₆ H ₃ -CH ₂ A.2672 nC ₃ H ₇ 2,4-Br ₂ -C ₆ H ₃ -CH ₂ A.2673 nC ₃ H ₇ 2,5-Br ₂ -C ₆ H ₃ -CH ₂ A.2674 nC ₃ H ₇ 2,6-Br ₂ -C ₆ H ₃ -CH ₂ A.2675 nC ₃ H ₇ 3,4-Br ₂ -C ₆ H ₃ -CH ₂ A.2676 nC ₃ H ₇ 3,5-Br ₂ -C ₆ H ₃ -CH ₂ A.2677 nC ₃ H ₇ 2-F, 3-C 1 -C ₆ H ₃ -CH ₂ A.2678 nC ₃ H ₇ 2-F, 4-C1-C ₆ H ₃ CH ₂ A.2679 nC ₃ H ₇ 2-F, 5-C 1-C ₆ H ₃ CH ₂ A.2680 nC ₃ H ₇ 2-F, 3-Br-C ₆ H ₃ CH ₂ A.2681 nC ₃ H ₇ 2-F, 4-Br-C ₆ H ₃ CH ₂ A.2682 nC ₃ H ₇ 2-F, 5-Br-C ₆ H ₃ CH ₂ A.2683 nC ₃ H ₇ 2-C1, 3-Br-C ₆ H ₃ CH ₂ A.2684 nC ₃ H ₇ 2-C1, 4-Br-C ₆ H ₃ CH ₂ A.2685 nC ₃ H ₇ 2-C1, 5-Br-C ₆ H ₃ CH ₂ A.2686 nC ₃ H ₇ 3-F, 4-C1-C ₆ H ₃ CH ₂ A.2687 nC ₃ H ₇ 3-F, 5-Cl-C ₆ H ₃ CH ₂ A.2688 nC ₃ H ₇ 3-F, 6-C 1 -C ₆ H ₃ -CH ₂ A.2689 nC ₃ H ₇ 3-F, 4-Br-C ₆ H ₃ CH ₂ A.2690 nC ₃ H ₇ 3-F, 5-Br-C ₆ H ₃ CH ₂ A.2691 nC ₃ H ₇ 3-F, 6-Br-C ₆ H ₃ CH ₂ A.2692 nC ₃ H ₇ 3-C1, 4-Br-C ₆ H ₃ CH ₂ A.2693 nC ₃ H ₇ 3-C1, 5-Br-C ₆ H ₃ CH ₂ A.2694 nC ₃ H ₇ 3-C1, 6-Br-C ₆ H ₃ CH ₂ A.2695 nC ₃ H ₇ 4-F, 5-Cl-C ₆ H ₃ CH ₂ A.2696 nC ₃ H ₇ 4-F, 6-Cl-C ₆ H ₃ CH ₂ A.2697 nC ₃ H ₇ 4-F, 5-Br-C ₆ H ₃ CH ₂ A.2698 nC ₃ H ₇ 4-F, 6-Br-C ₆ H ₃ CH ₂ A.2699 nC ₃ H ₇ 4-C1, 5-Br-C ₆ H ₃ CH ₂ A.2700 iC ₃ H ₇ 5-F, 6-C1-C ₆ H ₃ CH ₂ A.2701 iC ₃ H ₇ 5-F, 6-Br-C ₆ H ₃ CH ₂ A.2702 i iC ₃ H ₇ 5-C1, 6-Br-C ₆ H ₃ CH ₂

Nr. R ² R ⁴ A.2703 nC ₃ H ₇ 3-Br, 4-C1, 5-Br-C ₆ H ₂ CH ₂ A.2704 nC ₃ H ₇ 2-CN-C ₅ H ₄ -CH ₂ A.2705 nC ₃ H ₇ 3-CN-C ₆ H ₄ CH ₂ A.2706 nC ₃ H ₇ 4-CN-C ₆ H ₄ CH ₂ A.2707 nC ₃ H ₇ 2 -NO ₂ -C ₆ H ₄ -CH ₂ A.2708 nC ₃ H ₇ 3-NO ₂ -C ₆ H ₄ -CH ₂ A.2709 nC ₃ H ₇ 4-NO 2 -C ₆ H ₄ -CH ₂ A.2710 nC ₃ H ₇ 2-CH ₃ -C ₆ H ₄ -CH ₂ A.2711 nC ₃ H ₇ 3-CH ₃ -C ₆ H ₄ -CK ₂ A.2712 nC ₃ H ₇ 4-CH ₃ -C ₆ H ₄ -CH ₂ A.2713 nC ₃ H ₇ 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2714 nC ₃ H ₇ 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2715 nC ₃ H ₇ 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2716 nC ₃ H ₇ 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2717 nC ₃ H ₇ 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2718 11-C3H7 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2719 11-C3H7 2-C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2720 n-C3H7 3 -C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2721 nC ₃ H ₇ 4-C ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2722 n-C3H7 2-C ₃ H ₇ -C ₆ H ₄ -CH ₂ A.2723 nC ₃ H ₇ 3-C ₃ H ₇ -C ₆ H 4 -CH ₂ A.2724 nC ₃ H ₇ 4-C ₃ H ₇ -C ₆ H ₄ -CH ₂ A.2725 11-C3H7 2 -Cyclohexyl - C 8 H ₄ - CH ₂ A.2726 nC ₃ H ₇ 3 - Cyclohexyl - CGH ₄ -CH ₂ A.2727 11-C3H7 - Cyclohexyl - C 8 H ₄ - CH ₂ A.2728 nC ₃ H ₇ 2-Vinyl-C ₆ H ₄ -CH ₂ A.2729 T1-C3H7 3-Vinyl -C ₆ H ₄ -CH ₂ A.2730 J1-C3H7 4-Vinyl-C ₆ H ₄ CH ₂ A.2731 nC ₃ H ₇ 2-allyl-C ₆ H ₄ CH ₂ A. 2732 nC ₃ H ₇ 3-allyl-C ₆ H ₄ CH ₂ A. 2733 nC ₃ H ₇ 4-Allyl-C ₆ H ₄ CH ₂ A.2734 nC ₃ H ₇ 2-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.2735 nC ₃ H ₇ 3-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A.2736 n-C ₃ H ₇ 4-C ₆ H ₅ -C ₆ H ₄ -CH ₂ A. 2737 nC ₃ H ₇ 3-CH 3, 5-C ₄ H ₉ -C ₆ H ₃ -CH ₂ A.2738 nC ₃ H ₇ 2-OH-C ₆ H ₄ CH ₂ A.2739 C3H7 3-OH-C ₆ H ₄ CH ₂ A.2740 iC ₃ H ₇ i-oh-c ₆ h ₄ -ch ₂ A.2741 i iC ₃ H ₇ 2-OCH 3 -C ₆ H ₄ -CH ₂

Nr. R ² R ⁴ A.2742 nC ₃ H ₇ 3-OCH ₃ -C ₆ H ₄ -CH ₂ A.2743 nC ₃ H ₇ 4-OCH ₃ -C ₆ H ₄ -CH ₂ A.2744 n — C ₃ H ₇ 2,3- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2745 nC ₃ H ₇ 2,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2746 nC ₃ H ₇ 2,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2747 nC ₃ H ₇ 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2748 nC ₃ H ₇ 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ A.2749 nC ₃ H ₇ 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH ₂ A.2750 nC ₃ H ₇ 2-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2751 nC ₃ H ₇ 3-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2752 nC ₃ H ₇ 4-OC ₂ H ₅ -C ₆ H ₄ -CH ₂ A.2753 nC ₃ H ₇ 2-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A. 2754 nC ₃ H ₇ 3-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.2755 nC ₃ H ₇ 4-O- (nC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.2756 nC ₃ H ₇ 2-O- (iC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.2757 nC ₃ H ₇ 3-O- (iC ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.2758 nC ₃ H ₇ 4-O- (C ₃ H ₇ ) -C ₆ H ₄ -CH ₂ A.2759 nC ₃ H ₇ 4-O- (nC ₄ H ₉ ) -C ₆ H ₄ -CH ₂ A.2760 nC ₃ H ₇ 3-O- (t C ₄ H ₉ ) -C ₆ H ₄ -CH ₂ A.2761 nC ₃ H ₇ 4-O- (nC ₆ H ₃ ) -C ₆ H ₄ -CH ₂ A.2762 nC ₃ H ₇ 2-O-allyl-C ₆ H ₄ CH ₂ A.2763 nC ₃ H ₇ 3-O-allyl-C ₆ H ₄ CH ₂ A.2764 nC ₃ H ₇ 4-O-allyl-C ₆ H ₄ CH ₂ A.2765 nC ₃ H ₇ 2-CF ₃ -C ₆ H ₄ -CH ₂ A.2766 nC ₃ H ₇ 3 -CF ₃ -C ₆ H ₄ -CH ₂ A.2767 nC ₃ H ₇ 4-CF ₃ -C ₆ H ₄ -CH ₂ A.2768 nC ₃ H _{7 2-Acetyl-4 -CH2} -0δΗ A.2769 nC ₃ H ₇ 3-Acetyl-C ₆ H ₄ CH ₂ A.2770 nC ₃ H ₇ 4-Acetyl-C ₆ H ₄ CH ₂ A.2771 nC ₃ H ₇ 2-Methoxycarbonyl -C ₈ H ₄ -CH ₂ A.2772 nC ₃ H ₇ 3-Methoxycarbonyl - (½¾ -CH ₂ A.2773 nC ₃ H ₇ 4-Methoxycarbonyl - C ₆ H ₄ -CH ₂ A.2774 nC ₃ H ₇ 2-Aminocarbonyl -C ₈ H ₄ -CH ₂ A.2775 nC ₃ H ₇ 3-Aminocarbonyl -C ₈ H ₄ -CH ₂ A.2776 nC ₃ H ₇ 4-Aminocarbonyl -C ₆ H ₄ -CH ₂ A.2777 nC ₃ H ₇ 2-Dimethylaminocarbonyl-C 8 H ₄ -CH ₂ A.2778 iC ₃ H ₇ -Dimethylaminocarbonyl 3-C 6 H ₄ -CH ₂ A.2779 iC ₃ H ₇ 4-Dimethylaminocarbonyl -C ₈ H ₄ -CH ₂ A.2780 iC ₃ H ₇ 2- (N-Methylaminocarbonyl) -C ₆ H ₄ -CH ₂

W-

Nr. R ² R ⁴ A.2781 nC ₃ H ₇ 3- (N-Methylaminocarbonyl) -C ₆ H ₄ -CH ₂ A.2782 11-C3H7 4- (N-Methylaminocarbonyl) -C ₈ H ₄ -CH ₂ A.2783 nC ₃ H ₇ 2 -H ₂ NC ₆ H ₄ -CH ₂ A.2784 nC ₃ H ₇ 3-H ₂ NC ₆ H ₄ -CH ₂ S ~ ' A.2785 nC ₃ H ₇ 4 -H ₂ NC ₆ H ₄ -CH ₂ A.2786 nC ₃ H ₇ 2-Aminothiocarbonyl-C 6 H ₄ -CH ₂ A.2787 nC ₃ H ₇ 3-Aminothiocarbonyl-ββ ₄ -CH ₂ A.2788 nC ₃ H ₇ 4-Aminothiocarbonyl-C ₆ H ₄ -CH ₂ A.2789 nC ₃ H _{7 2-methoxyimino-methyl-4} CEH - _CH2 A.2790 n-C ₃ H 7 -Methoxyiminomethyl 3-C 6 H ₄ -CH ₂ A.2791 nC ₃ H ₇ 4-methoxyimino - C 6 H ₄ -CH ₂ A.2792 nC ₃ H ₇ 2 - Forms 1 - C 8 H ₄ - CH ₂ A.2793 nC ₃ H ₇ 3-Formyl-C ₆ H ₄ -CH ₂ A.2794 nC ₃ H ₇ 4-formyl-C ₆ H ₄ CH ₂ A.2795 nC ₃ H ₇ 2- (1'-Methoxyiminoeth-1'-yl) -C ₆ H ₄ -CH ₂ A.2796 nC ₃ H ₇ 3- (1'-Methoxyiminoeth-1'-yl) -C ₆ H ₄ -CH ₂ A.2797 nC ₃ H ₇ 4- (1'-Methoxyiminoeth-1'-yl) -C ₈ H ₄ -CH ₂ A. 2798 nC ₃ H ₇ 2-SCH ₃ -C ₆ H ₄ -CH ₂ A.2799 nC ₃ H ₇ 3 -SCH ₃ -C ₆ H ₄ -CH ₂ A.2800 nC ₃ H ₇ 4-SCH ₃ -C ₆ H ₄ -CH ₂ A.2801 nC ₃ H ₇ 2-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ A.2802 nC ₃ H ₇ 3 -SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ A.2803 nC ₃ H ₇ 4-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ A.2804 nC ₃ H ₇ 2-OCF ₃ -C ₆ H ₄ -CH ₂ A.2805 nC ₃ H ₇ 3 -OCF ₃ -C ₆ H ₄ -CH ₂ A.2806 nC ₃ H ₇ 4-OCF ₃ -C ₆ H ₄ -CH ₂ A.2807 nC ₃ H ₇ 2 -OCHF ₂ -C ₆ H ₄ -CH ₂ A.2808 nC ₃ H ₇ 3 -OCHF ₂ -C ₆ H ₄ -CH ₂ A.2809 nC ₃ H ₇ 4 -OCHF ₂ -C ₆ H ₄ -CH ₂ A.2810 nC ₃ H ₇ 3-CF ₃ , 4-OCF ₃ -C ₆ H ₃ -CH ₂ A.2811 nC ₃ H _{7 1-Naphthyl-CH2} A.2812 nC ₃ H ₇ 2-Naphthyl-CH ₂ A.2813 nC ₃ H ₇ 2-Phenoxyeth-1-yl A.2814 nC ₃ H ₇ 2- (2'-Chlorophenoxy) eth-1-yl A.2815 nC ₃ H ₇ 2- (3'-Chlorphenoxy) eth-l-yl A.2816 nC ₃ H ₇ 2- (4'-Chlorophenoxy) eth-1-yl A.2817 aC ₃ H ₇ 2- (3 ', 5'-Dichlorophenoxy) eth-1-yl A.2818 iC ₃ H ₇ 2- (2'-Cyanophenoxy) eth-1-yl A.2819 ic ₃ h ₇ 2- (3 ' -Cyanophenoxy) eth-1-yl

Nr. R ² R ⁴ A.2820 nC ₃ H ₇ 2- (4'-Cyanophenoxy) eth-l-yl A.2821 nC ₃ H ₇ 2- (2'-methylphenoxy) eth-l-yl A.2822 nC ₃ H ₇ 2- (3'-methylphenoxy) eth-l-yl A.2823 nC ₃ H ₇ 2- (4 * -Methylphenoxy) eth-l-yl A.2824 nC ₃ H ₇ 2- (3'-t-Butylphenoxy) eth-1-yl A.2825 nC ₃ H ₇ 2- (4'-t-Butylphenoxy) eth-1-yl A.2825 nC ₃ H ₇ 2- (2'-Nitrophenoxy) eth-l-yl A.2827 nC ₃ H ₇ 2- (3'-Nitrophenoxy) eth-l-yl A.2828 nC ₃ H ₇ 2- (4 * -Nitrophenoxy) eth-1-yl A.2829 nC ₃ H ₇ 2- (2-methoxyphenoxy) eth-l-yl A.2830 nC ₃ H ₇ 2- (3'-methoxyphenoxy) eth-1-yl A.2831 nC ₃ H ₇ 2- (4'-methoxyphenoxy) eth-l-yl A.2832 nC ₃ H ₇ 2- (2'-Trifluoromethylphenoxy) eth-1-yl j A.2833 nC ₃ H ₇ 2- (3'-Trifluoromethylphenoxy) eth-1-yl 1 A.2834 nC ₃ H ₇ 2- (4'-Trifluoromethylphenoxy) eth-1-yl A.2835 nC ₃ H ₇ 2- (2'-Acetylphenoxy) eth-1-yl; A.2836 nC ₃ H ₇ 2- (3'-Acetylphenoxy) eth-1-yl A.2837 nC ₃ H ₇ 2- (4'-Acetylphenoxy) eth-1-yl; A.2838 nC ₃ H ₇ 2- (2'-Methoxycarbonyl) eth-1-yl! A.2839 nC ₃ H ₇ 2- (3'-Methoxycarbonyl) eth-1-yl A.2840 nC ₃ H ₇ 2- (4'-methoxycarbonyl) eth-l-yl A.2841 nC ₃ H ₇ 2- (2'-Dimethylaminocarbonyl) eth-1-yl A.2842 nC ₃ H ₇ 2- (3'-Dimethylaminocarbonyl) eth-1-y1 A.2843 nC ₃ H ₇ 2- (4'-Dimethylaminocarbonyl) eth-1-y1 A.2844 nC ₃ H ₇ 2- (2-Aminothiocarbonyl) eth-1-yl A.2845 nC ₃ H ₇ 2- (3'-Aminothiocarbonyl) eth-1-yl A.2846 nC ₃ H ₇ 2- (4'-Aminothiocarbonyl) eth-1-yl A.2847 nC ₃ H ₇ 2- (2'-Methylsulfonyl) eth-1-yl A.2848 nC ₃ H ₇ 2- (3'-methylsulfonyl) eth-l-yl A.2849 nC ₃ H ₇ 2- (4'-Methylsulfonyl) eth-1-yl A.2850 nC ₃ H ₇ 3-Phenoxyprop-1-yl A.2851 nC ₃ H ₇ 3- (2'-Chlorophenoxy) prop-1-yl A.2852 nC ₃ H ₇ 3- (3'-Chlorophenoxy) prop-1-yl A.2853 nC ₃ H ₇ 3- (4'-Chlorophenoxy) prop-1-yl A.2854 nC ₃ H ₇ 3- (3 *, 5 ', Dichlorophenoxy) prop-1-yl A.2855 aC ₃ H ₇ 3- (2'-Cyanophenoxy) prop-1-yl A.2856 iC ₃ H ₇ 3- (3'-Cyanophenoxy) prop-1-yl A.2857 IC ₃ H ₇ 3- (4'-Cyanophenoxy) prop-l-yl A.2858 i iC ₃ H ₇ 3 * (2'-methylphenoxy) prop-1-yl

W-

Nr. R ² R ⁴ A.2859 nC ₃ H ₇ 3- (3'-methylphenoxy) prop-1-yl A.2860 nC ₃ H ₇ 3- (4'-methylphenoxy) prop-l-yl A.2861 nC ₃ H ₇ 3- (2'-Methoxyphenoxy) prop-1-yl A.2862 nC ₃ H ₇ 3- {3 ' methoxyphenoxy) prop-1-yl A.2863 nC ₃ H ₇ 3- (4'-methoxyphenoxy) prop-1-yl A.2864 nC ₃ H ₇ 3- (2'-Trifluoromethylphenoxy) prop-1-yl A.2865 nC ₃ H ₇ 3- (3 ' Trifluormethylphenoxy) prop-1-yl A.2866 nC ₃ H ₇ 3- (4'-Trifluormethylphenoxy) prop-l-yl A.2867 nC ₃ H ₇ 4-Phenoxybut-1-yl A.2868 nC ₃ H ₇ 2-Phenyleth-1-yl A.2869 nC ₃ H ₇ 2- (2'-Chlorophenyl) eth-1-yl A.2870 nC ₃ H ₇ 2- (3'-Chlorphenyl) eth-1-yl A.2871 nC ₃ H ₇ 2- (4'-Chlorophenyl) eth-1-yl A.2872 nC ₃ H ₇ 2- (3 ', 5'-Dichlorphenyl) eth-l-yl A.2873 nC ₃ H ₇ 2- (2'-cyanophenyl) eth-l-yl A.2874 nC ₃ H ₇ 2- (3'-Cyanophenyl) eth-1-yl A.2875 nC ₃ H ₇ 2- (4'-cyanophenyl) eth-l-yl A.2876 nC ₃ H ₇ 2- (2'-Methylphenyl) eth-1-yl A.2877 nC ₃ H ₇ 2- (3'-Methylphenyl) eth-l-yl A. 2878 nC ₃ H ₇ 2- (4'-Methylphenyl) eth-1-yl A. 2879 nC ₃ H ₇ 2- (2'-Methoxyphenyl) eth-1-yl A.2880 nC ₃ H ₇ 2- (3'-Methoxyphenyl) eth-1-yl A.2881 nC ₃ phi ₇ 2- (4'-Methoxyphenyl) eth-l-yl A.2882 nC ₃ H ₇ 2- (2 ' Trifluormethylphenyl) eth-l-yl A.2883 nC ₃ H ₇ 2- (3 ' Trifluormethylphenyl) eth-l-yl A.2884 nC ₃ H ₇ 2- (4'-Trifluoromethylphenyl) eth-1-yl A.2885 nC ₃ H ₇ 3-Phenylprop-1-yl A.2886 nC ₃ H ₇ 3- (2-Chlorphenyl) prop-1-yl A.2887 nC ₃ H ₇ 3- (3'-Chlorophenyl) prop-1-yl A.2888 nC ₃ H ₇ 3- (4'-Chlorphenyl) prop-1-yl A.2889 nC ₃ H ₇ 3- (2'-Cyanophenyl) prop-1-yl A.2890 nC ₃ H ₇ 3- (3'-Cyanophenyl) prop-1-yl A.2891 nC ₃ H ₇ 3- (4'-cyanophenyl) prop-1-yl A.2892 nC ₃ H ₇ 3- (2-Trifluormethylphenyl) prop-1-yl A.2893 nC ₃ H ₇ 4-Phenylbut-1-yl A.2894 nC ₃ H ₇ 4- (4'-Chlorphenyl) but-1-yl A.2895 nC ₃ H ₇ 5- (4'-Chlorphenyl) hex-1-yl A.2896 nC ₃ H ₇ 2-pyridylmethyl A.2897 nC ₃ H ₇ 1-Pyridylmethyl

Nr. R ² R ⁴ A.2898 nC ₃ H ₇ 4-pyridylmethyl A.2899 nC ₃ H ₇ 4-Chloropyridin-2-ylmethyl A.2900 nC ₃ H ₇ 5-Chloro-pyridin-2-ylmethyl A.2901 nC ₃ H ₇ 6-Chloropyridin-2-ylmethyl | A.2902 nC ₃ H ₇ 5-Chloropyridin-3-ylmethyl j A.2903 nC ₃ H ₇ 6-Chloropyridin-3-ylmethyl j A.2904 nC ₃ H ₇ 2-Chloropyridin-4-ylmethyl A.2905 nC ₃ H ₇ 2-pyrimidinylmethyl A.2906 nC ₃ H ₇ 4-Chloropyrimidin-2-ylmethyl A.2907 nC ₃ H ₇ 5-Chloropyrimidin-2-ylmethyl A.2908 nC ₃ H ₇ 2-Chloropyrimidin-4-ylmethyl j A.2909 nC ₃ H ₇ 6-Chloropyrimidin-4-ylmethyl; A.2910 nC ₃ H ₇ 2-Chloropyrimidin-5-ylmethyl j A.2911 nC ₃ H ₇ 4-Pyridazinylmethyl A.2912 nC ₃ H ₇ 2-Pyrazinylmethyl A.2913 nC ₃ H ₇ 5-Chloropyrazin-2-ylmethyl A.2914 nC ₃ H ₇ 6-Chloropyrazin-2-ylmethyl A.2915 nC ₃ H ₇ 3-Pyridazinylmethyl ί A.2916 nC ₃ H ₇ 6-Chloropyridazin-3-ylmethyl 1 JA.2917 nC ₃ H ₇ 1,3,5-Triazinylmethyl! (ä.2918 nC ₃ H ₇ 2-Furylmethyl ’ A.2919 nC ₃ H ₇ 3-Furylmethyl! A.2920 nC ₃ H ₇ 4-Bromofur-2-ylmethyl j A.2921 nC ₃ H ₇ 5-Chlorofuran-2-ylmethyl A.2922 nC ₃ H ₇ 2-Thienylmethyl; A.2923 nC ₃ H ₇ thienylmethyl ( A.2924 nC ₃ H ₇ 5-methyl-thien-3-ylmethyl A.2925 nC ₃ H ₇ 5-Chlorothien-2-ylmethyl A.2926 nC ₃ H ₇ 2-Chlorothien-4-ylmethyl A.2927 nC ₃ H ₇ 2-Pyrroles methyl A.2928 nC ₃ H ₇ 3-pyrrolylmethyl A.2929 nC ₃ H ₇ 2-Oxazolylmethyl j A.2930 nC ₃ H ₇ 4-Methyl-oxazol-2-ylmethyl A.2931 nC ₃ H ₇ 5-Methyl-oxazol-2-ylmethyl A.2932 nC ₃ H ₇ 4-Chlorooxazol-2-ylmethyl; A.2933 nC ₃ H ₇ 5-Chlorooxazol-2-ylmethyl A.2934 n — C ₃ H ₇ 4-Oxazolylmethyl A.2935 iC ₃ H ₇ 2-Methyl-oxazol-4-ylmethyl A.2936 iC ₃ H ₇ 5-Methyl-oxazol-4-ylmethyl

Nr. R ² R ⁴ A.2937 nC ₃ H ₇ 2-chlorooxazole-4-ylmethyl A.2938 nC ₃ H ₇ 5-chlorooxazole-4-ylmethyl A.2939 nC ₃ H ₇ 5-oxazolylmethyl A.2940 nC ₃ H ₇ 2-Methyl-oxazol-5-ylmethyl A.2941 nC ₃ H ₇ 4-Methyl-oxazol-5-ylmethyl A.2942 nC ₃ H ₇ 2-chlorooxazole-5-ylmethyl A.2943 nC ₃ H ₇ 4-Chlorooxazol-5-ylmethyl A.2944 nC ₃ H ₇ 2-thiazolylmethyl A.2945 nC ₃ H ₇ 4-Methyl-thiazol-2-ylmethyl A.2946 n — C ₃ H ₇ 5-Methyl-thiazol-2-ylmethyl A.2947 nC ₃ H ₇ 4-Chloro-thiazol-2-ylmethyl A.2948 nC ₃ H ₇ 5-Chlorothiazol-2-ylmethyl A.2949 nC ₃ H ₇ 4-thiazolylmethyl A.2950 nC ₃ H ₇ 2-Methyl-thiazol-4-ylmethyl A.2951 nC ₃ H ₇ 5-Methylthiazol-4-ylmethyl A.2952 nC ₃ H ₇ 2-Chloro-thiazol-4-ylmethyl A.2953 nC ₃ H ₇ 5-Chloro-thiazol-4-ylmethyl A.2954 nC ₃ H ₇ 5thiazolylmethyl A.2955 nC ₃ H ₇ 2-Methylthiazol-5-ylmethyl A.2956 nC ₃ H ₇ 4-Methylthiazol-5-ylmethyl A.2957 nC ₃ H ₇ 2-Chlorothiazol-5-ylmethyl A.2958 nC ₃ H ₇ 4-Chloro-thiazol-5-ylmethyl A.2959 nC ₃ H ₇ 3-Isoxazolylmethyl A.2960 nC ₃ H ₇ 4-Methylisoxazol-3-ylmethyl A.2961 nC ₃ H ₇ 5-Methylisoxazol-3-ylmethyl A.2962 nC ₃ H ₇ 4-Chloroisoxazol-3-ylmethyl A.2963 nC ₃ H ₇ 5-Chloroisoxazol-3-ylmethyl A.2964 nC ₃ H ₇ 4-Isoxazolylmethyl A.2965 nC ₃ H ₇ 3-Methyl-isoxazol-4-ylmethyl A.2966 nC ₃ H ₇ 5-Methylisoxazol-4-ylmethyl A.2967 nC ₃ H ₇ 3-Chloroisoxazol-4-ylmethyl A.2968 nC ₃ H ₇ 5-Chloroisoxazol-4-ylmethyl A.2969 nC ₃ H ₇ 5 - Isoxazolylmethyl A.2970 nC ₃ H ₇ 3-Methyl-isoxazol-5-ylmethyl A.2971 nC ₃ H ₇ 4-Methylisoxazol-5-ylmethyl A.2972 ac ₃ H ₇ 3-Chloroisoxazol-5-ylmethyl A.2973 i ~ C ₃ H ₇ 1-Chloroisoxazol-5-ylmethyl A.2974 iC ₃ H ₇ i-Isothiazolylmethyl A.2975 l ic ₃ h ₇ 1-Methylisothiazol-3-ylmethyl

22 ^ (^

Nr. R ² R ⁴ A.2976 nC ₃ H ₇ 5-Methylisothiazol-3-ylmethyl A.2977 nC ₃ H ₇ 4-Chloroisothiazol-3-ylmethyl A.2978 nC ₃ H ₇ 5-Chlorisothiazol-3-ylmethyl A.2979 nC ₃ H ₇ 4-Isothiazolylmethyl A.2980 nC ₃ H ₇ 3-Methylthio and 1,4-methylmethyl A.2981 nC ₃ H ₇ 5-Methylisothiazol-4-ylmethyl A.2982 nC ₃ H ₇ 3-Chlorisothiazol-4-ylmethyl A.2983 nC ₃ H ₇ 5-Chlorisothiazol-4-ylmethyl A.2984 nC ₃ H ₇ 5 - Isothiazolylmethyl A.2985 nC ₃ H ₇ 3-Methylisothiazol-5-ylmethyl A.2986 nC ₃ H ₇ 4-methylisothiazol-5-ylmethyl A.2987 nC ₃ H ₇ 3-Chloroisothiazol-5-ylmethyl A.2988 nC ₃ H ₇ 4-Chloroisothiazol-5-ylmethyl A.2989 nC ₃ H ₇ 4-Imidazolylmethyl A.2990 nC ₃ H ₇ 1-Phenylpyrazol-3-ylmethyl A.2991 nC ₃ H ₇ 1-Methylimidazol-4-ylmethyl A.2992 nC ₃ H ₇ 1-Phenyl-1,2,4-triazol-3-ylmethyl A.2993 nC ₃ H ₇ 1,2,4-oxadiazol-3-ylmethyl A.2994 nC ₃ H ₇ 5-Chloro-1,2,4-oxadiazol-3-ylmethyl A.2995 nC ₃ H ₇ 5-Methyl-1,2,4-oxadiazol-3-ylmethyl A.2996 nC ₃ H ₇ 5-Trifluoromethyl-1,2,4-oxadiazol-3-ylmethyl A.2997 nC ₃ H ₇ 1,3,4-Oxadiazol-2-ylmethyl A.2998 nC ₃ H ₇ 5-Chloro-1,3,4-oxadiazol-2-ylmethyl A.2999 nC ₃ H ₇ 5-Methyl-1,3,4-oxadiazol-2-ylmethyl A.3000 nC ₃ H ₇ 5-methoxy-1,3,4-oxadiazol-2-ylmethyl A.3001 nC ₃ H ₇ 1,2,4-thiadiazol-3-ylmethyl A.3002 nC ₃ H ₇ 5-Chloro-1,2,4-thiadiazol-3-ylmethyl A.3003 nC ₃ H ₇ 5-Methyl-1,2,4-thiadiazol-3-ylmethyl A.3004 nC ₃ H ₇ 1,3,4-Thiadiazol-2-ylmethyl A.3005 nC ₃ H ₇ 5-chloro-1,3,4-thiadiazol-2-ylmethyl A.3006 nC ₃ H ₇ 5-methyl-1,3,4-thiadiazol-2-ylmethyl A.3007 nC ₃ H ₇ 5-Cyano-1,3,4-thiadiazol-2-ylmethyl A.3008 nC ₃ H ₇ 2- (2'-Pyridinyloxy) eth-l-yl A.3009 nC ₃ H ₇ 2- (3'-Pyridinyloxy) eth-1-yl A.3010 nC ₃ H ₇ 2- (4'-Pyridinyloxy) eth-1-yl A.3011 nC ₃ H ₇ 2- (2'-pyrimidinyloxy) eth-1-yl A.3012 nc ₃ H ₇ 2- (4'-Pyrimidinyloxy) eth-1-yl A.3013 nC ₃ H ₇ : 2 '- (5'-Pyrimidinyloxy) eth-1-yl A.3014 _{7 -} c ₃ h ₇ : ! - (2'-Pyrazinyloxy) eth-1-yl

-//from-

Nr. R ² R ⁴ A.3015 nC ₃ H ₇ 2- (2'-pyridazinyloxy) eth-1-yl A.3016 nC ₃ H ₇ 2- (3'-Pyridazinyloxy) eth-1-yl A.3017 nC ₃ H ₇ 2- (1 ', 3', 5'-Triazinyloxy) eth-1-yl A.3018 nC ₃ H ₇ 2- (5'-methylisoxazole-3'-yloxy) eth-1-yl A.3019 nC ₃ H ₇ 2- (5 ' Chlorisoxazol-3'-yloxy) eth-l-yl A.3020 nC ₃ H ₇ 2- (2'-Methoxythiazol-4'-yloxy) eth-1-yl A.3021 nC ₃ H ₇ 2- (4'-chlorooxazole-2-yloxy) eth-l-yl A.3022 nC ₃ H ₇ 2- (1'-Phenyl-1'H-1 ', 2', 4'-triazol-3'-yloxy) eth-1-yl A.3023 nC ₃ H ₇ 2- (1'-Phenylpyrazol-3'-yloxy) eth-1-yl A.3024 nC ₃ H ₇ c ₆ h ₅ A.3025 nC ₃ H ₇ 2-Cl-C ₆ H ₄ A.3026 nC ₃ H ₇ 3-Cl-C ₆ H ₄ A.3027 nC ₃ H ₇ 4-Cl-C ₆ H ₄ A.3028 nC ₃ H ₇ 2,3-Cl ₂ -C ₆ H ₃ A.3029 nC ₃ H ₇ 2,4-Cl ₂ -C ₆ H ₃ A.3030 nC ₃ H ₇ 2,5-Cl ₂ -C ₆ H ₃ A.3031 nC ₃ H ₇ 3,4-Cl ₂ -C ₆ H ₃ A.3032 nC ₃ H ₇ 3,5-Cl ₂ -C ₆ H ₃ A.3033 nC ₃ H ₇ 4-CN-C ₆ H ₄ A.3034 nC ₃ H ₇ 2-NO ₂ -C ₆ H ₄ A.3035 nC ₃ H ₇ 3-NO ₂ -C ₆ H ₄ A.3036 nC ₃ H ₇ 4-NO ₂ -C ₆ H ₄ A.3037 nC ₃ H ₇ 2,4- (NO ₂ ) ₂ -C ₆ H ₃ A.3038 nC ₃ H ₇ 2-CH ₃ -C ₆ H ₄ A.3039 nC ₃ H ₇ 3-CH ₃ -C ₆ H ₄ A.3040 nC ₃ H ₇ 4-CH ₃ -C ₆ H ₄ A.3041 nC ₃ H ₇ 2,3- (CH ₃ ) ₂ -C ₆ H ₃ A.3042 nC ₃ H ₇ 2,4- (CH ₃ ) ₂ -C ₆ H ₃ A.3043 nC ₃ H ₇ 2,5- (CH ₃ ) ₂ -C ₆ H ₃ A.3044 nC ₃ H ₇ 2,6- (CH ₃ ) ₂ -C ₆ H ₃ A.3045 nC ₃ H ₇ 2-C 6 H ₄ -C6fÍ5 A.3046 nC ₃ H ₇ 3-C ₆ H ₅ -C ₆ H ₄ A.3047 nC ₃ H ₇ 4-C ₆ H ₅ -C ₆ H ₄ A.3048 nC ₃ H ₇ 3-OCH ₃ -C ₆ H ₄ A.3049 nC ₃ H ₇ 1-OCH ₃ -C ₆ H ₄ A.3050 nC ₃ H ₇ 3-Acetyl-C 6 H ₄ A.3051 nC ₃ H _{7 1-Acetyl-4} CGH A.3052 ^ -c ₃ h ₇ and -Methoxycarbonyl-C 6 H ₄

Nr. R ² R ⁴ A.3053 nC ₃ H ₇ 4-C 6 H ₄ -Methoxycarbonyl A.3054 nC ₃ H ₇ 3-CF ₃ -C ₆ H ₄ A.3055 nC ₃ H ₇ 4-CF ₃ -C ₆ H ₄ A.3056 nC ₃ H ₇ 2 - Naphthyl A.3057 nC ₃ H ₇ 6-chloropyridazine-3-yl A.3058 nC ₃ H ₇ 5-Chlorpyra from in-2-y1 A.3059 nC ₃ H ₇ Quinolin-2-yl A.3060 nC ₃ H ₇ 2,5-Dimethylpyrazine-3-yl A.3061 nC ₃ H ₇ Pyrazin-2-yl A.3062 nC ₃ H ₇ 3-Chloropyrid-2-yl A.3063 nC ₃ H ₇ 6-chloropyrid-2-yl A.3064 nC ₃ H ₇ 4-Trifluoromethyl, 6-chloropyrid-2-yl A.3065 nC ₃ H ₇ 4-trifluoromethylpyrid-2-yl A.3066 nC ₃ H ₇ 6-trifluoromethylpyrid-2-yl A.3067 nC ₃ H ₇ 6-methoxypyridin-2-yl A.3068 nC ₃ H ₇ 5-Chloropyridin-2-yl A.3069 nC ₃ H ₇ Pyridin-2-yl A.3070 nC ₃ H ₇ Benzothiazol-2-yl A.3071 nC ₃ H ₇ 7-Chloro-quinolin-4-yl A.3072 nC ₃ H ₇ 3-nitro-pyridin-2-yl A.3073 nC ₃ H ₇ Pyrrole-3-yl A.3074 nC ₃ H ₇ Pyrrol-2-yl A.3075 nC ₃ H ₇ 2,6-Dioctylpyrid-4-yl A.3076 nC ₃ H ₇ 5-nitro-pyridin-2-yl A.3077 nC ₃ H ₇ Pyridin-4-yl A.3078 nC ₃ H ₇ Pyridin-3-yl A. 3079 nC ₃ H ₇ Pyrimidin-2-yl A.3080 nC ₃ H ₇ Pyrimidin-4-yl A.3081 nC ₃ H ₇ Quinazolin-4-yl A.3082 nC ₃ H ₇ 6-Chloro-pyrimidin-4-yl A.3083 nC ₃ H ₇ 6-Methoxy-pyrimidin-4-yl A.3084 nC ₃ H ₇ 2,5,6-Trichloro-4-yl A.3085 nC ₃ H ₇ 2,6-dimethyl-pyrimidin-4-yl A.3086 nC ₃ H ₇ 2-Methyl, 6-chloropyrimidin-4-yl A.3087 nC ₃ H ₇ 2-Methyl, 6-Ethoxy-pyrimidin-4-yl A.3088 nC ₃ H ₇ 4,5,6-trichloro-2-yl A.3089 nC ₃ H ₇ 4,6-Dimethoxy-pyrimidin-2-yl A.3090 i ^- C ₃ H ₇ 4,6-dimethyl-2-yl A.3091 nC ₃ H ₇ 4,6-Dichloropyrimidin-2-yl

Nr. R ² R ⁴ A.3092 nC ₃ H ₇ 4-Methyl, 6-methoxy-pyrimidin-2-yl A.3093 nC ₃ H ₇ 4-Chloro-6-methoxypyrimidin-2-yl A.3094 nC ₃ H ₇ 6-Chloroquinoxalin-2-yl A.3095 nC ₃ H ₇ 3,6-Dichloro-1,2,4-triazin-5-yl A.3096 nC ₃ H ₇ 4-Methoxy-1,3,5-triazin-2-yl; A.3097 nC ₃ H ₇ 4-Ethoxy-1,3,5-triazin-2-yl A.3098 nC ₃ H ₇ 4,6-dichloro-1,3,5-triazin-2-yl A.3099 nC ₃ H ₇ 4-Ethoxy, 6-Chloro-1,3,5-triazin-2-yl A.3100 nC ₃ H ₇ Isoxazol-3-yl A.3101 nC ₃ H ₇ Thien-2-yl A.3102 nC ₃ H ₇ Fur-2-yl A.3103 nC ₃ H ₇ Thiatriazole-5-yl A.3104 nC ₃ H ₇ (E) -l-chloropropene-3-yl A.3105 nC ₃ H ₇ (E) -4- (4'-Chlorphenyl) but-2-en-1-yl A.3106 nC ₃ H ₇ Propyn-3-yl A.3107 nC ₃ H ₇ Methylcarbonyl A.3108 n-C ₃ H ₇ Ethyl carbones 1 A.3109 nC ₃ H ₇ n-Propy lcarbones 1 A.3110 nC ₃ H ₇ i - Propylcarbones 1 A.3111 nC ₃ H ₇ n-Butylcarbonyl A.3112 nC ₃ H ₇ p-Butylcarbonyl A.3113 nC ₃ H ₇ i-Butylcarbonyl A.3114 nC ₃ H ₇ t-Butylcarbonyl A.3115 nC ₃ H ₇ n Pentylcarbonyl A.3116 nC ₃ H ₇ i-Pentylcarbonyl A.3117 nC ₃ H ₇ neo-Pentylcarbonyl A.3118 nC ₃ H ₇ n Hexylcarbonyl A. 3119 nC ₃ H ₇ n Octylcarbony1 A.3120 nC ₃ H ₇ 1-Propenylcarbonyl A. 3121 nC ₃ H ₇ 2-Penten-1-yl-carbonyl A.3122 nC ₃ H ₇ 2,5-heptadiene-yl-carbonyl A. 3123 nC ₃ H ₇ benzoyl A.3124 nC ₃ H ₇ 2-chlorobenzoyl A.3125 nC ₃ H ₇ 3-chlorobenzoyl A. 3126 nC ₃ H ₇ -Chlorbenzoyl A.3127 nC ₃ H ₇ 2 - Cyanobenzoyl A.3128 nC ₃ H ₇ -Cyanobenzoyl A.3129 nC ₃ H ₇ -Cyanobenzoyl A.3130 nC ₃ H ₇ t methoxybenzoyl

- 2W-

Nr. R ² R ⁴ A.3131 nC ₃ H ₇ 2 -Pyridylcarbonyl A.3132 nC ₃ H ₇ 3 -Pyridylcarbonyl A.3133 nC ₃ H ₇ 4-Pyridylcarbonyl A.3134 nC ₃ H ₇ 2 -Pyrimidinylcarbonyl A.3135 nC ₃ H ₇ 2-Oxazolylcarbonyl A.3136 nC ₃ H ₇ 4-Methyl-isoxazol-5-ylcarbonyl A.3137 nC ₃ H ₇ methylsulfonyl A.3138 nC ₃ H ₇ ethylsulfonyl A.3139 nC ₃ H ₇ n-propylsulfonyl A.3140 nC ₃ H ₇ i-propylsulfonyl A.3141 nC ₃ H ₇ n-butylsulfonyl A.3142 nC ₃ H ₇ t-butylsulfonyl A.3143 nC ₃ H ₇ n-pentylsulfonyl A.3144 nC ₃ H ₇ neo-pentylsulfonyl A.3145 nC ₃ H ₇ n-hexylsulfonyl A.3146 nC ₃ H ₇ n-Oc tylsu1f onyl A.3147 nC ₃ H ₇ phenylsulfonyl A.3148 nC ₃ H ₇ 2-Chlorphenylsulfonyl A.3149 nC ₃ H ₇ 3-Chlorphenylsulfonyl A.3150 nC ₃ H ₇ 4-Chlorophenylsulfonyl A.3151 nC ₃ H ₇ 2-Cyanophenylsulfonyl A.3152 nC ₃ H ₇ 3-Cyanophenylsulfonyl A.3153 nC ₃ H ₇ 4 -Cyanophenylsulfonyl A.3154 nC ₃ H ₇ 2-Pyridylsulfonyl A.3155 nC ₃ H ₇ 3-Pyridylsulfonyl A.3156 nC ₃ H ₇ 4-Pyridylsulfonyl A.3157 nC ₃ H ₇ 2 -Pyrimidinylsulfonyl A.3158 nC ₃ H ₇ 4-Oxazolylsulfonyl A.3159 nC ₃ H ₇ 5-Chlorothiazol-2-ylsulfonyl j A.3160 nC ₃ H ₇ 2 -tC ₄ H ₉ -C ₆ H ₄ -CH ₂ · A.3161 nC ₃ H ₇ 3-C ₄ H ₉ -C ₆ H ₄ -CH ₂ ; A.3162 nC ₃ H ₇ 4-C ₄ H ₉ -C ₆ H ₄ -CH ₂ j A.3163 nC ₃ H ₇ 2- (4'-Chlorothiazol-2'-yloxy) eth-1-yl; A, 3164 nC ₃ H ₇ 2- (1'-Methylpyrazol-4'-yloxy) eth-1-yl ¹ A.3165 n. ^- C ₃ H ₇ 4-Br-C ₆ H _4; A.3166 nC ₃ H ₇ 3,5- (CH ₃ ) ₂ -C ₆ H ₃ A.3167 ₇ —c ₃ h ₇ 4-C ₂ H ₅ -C ₆ H ₄ A.3168 iC ₃ H ₇ 3-Dimethylaminocarbonyl-C 8 H ₄ A.3169 iC ₃ H ₇ 4-Dimethylaminocarbonyl -C ₆ H ₄

- Ζ5Ί-

Nr. R ² R ⁴ A.3170 nC ₃ H ₇ 2-Hydroxyprop-1-yl A.3171 nC ₃ H ₇ 6-Hydroxy-2-methyl-pyrimidin-4-ylmethyl A.3172 nC ₃ H ₇ [6-OH, 2-CH (CH ₃ ) 2 -pyrimidin-4-yl] -CH 2 A.3173 nC ₃ H ₇ [6-OH, 2-CH (CH ₂ ) ₂ -pyrimidin-4-yl] -CH ₂ A.3174 nC ₃ H ₇ 5- (2'-Furan) -pent-1-yl A.3175 nC ₃ H ₇ 5- (2'-N-Methyl-pyrrole) -pent-1-yl A.3176 nC ₃ H ₇ [2- (4-Cl-C ₆ H ₄₎ -oxazole-4-yl] _-CH2 A.3177 nC ₃ H ₇ 3 -CF ₃ -pyridin-2-yl A.3178 nC ₃ H ₇ 5 -CF _3- pyridin-2-yl A.3179 nC ₃ H ₇ 6- (2'-Thienyl) hex-yl A.3180 nC ₃ H ₇ (E) -3-chloro-but-2-en-1-yl A.3181 nC ₃ H ₇ (Z) -3-chloro-but-2-en-l-yl A.3182 nC ₃ H ₇ (E) -2-bromo-but-2-en-l-yl A.3183 nC ₃ H ₇ (Z) -2-bromo-but-2-en-l-yl A.3184 nC ₃ H ₇ (E) -l-chloro-prop-l-en-3-yl A.3185 nC ₃ H ₇ (Z) -l-chloro-prop-l-en-3-yl A.3186 nC ₃ H ₇ But-en-3-yl A.3187 nC ₃ H ₇ CH ₂ CH ₂ Br A.3188 nC ₃ H ₇ CH ₂ CH ₂ CH ₂ Br A.3189 nC ₃ H ₇ CH ₂ CH ₂ CH ₂ CH ₂ Br A.3190 nC ₃ H ₇ Methylprop-2-yl A.3191 nC ₃ H ₇ 2-Ethoxyprop-1-yl A.3192 nC ₃ H ₇ 2-I sopropoxypropyl 1 A.3193 nC ₃ H ₇ But-yn-3-yl A.3194 nC ₃ H ₇ But-in-4-yl A.3195 nC ₃ H ₇ But-2-yn-4-yl A.3196 nC ₃ H ₇ Pent-lin-4-yl A.3197 nC ₃ phi ₇ Pent-2-yn-4-yl A.3198 nC ₃ H ₇ Pent-yn-5-yl A.3199 nC ₃ H ₇ Pent-2-yn-5-yl A.3200 nC ₃ H ₇ E-2-chloro-but-2-en-l-yl A.3201 nC ₃ H ₇ Z, 2-chloro-but-2-en-yl A.3202 nC ₃ H ₇ Z-l-chloro-prop-l-en-3-yl A.3203 nC ₃ H ₇ 2-Methylpiper-1-en-3-yl A.3204 nC ₃ H ₇ 2-chloro-prop-l-en-3-yl A.3205 nC ₃ H ₇ 2-bromoprop-l-en-3-yl A.3206 aC ₃ H ₇ 3UT-en-2-yl A.3207 iC ₃ H ₇ I 3UT-en-3-yl A.3208 iC ₃ H ₇ L-Iodprop-yn-3-yl

'čýľ -

Nr. R ² R ⁴ A.3209 nC ₃ H ₇ E-3-bromo-but-2-en-l-yl A.3210 nC ₃ H ₇ Z-3-bromo-but-2-en-l-yl A.3211 nC ₄ Hg H A.3212 nC ₄ Hg ch ₃ A.3213 nC ₄ Hg C2H5 A.3214 nC ₄ Hg nC ₃ H ₇ A.3215 nC ₄ H ₉ iC ₃ H ₇ A.3216 n ~ C ₄ Hg cyclopropyl A.3217 nC ₄ Hg nC ₄ Hg A.3218 nC ₄ Hg SC ₄ Hg A.3219 nC ₄ Hg 1-C ₄ Hg A.3220 nC ₄ Hg t ₄ C ₄ Hg A.3221 nC ₄ Hg CH ₂ CH ₂ Cl A.3222 nC ₄ Hg ch ₂ ch ₂ ch ₂ ci A.3223 nC ₄ Hg CH ₂ CH ₂ Br A.3224 nC ₄ Hg CH ₂ CH ₂ CH ₂ Br A.3225 nC ₄ H9 ch ₂ ch ₂ cn A.3226 nC ₄ Hg ch ₂ ch ₂ ch ₂ cn A.3227 nC ₄ Hg cyclopropylmethyl A.3228 nC ₄ H9 2-Cyclopropyleth-1-yl A.3229 nC ₄ H9 2-methoxyethyl-1-yl A.3230 nC ₄ H9 2-ethoxyethanol-1-yl A.3231 nC ₄ H ₉ 2-Isopropoxyeth-yl A.3232 nC ₄ Hg 3-methoxypropyl-1-yl A.3233 nC ₄ Hg 3-ethoxypropyl-1-yl A.3234 nC ₄ Hg 3-isopropoxypropanoic-1-yl A.3235 n.-C ₄ Hg 4methoxybut-1-yl A.3236 nC ₄ H ₉ 4-Isopropoxybut-1-yl A.3237 nC ₄ Hg Propen-3-yl A.3238 nC ₄ H ₉ But-2-en-1-yl A.3239 nC ₄ 19 2-methylprop-1-y1 A.3240 nC ₄ Hg 2-ethoxypropyl-1-yl A.3241 nC ₄ H ₉ 2-sopropoxyp rop-1-yl A.3242 nC ₄ Hg But-in-3-yl A.3243 nC ₄ H ₉ But-in-4-yl A.3244 nC ₄ H ₉ 3UT-2-yn-4-yl A.3245 1-C ₄ Hg Pent-in-4-yl A.3246 IC ₄ Hg ? Ent-2-yn-4-yl A.3247 1-C4H9 ? Ent-l-yn-5-yl

-ζπ-

Nr. R ² R ⁴ A.3248 II-C4H9 Pent-2-yn-5-yl A.3249 II-C4H9 E-2-chloro-but-2-en-l-yl A.3250 nC ₄ Hg Z-2-chloro-but-2-en-l-yl A.3251 nC ₄ Hg E-l-chloro-prop-l-en-3-yl A.3252 nC ₄ H9 2-methyl-prop-l-en-3-yl A.3253 nC ₄ H ₉ 2-chloro-prop-l-en-3-yl A.3254 nC ₄ Hg 2-bromoprop-l-en-3-yl A.3255 n C ₄ H ₉ But-2-en-l-yl A.3256 nC ₄ H ₉ But-3-en-l-yl A.3257 nC ₄ H ₉ l-Iodprop-l-yn-3-yl A.3258 nC ₄ H ₉ propargyl A.3259 i-C ₄ Hg H A.3260 iC ₄ H ₉ ch ₃ A.3261 n-C ₄ H ₉ C ₂ H ₅ A.3262 n-C ₄ H ₉ nC ₃ H ₇ A.3263 iC ₄ H ₉ iC ₃ H ₇ A.3264 t-c ₄ h ₉ cyclopropyl A.3265 Í ~ C ₄ H ₉ nC ₄ Hg A.3266 t-c ₄ h ₉ S * C ₄ H 9 A.3267 n-C ₄ H ₉ iC ₄ H ₉ A.3268 n-C ₄ H ₉ tC ₄ H ₉ A.3269 n-C ₄ H ₉ CH ₂ CH ₂ Cl A.3270 n-C ₄ H ₉ ch ₂ ch ₂ ch ₂ ci A.3271 n-C ₄ H ₉ CH ₂ CH ₂ Br A.3272 n-C ₄ H ₉ CH ₂ CH ₂ CH ₂ Br A.3273 : .- C ₄ H ₉ CH ₂ CH ₂ CN A.3274 n-C ₄ H ₉ ch ₂ ch ₂ ch ₂ cn A.3275 n-C ₄ H ₉ cyclopropylmethyl A.3276 n-C ₄ H ₉ 2-Cyclopropylth-1-yl A.3277 n-C ₄ H ₉ 2-Me thoxye th-1-yl A.3278 n-C ₄ H ₉ 2-E thoxy-th-1-yl A.3279 iC ₄ H ₉ 2-Isopropoxy-eth-1-yl A.3280 ic ₄ h ₉ 3-methoxypropyl-1-yl A.3281 n-C ₄ H ₉ 3-ethoxypropyl-yl A.3282 n-C ₄ H ₉ 3-1sopropoxyprop-1-yl A.3283 n-C ₄ H ₉ 4-methoxy-but yl A.3284 iC ₄ H ₉ 1-Isopropoxybut-1-yl A.3285 iC ₄ H ₉ ? Ropen-3-yl A.3286 iC ₄ H ₉ 1 But-2-en-1-yl

- m-

Nr. R ² R ⁴ A.3287 I-C4H9 2-methylprop-1-y1 A.3288 I-C4H9 2-Ethoxyprop-1-yl A.3289 I-C4H9 2-isopropoxypropanoic-yl A.3290 iC ₄ H ₉ But-in-3-yl A.3291 I-C4H9 But-in-4-yl A.3292 I-C4H9 But-2-yn-4-yl A.3293 I-C4H9 Pent-in-4-yl A.3294 I-C4H9 Pent-2-yn-4-yl A.3295 I-C4H9 Pent-in-5-yl A.3296 I-C4H9 Pent-2-yn-5-yl A.3297 I-C4H9 E-2-chloro-but-2-en-l-yl A.3298 I-C4H9 Z-2-chloro-but-2-en-l-yl A.3299 I-C4H9 E-l-chloro-prop-l-en-3-yl A.3300 i ^- C4H9 2-methyl-prop-l-en-3-yl A.3301 t-C4H9 2-chloro-prop-l-en-3-yl A.3302 I-C4H9 2-bromoprop-1-en-3-y1 A.3303 I-C4H9 But-2-en-l-yl A.3304 I-C4H9 But-3-en-l-yl A.3305 I-C4H9 l-Iodprop-l-yn-3-yl A.3306 I-C4H9 propargyl A.3307 n CsHu H A.3308 n CsHu ch ₃ A.3309 n CsHu C ₂ H ₅ A.3310 n CSHN nC ₃ H ₇ A.3311 n CsHu I-C3H7 A.3312 n CSHN cyclopropyl A.3313 n CSHN n-C4H9 A.3314 n CSHN S-C4H9 A.3315 n CsHu -C4H9 A.3316 n CSHN tC ₄ H ₉ A.3317 n CSHN CH ₂ CH ₂ Cl A.3318 nc ₅ Hn ch ₂ ch ₂ ch ₂ ci A.3319 n CSHN CH ₂ CH ₂ Br A.3320 n CSHN CH ₂ CH ₂ CH ₂ Br A.3321 n ^- C 5 H 1 X CH ₂ CH ₂ CN A.3322 n CsHu CH ₂ CH ₂ CH ₂ CN A.3323 Π-ϋςΗχχ Cyclopropylme thyl A.3324 I-C5HXX 2-Cyclopropyleth-yl A.3325 I-C5H1X 2-methoxyethyl-1-yl

-Ζ5Τ-

Nr. R ² R ⁴ A. 3326 n CSHN 2-ethoxyethanol-1-yl A.3327 n CSHN 2-1-propropoxy-th-1-yl A.3328 11-C5H11 3-methoxypropyl-1-yl A.3329 n CSHN 3-ethoxypropyl-1-yl A.3330 n CSHN 3-lsopropoxyprop-1-yl A.3331 n CSHN 4methoxybut-1-yl A.3332 n CSHN 4-1sopropoxybut-1-yl A.3333 n CSHN Propen-3-yl A.3334 n CSHN But-2-en-yl A.3335 n CSHN 2-Methoxyprop-yl A.3336 n CSHN 2-E-thoxyprop-1-yl A.3337 n CSHN 2-1sopropoxyprop-1-y1 A.3338 n CSHN But-in-3-yl A.3339 11-C5H11 But-in-4-yl A.3340 nC _with H _u But-2-yn-4-yl A.3341 n CSHN Pent-yn-4-yl A.3342 n CSHN Pent-2-yn-4-yl A.3343 n CSHN Pent-yn-5-yl A.3344 nC ₅ Hn Pent-2-yn-5-yl A.3345 n CSHN E-2-chloro-but-2-en-yl A.3346 nC ₅ Hn Z-2-chloro-but-2-en-l-yl A.3347 nC ₅ Hu E-l-chloro-prop-l-en-3-yl A.3348 nC ₅ Hn 2-methyl-prop-3-yl A.3349 n CSHN 2-chloro-prop-l-en-3-yl A.3350 nC ₅ Hu 2-bromoprop-l-en-3-yl A.3351 n CSHN But-2-en-yl A.3352 n CSHN But-3-en-l-yl A.3353 n CSHN 1 'Iprprop-1'-in-3-y 1 A.3354 n CSHN propargyl A.3355 Cyclo-C ₅ H ₉ H A.3356 Cyclo-CsHg ch ₃ A.3357 Cyclo-CsH ₉ c ₂ h ₅ A.3358 Cyclo-CsHg nC ₃ H ₇ A.3359 Cyclo-CsHg i C ₃ H ₇ A.3360 3Cyclo-CsH ₉ cyclopropyl A.3361 ľyclo-CsHg 1 - c ₄ h ₉ A.3362 lyclo-CsHg 3-C ₄ H ₉ A.3363 ľyclo-C5H3 L - C ₄ H ₉ A.3364 ( ľyclo-CsHg with -C ₄ H ₉

'2-56-

Nr. R ² R ⁴ A.3365 Cyclo-CsHg CH ₂ CH ₂ Cl A.3366 Cyclo-CsHg ch ₂ ch ₂ ch ₂ ci A.3367 Cyclo-CsHg CH ₂ CH ₂ Br A.3368 CYEL-CsHg CH ₂ CH ₂ CH ₂ Br A.3369 Cyclo-CsHg CH ₂ CH ₂ CN A.3370 Cyclo-C ₅ Hg ch ₂ ch ₂ ch ₂ cn A.3371 Cyclo-C ₅ Hg cyclopropylmethyl A.3372 Cyclo-CsHg 2-Cyclopropyleth-1-yl A.3373 Cyclo-CsHg 2-methoxyethyl-1-yl A.3374 Cyclo-CsHg 2-ethoxyethanol-yl A.3375 Cyclo-CsHg 2-Isopropoxy-eth-1-yl A.3376 Cyclo-CsHg 3-Methoxyprop-1-yl A.3377 Cyclo-CsHg 3-ethoxypropyl-1-yl A.3378 Cyclo-CsHg 3-Isopropoxyprop-1-yl A.3379 Cyclo-CsHg 4methoxybut-1-yl A.3380 Cyclo-C ₅ H ₉ 4-Isopropoxy-but-1-yl A.3381 Cyclo-CsHg Propen-3-yl A.3382 Cyclo-CsHg But-2-en-l-yl A.3383 Cyclo-CsHg Methylprop-2-yl A.3384 Cyclo-CsHg 2-Ethoxyprop-1-yl A.3385 Cyclo-CsHg 2-1 sopropoxyp rop-1-yl A.3386 Cyclo-CsHg But-in-3-yl A.3387 Cyclo-CsHg But-in-4-yl A.3388 Cyclo-CsHg But-2-yn-4-yl A.3389 Cyclo-CsHg Pent-in-4-yl A.3390 Cyclo-CsHg Pent-2-yn-4-yl A.3391 Cyclo-CsHg Pent-in-5-yl A.3392 Cyclo-CsHg Pent-2-yn-5-yl A.3393 Cyclo-CsHg E-2-chloro-but-2-en-l-yl A.3394 Cyclo-CsHg Z-2-Chlorobut-2-en-1-yl j A.3395 Cyclo-CsHg E-1-Chlorprop-1-en-3-yl; j A.3396 Cyclo-CsHg 2-Methylprop-1-en-3-yl A.3397 Cyclo-CsHg 2-Chloroprop-1-en-3-yl; A.3398 Cyclo-C5H9 2-bromoprop-l-en-3-yl A.3399 Cyclo-CsHg But-2-en-1-yl; A.3400 Cyclo-C5H9 But-3-en-1-yl A.3401 Cyclo-CsHg l-Iodprop-l-yn-3-yl A.3402 Cyclo-CsHg propargyl A.3403 1-C ₆ H ₁₃

- Z.> 7-

Nr. R ² R ⁴ A.3404 n CgHi3 ch ₃ A.3405 n-C6Hi3 C ₂ H ₅ A.3406 n-C6Hi3 nC ₃ H ₇ A.3407 n-C6Hi3 iC ₃ H ₇ A.3408 n-C6H ₁₃ cyclopropyl A.3409 n-C ₆ H 13 nC ₄ Hg A.3410 n-C6Hi3 S-C4H9 A.3411 n-C6Hi3 1-C4H9 A.3412 n-C6Hi3 tC ₄ H ₉ A.3413 n-C6Hi3 CH ₂ CH ₂ Cl A.3414 n-C6H ₁₃ ch ₂ ch ₂ ch ₂ ci A.3415 n-C ₆ H 13 CH ₂ CH ₂ Br A.3416 n-C ₆ H 13 CH ₂ CH ₂ CH ₂ Br A.3417 n-C ₆ H 13 CH ₂ CH ₂ CN A.3418 n-C ₈ H 13 ch ₂ ch ₂ ch ₂ cn A.3419 n-C ₆ H 13 Cyclopropylme thyl A.3420 n-C ₆ H 13 2-Cyclopropyleth-1-yl A.3421 n-C6Hl3 2-methoxyethyl-1-yl A.3422 n-C ₆ H 13 2-ethoxyethanol-1-yl A. 3423 n-C ₆ H 13 2-lsopropoxyeth-yl A.3424 ⁿ -C6Hx ₃ 3-methoxypropyl-1-yl A.3425 n-C ₆ H 13 3-ethoxypropyl-yl A. 3426 n-C6Hi3 3-isopropoxypropanoic-1-yl A.3427 n-C ₆ H 13 4methoxybut-1-yl A.3428 n-C ₆ H 13 4-Isopropoxy-but-1-yl A.3429 n-C6Hi3 Propen-3-yl A.3430 n-C ₆ H 13 But-2-en-l-yl A.3431 _n-3 C6Hx 2-methylprop-1-yl A.3432 n-COHN Ethoxypropyl-2-yl A.3433 n-C ₆ H 13 2-1sopropoxyprop-1-yl A.3434 n-C ₆ H 13 But-in-3-yl A.3435 n-C ₆ H 13 But-in-4-yl A.3436 n-C6Hi3 But-2-yn-4-yl A.3437 nC ₆ Hi ₃ Pent-in-4-yl A.3438 nC ₆ Hi ₃ Pent-2-yn-4-yl A.3439 n — C6H3 ₃ Pent-in-5-yl A.3440 ^ - C6H3 ₃ Pent-2-yn-5-yl A.3441 i 1 ~ C6Hi ₃ 3-2-chloro-but-2-en-l-yl A.3442 I l 'C6Hi3 2-2-chloro-but-2-en-l-yl

-2 / 2

Nr. R ² R ⁴ A.3443 nC ₆ H ₁₃ E-l-chloro-prop-l-en-3-yl A.3444 n-C ₈ H 13 2-methyl-prop-l-en-3-y1 A.3445 X 1 -C 6 H ₃ 2-chloro-prop-l-en-3-yl A.3446 n-C ₈ H 13 2-bromoprop-l-en-3-y1 A.3447 n-C6Hi3 But-2-en-l-yl A.3448 nC ₆ H ₁₃ But-3-en-l-yl A. 3449 n-C ₆ H ₃ l-lodprop-l-yn-3-yl A.3450 n-C ₈ H 13 propargyl A. 3451 Cyclo-CgHu H A.3452 Cyclo-CgHu ch ₃ A.3453 Cyclo-C ₆ Hn c ₂ h ₅ A.3454 Cyclo-C ₅ Hn nC ₃ H ₇ A.3455 Cyclo-CgHu iC ₃ H ₇ A.3456 Cyclo-CgHu cyclopropyl A.3457 Cyclo-C ₆ Hn n -C 4 H 9 A.3458 Cyclo-CgHii S-C4H9 A.3459 Cyclo-C6Hn I-C4H9 A.3460 Cyclo-CgHu tC ₄ H ₉ A.3461 Cyclo-CgHu CH ₂ CH ₂ Cl A.3462 Cyclo-CSHN CH ₂ CH ₂ CH ₂ Cl A.3463 Cyclo-C6Hn CH ₂ CH ₂ Br A.3464 Cyclo-CgHu CH ₂ CH ₂ CH ₂ Br A.3465 Cyclo-CgHu CH ₂ CH ₂ CN A.3466 Cyclo-CgHu CH ₂ CH ₂ CH ₂ CN A.3467 Cyclo-CgHu cyclopropylmethyl A.3468 Cyclo-CgHu 2-Cyclopropyleth-1-yl A.3469 Cyclo-C ₆ Hn 2-methoxyethyl-yl A.3470 Cyclo-C ₆ Hn 2-ethoxyethanol 1-y1 A.3471 Cyclo-CgHii 2-1-propropoxy-th-1-yl A.3472 Cyclo-C ₆ Hn 3-methoxypropyl-1-yl A.3473 Cyclo-CgHu 3-Ethoxyprop-1-yl A.3474 Cyclo-C ₆ Hn 3-1sopropoxyprop-1-yl A.3475 Cyclo-CgHu 4-methoxy-but yl A.3476 Cyclo-CgHu i-Isopropoxybut-yl A.3477 Cyclo-CgHu Propen-3-yl A.3478 Cyclo-CSHN 3UT-2-en-l-yl A.3479 Cyclo-CgHu Methylprop-2-yl A.3480 Cyclo-CgHu i Ϊ-E thoxyprop-1-yl A.3481 ( Cyclo-CgHu1 -Isopropoxyprop-1-yl

Nr. R ² R ⁴ A.3482 Cyclo-CgHii But-in-3-yl A.3483 Cyclo-CgHu But-in-4-yl A.3484 Cyclo-C6Hu But-2-yn-4-yl A.3485 Cyclo-C6Hn Pent-in.-4-yl A.3486 Cyclo-CgHu Pent-2-yn-4-yl A.3487 Cyclo-CgHu Pent-in-5-yl A.3488 Cyclo-CgHii Pent-2-yn-5-yl A.3489 Cyclo-Cehula E-2-chloro-but-2-en-l-yl A.3490 Cyclo-C6Hn Z-2-chloro-but-2-en-l-yl A.3491 Cyclo-CgHii E-l-chloro-prop-l-en-3-yl A.3492 Cyclo-CSHN 2-methyl-prop-l-en-3-yl A.3493 Cyclo-CgHii 2-chloro-prop-l-en-3-yl A.3494 Cyclo-CgHu 2-bromoprop-l-en-3-yl A.3495 Cyclo-CgHu But-2-en-l-yl A.3496 Cyclo-CgHu But-3-en-l-yl A.3497 Cyclo-CgHii l-Iodprop-l-yn-3-yl A.3498 Cyclo-CgHii propargyl A.3499 H H A.3500 H ch ₃ A.3501 H c ₂ h ₅ A.3502 H nC ₃ H ₇ A.3503 H iC ₃ H ₇ A.3504 H cyclopropyl A.3505 H n-C4H9 A.3506 H S-C4H9 A.3507 H -C4H9 A.3508 H t -C4H9 A.3509 H ch ₂ ch ₂ ci A.3510 H CH2CH2CH2C A.3511 H CH ₂ CH ₂ Br A.3512 H CH ₂ CH ₂ CH ₂ Br A.3513 H CH ₂ CH ₂ CN A.3514 H CH ₂ CH ₂ CH ₂ CN A.3515 H 3yclopropylmethyl A.3516 H 2-Cyclopropyleth-1-yl A.3517 and 2-methoxyethyl-1-yl A.3518 2-ethoxyethanol-1-yl A.3519 and 2-Isopropoxyeth-1-yl A.3520 i: J-methoxypropyl-1-yl

Z'6 v-

Nr. R ² R ⁴ A.3521 H 3-Ethoxyprop-1-yl A.3522 H 3-isopropoxypropanoic-yl A.3523 H 4-Methoxybut-1-yl A.3524 H 4-Isopropoxybut-1-yl A.3525 H Propen-3-yl A.3526 H But-2-en-1-yl A.3527 H 2-Methoxyprop-yl A.3528 H 2-Ethoxyprop-1-yl A.3529 H 2-yl-isopropoxypropanoic A.3530 H But-yn-3-yl A.3531 H But-in-4-yl A.3532 H But-2-yn-4-yl A.3533 H Pent-yn-4-yl A.3534 H Pent-2-yn-4-yl A.3535 H Pent-yn-5-yl A.3536 H Pent-2-yn-5-yl A.3537 H E-2-chloro-but-2-en-yl A.3538 H Z-2-chloro-but-2-en-l-yl A.3539 H E-1-chloro-prop-1-en-3-yl A.3540 H 2-methyl-prop-l-en-3-yl A.3541 H 2-chloro-prop-l-en-3-yl A.3542 H 2-bromoprop-l-en-3-yl A.3543 H But-2-en-1-yl A.3544 H But-3-en-l-yl A.3545 H l-Iodprop-l-yn-3-yl A.3546 H propargyl A.3547 cyclo-C ₄ H ₇ H A.3548 cyclo-C ₄ H ₇ ch ₃ A.3549 cyclo-C ₄ H ₇ c ₂ h _p A.3550 cyclo-C ₄ H ₇ nC ₃ H ₇ A.3551 cyclo-C ₄ H ₇ iC ₃ H ₇ A.3552 cyclo-C ₄ H ₇ cyclopropyl A.3553 cyclo-C ₄ H ₇ nC ₄ H ₉ A.3554 cyclo-C ₄ H ₇ S -C ₄ Hg A.3555 cyclo-C ₄ H ₇ iC ₄ H ₉ A.3556 cyclo-C ₄ H ₇ tC ₄ H ₉ A.3557 cyclo-C ₄ H ₇ CH ₂ CH ₂ Cl A.3558 oyclo-C ₄ H ₇ CH ₂ CH ₂ CH ₂ Cl A.3559 3Cyclo-C ₄ H ₇ CH ₂ CH ₂ Br

- 2b1-

Nr. R ² R ⁴ A.3560 cyclo-C ₄ H ₇ CH ₂ CH ₂ CH ₂ Br A.3561 cyclo-C ₄ H ₇ CH ₂ CH ₂ CN A.3562 Cyclo-C ₄ H ₇ ch ₂ ch ₂ ch ₂ cn A.3563 Cyclo-C ₄ H ₇ Cyclopropy1methyl A.3564 Cyclo-C ₄ H ₇ 2-Cycloopropyleth-1-y1 A.3565 Cyclo-C ₄ H7 2-methoxyethyl-1-yl A.3566 Cyclo-C ₄ H ₇ 2-ethoxyethanol 1-y1 A.3567 Cyclo-C ₄ H ₇ 2-1-propropoxy-th-1-yl A.3568 Cyclo-C ₄ H ₇ 3-methoxypropyl-1-yl A.3569 Cyclo-C ₄ H ₇ 3-Ethoxyprop-1-yl A.3570 Cyclo-C ₄ H ₇ 3-lsopropoxyprop-1-yl A.3571 Cyclo-C ₄ H ₇ 4methoxybut-1-yl A.3572 Cyclo-C ₄ H ₇ 4-Isopropoxybut-1-yl A.3573 Cyclo-C ₄ H ₇ Propen-3-yl A.3574 Cyclo-C ₄ H ₇ But-2-en-l-yl A.3575 Cyclo-C ₄ H ₇ 2-yl-methoxy-propyl A.3576 Cyclo-C ₄ H ₇ 2-Ethoxyprop-1-yl A.3577 Cyclo-C ₄ H ₇ 2-1sopropoxyprop-1-yl A.3578 Cyclo-C ₄ H ₇ But-in-3-yl A.3579 Cyclo-C ₄ H ₇ But-in-4-yl A.3580 CyclO'C ₄ H ₇ But-2-yn-4-yl A.3581 Cyclo-C ₄ H ₇ Pent-yn-4-yl A.3582 Cyclo-C ₄ H ₇ Pent-2-yn-4-yl A.3583 Cyclo-C ₄ H ₇ Pent-in-5-yl A.3584 Cyclo-C ₄ H ₇ Pent-2-yn-5-yl A.3585 Cyclo-C ₄ H ₇ E-2-chloro-but-2-en-l-yl A.3586 Cyclo-C ₄ H ₇ Z-2-chloro-but-2-en-l-yl A.3587 Cyclo-C ₄ H ₇ E-ľChlorprop ľen.-3-yl A.3588 Cyclo-C ₄ H ₇ 2-methyl-prop-3-yl A.3589 Cyclo-C ₄ H ₇ 2-chloro-prop-en-3-yl A.3590 Cyclo-C ₄ H ₇ 2-bromoprop-l-en-3-yl A.3591 Cyclo-C ₄ H ₇ But-2-en-yl A.3592 Cyclo-C ₄ H ₇ But-3-en-l-yl A.3593 Cyclo-C ₄ H ₇ l-Iodprop-yn-3-yl A.3594 : yclo-C ₄ H ₇ propargyl

Table B

Nr. R ³ B.l. CH ₂ CN B.2 (CH ₂ ) ₂ CN B.3 (ch ₂ ) ₃ cn B.4 (CH ₂ ) ₄ CN B.5 ch ₂ no ₂ B.6 (CH ₂ ) ₂ NO ₂ B.7 (ch ₂ ) ₂ no ₂ B.8 (CH ₂ ) ₄ NO ₂ B.9 ch ₂ oh B.10 (CH ₂ ) ₂ OH B.11 (CH ₂ ) ₃ OH B.12 (ch ₂ ) ₄ oh B.13 ch ₂ nh ₂ B.14 (CH ₂ ) ₂ NH ₂ B.15 (ch ₂ ) ₃ nh ₂ B.16 (CH ₂ ) ₄ NH ₂ B.17 ch ₂ nhch ₃ B.18 (CH ₂ ) ₂ NHCH ₃ B.19 (CH ₂ ) ₃ NHCH ₃ B.20 (ch ₂ ) ₄ nhch ₃ B.21 CH ₂ N (CH ₃ ) ₂ B.22 (CH ₂ ) ₂ N (CH ₃ ) ₂ B.23 <CH ₂ ) ₃ N (CH ₃ ) ₂ B.24 (CH ₂ ) ₄ N (CH ₃ ) ₂ B.25 ch ₂ n (ch ₂ ch ₃ ) ₂ B.26 (CH ₂ ) ₂ N (CH ₂ CH ₃ ) ₂ B.27 (CH ₂ ) ₃ N (CH ₂ CH ₃ ) 2 B.28 (CH ₂ ) ₄ N (CH ₂ CH ₃ ) ₂ B.29 ch ₂ and ₃ B.30 (CH ₂ ) ₂ OCH ₃ B.31 (ch ₂ ) ₃ OCH ₃ B.32 (CH ₂ ) ₄ OCH ₃ B.33 ch ₂ and ₂ ch ₃ B.34 (CH ₂ ) ₂ OCH ₂ CH ₃ B.35 (CH ₂ ) ₃ OCH ₂ CH ₃ B.36 (ch ₂ ) ₄ and ₂ ch ₃ B.37 ch ₂ o (CH ₂ ) ₂ ch ₃

Nr. R ³ B.38 (ch ₂ ) ₂ o (ch ₂ ) ₂ ch ₃ B.39 (CH ₂ ) ₃ O (CH ₂ ) ₂ CH ₃ B.40 (CH ₂ ) ₄ O (CH ₂ ) ₂ CH ₃ B.41 CH ₂ OCH (CH ₃ ) ₂ B.42 (CH ₂ ) ₂ OCH (CH ₃ ) ₂ B.43 (CH ₂ ) ₃ OCH (CH ₃ ) ₂ B.44 (CH ₂ ) ₄ OCH (CH ₃ ) ₂ B.45 CH ₂ OC (CH ₃ ) ₃ B.46 (CH ₂ ) ₂ C (CH ₃ ) ₃ B.47 (CH ₂ ) ₃ OC (CH ₃ ) ₃ B.48 (CH ₂ ) ₄ OC (CH ₃ ) ₃ B.49 ch ₂ ocf ₃ B.50 (CH ₂ ) ₂ OCF ₃ B.51 (CH ₂ ) ₃ OCF ₃ B.52 (CH ₂ ) ₄ OCF ₃ B.53 CH2SCH3 B.54 (CH ₂ ) ₂ SCH ₃ B.55 <ch ₂ ) ₃ sch ₃ B.56 (CH ₂ ) ₄ SCH ₃ B.57 ch ₂ statues ₃ B.58 (CH ₂ ) ₂ SOCH ₃ B.59 (CH ₂ ) ₃ SOCH ₃ B.60 (CH ₂ ) ₄ SOCH ₃ B.61 ch ₂ so ₂ ch ₃ B.62 (CH ₂ ) ₂ SO ₂ CH ₃ B.63 (CH ₂ ) ₃ SO ₂ CH ₃ B.64 (CH ₂ ) ₄ SO ₂ CH ₃ B.65 _CH2 -cyclopropyl B.66 (CH ₂ ) ₂ -cyclopropyl B.67 ¹ CH ₂ ) ₃ -cyclopropyl B.68 (CH ₂ ) ₄ -cyclopropyl B.69 CH ₂ -cyclopentyl B.70 (CH ₂ ) ₂ -cyclopentyl B.71 (CH ₂ ) ₃ "cyclopentyl B.72 (CH ₂ ) ₄ -cyclopentyl B.73 1 H ₂ -cyclohexyl B.74 (CH ₂ ) ₂ -cyclohexyl B.75 (CH ₂ ) ₃ -cyclohexyl B.76 (CH ₂ ) ₄ -cyclohexyl

£ 64-

Nr. R ³ B.77 chf ₂ B.78 cf ₃ B.79 ch ₂ chf ₂ B.80 ch ₂ cf ₃ B.81 chfchf ₂ B.82 ch ₂ ch ₂ f B.83 chfch ₃ B.84 chfcf ₃ B. 85 CF ₂ CF ₂ B.86 cf ₂ chfcf ₃ B.87 ch ₂ cci ₃ B.88 cf ₂ i want ₂ B.89 cf ₂ chfci B.90 CF ₂ CHFBr B.91 CH (CF ₃ ) ₂ B.92 CH (CF ₃ ) CH ₃ B.93 ch ₂ ch ₂ cf ₃ B.94 ch ₂ chfch ₃ B.95 ch ₂ cf ₂ cf ₃ B.96 CH ₂ CH ₂ CH ₂ F B.97 CH ₂ CF ₂ CF ₂ CF ₃ B.98 ch ₂ ch ₂ chfch ₃ B.99 ch ₂ ch ₂ ch ₂ ch ₂ f B.100 ch ₂ ci B.101 ch ₂ ch ₂ ci B.102 ch ₂ want ₃ B.103 ch ₂ ch ₂ ch ₂ ci B.104 ch ₂ ch ₂ want ₃ B.105 ch ₂ ch ₂ ch ₂ ch ₂ ci B.106 CH ₂ Br B.107 CH ₂ CH ₂ Br B.108 CH ₂ CHBrCH ₃ B.109 CH ₂ CH ₂ CH ₂ Br B.110 CH ₂ CH ₂ CHBrCH ₃ B.111 CH ₂ CH ₂ CH ₂ CH ₂ Br B.112 ch ₂ -c ₆ h ₅ B.113 : h ₂ -oc ₆ h ₅ B.114 : h (ch ₃ ) cn B.115 : h (ch ₃ ) ch ₂ cn

Nr. R ³ B.116 CH ₂ CH (CH ₃ ) CN B.117 CH _(CH3) CH _(CH3) CN B.118 CH (CH ₃ ) (CH ₂ ) ₂ CN B.119 ch ₂ ch (ch ₃ ) ch ₂ cn B.120 (CH ₂ ) ₂ CH (CH ₃ ) CN B.121 CH (CH ₃ ) CH (CH ₃ ) CH ₂ CN B.122 CH (CH ₃ ) CH ₂ CH (CH ₃ ) CN B.123 CH ₂ CH (CH ₃ ) CH (CH ₃ ) CN B.124 CH _(CH3) CH _(CH3) CH _(CH3) CN B.125 CH (CH ₃ ) (CH ₂ ) ₃ CN B.126 CH (CH _{3) 2} NO B.127 CH (CH ₃ ) CH ₂ NO ₂ B.128 CH ₂ CH (CH ₃ ) NO ₂ B.129 CH (CH ₃ ) CH (CH ₃ ) NO ₂ B.130 CH (CH ₃ ) (CH ₂ ) ₂ NO ₂ B.131 CH ₂ CH (CH ₃ ) CH ₂ NO ₂ B.132 (CH ₂ ) ₂ CH (CH ₃ ) NO ₂ B.133 CH (CH ₃ ) CH (CH ₃ ) CH ₂ NO ₂ B.134 CH (CH ₃ ) CH ₂ CH (CH ₃ ) NO ₂ B.135 CH ₂ CH (CH ₃ ) CH (CH ₃ ) NO ₂ B.136 CH _(CH3) CH _(CH3) CH _{(CH3) 2} no B.137 CH (CH ₃ ) (CH ₂ ) ₃ NO ₂ B.138 CH _(CH3) OH B.139 CH (CH ₃ ) CH ₂ OH B.140 CH ₂ CH (CH ₃ ) OH B.141 CH _(CH3) CH _(CH3) OH B.142 CH (CH ₃ ) (CH ₂ ) ₂ OH B.143 CH ₂ CH (CH ₃ ) CH ₂ OH B.144 (CH ₂ ) ₂ CH (CH ₃ ) OH B.145 CH (CH ₃ ) CH (CH ₃ ) CH ₂ OH B.146 CH (CH ₃ ) CH ₂ CH (CH ₃ ) OH B.147 CH ₂ CH (CH ₃ ) CH (CH ₃ ) OH B.148 CH _(CH3) CH _(CH3) CH _(CH3) OH B.149 CH (CH ₃ ) (CH ₂ ) ₃ OH B.150 CH _{(CH3) OCH3} B.151 CH (CH ₃ ) CH ₂ OCH ₃ B.152 CH ₂ CH (CH ₃ ) OCH ₃ B.153 CH _(CH3) CH _{(CH3) OCH3} B.154 CH (CH ₃ ) (CH ₂ ) ₂ OCH ₃

7.66-

1 Nr. R ³ 1 B.155 CH 2 CH (CH ₃ ) CH ₂ OCH ₃ J B.156 (CH ₂ ) ₂ CH (CH ₃ , OCH ₃₎ J B.157 CH (CH ₃ ) CH (CH ₃ ) CH ₂ OCH ₃ J B.158 CH (CH ₃ ) CH ₂ CH (CH ₃ ) OCH ₃ J B.159 CH ₂ CH (CH ₃ ) CH (CH ₃ ) OCH ₃ J B.160 CH _(CH3) CH _(CH3) CH _{(CH3) OCH3} 1 B.161 CH (CH ₃ ) (CH ₂ ) ₃ OCH ₃ 1 B.162 CH (CH ₃ ) OCH ₂ CH ₃ 1 B.163 CH (CH ₃ ) CH ₂ OCH ₂ CH ₃ J B.164 CH ₂ CH (CH ₃ ) OCH ₂ CH ₃ J B.165 CH (CH ₃ ) CH (CH ₃ ) OCH ₂ CH ₃ J B.166 CH _{(CH3) <CH2) 2 OCH2 CH3} j B.167 ch ₂ ch (ch ₃ ) ch ₂ and ₂ ch ₃ | B.168 (CH ₂ ) ₂ CH (CH ₃ ) OCH ₂ CH ₃ J B.169 CH (CH ₃ ) CH (CH ₃ ) CH ₂ OCH ₂ CH ₃ J B.170 CH (CH ₃ ) CH ₂ CH (CH ₃ ) OCH ₂ CH ₃ j B.171 CH ₂ CH (CH ₃ ) CH (CH ₃ ) OCH ₂ CH ₃ 1 B.172 CH (CH ₃ ) CH (CH ₃ ) CH (CH ₃ ) OCH ₂ CH ₃ j B.173 CH (CH ₃ ) (CH ₂ ) ₃ OCH ₂ CH ₃ 1 B.174 CH (CH ₃ ) CH ₂ O (CH ₂ ) ₂ CH ₃ j B.175 CH ₂ CH (CH ₃ ) O (CH ₂ ) ₂ CH ₃ 1 B.176 CH (CH ₃ ) CH (CH ₃ ) 0 (CH ₂ ) ₂ CH ₃ j B.177 CH (CH ₃ ) (CH ₂ ) ₂ O (CH ₂ ) ₂ CH ₃ J B.178 CH ₂ CH (CH ₃₎ CH ₂ O (CH _{2) 2} CH ₃ j B.179 (CH _{2) 2} CH _(CH3) 0 _{(CH2) 2 CH3} 1 B.180 CH (CH ₃ ) CH (CH ₃ ) CH ₂ O (CH ₂ ) ₂ ch ₃ J B.181 CH (CH ₃ ) CH ₂ CH (CH ₃ ) 0 (CH ₂ ) ₂ ch ₃ 1 B.182 _CH2 CH _(CH3) CH _(CH3) 0 _{(CH2) 2 CH3} J B.183 CH (CH ₃ ) CH (CH ₃ ) CH (CH ₃ ) 0 (CH ₂ ) ₂ CH ₃ j B.184 CH (CH ₃ ) (CH ₂ ) ₃ O (CH ₂ ) ₂ CH ₃ J B.185 CH (CH ₃₎ OCH (CH _{3) 2} j B.186 CH (CH ₃ ) CH ₂ OCH (CH ₃ ) ₂ J B.187 CH ₂ CH (CH ₃ ) OCH (CH ₃ ) ₂ J B.188 CH (CH ₃₎ CH (CH ₃₎ OCH _{<CH3) 2} J B.189 < CH (CH ₃ ) (CH ₂ ) ₂ OCH (CH ₃ ) ₂ J B.190 ( CH ₂ CH (CH ₃ ) CH ₂ OCH (CH ₃ ) 2 J B.191 (CH ₂ ) ₂ CH (CH ₃ ) OCH (CH ₃ ) 2 1 B.192 C CH (CH ₃ ) CH (CH ₃ ) CH ₂ OCH (CH ₃ ) 2 | B.193 C CH (CH ₃ ) CH ₂ CH (CH ₃ ) OCH (CH ₃ ) ₂

- 26? -

Nr. R3 B.194 CH ₂ CH (CH ₃ ) CH (CH ₃ ) OCH (CH ₃ is ₂ B.195 CH (CH ₃₎ CH (CH ₃₎ CH (CH ₃₎ OCH (CH _{3) 2} B.196 CH (CH ₃ ) (CH ₂ ) ₃ OCH (CH ₃ ) ₂ B.197 CH _(CH3) OC _{(CH3) 3} B.198 CH (CH ₃ ) CH ₂ OC (CH ₃ ) 3 B.199 CH ₂ CH (CH ₃ ) OC (CH ₃ ) ₃ B.200 CH _(CH3) CH _(CH3) OC _{(CH3) 3} B.201 CH (CH ₃ ) (CH ₂ ) ₂ OC (CH ₃ ) 3 B.202 CH ₂ CH (CH ₃ ) CH ₂ OC (CH ₃ ) ₃ B.203 (CH ₂ ) ₂ CH (CH ₃ ) OC (CH ₃ ) ₃ B.204 CH (CH ₃ ) CH (CH ₃ ) CH ₂ OC (CH ₃ ) ₃ B.205 CH (CH ₃ ) CH ₂ CH (CH ₃ ) OC (CH ₃ ) 3 B.206 _CH2 CH _(CH3) CH _(CH3) OC _(CH3) 3 B.207 CH _(CH3) CH _(CH3) CH _(CH3) OC _{(CH3) 3} B.208 CH (CH ₃ ) (CH ₂ ) ₃ OC (CH ₃ ) ₃ B.209 CH _{(CH3) OCF3} B.210 CH (CH ₃ ) CH ₂ OCF ₃ B.211 CH ₂ CH (CH ₃ ) OCF ₃ B.212 CH _(CH3) CH _{(CH3) OCF3} B.213 CH (CH ₃ ) (CH ₂ ) ₂ OCF ₃ B.214 CH ₂ CH (CH ₃ ) CH ₂ OCF ₃ B.215 (CH ₂ ) ₂ CH (CH ₃ ) OCF ₃ B.216 CH (CH ₃ ) CH (CH ₃ ) CH ₂ OCF ₃ B.217 CH (CH ₃ ) ₂ CH (CH ₃ ) 0 CF ₃ B.218 _CH2 CH _(CH3) CH _{(CH3) OCF3} B.219 CH _(CH3) CH _(CH3) CH _{(CH3) OCF3} B.220 CH (CH ₃ ) (CH ₂ ) ₃ OCF ₃ B.221 ch (ch ₃ ) sch ₃ B.222 CH (CH ₃ ) CH ₂ SCH ₃ B.223 CH ₂ CH (CH ₃ ) SCH ₃ B.224 CH _(CH3) CH _{(CH3) SCH3} B.225 CH (CH ₃ ) (CH ₂ ) ₂ SCH ₃ B.226 CH ₂ CH (CH ₃ ) CH ₂ SCH ₃ B.227 (CH ₂ ) ₂ CH (CH ₃ ) SCH ₃ B.228 CH (CH ₃ ) CH (CH ₃ ) CH ₂ SCH ₃ B.229 CH (CH ₃ ) ch ₂ ch (ch ₃ ) sch ₃ B.230 CH ₂ CH (CH ₃ ) ch (ch ₃ ) sch ₃ B.231 ( CH _(CH3) CH _(CH3) CH _{(CH3) SCH3} B.232 ( H (CH ₃₎ (CH _{2) 3} SCH ₃

- w-

Nr. R ³ B.233 CH (CH ₃ ) statues ₃ B.234 CH (CH ₃ ) CH ₂ SOCH ₃ B.235 CH ₂ CH (CH ₃ ) SOCH ₃ B.236 CH (CH ₃₎ CH (CH _{3) 3} SOC B.237 CH (CH ₃ ) (CH ₂ ) ₂ SOCH ₃ B.238 CH ₂ CH (CH ₃ ) CH ₂ SOCH ₃ B.239 (CH ₂ ) ₂ CH (CH ₃ ) SOCH ₃ B.240 CH (CH ₃ ) CH (CH ₃ ) CH ₂ SOCH ₃ B.241 CH (CH ₃ ) CH ₂ CH (CH ₃ ) statues ₃ B.242 ch ₂ ch (ch ₃ ) CH (ch ₃ ) statues ₃ B.243 CH (CH ₃₎ CH (CH ₃₎ CH (CH _{3) 3} SOC B.244 CH (CH ₃ ) (CH ₂ ) ₃ SOCH ₃ B.245 CH (CH ₃ ) SO ₂ CH ₃ B.246 CH (CH ₃ ) CH ₂ SO ₂ CH ₃ B.247 CH (CH ₃ ) (CH ₂ ) ₃ SO ₂ CH ₃ B.248 CH ₂ CH (CH ₃ ) SO ₂ CH ₃ B.249 CH (CH ₃ ) CH (CH ₃ ) SO ₂ CH ₃ B.250 CH (CH ₃ ) (CH ₂ ) ₂ SO ₂ CH 3 B.251 CH ₂ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ B.252 (CH ₂ ) ₂ CH (CH ₃ ) SO ₂ CH ₃ B.253 CH (CH ₃ ) CH (CH ₃ ) CH ₂ SO ₂ CH ₃ B.254 CH (CH ₃ ) ch ₂ ch (ch ₃ ) with ₂ ch ₃ B.255 _CH2 CH _(CH3) CH _{(CH3) SO2 CH3} B.256 CH (CH ₃ ) CH (CH ₃ ) CH (CH ₃ ) SO ₂ CH ₃ B.257 CH (CH ₃ ) (CH ₂ ) ₃ SO ₂ CH ₃ B.258 CH _(CH3) -cyclopropyl B.259 CH _{(CH3) 2-cyclopropyl} B.260 CH ₂ CH (CH ₃ ) -cyclopropyl B.261 CH _(CH3) CH _(CH3) -cyclopropyl B.262 CH (CH ₃ ) (CH ₂ ) ₂ -cyclopropyl B.263 CH ₂ CH (CH ₃ ) CH ₂ -cyclopropyl B.264 (CH ₂ ) ₂ CH (CH ₃ ) -cyclopropyl B.265 CH (CH ₃ ) CH (CH ₃ ) CH ₂ -cyclopropyl B.266 CH (CH ₃ ) CH ₂ CH (CH ₃ ) -cyclopropyl B.267 CH ₂ CH (CH ₃ ) CH (CH ₃ ) -cyclopropyl B.268 CH _(CH3) CH _(CH3) CH _(CH3) -cyclopropyl B.269 CH (CH ₃ ) (CH ₂ ) ₃ -cyclopropyl B.270 CH (CH ₃₎ -cyclopentyl B.271 CH _{(CH3) CH2} -cyclopentyl

-26 $ -

Nr. R ³ B.272 CH ₂ CH (CH ₃ ) -cyclopentyl B.273 CH (CH ₃₎ CH (CH ₃₎ -cyclopentyl B.274 CH (CH ₃ ) (CH ₂ ) ₂ -cyclopentyl B.275 CH ₂ CH (CH ₃ ) CH ₂ -cyclopentyl B.276 (CH ₂ ) ₂ CH (CH ₃ ) -cyclopentyl B.277 CH (CH ₃ ) CH (CH ₃ ) CH ₂ -cyclopentyl B.278 CH (CH ₃ ) CH ₂ CH (CH ₃ ) -cyclopentyl B.279 CH ₂ CH (CH ₃ ) CH (CH ₃ ) -cyclopentyl B.280 CH (CH ₃₎ CH (CH ₃₎ CH (CH ₃₎ -cyclopentyl B. 281 CH (CH ₃ ) (CH ₂ ) ₃ -cyclopentyl B.282 CH _(CH3) -cyclohexyl B.283 CH (CH ₃ ) CH ₂ -cyclohexyl B.284 CH ₂ CH (CH ₃ ) -cyclohexyl B.285 CH _(CH3) CH _(CH3) -cyclohexyl B.286 CH (CH ₃ ) (CH ₂ ) ₂ -cyclohexyl B.287 CH ₂ CH (CH ₃ ) CH ₂ -cyclohexyl B.288 (CH ₂ ) ₂ CH (CH ₃ ) -cyclohexyl B.289 CH (CH ₃ ) CH (CH ₃ ) CH ₂ -cyclohexyl B.290 CH (CH ₃ ) CH ₂ CH (CH ₃ ) -cyclohexyl B.291 CH ₂ CH (CH ₃ ) CH (CH ₃ ) -cyclohexyl B.292 CH _(CH3) CH _(CH3) CH _(CH3) -cyclohexyl B.293 CH (CH ₃ ) (CH ₂ ) ₃ -cyclohexyl B.294 CH (CH ₃ ) CHF ₂ B.295 CF (CH ₃ ) CHF ₂ B.296 CH (CH ₃ ) CH ₂ F B.297 CF _{(CH3) 3} B.298 CF (CH ₃ ) CF ₃ B.299 CH _(CH3) CC1 ₃ B.300 CH _{(CH3) CF3} B.301 ch (ch ₃ ) ch ₂ cf ₃ B.302 ch ₂ ch (ch ₃ ) cf ₃ B.303 CH _(CH3) CH _{(CH3) CF3} B.304 CH (CH ₃₎ CF ₂ CF ₃ B.305 CH _(CH3) Br B.306 CH _{(CH3) CH2} Br B.307 CH (CH ₃ ) (CH ₂ ) ₂ Br B.308 2 H (CH ₃₎ (CH _{2) 3} Br B.309 ĽH (CH ₃₎ C 1 -C B.310 ( h (ch ₃ ) ch ₂ ci

- Ζ ^ ν-

Nr. R ³ B.311 CH (CH ₃₎ (CH _{2) 2} C1 B.312 CH (CH ₃ ) (CH ₂ ) ₃ Cl B.313 CH _{(CH3) OCF3} B. 314 CH (CH ₃ ) CH ₂ OCF ₃ B.315 CH (CH ₃ ) (CH ₂ ) ₂ OCF ₃ B. 316 CH (CH ₃ ) (CH ₂ ) ₃ ocf ₃ B.317 CH (CH ₃₎ F B.318 CH (CH ₃ ) CH ₂ F B.319 CH (CH ₃ ) (CH ₂ ) ₂ f B.320 CH (CH ₃ ) (CH ₂ ) ₃ F B.321 CH _(CH3) aminophenol 1 B.322 CH _{(CH3) 2} 1 aminophenol B.323 CH ₂ CH (CH ₃ ) -phenyl B.324 CH _(CH3) CH _(CH3) -phenyl B.325 CH (CH ₃ ) (CH ₂ ) ₂ -phenyl B.326 CH ₂ CH (CH ₃ ) CH ₂ -phenyl B.327 (CH ₂ ) ₂ CH (CH ₃ ) -phenyl B.328 CH (CH ₃ ) CH (CH ₃ ) CH ₂ -phenyl B.329 CH (CH ₃ ) CH ₂ CH (CH ₃ ) -phenyl B.330 CH ₂ CH (CH ₃ ) CH (CH ₃ ) -phenyl B.331 CH _(CH3) CH _(CH3) CH _(CH3) -phenyl B. 332 CH (CH ₃ ) (CH ₂ ) ₃ -phenyl B.333 2-FC ₆ H ₄ -CH ₂ B.334 3-FC ₆ H ₄ -CH ₂ B.335 4-FC ₆ H ₄ -CH ₂ B.336 2,3-F ₂ -C ₆ H ₃ -CH ₂ B.337 2,4-F ₂ -C ₆ H ₃ -CH ₂ B.338 2,5-F ₂ -C ₆ H ₃ -CH ₂ B.339 2,6-F ₂ -C ₆ H ₃ -CH ₂ B.340 3.4-F ₂ -C ₆ H ₃ -CH ₂ B.341 3,5-F ₂ -C ₆ H ₃ -CH ₂ B.342 2-Cl-C ₆ H ₄ CH ₂ B.343 3-Cl-C ₆ H ₄ CH ₂ B.344 4-Cl-C ₆ H ₄ CH ₂ B.345 2,3-Cl ₂ -C ₆ H ₃ -CH ₂ B.346 2.4-Cl ₂ -C ₆ H ₃ -CH ₂ B.347 2,5-Cl ₂ -C ₆ H ₃ -CH ₂ ä B.348 2,6-Cl ₂ -C ₆ H ₃ -CH ₂ ; B.349 3,4-Cl ₂ -C ₆ H ₃ -CH ₂ i

i V

Nr. R ³ B.350 3,5-Cl ₂ -C ₆ H ₃ -CH ₂ B.351 2,3,4-Cl ₃ -C ₆ H ₂ -CH ₂ B.352 2,3,5-Cl ₃ -C ₆ H ₂ -CH ₂ B.353 2,3,6-Cl ₃ -C ₆ H ₂ -CH ₂ B.354 2,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ B.355 2,4,6-Cl ₃ -C ₆ H ₂ -CH ₂ B.356 3,4,5-Cl ₃ -C ₆ H ₂ -CH ₂ B.357 2-Br-C ₆ H ₄ CH ₂ B.358 3-Br-C ₆ H ₄ CH ₂ B.359 4-Br-C ₆ H ₄ CH ₂ B.360 2,3-Br ₂ -C ₆ H ₃ -CH ₂ B.361 2,4-Br ₂ -C ₆ H ₃ -CH ₂ B.362 2,5-Br ₂ -C ₆ H ₃ -CH ₂ B.363 2,6-Br ₂ -C ₆ H ₃ -CH ₂ B.364 3,4-Br ₂ -C ₆ H ₃ -CH ₂ B.365 3,5-Br ₂ -C ₆ H ₃ -CH ₂ B.366 2-F, 3-Cl-C ₆ H ₃ CH ₂ B.367 2-F, 4-Cl-C ₆ H ₃ CH ₂ B.368 2-F, 5-Cl-C ₆ H ₃ CH ₂ B.369 2-F, 3-Br-C ₆ H ₃ CH ₂ B.370 2-F, 4-Br-C ₆ H ₃ CH ₂ B.371 2-F, 5-Br-C ₆ H ₃ CH ₂ B.372 2-Cl, 3-FC ₆ H ₃ -CH ₂ B.373 2-Cl, 4-FC ₆ H ₃ -CH ₂ B.374 2-Cl, 5-FC ₆ H ₃ -CH ₂ B.375 2-C1, 3-Br-C ₆ H ₃ CH ₂ B.376 2-C1, 4-Br-C ₆ H ₃ CH ₂ B.377 2-C1, 5-Br-C ₆ H ₃ CH ₂ B.378 2-Br, 3-FC ₆ H ₃ -CH ₂ B.379 2-Br, 4-FC ₆ H ₃ -CH ₂ B.380 2-Br, 5-FC ₆ H ₃ -CH ₂ B.381 2-Br, 3-7Cl-C ₆ H ₃ CH ₂ B.382 2-Br, 4-Cl-C ₆ H ₃ CH ₂ B.383 2-Br, 5-Cl-C ₆ H ₃ CH ₂ B.384 4-C 1, 3,5-Br ₂ -C ₆ H ₂ -CH ₂ B.385 2-CN-cei? -C? B.386 J-CN-C ₆ H ₄ CH ₂ B.387 i-cn-c ₆ h ₄ -ch ₂ B.388 I j-no ₂ -c ₆ h ₄ -ch ₂

'in-

Nr. R ³ B.389 3-NO ₂ -C ₆ H ₄ -CH ₂ B.390 4-NO ₂ -C ₆ H ₄ -CH ₂ B.391 2-CH ₃ -C ₅ H ₄ -CH ₂ B.392 3-CH ₃ -C ₆ H ₄ -CH ₂ B.393 4-CH ₃ -C ₆ H ₄ -CH ₂ B.394 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.395 2,4- (CH ₃ ) ₂ -C ₆ H ₃ 'CH ₂ B.396 2,5- (CH ₃ ) 2 -C ₆ H ₃ -CH ₂ B.397 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.398 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.399 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.400 2-CH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.401 3-CH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.402 4-CH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.403 2-CH (CK ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.404 3-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.405 4-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.406 3-C (CH ₃ ) ₃ -C ₆ H ₄ -CH ₂ B.407 4-C (CH ₃ ) ₃ -C ₆ H ₄ -CH ₂ B.408 2-C ₆ H 5 -C ₆ H ₄ -CH ₂ B.409 3-C ₆ H ₅ -C ₆ H ₄ -CH ₂ B.410 4-C ₆ H ₅ -C ₆ H ₄ -CH ₂ B.411 2-OCH ₃ -C ₆ H ₄ -CH ₂ B.412 3-OCH ₃ -C ₆ H ₄ -CH ₂ B.413 4-OCH ₃ -C ₆ H ₄ -CH ₂ B.414 2,3- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.415 2,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.416 2,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.417 2,6- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.418 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.419 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH ₂ B.420 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH ₂ B.421 2-OCH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.422 3-OCH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.423 4-OCH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.424 2-O (CH ₂ ) ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.425 3-0 (CH ₂ ) ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.426 1 - 0 (ch ₂ ) ₂ ch _{3 -} c ₆ h ₄ - ch ₂ B.427 2-OCH (CH ₃ ) 2 -C _with H ₄ -CH ₂

- ľn ~

Nr. R ³ B.428 3-OCH (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.429 4-OCH (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.430 3-OC (CH ₃ ) ₃ -C ₆ H ₄ -CH ₂ B.431 4-OC (CH ₃ ) ₃ -C ₆ H ₄ -CH ₂ B.432 2-OCH ₂ CH = CH ₂ -C ₆ H ₄ -CH ₂ B.433 3-ch ₂ ch = ch ₂ -c ₆ h ₄ -ch ₂ B.434 4-OCH ₂ CH = CH ₂ -C ₆ H ₄ -CH ₂ B.435 2-CF ₃ -C ₆ H ₄ -CH ₂ B.436 3-CF ₃ -C ₆ H ₄ -CH ₂ B.437 4-CF ₃ -C ₆ H ₄ -CH ₂ B.438 2-CO ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.439 3-CO ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.440 4-CO ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.441 2-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.442 3-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.443 4-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.444 2-CONH ₂ -C ₆ H ₄ -CH ₂ B.445 3-CONH ₂ -C ₆ H ₄ -CH ₂ B.446 4-CONH ₂ -C ₆ H ₄ -CH ₂ B.447 2-CON (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.448 3-CON (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.449 4-CON (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.450 2-CONHCH ₃ -C ₆ H ₄ -CH ₂ B.451 3-CONHCH ₃ -C ₆ H ₄ -CH ₂ B.452 4-CONHCH ₃ -C ₆ H ₄ -CH ₂ B.453 2-NH ₂ -C ₆ H ₄ -CH ₂ B.454 3-NH ₂ -C ₆ H ₄ -CH ₂ B.455 4-NH ₂ -C ₆ H ₄ -CH ₂ B.456 2-N (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.457 3-N (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.458 4-N (CH ₃ ) ₂ -C ₆ H ₄ -CH ₂ B.459 2-NHCH ₃ -C ₆ H ₄ -CH ₂ B.460 3-NHCH ₃ -C ₆ H ₄ -CH ₂ B.461 4-NHCH ₃ -C ₆ H ₄ -CH ₂ B.462 2-CSNH ₂ -C ₆ H ₄ -CH ₂ B.463 3-CSNH ₂ -C ₆ H ₄ -CH ₂ B.464 i-csnh ₂ -c ₆ h ₄ -ch ₂ B.465 2-SCH ₃ -C ₆ H ₄ -CH ₂ B.466 s-sch _{3 -} c ₆ h _{4 -} ch ₂

I

I

Nr. R ³ B.467 4-SCH ₃ -C ₆ H ₄ -CH ₂ B.468 2-SOCH ₃ -C ₆ H ₄ -CH ₂ B.469 3-SOCH ₃ -C ₆ H ₄ -CH ₂ B.470 4-SOCH ₃ -C ₆ H ₄ -CH ₂ B.471 2-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.472 3-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.473 4-SO ₂ CH ₃ -C ₆ H ₄ -CH ₂ B.474 2-OCF ₃ -C ₆ H ₄ -CH ₂ B.475 3-OCF ₃ -C ₅ H ₄ -CH ₂ B.476 4-OCF ₃ -C ₆ H ₄ -CH ₂ B.477 2-OCHF ₂ -C ₆ H ₄ -CH ₂ B.478 3-OCHF ₂ -C ₆ H ₄ -CH ₂ B.479 4-OCHF ₂ -C ₆ H ₄ -CH ₂ B.480 3-CF ₃ , 4-OCF ₃ -C ₆ H ₃ -CH ₂ B.481 2-CH ₂ CH ₂ FC ₆ H ₄ -CH ₂ B.482 3-CH ₂ CH ₂ FC ₆ H ₄ -CH ₂ B.483 4-CH ₂ CH ₂ FC ₆ H ₄ -CH ₂ B.484 2-CH ₂ CF ₃ -C ₆ H ₄ -CH ₂ B.485 3-CH ₂ CF ₃ -C ₆ H ₄ -CH ₂ B.486 4-CH ₂ CF ₃ -C ₆ H ₄ -CH ₂ B.487 2-CF ₂ CHF ₂ -C ₆ H ₄ -CH ₂ B.488 3-CF ₂ CHF ₂ -C ₆ H ₄ -CH ₂ B.489 4-CF ₂ CHF ₂ -C ₆ H ₄ -CH ₂ B.490 2-CHF ₂ -C ₆ H ₄ -CH ₂ B.491 3-CHF ₂ -C ₆ H ₄ -CH ₂ B.492 4-CHF ₂ -C ₆ H ₄ -CH ₂ B.493 _{naphthalin-l-yl-CH2} B.494 _{naphthalin-2-yl-CH2} B.495 _{pyridin-2-yl-CH2} B.496 _{pyridin-3-yl-CH2} B.497 _{pyridin-4-yl-CH2} B.498 5-CH ₃ -pyridin-2-yl-CH ₂ B.499 _{6-CH3-pyridin-2-yl-CH2} B.500 _{5-CH3-pyridin-3-yl-CH2} B.501 _{6-CH3-pyridin-3-yl-CH2} B.502 5-OCH ₃ -pyridin-2-ylCH ₂ B.503 S-OCH ₃ -pyridin-2-yl-CH ₂ B.504 □ -OCH ₃ -pyridin-3-yl-CH ₂ B.505 5-OCH ₃ -pyridin-3-ylCH ₂

- 5 ~ -

Nr. R ³ B.506 _{4-Cl-pyridin-2-yl-CH2} B.507 _{5-Cl-pyridin-2-yl-CH2} B.508 _{6-Cl-pyridin-2-yl-CH2} B.509 _{2-Cl-pyridin-3-yl-CH2} B.510 _{5-Cl-pyridin-3-yl-CH2} B.511 _{6-Cl-pyridin-3-yl-CH2} B.512 _{2-Cl-pyridin-4-yl-CH2} B.513 _{3,5-Cl-pyridin-2-yl-CH2} B.514 _{pyrimidin-2-yl-CH2} B.515 _{4-Cl-pyrimidin-2-yl-CH2} B.516 _{5-Cl-pyrimidin-2-yl-CH2} B.517 4-CH ₃ -pyrimidin-2-yl-CH ₂ B.518 5-CH ₃ -pyrimidin-2-yl-CH ₂ B.519 4-OCH ₃ -pyrimidin-2-yl-CH ₂ B.520 5-OCH ₃ -pyrimidin-2-yl-CH ₂ B.521 4-OCH ₂ CH ₃ -pyrimidin-2-yl-CH ₂ B.522 5-OCH ₂ CH ₃ -pyrimidin-2-yl-CH ₂ B.523 _{pyrimidin-4-yl-CH2} B.524 _{2-Cl-pyrimidin-4-yl-CH2} B.525 _{6-Cl-pyrimidin-4-yl-CH2} B.526 2,6-Cl ₂ -pyrimidin-4-yl-CH ₂ B. 527 2-CH ₃ -pyrimidin-4-yl-CH 2 B.528 6-CH ₃ -pyrimidin-4-yl-CH 2 B.529 2-OCH ₃ -pyrimidin-4-yl-CH ₂ B.530 6-OCH ₃ -pyrimidin-4-yl-CH ₂ B.531 2-OCH ₂ CH ₃ -pyrimidin-4-yl-CH ₂ B.532 6-OCH ₂ CH ₃ -pyrimidin-4-yl-CH ₂ B.533 _{pyrimidin-5-yl-CH2} B.534 _{2-Cl-pyrimidin-5-yl-CH2} B.535 2-CH ₃ -pyrimidin-5-yl-CH ₂ B.536 2-OCH ₃ -pyrimidin-5-yl-CH ₂ B.537 2-OCH ₂ CH ₃ -pyrimidin-5-yl-CH ₂ B.538 _{furan-2-yl-CH2} B.539 _{4-Br-furan-2-yl-CH2} B.540 _{4-C1-furan-2-y1-CH2} B.541 _{4-CN-furan-2-y1-CH2} B.542 4-CH ₃ -furan-2-yl-CH ₂ B.543 _{5-Br-furan-2-y1-CH2} B.544 _{5-Cl-furan-2-yl-CH2}

- Zfí-

Nr. R ³ B.545 5-CN-furan-2-yľCH2 B.546 _{5-CH3-furan-2-2} yľCH B.547 furan-3-ylCH ₂ B.548 5-Br-furan-3-ylCH ₂ B.549 5-Cifuran-3-ylCH ₂ B.550 5-CN-furan-3-ylCH ₂ B.551 _{5-CH3-furan-3-2} yľCH B.552 _{thien-2-yl-CH2} B.553 _{4-Br-thien-2-2} yľCH B.554 _{4-Cľthien-2-2} yľCH B.555 4-CN-thien-2-ylCH ₂ B.556 4-CH ₃ -thien-2-ylCH ₂ B.557 _{5-Br-thien-2-2} yľCH B.558 _{5-Cľthien-2-2} yľCH B.559 5-CN-thien-2-ylCH ₂ B.560 5-CH ₃ -thien-2-ylCH ₂ B.561 _thien-3-2 yľCH B.562 5-Br-thien-3-ylCH ₂ B.563 _{5-Cľthien-3-2} yľCH B.564 _{5-CN-thien-3-yl-CH2} B.565 5-CH ₃ -thien-3-ylCH ₂ B.566 oxazol- ₂ -yl-CH2 B.567 4-Br-oxazol- ₂ -ylCH2 B.568 4-Coxazol- ₂ -yl-CH2 B.569 _{4-CN-oxazol-2-yl-CH2} B.570 4-CH ₃ -oxazol-2-ylCH ₂ B.571 _{5-Br-oxazol-2-yl-CH2} B.572 _{5-Cľoxazol-2-yl-CH2} B.573 5-CN-oxazol- ₂ -ylCH ₂ B.574 _{5-CH3--oxazoľ2} yľCH ₂ B.575 _{oxazol-4-yl-CH2} B.576 2-Br-oxazol-4-ylCH ₂ B.577 2-Coxazol-4-ylCH ₂ B.578 2-CN-oxazol-4-ylCH ₂ B.579 2-CH ₃ -oxazol-4-ylCH ₂ B.580 2-C ₆ H _5--oxazoľ4 yľCH ₂ B.581 5-Br-oxazol-4-ylCH ₂ B.582 _{5-Cl-oxazol-4-yl-CH2} B.583 5-CN-oxazol-4-ylCH ₂

Nr. R ³ B.584 _{5-CH3-oxazol-4-yl-CH2} B.585 _{oxazol-5-yl-CH2} B.586 _{4-Br-oxazol-5-yl-CH2} B.587 _{4-Cl-oxazol-5-yl-CH2} B.588 _{4-CN-oxazol-5-yl-CH2} B. 589 4-CH ₃ -oxazol-5-yl-CH ₂ B.590 _{2-Br-oxazol-5-yl-CH2} B. 591 _{2-Cl-oxazol-5-yl-CH2} B.592 _{2-CN-oxazol-5-yl-CH2} B.593 2-CH ₃ -oxazol-5-yl-CH ₂ B.594 _{isoxazol-3-yl-CH2} B.595 _{4-Br-isoxazol-3-yl-CH2} B.596 _{4-Cl-isoxazol-3-yl-CH2} B.597 _{4-CN-isoxazol-3-yl-CH2} B.598 _{4-CH3 isoxazol-3-yl-CH2} B.599 _{5-Br-isoxazol-3-yl-CH2} B.600 _{5-Cl-isoxazol-3-yl-CH2} B.601 _{5-CN-isoxazol-3-yl-CH2} B.602 5-CH ₃ -isoxazol-3-yl-CH ₂ B.603 _{isoxazol-4-yl-CH2} B.604 _{3-Br-isoxazol-4-yl-CH2} B.605 _{3-Cl-isoxazol-4-yl-CH2} B.606 _{3-CN-isoxazol-4-yl-CH2} B.607 3-CH ₃ -isoxazol-4-yl-CH ₂ B.608 _{5-Br-isoxazol-4-yl-CH2} B.609 _{5-Cl-isoxazol-4-yl-CH2} B.610 _{5-CN-isoxazol-4-yl-CH2} B.611 5-CH ₃ -isoxazol-4-yl-CH ₂ B.612 3,5- (CH ₃ ) ₂ -isoxazol-4-yl-CH ₂ B.613 _{isoxazol-5-yl-CH2} B.614 _{3-Br-isoxazol-5-yl-CH2} B.615 _{3-Cl-iaoxazol-5-yl-CH2} B.616 _{3-CN-isoxazol-5-yl-CH2} B.617 3-CH ₃ -isoxazol-5-yl-CH ₂ B.618 _{3-C6H5-isoxazol-5-yl-CH2} B.619 4-C1-C 6 H _{3-isoxazol-5-yl-CH2} B.620 4-Br, _{3-C6H5-isoxazol-5-yl-CH2} B.621 _{4-Br-isoxazol-5-yl-CH2} B.622 _{l-Cl-isoxazol-5-yl-CH2}

Nr.

R ³

B.623

_{4-CN-isoxazol-5-yl-CH2}

B.624

14-CH ₃ -isoxazol-5-yl-CH 2

B.625

_{Ithiazol-2-yl-CH2}

B.626

_{4-Br-thiazol-2-yl-CH2}

B.627

_{4-Cl-thiazol-2-yl-CH2}

B.628

_{4-CN-thiazol-2-yl-CH2}

B.629

4-CH ₃ -thiazol-2-yl-CH 2

B. 630

_{5-Br-thiazol-2-yl-CH2}

B.631

5-Cl-thiazol-2-yl-CH2

B.632

_{5-CN-thiazol-2-yl-CH2}

B.633

5-CH 3 -thiazol-2-yl-CH ₂

B.634 _{thiazol-4-yl-CH2}

B.635

_{2-Br-thiazol-4-yl-CH2}

B.636

_{2-Cl-thiazol-4-yl-CH2}

B.637

2-CN-thiazol-4-yl-CH ₂

B.638

2-CH ₃ -thiazol-4-yl-CH ₂

B.639

_{5-Br-thiazol-4-yl-CH2}

B.640 15-Cl-thiazol-4-yl-CH ₂

B.641

_{5-CN-thiazole-4-yl-CH2}

B.642

5-CH ₃ -thiazol-4-yl-CH ₂

B.643 _{thiazol-5-yl-CH2}

B.644

_{4-Br-thiazol-5-yl-CH2}

B.645

_{4-Cl-thiazol-5-yl-CH2}

B.646

_{4-CN-thiazol-5-yl-CH2}

B.647

4-CH ₃ -thiazol-5-yl-CH ₂

B.648

_{2-Br-thiazol-5-yl-CH2}

B.649

12-Cl-thiazol-5-yl-CH ₂

B.650

2-CN-thiazol-5-yl-CH ₂

B.651

2-CH ₃ -thiazol-5-yl-CH ₂

B.652 _{isothiazol-3-yl-CH2}

B.653

_{I4-Br-isothiazol-3-yl-CH2}

B.654

_{4-Cl-isothiazol-3-yl-CH2}

B.655

_{4-CN-isothiazol-3-yl-CH2}

B.656

_{4-CH3-isothiazol-3-yl-CH2}

B.657

_{5-Br-isothiazol-3-yl-CH2}

B.658

_{5-Cl-isothiazol-3-yl-CH2}

B.659

_{5-CN-isothiazol-3-yl-CH2}

B.660

5-CH 3 -isothiazol-3-yl-CH ₂

B.661 _{isothiazol-4-yl-CH2}

-NO-

Nr. R ³ B.662 _3-Br-2 -isothiazole-4-yľCH B.663 3-Isothiazol-4-ylCH ₂ B.664 3-CN-isothiazol-4-ylCH ₂ B.665 3-CH ₃ -isothiazol-4-ylCH ₂ B.666 _5-Br-2 -isothiazole-4-yľCH B.667 5-Isothiazol-4-ylCH ₂ B.668 5-CN-isothiazol-4-ylCH ₂ B.669 _{5-CH3--isothiazoľ4} yľCH ₂ B.670 3,5- _{(CH3) 2-isothiazol-4-yl-CH2} B.671 isothiazol-5-ylCH ₂ B.672 3-Br-isothiazol-5-ylCH ₂ B.673 _{3-Cľisothiazol-5-2} yľCH B.674 3-CN-isothiazol-5-ylCH ₂ B.675 3-CH ₃ -isothiazol-5-ylCH ₂ B.676 _4-Br-2 isothiazoľ5-yľCH B.677 _{4-Cl-isothiazol-5-2} yľCH B.678 4-CN-isothiazol-5-ylCH ₂ B.679 _{4-CH3--isothiazoľ5} yľCH ₂ B.680 imidazol- ₂ -ylCH ₂ B.681 1'-imidazol- ₂ -ylCH ₂ B.682 l-Br-imidazol-2-yl-CH2 B.683 1-CN-imidazol- ₂ -ylCH ₂ B.684 1'CH ₃ -imidazol- ₂ -yl-CH ₂ B.685 4-Cl-imidazol- ₂ -ylCH2 B.686 4-Br-imidazol- ₂ -ylCH2 B.687 4-CN-imidazol- ₂ -ylCH2 B.688 4-CH ₃ -imidazol- ₂ -ylCH ₂ B.689 1-CH ₃ , 5-Climidazol- ₂ -ylCH ₂ B.690 1,4- (CH ₃ ) ₂ -imidazol- ₂ -ylCH ₂ B.691 1,5- (CH ₃ ) ₂ -imidazol- ₂ -ylCH ₂ B.692 _{imidazol-4-yl-CH2} B.693 2-Climidazol-4-ylCH ₂ B.694 2-Br-imidazol-4-ylCH ₂ B.695 2-CN-imidazol-4-ylCH ₂ B.696 1'CH ₃ -imidazol-4-yl-CH ₂ B.697 2-CH ₃ -imidazol-4-ylCH ₂ B.698 _{5-Cl-imidazol-4-yl-CH2} B.699 _{5-Br-imidazol-4-2} yľCH B.700 _{5-CN-imidazol-4-2} yľCH

Nr. R ³ B.701 5-CH ₃ -imidazol-4-ylCH ₂ B.702 1-CH ₃ , 5-Cl-imidazol-4-yl-CH ₂ B.703 1,2- (CH ₃ ) ₂ -imidazol-4-yl-CH ₂ B.704 1,5- (CH ₃ ) ₂ -imidazol-4-yl-CH ₂ B.705 _{pyrazol-3-yl-CH2} B.706 _{5-Br-pyrazol-3-yl-CH2} 07 _{5-Cl-pyrazol-3-yl-CH2} B.708 5-CN-pyrazol-3-yl-CH ₂ B.709 5-CH ₃ -pyrazol-3-yl-CH ₂ B.710 1-C 8 H 5 -pyrazol-3-yl-CH ₂ B.711 _{4-Br-pyrazol-3-2} yľCH B.712 _{4-Cľpyrazol-3-2} yľCH B.713 _{4-CN-pyrazol-3-yl-CH2} B.714 4-CH ₃ -pyrazol-3-yl-CH ₂ B.715 1-CH ₃ -pyrazol-3-yl-CH ₂ B.716 1,4- (CH ₃ ) ₂ -pyrazol-3-yl-CH ₂ B.717 1,5- (CH ₃ ) ₂ -pyrazol-3-yl-CH ₂ B.718 1-CH ₃ , 4-Cl-pyrazol-3-yl-CH ₂ B.719 1-CH ₃ , 5-Cl-pyrazol-3-yl-CH ₂ B.720 _{pyrazol-4-yl-CH2} B.721 _{3-Br-pyrazol-4-yl-CH2} B.722 3-C 1 -pyrazol-4-yl-CH ₂ B.723 3-CN-pyrazol-4-ylCH ₂ B.724 3-CH ₃ -pyrazol-4-yl-CH ₂ B.725 1-CH ₃ -pyrazol-4-yl-CH ₂ B.726 1,5- (CH ₃ ) ₂ -pyrazol-4-yl-CH ₂ B.727 1,3- (CH ₃ ) ₂ -pyrazol-4-yl-CH ₂ B.728 1-CH ₃ , 3-C 1 -pyrazol-4-yl-CH ₂ B.729 1-CH _3,5 -C ₁ -pyrazol-4-yl-CH ₂ B.730 _{pyrazol-5-yl-CH2} B.731 _{3-Br-pyrazol-5-yl-CH2} B.732 _{3-Cl-pyrazol-5-yl-CH2} B.733 3-CN-pyrazol-5-yl-CH ₂ B.734 3-CH ₃ -pyrazol-5-yl-CH ₂ B.735 1'CH ₃ -pyrazol-5-yl-CH ₂ B.736 _{4-Br-pyrazol-5-yl-CH2} B.737 _{4-Cl-pyrazol-5-yl-CH2} B.738 _{4-CN-pyrazol-5-yl-CH2} B.739 4-CH ₃ -pyrazol-5-yl-CH ₂

7č 1 -

Nr. R ³ B.740 5-CH 3 -1,2,4-thiadiazol-3-yl-CH = CH ⁵ B.741 5-CF 3 -1,2,4-thiadiazol-3-yl CH = CH B.742 5-OCH 3 -1,2,4-thiadiazol-3-yl CH = CH B.743 5-thiadiazole-3-C1-1,2,4 yľCH CH B.744 5-CH (CH ₃ ) 2-1 / 2,4-thiadiazol-3-yl-CH = CH B.745 pyrrol-2-yl-CH = CH B.746 4-Cľpyrroľ2 yľCH-CH B.747 4-Br-pyrrol-2-yl-CH = CH B.748 _{4-CH3--pyrroľ2} yľCH CH B.749 4-C6H5-pyrrol-2-yl-CH = CH B.750 benzimidazol-2-yl-CH = CH B.751 quinolin-2-y1-CH = CH B.752 2-FC ₆ H ₄ -CH = C (CH ₃ ) B.753 3-FC ₆ H ₄ -CH = C (CH ₃ ) B.754 4-FC ₆ H ₄ -CH = C (CH ₃ ) B.755 2,3-F ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.756 2,4-F ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.757 2,5-F ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.758 2,6-F ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.759 3,4-F ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.760 3,5-F ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.761 2-Cl-C ₆ H ₄ -CH = C (CH ₃₎ B.762 3-Cl-C ₆ H ₄ -CH = C (CH ₃₎ B.763 4-Cl-C ₆ H ₄ -CH = C (CH ₃ ) B.764 2,3-Cl ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.765 2,4-Cl ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.766 2,5-Cl ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.767 2,6-Cl ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.768 3,4-Cl ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.769 3,5-Cl ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.770 2,3,4-Cl ₃ -C ₆ H ₂ -CH = C (CH ₃ ) B.771 2,3,5-Cl ₃ -C ₆ H ₂ -CH = C (CH ₃ ) B.772 2,3,6-Cl ₃ -C ₆ H ₂ -CH = C (CH ₃ ) B.773 2,4,5-Cl ₃ -C ₆ H ₂ -CH = C (CH ₃ ) B.774 2,4,6-Cl ₃ -C ₆ H ₂ -CH = C (CH ₃ ) B.775 3,4,5-Cl ₃ -C ₆ H ₂ -CH = C (CH ₃ ) B.776 2-Br-C ₆ H ₄ -CH = C (CH ₃₎ B.777 3-Br-C ₆ H ₄ -CH = C (CH ₃₎

5 0 5 0 Nr. R ³ B.778 4-Br-C ₆ H ₄ -CH = C (CH ₃ ) B.779 2,3-Br ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.780 2,4-Br ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.781 2,5-Br ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.782 2,6-Br ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.783 3,4-Br ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.784 3,5-Br ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.785 2-F, 3-Cl-C ₆ H ₃ -CH-C _(CH3) B.786 2-F, 4-Cl-C ₆ H ₃ -CH-C _(CH3) B.787 2-F, 5-Cl-C ₆ H ₃ -CH-C _(CH3) B.788 2-F, 3-Br-C ₆ H ₃ -CH-C _(CH3) B.789 2-F, 4-Br-C ₆ H ₃ -CH-C _(CH3) B.790 2-F, 5-Br-C ₆ H ₃ -CH-C _(CH3) B.791 2-C1, 3-FC ₆ H ₃ -CH = C (CH ₃ ) B.792 2-C1, 4-FC ₆ H ₃ -CH = C (CH ₃ ) B.793 2-C1,5-FC ₆ H ₃ -CH = C (CH ₃ ) B.794 2-C1, 3-Br-C ₆ H ₃ -CH-C _(CH3) B.795 2-C1, 4-Br-C ₆ H ₃ -CH-C _(CH3) B.796 2-C1, 5-Br-C ₆ H ₃ -CH-C _(CH3) B.797 2-Br, 3-FC ₆ H ₃ -CH = C (CH ₃ ) B.798 2-Br, 4-FC ₆ H ₃ -CH = C (CH ₃ ) B.799 2-Br, 5-FC ₆ H ₃ -CH = C (CH ₃ ) B.800 2-Br, 3-Cl-C ₆ H ₃ -CH-C _(CH3) B.801 2-Br, 4-Cl-C ₆ H ₃ -CH-C _(CH3) B.802 2-Br, 5-Cl-C ₆ H ₃ -CH-C _(CH3) B.803 4-Cl, 3,5-Br ₂ -C ₆ H ₂ -CH = C (CH ₃ ) B.804 2-CN-C ₆ H ₄ -CH = C (CH ₃₎ B.805 3-CN-C ₆ H ₄ -CH = C (CH ₃₎ B.806 4-CN-C ₆ H ₄ -CH = C (CH ₃₎ B.807 2-NO ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.808 3-NO ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.809 4-NO ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.810 2-CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.811 3-CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) [ B.812 4-CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) ( B.813 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) i B.814 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) i B.815 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) i B.816 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) i

Nr. R ³ B.817 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.818 3,5- (CH ₃ ) 2 -C ₆ H ₃ -CH = C (CH ₃ ) B.819 2-CH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.820 3-CH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.821 4-CH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.822 2-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.823 3-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.824 4-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.825 3-C (CH ₃ ) ₃ -c ₆ h ₄ -ch = c (ch ₃ ) B.826 4-C (CH ₃ ) ₃ -c ₆ h ₄ -ch = c (ch ₃ ) B.827 2-C ₆ H ₅ -C ₆ H ₄ -CH = C (CH ₃₎ B.828 3-C ₆ H ₅ -C ₆ H ₄ -CH = C (CH ₃ ) B.829 4-C ₆ H _with -C ₆ H ₄ -CH = C (CH ₃ ) B.830 2-OCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.831 3-OCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.832 4-OCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.833 2,3- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B. 834 2,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.835 2,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.836 2,6- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.837 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.838 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = C (CH ₃ ) B.839 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH = C (CH ₃ ) B.840 2-OCH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.841 3-OCH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.842 4-OCH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.843 2-0 (ch ₂ ) ₂ ch ₃ -c ₆ h ₄ -ch = c (ch ₃ ) B.844 3-O (CH ₂ ) ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.845 4-0 (ch ₂ ) ₂ ch _{3 -} c ₆ h ₄ - ch = c (ch ₃ ) B.846 2-OCH (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (ch ₃ ) B.847 3-OCH (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.848 4-OCH (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.849 3-OC (CH ₃ ) ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.850 4-OC (CH ₃ ) ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B. 851 2-OCH ₂ CH = CH ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.852 3-OCH ₂ CH = CH ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.853 4-OCH ₂ CH = CH ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.854 2 -CF ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.855 3-CP ₃ -C ₆ H ₄ -CH = C (CH ₃ )

Nr. R ³ B.856 4-CF ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.857 2-co ₂ ch ₃ -c ₆ h ₄ -ch = c (CH ₃ ) j B.858 3-CO ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.859 4-CO ₂ CH ₃ -C ₆ H ₄ -CH = C (ch ₃ ) B.860 2-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.861 3-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) i B.862 4-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) 1 j B.863 2-CONH ₂ -C ₆ H ₄ -CH = C (CH ₃ ) 1 B.864 3-conh ₂ -c ₆ h ₄ -ch = c (ch ₃ ); B.865 4-CONH ₂ -C ₆ H ₄ -CH = C (CH ₃ ); B.866 2-con (ch ₃ ) ₂ -c ₆ h ₄ -ch = c (ch ₃ ); B.867 3-CON (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) - B.868 4-CON (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) 1 B.869 2-conhch ₃ -c ₆ h ₄ -ch = c (ch ₃ ) < B.870 3-CONHCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) i B.871 4-CONHCH ₃ -C ₆ H ₄ -CH = C _(CH3); B.872 2-NH ₂ -C ₆ H ₄ -CH = C (CH ₃ ): B.873 3-NH ₂ -C ₆ H ₄ -CH = C (CH ₃ )! B.874 4-NH ₂ -C ₆ H ₄ -CH = C (CH ₃ ) i B.875 2-N (CH ₃ ) ₂ -c ₆ h ₄ -ch = c (CH ₃ ) 1 B.876 3-N (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.877 4-N (CH ₃ ) ₂ -C ₆ H ₄ -CH = C (CH ₃ ) and s B.878 2-NHCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.879 3-NHCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.880 4-NHCH ₃ -C ₆ H ₄ -CH = C (ch ₃ ) B.881 2-CSNH ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.882 3 -csnh ₂ -c ₆ h ₄ -CH = C (CH ₃ ) B.883 4-CSNH ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.884 2-sch _{3 -} c ₆ h ₄ - ch = c (ch ₃ ) B.885 3-SCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.886 4-SCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) i B.887 2-SOCH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) 1 B.888 3-sculpture ₃ -c ₆ h ₄ -ch = c (CH ₃ ) B.889 4-SOCH ₃ -C ₆ H ₄ -CH = C (ch ₃ ) B.890 2-Sat ₂ ch ₃ -c ₆ h ₄ -ch = c (CH ₃ ) B.891 3-SO ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) 1 B.892 4-SO ₂ CH ₃ -C ₆ H ₄ -CH = C (CH ₃ ) [ B.893 2-OCF ₃ -C ₆ H ₄ -CH = C (CH ₃ ) J B.894 3-OCF ₃ -C ₆ H ₄ -CH = C (CH ₃ ) 1

-Ztf-

Nr. R ³ B.895 4-OCF ₃ -C ₆ H ₄ -CH = C (ch ₃ ) B.896 2 -ochf ₂ -c ₆ h ₄ -CH = C (CH ₃ ) ₅ B.897 3-OCHF ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.898 4-OCHF ₂ -C ₆ H ₄ -CH = C (CH ₃ ) B.899 3-CF ₃ , 4-OCF ₃ -C ₆ H ₃ -CH = C (CH ₃ ) B.900 2-CH ₂ CH ₂ FC ₆ H ₄ -CH = C (CH ₃ ) B.901 3-CH ₂ CH ₂ FC ₆ H ₄ -CH = C (CH ₃ ) B.902 4-CH ₂ CH ₂ FC ₆ H ₄ -CH = C (CH ₃ ) B.903 2-CH ₂ CF ₃ -C ₆ H ₄ -CH = C (CH ₃ ) B.904 3-ch ₂ cf ₃ -c ₆ h ₄ -ch = c (CH ₃ ) B.905 4 -CH ₂ CF ₃ -C ₆ H ₄ -CH = C (CH ₃₎ B.906 2-CF ₂ CHF ₂ -C ₆ H ₄ -CH = C _(CH3) B.907 3-CF ₂ CHF ₂ -C ₆ H ₄ -CH = C _(CH3) B.908 4-CHF ₂ CF ₂ -C ₆ H ₄ -CH = C _(CH3) B.909 2-CHF ₂ -C ₆ H ₄ -CH = C _(CH3) B.910 3-CHF ₂ -C ₆ H ₄ -CH = C _(CH3) B.911 4-CHF ₂ -C ₆ H ₄ -CH = C _(CH3) B.912 naphthalin-l-yl-CH = C (CH ₃₎ B.913 naphthalin-2-yl-CH = C (CH ₃₎ B.914 pyridin-2-yl-CH = C (CH ₃₎ B.915 pyridin-3-yl-CH = C (CH ₃₎ B.916 pyridin-4-yl-CH = C (CH ₃₎ B.917 _{5-CH3-pyridin-2-yl-CH} = C (CH ₃₎ B.918 6-CH ₃ -pyridin-2-yl-CH = C (CH ₃ ) B.919 _{5-CH3-pyridin-3-yl-CH} = C (CH ₃₎ B.920 _{6-CH3-pyridin-3-yl-CH} = C (CH ₃₎ B.921 5-OCH ₃ -pyridin-2-yl-CH = C (CH ₃ ) B.922 6-OCH ₃ -pyridin-2-yl-CH = C (CH ₃ ) B.923 _{5-OCH3-pyridin-3-yl-CH} = C (CH ₃₎ B.924 6-OCH ₃ -pyridin-3-yl-CH = C (CH ₃ ) B.925 4-Cl-pyridin-2-yl-CH = C (CH ₃₎ B.926 5-Cl-pyridin-2-yl-CH = C (CH ₃₎ B.927 6-Cl-pyridin-2-yl-CH = C (CH ₃₎ B.928 2-Cl-pyridin-3-yl-CH = C (CH ₃₎ B.929 5-Cl-pyridin-3-yl-CH = C (CH ₃₎ B.930 6-Cl-pyridin-3-yl-CH = C (CH ₃₎ B.931 2-Cl-pyridin-4-yl-CH = C (CH ₃₎ B.932 3,5-Cl ₂ -pyridin-2-yl-CH = C (CH ₃₎ B.933 j 3yrimidin-2-yl-CH = C (CH ₃₎

- 7Μ-

5 0 5 0 Nr. R ³ B.934 4-Cl-pyrimidin-2-yl-CH = C (CH ₃₎ B.935 5-Cl-pyrimidin-2-yl-CH = C (CH ₃₎ B.936 4-CH ₃ -pyrimidin-2-yl-CH = C (CH ₃ ) B.937 5-CH ₃ -pyrimidin-2-yl-CH = C (CH ₃ ) B.938 4-OCH 3 -pyrimidin-2-yl-CH = C (CH ₃ ) B.939 5-OCH ₃ -pyrimidin-2-yl-CH = C (CH ₃ ) B.940 pyrimidin-4-yl-CH = C (CH ₃₎ B.941 2-Cl-pyrimidin-4-yl-CH = C (CH ₃₎ B.942 6-Cl-pyrimidin-4-yl-CH = C (CH ₃₎ B.943 2,6-Cl 2 -pyrimidin-4-yl-CH = C (CH ₃ ) B.944 2-CH ₃ -pyrimidin-4-yl-CH = C (CH ₃ ) B.945 6-CH ₃ -pyrimidin-4-yl-CH = C (CH ₃ ) B.946 2-OCH ₃ -pyrimidin-4-yl-CH = C (CH ₃ ) B.947 6-OCH ₃ -pyrimidin-4-yl-CH = C (CH ₃ ) B.948 pyrimidin-5-yl-CH = C (CH ₃₎ B.949 2-Cl-pyrimidin-5-yl-CH = C (CH ₃₎ B.950 2-CH ₃ -pyrimidin-5-yl-CH = C (CH ₃ ) B.951 2-OCH ₃ -pyrimidin-5-yl-CH = C (CH ₃ ) B.952 furan-2-yl-CH = C (CH ₃₎ B.953 4-Br-furan-2-yl-CH = C (CH ₃₎ B.954 4-Cl-furan-2-yl-CH = C (CH ₃₎ B.955 4-CN-furan-2-yl-CH = C (CH ₃₎ B.956 _{4-CH3-furan-2-yl-CH} = C (CH ₃₎ B.957 5-Br-furan-2-yl-CH = C (CH ₃₎ B.958 5-Cl-furan-2-yl-CH = C (CH ₃₎ B.959 5-CN-furan-2-yl-CH = C (CH ₃₎ B.960 _{5-CH3-furan-2-yl-CH} = C (CH ₃₎ B.961 furan-3-yl-CH = C (CH ₃₎ B.962 5-Br-furan-3-yl-CH = C (CH ₃₎ B.963 5-Cl-furan-3-yl-CH = C (CH ₃₎ B.964 5-CN-furan-3-yl-CH = C (CH ₃₎ B.965 5-CH ₃ -furan-3-yl-CH = C (CH ₃ ); B.966 thien-2-yl-CH = C (CH ₃₎ B.967 4-Br-thien-2-yl-CH = C (CH ₃₎ B.968 4-Cl-thien-2-yl-CH = C (CH ₃₎ B.969 4-CN-thien-2-yl-CH = C (CH ₃₎ B.970 4-CH ₃ -thien-2-yl-CH = C (CH ₃ ) B.971 5-Br-thien-2-yl-CH = C (CH ₃₎ B.972 5-Cl-thien-2-yl-CH = C (CH ₃₎

Nr. R ³ B.973 5-CN-thien-2-yl-CH = C (CH ₃₎ B.974 5-CH ₃ -thien-2-yl-CH = C (CH ₃ ) ₅ B.975 thien-3-yľCH = C (CH ₃₎ B.976 5-Br-thien-3-yľCH = C (CH ₃₎ B.977 5-Cľthien-3-yľCH = C (CH ₃₎ B.978 5-CN-thien-3-yľCH = C (CH ₃₎ B.979 J 5-CH ₃ -thien-3-ylCH = C (CH ₃ ) B.980 oxazol-2-yľCH = C (CH ₃₎ B.981 4-Br-oxazol-2-ylCH = C (CH ₃ ) B.982 4-Cl-oxazol-2-yl-CH = C _<CH3) B.983 4-CN-oxazol-2-ylCH = C (CH ₃ ) B.984 _{4-CH3-oxazol-2-yl-CH} = C (CH ₃₎ B.985 5-Br-oxazol-2-ylCH = C (CH ₃ ) B.986 5-Cl-oxazol-2-ylCH = C (CH ₃ ) B.987 5-CN-oxazol-2-yl-CH = C (CH ₃₎ B.988 _{5-CH3-oxazol-2-yl-CH} = C (CH ₃₎ B.989 Oxazol-4-yl-CH = C (CH ₃₎ B.990 2-Br-oxazo1-4-yl-CH = C (CH ₃₎ B.991 2-Cl-oxazol-4-ylCH = C (CH ₃ ) B.992 2-CN-oxazol-4-ylCH = C (CH ₃ ) B.993 2-CH ₃ -oxazol-4-ylCH = C (CH ₃ ) B.994 2 -C 8 H -oxazol-4-yl-CH = C (CH ₃ ) B.995 5-Br-oxazol-4-yl-CH = C (CH ₃₎ B.996 5-Cľoxazol-4-yl-CH = C (CH ₃₎ B.997 5-CN-oxazol-4-yl-CH = C (CH ₃₎ B.998 5-CH ₃ -oxazol-4-yl-CH = C (CH ₃ ) B.999 oxazol-5-yl-CH = C (CH ₃₎ B.lOOO 4-Br-oxazol-5-yl-CH = C (CH ₃₎ B.1001 4-C 1 -oxazol-5-yl-CH = C (CH ₃ ) B.1002 4-CN-oxazol-5-yl-CH = C (CH ₃₎ B.1003 4-CH ₃ -oxazol-5-ylCH = C (CH ₃ ) B.1004 2-Br-oxazol-5-yl-CH = C (CH ₃₎ B.1005 2-Cl-oxazol-5-yl-CH = C (CH ₃₎ B.1006 2-CN-oxazol-5-yl-CH = C (CH ₃₎ B.1007 _{2-CH3-oxazol-5-yl-CH} = C (CH ₃₎ B.1008 isoxazol-3-yl-CH = C (CH ₃₎ B.1009 4-Br-isoxazol-3-yl-CH = C (CH ₃₎ B.1010 4-Cl-isoxazol-3-yl-CH = C (CH ₃₎ B.1011 4-CN-isoxazol-3-yl-CH = C (CH ₃₎

5 0 5 0 Nr. R ³ B.1012 4-CH 3 -isoxazol-3-yl-CH = C (CH ₃ ) B.1013 5-Br-isoxazol-3-yl-CH = C (CH ₃₎ B.1014 5-Cl-isoxazol-3-yl-CH = C (CH ₃₎ B.1015 5-CN-isoxazol-3-yl-CH = C (CH ₃₎ B.1016 5-CH ₃ -isoxazol-3-yl-CH = C (CH ₃ ) B.1017 isoxazol-4-yl-CH = C (CH ₃₎ B.1018 3-Br-isoxazol-4-yl-CH = C (CH ₃₎ B.1019 3-Cl-isoxazol-4-yl-CH = C (CH ₃₎ B.1020 3-CN-isoxazol-4-yl-CH = C (CH ₃₎ B.1021 3-CH ₃ -isoxazol-4-yl-CH = C (CH ₃ ) B.1022 5-Br-isoxazol-4-yl-CH = C (CH ₃₎ B.1023 5-Cl-isoxazol-4-yl-CH = C (CH _3); B.1024 5-CN-isoxazol-4-yl-CH = C (CH ₃ ) δ B.1025 5-CH ₃ -isoxazol-4-yl-CH = C (CH ₃ ) | B.1026 3,5- (CH ₃ ) ₂ 'isoxazol-4-yl-CH = C (CH ₃ ) 1 B.1027 isoxazol-5-yl-CH = C (CH ₃ ) 1 B.1028 3-Br-isoxazol-5-yl-CH = C (CH ₃ ) i B.1029 3-Cl-isoxazol-5-yl-CH = C (CH ₃₎ B.1030 3-CN-isoxazol-5-yl-CH = C (CH ₃₎ B.1031 3-CH ₃ -isoxazol-5-yl-CH = C (CH ₃ ) B.1032 3-C ₆ H 5-isoxazol-5-yl-CH = C (CH ₃₎ B.1033 4-Cl-C 6 H 3-isoxazol-5-yl-CH = C (CH ₃₎ B.1034 4-Br, 3-C 6 H 5 -isoxazol-5-yl-CH = C (CH ₃ ) B.1035 4-Br-isoxazol-5-yl-CH = C (CH ₃₎ B.1036 4-Cl-isoxazol-5-yl-CH = C (CH ₃₎ B.1037 4-CN-isoxazol-5-yl-CH = C (CH ₃₎ B.1038 4-CH ₃ -isoxazol-5-yl-CH = C (CH ₃ ) B.1039 thiazol-2-yl-CH = C (CH ₃₎ B.1040 4-Br-thiazol-2-yl-CH = C (CH ₃₎ B.1041 4-Cl-thiazol-2-yl-CH = C (CH ₃₎ B.1042 4-CN-thiazol-2-yl-CH = C (CH ₃₎ B.1043 4-CH ₃ -thiazol-2-yl-CH = C (CH ₃ ) B.1044 5-Br-thiazol-2-yl-CH = C (CH ₃₎ B.1045 5-Cl-thiazol-2-yl-CH = C (CH ₃₎ B.1046 5-CN-thiazol-2-yl-CH = C (CH ₃₎ B.1047 5-CH ₃ -thiazol-2-yl-CH = C (CH ₃ ) B.1048 thiazol-4-yl-CH = C (CH ₃₎ B.1049 2-Br-thiazol-4-yl-CH = C (CH ₃₎ B.1050 2-Cl-thiazol-4-yl-CH = C (CH ₃₎

Nr. R ³ B.1051 2-CN-thiazol-4-yl-CH = C (CH ₃₎ B.1052 2-CH ₃ -thiazol-4-yl-CH = C (CH ₃ ) ₅ B.1053 5-Br-thiazol-4-yl-CH = C (CH ₃₎ • B.1054 5-Cl-thiazol-4-yl-CH = C (CH ₃₎ B.1055 5-CN-thiazol-4-yl-CH = C (CH ₃₎ B.1056 5-CH ₃ -thiazol-4-yl-CH = C (CH ₃ ) B.1057 J thiazol-5-yl-CH = C (CH ₃₎ B.1058 4-Br-thiazol-5-yl-CH = C (CH ₃₎ B.1059 4-Cl-thiazol-5-yl-CH = C (CH ₃₎ B.1060 4-CN-thiazol-5-yl-CH = C (CH ₃₎ B.1061 4-CH ₃ -thiazol-5-yl-CH = C (CH ₃ ) B.1062 2-Br-thiazol-5-yl-CH = C (CH ₃₎ B.1063 2-Cl-thiazol-5-yl-CH = C (CH ₃₎ B.1064 2-CN-thiazol-5-yl-CH = C (CH ₃₎ B.1065 2-CH ₃ -thiazol-5-yl-CH = C (CH ₃ ) B.1066 isothiazol-3-yl-CH = C (CH ₃₎ B.1067 4-Br-isothiazol-3-yl-CH = C (CH ₃₎ B.1068 4-Cl-isothiazol-3-yl-CH = C (CH ₃₎ B.1069 4-CN-isothiazol-3-yl-CH = C (CH ₃₎ B.1070 4-CH ₃ -isothiazol-3-yl-CH = C (CH ₃ ) B.1071 5-Br-isothiazol-3-yl-CH = C (CH ₃₎ B.1072 5-Cl-isothiazol-3-yl-CH = C (CH ₃₎ B.1073 5-CN-isothiazol-3-yl-CH = C (CH ₃₎ B.1074 5-CH ₃ -isothiazol-3-yl-CH = C (CH ₃ ) B.1075 isothiazol-4-yl-CH = C (CH ₃₎ B.1076 3-Br-isothiazol-4-yl-CH = C (CH ₃₎ B.1077 3-Cl-isothiazol-4-yl-CH = C (CH ₃₎ B.1078 3-CN-isothiazol-4-yl-CH = C (CH ₃₎ B.1079 3-CH ₃ -isothiazol-4-yl-CH = C (CH ₃ ) B.1080 5-Br-isothiazol-4-yl-CH = C (CH ₃₎ B.1081 5-Cl-isothiazol-4-yl-CH = C (CH ₃₎ B.1082 5-CN-isothiazol-4-yl-CH = C (CH _3; B.1083 5-CH ₃ -isothiazol-4-yl-CH = C (CH ₃ ) B.1084 3,5- (CH ₃ ) ₂ -isothiazol-4-yl-CH = C (CH ₃ ) B.1085 Isothiazol-5-yl-CH = C (CH ₃ ) B.1086 3-Br-isothiazol-5-yl-CH = C (CH ₃₎ B.1087 i-Cl-isothiazol-5-yl-CH = C (CH ₃₎ B.1088; and-CN-isothiazol-5-yl-CH = C (CH ₃₎ B.1089: $ -CH ₃ -isothiazol-5-yl-CH = C (CH ₃ )

-2 <3 ο-

5 0 5 3 Nr. R ³ B.1090 4-Br-isothiazol-5-yl-CH = C (CH ₃₎ B.1091 4-Cl-isothiazol-5-yl-CH = C (CH ₃₎ B.1092 4-CN-isothiazol-5-yl-CH = C (CH ₃ ) i B.1093 4-CH ₃ -isothiazol-5-yl-CH = C (CH ₃ ) B.1094 imidazol-2-yl-CH = C (CH ₃ ) B.1095 l-Cl-imidazol-2-yl-CH = C (CH ₃₎ B.1096 l-Br-imidazol-2-yl-CH = C (CH ₃₎ B.1097 L-CN-imidazol-2-yl-CH = C (CH ₃₎ B.1098 1-CH ₃ -imidazol-2-yl-CH = C (CH ₃ ) B.1099 4-Cl-imidazol-2-yl-CH = C (CH ₃₎ B.1100 4-Br-imidazol-2-yl-CH = C (CH ₃₎ B.1101 4-CN-imidazol-2-yl-CH = C (CH ₃₎ B.1102 4-CH ₃ -imidazol-2-yl-CH = C (CH ₃ ) B.1103 1-CH _3,5 -imidazol-2-yl-CH = C (CH ₃ ) B.1104 1,4- (CH ₃ ) ₂ -imidazol-2-yl-CH = C (CH ₃ ) B.1105 1,5- (CH ₃ ) ₂ -imidazol-2-yl-CH = C (CH ₃ ) B.1106 imidazol-4-yl-CH = C (CH ₃₎ B.1107 2-Cl-imidazol-4-yl-CH = C (CH ₃₎ B.1108 2-Br-imidazol-4-yl-CH = C (CH ₃₎ B.1109 2-CN-imidazol-4-yl-CH = C (CH ₃₎ B.1110 1-CH ₃ -imidazol-4-yl-CH = C (CH ₃ ) B.llll 2-CH ₃ -imidazol-4-yl-CH = C (CH ₃ ) B.1112 5-Cl-imidazol-4-yl-CH = C (CH ₃₎ B.1113 5-Br-imidazol-4-yl-CH = C (CH ₃₎ B.1114 5-CN-imidazol-4-yl-CH = C (CH ₃₎ B.1115 5-CH ₃ -imidazol-4-yl-CH = C (CH ₃ ) B.1116 _1-CH3, 5-Cl-imidazol-4-yl-CH = C (CH ₃₎ B.1117 1,2- (CH ₃ ) ₂ -imidazol-4-yl-CH = C (CH ₃ ) B.1118 1,5- (CH ₃ ) ₂ -imidazol-4-yl-CH = C (CH ₃ ) B.1119 pyrazol-3-yl-CH = C (CH ₃₎ B.1120 5-Br-pyrazol-3-yl-CH = C (CH ₃₎ B.1121 5-Cl-pyrazol-3-yl-CH = C (CH ₃₎ B.1122 5-CN-pyrazol-3-yl-CH = C (CH ₃₎ B.1123 5-CH ₃ -pyrazol-3-yl-CH = C (CH ₃ ) B.1124 L-C 6 H ₅ -pyrazol-3-yl-CH = C (CH ₃ ) B.1125 and-Br-pyrazol-3-yl-CH = C (CH ₃₎ B.1126 l-Cl-pyrazol-3-yl-CH = C (CH ₃₎ B.1127 L-CN-pyrazol-3-yl-CH = C (CH ₃₎ B.1128 i 1-CH ₃ -pyrazol-3-yl-CH = C (CH ₃ )

Nr. R ³ B.1129 1-CH 3 -pyrazol-3-yl-CH = C (CH ₃ ) B.1130 1,4- (CH ₃ ) ₂ -pyrazol-3-yl-CH = C (CH ₃ ) B.1131 1,5- (CH ₃ ) ₂ -pyrazol-3-yl-CH = C (CH ₃ ) B.1132 _1-CH3, 4-Cl-pyrazol-3-yl-CH = C (CH ₃₎ B.1133 _1-CH3, 5-Cl-pyrazol-3-yl-CH = C (CH ₃₎ B.1134 pyrazol-4-yl-CH = C (CH ₃₎ B.1135 3-Br-pyrazol-4-yl-CH = C (CH ₃₎ B.1136 3-Cl-pyrazol-4-yl-CH = C (CH ₃₎ B.1137 3-CN-pyrazol-4-yl-CH = C (CH ₃₎ B.1138 3-CH ₃ -pyrazol-4-yl-CH = C (CH ₃ ) B.1139 1-CH ₃ -pyrazol-4-yl-CH = C (CH ₃ ) B.1140 1,5- (CH ₃ ) ₂ -pyrazol-4-yl-CH = C (CH ₃ ) B.1141 1,3- (CH ₃ ) ₂ -pyrazol-4-yl-CH = C (CH ₃ ) B.1142 1-CH _{3 R} 3-Cl-pyrazol-4-yl-CH = C (CH ₃₎ B.1143 1-CH ₃ , 5-Cl-pyrazol-4-yl-CH = C (CH ₃ ) B.1144 pyrazol-5-yl-CH = C (CH ₃₎ B.1145 3-Br-pyrazol-5-yl-CH = C (CH ₃₎ B.1146 3-Cl-pyrazol-5-yl-CH = C (CH ₃₎ B.1147 3-CN-pyrazol-5-yl-CH = C (CH ₃₎ B.1148 3 -CH ₃ -pyrazol-5-yl-CH = C (CH ₃ ) B.1149 1-CH ₃ -pyrazol-5-yl-CH = C (CH ₃ ) B.1150 4-Br-pyrazol-5-yl-CH = C (CH ₃₎ B.1151 4-Cl-pyrazol-5-yl-CH = C (CH ₃₎ B.1152 4-CN-pyrazol '5-yl-CH = C (CH ₃₎ B.1153 4-CH ₃ -pyrazol-5-yl-CH = C (CH ₃ ) B.1154 1,3- (CH ₃ ) ₂ -pyrazol-5-yl-CH = C (CH ₃ ) B.1155 1,4- (CH ₃ ) ₂ -pyrazol-5-yl-CH = C (CH ₃ ) B.1156 1-CH ₃ , 3-Cl-pyrazol-5-yl-CH = C (CH ₃ ) B.1157 _1-CH3, 4-Cl-pyrazol-5-yl-CH = C (CH ₃₎ B.1158 1,3,4-oxadiazol-5-yl-CH = C (CH ₃₎ B.1159 2-CH 3 -1,3,4-oxadiazol-5-yl-CH = C (CH ₃ ) B.1160 2-CF ₃ -1,3,4-oxadiazol-5-yl-CH = C (CH ₃ ) B.1161 2-OCH 3 -1,3,4-oxadiazol-5-yl-CH = C (CH ₃ ) B.1162 2-C1-1,3,4-oxadiazol-5-yl-CH = C (CH ₃₎ B.1163 2-CH (CH ₃ ) ₂ -1,3,4-oxadiazol-5-yl-CH = C (CH ₃ ) B.1164 1,3,4-oxadiazol-2-yl-CH = C (CH ₃₎ B.1165 5-CH ₃ -1,3,4-oxadiazol-2-yl-CH = C (CH ₃ ) B.1166 5-CF ₃ -1,3,4-oxadiazol-2-yl-CH = C (CH ₃ ) B.1167 5-OCH ₃ -1,3,4-oxadiazol-2-yl-CH = C (CH ₃ )

Nr. R ³ B.1168 5-C1-1,3,4-oxadiazol-2-yl-CH = C (CH ₃₎ B.1169 5-CH (CH ₃ ) 2 -1,4,4-oxadiazol-2-yl-CH = C (CH ₃ ) ₅ B.1170 5-C6H5-I, 3,4-oxadiazol-2-yl-CH = C (CH ₃₎ B.1171 1,2,4-oxadiazol-3-yl-CH = C (CH ₃₎ B.1172 5-CH ₃ -1,2,4-oxadiazol-3-yl-CH = C (CH ₃ ) B.1173 5-CF ₃ -1,2,4-oxadiazol-3-yl-CH = C (CH ₃ ) B.1174 5-C1-1.2,4-oxadiazol-3-yl-CH = C (CH ₃₎ B.1175 5-CH (CH ₃ ) 2-1,2,4-oxadiazol-3-yl-CH = C (CH ₃ ) B.1176 1,2,4-triazol-3-yl-CH = C (CH ₃₎ B.1177 1-CH ₃ -1,2,4-triazol-3-yl-CH = C (CH ₃ ) B.1178 5-CH ₃ -1,2,4-triazol-3-yl-CH = C (CH ₃ ) > B.1179 5-CF ₃ -1,2,4-triazol-3-yl-CH = C (CH ₃ ) B.1180 5-OCH ₃ -1,2,4-triazol-3-yl-CH = C (CH ₃ ) B.1181 5-Cl-l, 2,4-triazol-3-yl-CH = C (CH ₃₎ B.1182 5-CH _(CH3) 2-1,2,4-trxazol-3-yl-CH = C (CH ₃₎ B.1183 1-C ₆ H ₅ -1,2,4-triazol-3-yl-CH = C (CH ₃ ) B.1184 1,3,4-thiadiazol-5-yl-CH = C (CH ₃₎ B.1185 2-CH ₃ -1,3,4-thiadiazol-5-yl-CH = C (CH ₃ ) B.1186 2-CF ₃ -1,3,4-thiadxazol-5-yl-CH = C (CH ₃ ) B.1187 2-OCH 3 -1,3,4-thiadiazol-5-yl-CH = C (CH ₃ ) B.1188 2-Cl-l, 3,4-thiadiazol-5-yl-CH = C (CH ₃₎ B.1189 2-CH _(CH3) 2-1,3,4-thiadiazol-5-yl-CH = C (CH ₃₎ B.1190 1,3,4-thiadiazol-2-yl-CH = C (CH ₃₎ B.1191 5-CH ₃ -1,3,4-thxadxazol-2-yl-CH = C (CH ₃ ) B.1192 5-CF 3 -1,3,4-thiadiazol-2-yl-CH = C (CH ₃ ) B.1193 5-OCH ₃ -1,3,4-thiadxazol-2-yl-CH = C (CH ₃ ) B.1194 5-C1-1,3,4-thiadiazol-2-yl-CH = C (CH ₃₎ B.1195 5-CH _(CH3) 2-1,3,4-thiadiazol-2-yl-CH = C (CH ₃₎ B.1196 5-C6H5-I, 3,4-thiadiazol-2-yl-CH = C (CH ₃₎ B.1197 1,2,4-thiadxazol-3-yl-CH = C (CH ₃₎ B.1198 5-CH ₃ -1,2,4-thiadiazol-3-yl-CH = C (CH ₃ ) B.1199 5-CF 3 -1,2,4-thiadiazol-3-yl-CH = C (CH ₃ ) B.1200 5-OCH ₃ -1,2,4-thiadiazol-3-yl-CH = C (CH ₃ ) B.1201 5-C1-1,2,4-thiadiazol-3-yl-CH = C (CH ₃₎ B.1202 5-CH _(CH3) 2-1,2,4-thiadiazol-3-yl-CH = C (CH ₃₎ B.1203 R yrrol-2-yl-CH = C (CH ₃ ) B.1204 J-C-pyrro1-2-yl-CH = C (CH ₃₎ B.1205 l-Br-pyrrol-2-yl-CH = C (CH ₃₎ B.1206 1-CH ₃ -pyrrol-2-yl-CH = C (CH ₃ )

'213-

Nr. R ³ B.1207 4-C6H5-pyrrol-2-yľCH = C (CH ₃₎ B.1208 benzimidazol-2-yl-CH = C (CH _{3) 5} B.1209 quinolin-2-y 1 CH = C (CH ₃ ) B.1210 C = CH B.1211 ch ₂ c = ch B.1212 ch ₂ cscci B.1213 • CH ₂ C = CBr B.1214 ch ₂ c = ci B.1215 ch ₂ cscch ₃ B.1216 ch ₂ c ^ cch ₂ ch ₃ B.1217 ch ₂ c = cch ₂ oh B.1218 CH ₂ CSCH ₂ NH ₂ B.1219 ch ₂ c = cch ₂ ci B.1220 CH ₂ Cs = CCH ₂ OCH ₃ B.1221 ch ₂ c = cch ₂ and ₂ ch ₃ B.1222 ch ₂ c = cch ₂ sch ₃ B.1223 CH ₂ CSCH ₂ N (CH ₃ ) ₂ B.1224 ch ₂ c = cc ₆ h ₅ B.1225 ch ₂ ch ₂ c = ch B.1226 CH ₂ CH ₂ CSCC 1 B.1227 CH ₂ CH ₂ C = CBr B.1228 ch ₂ ch ₂ c = ci B.1229 CH ₂ CH ₂ CSCCH ₃ B.1230 ch ₂ ch ₂ c = cch ₂ ch ₃ B.1231 CH ₂ CH ₂ CBCCH ₂ OH B.1232 CH ₂ CH ₂ Cs = CCH ₂ NH ₂ B.1233 CH ₂ CH ₂ C = CCH ₂ C B.1234 ch ₂ ch ₂ c = cch ₂ and ₃ B.1235 ch ₂ ch ₂ c S cch ₂ and ₂ ch ₃ B.1236 CH ₂ CH ₂ CsCCH ₂ SCH ₃ B.1237 ch ₂ ch ₂ c = c ₂ n (ch ₃ ) 2 B.1238 CH ₂ CH ₂ C = CC ₆ H ₅ B.1239 CH ₂ CH ₂ CH ₂ Cs = CH B.1240 ZH ₂ CH ₂ CH ₂ CsCl 1 B.1241 CH ₂ CH ₂ CH ₂ C = CBr B.1242 ( h ₂ ch ₂ ch ₂ c = ci B.1243 ( h ₂ ch ₂ ch ₂ c = cch ₃ B.1244 C : h ₂ ch ₂ ch ₂ en cch ₂ ch ₃ B.1245 C h ₂ ch ₂ ch ₂ c = cch ₂ oh

-L FR-

Nr. R ³ B.1246 CH ₂ CH ₂ CH ₂ C = CCH ₂ NH ₂ B.1247 CH ₂ CH ₂ CH ₂ C = CCH ₂ Cl B.1248 CH ₂ CH ₂ CH ₂ C = CCH ₂ OCH ₃ B.1249 CH ₂ CH ₂ CH ₂ C with CCH ₂ OCH ₂ CH ₃ B.1250 CH ₂ CH ₂ CH ₂ C Ξ cch ₂ sch ₃ B.1251 ch ₂ ch ₂ ch ₂ c S cch ₂ n (CH ₃ ) 2 B.1252 CH ₂ CH ₂ CH ₂ CSCC ₆ H ₅ B.1253 CH _(CH3) C-CH B.1254 CH _(CH3) C = cci B.1255 CH (CH ₃ ) C = CBr B.1256 CH (CH ₃ ) C = Cl B.1257 CH (CH ₃ ) C = CCH ₃ B.1258 CH (CH _{3) 2} CH ₃ CSCCH B.1259 CH _{(CH3) 2} OH CSCCH B.1260 CH (CH ₃ ) C = CCH ₂ NH ₂ B.1261 CH (CH _{3) 2} C 1 CSCCH B.1262 CH (CH ₃ ) C = CCH ₂ OCH ₃ B.1263 CH (CH ₃ ) C = CCH ₂ OCH ₂ CH ₃ B.1264 CH (CH ₃ ) c = cch ₂ sch ₃ B.1265 CH _(CH3) E CCH ₂ N (CH ₃₎ 2 B.1266 CH (CH ₃ ) CSCC ₆ H ₅ B.1267 ch = ch-c ₆ h ₅ B.1268 C (CH ₃ ) = ch-c ₆ h ₅ B.1269 CSCC ₆ H ₅

Nr. R ³ B.1270 1,3- (CH ₃ ) 2 -pyrazol-5-yl-CH 2 B.1271 1,4- _{(CH3) 2-pyrazol-5-yl-CH2} B.1272 1-CH ₃ , 3-Cl-pyrazol-5-yl-CH ₂ B.1273 1-CH ₃ , 4-Cl-pyrazol-5-yl-CH ₂ B.1274 _{1,3,4-oxadiazol-5-yl-CH2} B.1275 2-CH ₃ -1,3,4-oxadiazol-5-yl-CH ₂ B.1276 2-CF ₃ -1,3,4-oxadiazol-5-yl-CH ₂ B.1277 2-OCH ₃ -1,3,4-oxadiazol-5-yl-CH ₂ B.1278 _{2-C1-1,3,4-oxadiazol-5-yl-CH2} B.1279 2-CH (CH ₃ ) ₂ -1,3,4-oxadiazol-5-yl-CH ₂ B.1280 1, _{3,4-oxadiazol-2-yl-CH2} B.1281 5-CH ₃ -1,3,4-oxadiazol-2-yl-CH ₂ B.1282 5-CF ₃ -1,3,4-oxadiazol-2-yl-CH ₂ B.1283 5-OCH ₃ -1,3,4-oxadiazol-2-yl-CH ₂ B.1284 _{5-C1-1,3,4-oxadiazol-2-yl-CH2} B.1285 5-CH (CH ₃ ) ₂ -1,3,4-oxadiazol-2-yl-CH ₂ B.1286 5-C6H5-I, _{3,4-oxadiazol-2-yl-CH2} B.1287 _{1,2,4-oxadiazol-3-yl-CH2} B.1288 5-CH 3 -1,2,4-oxadiazol-3-yl-CH ₂ B.1289 5-CF ₃ -1,2,4-oxadiazol-3-yl-CH ₂ B.1290 5-OCH ₃ -1,2,4-oxadiazol-3-yl-CH ₂ B.1291 _{5-C1-1,2,4-oxadiazol-3-yl-CH2} B.1292 5-CH (CH ₃ ) ₂ -1,2,4-oxadiazol-3-yl-CH ₂ B.1293 _{1,2,4-triazol-3-yl-CH2} B.1294 1-CH ₃ -1,2,4-triazol-3-yl-CH ₂ B.1295 5-CH ₃ -1,2,4-triazol-3-yl-CH ₂ B.1296 5-CF ₃ -1,2,4-triazol-3-yl-CH ₂ B.1297 5-OCH ₃ -1,2,4-triazol-3-yl-CH ₂ B.1298 _{5-C1-1,2,4-triazol-3-yl-CH2} B.1299 5-CH (CH ₃ ) ₂ -1,2,4-triazol-3-yl-CH ₂ B.1300 I-C6H5-I, _{'2,4-triazol-3-yl-CH2} B.1301 _{1,3,4-thiadiazol-5-yl-CH2} B.1302 2-CH ₃ -1,3,4-thiadiazol-5-yl-CH ₂ B.1303 2-CF ₃ -1,3,4-thiadiazol-5-yl-CH ₂ B.1304 2-OCH ₃ -1,3,4-thiadiazol-5-yl-CH ₂ B.1305 2-CH ₂ OCH ₃ -1,3,4-thiadiazol-5-yl-CH ₂ B.1306 _{2-C1-1,3,4-fchiadiazol-5-yl-CH2} B.1307 2-CH (CH ₃ ) ₂ -1,3,4-thiadiazol-5-yl-CH ₂

Nr.

R ³

B.1308

B.1309

B.1310

B.1311

B.1312

B.1313

B.1314

B.1315

_{-tyé1,3,4-thiadiazol-2-yl-CH2}

5-CH 3 -1,3,4-thiadiazol-2-ylCH ₂

5-CF 3 -1,3,4-thiadiazol- ₂ -ylCH ₂

5-OCH 3 -1,3,4-thiadiazol-2-ylCH 2

5-Cl, 3,4-thiadiazol- ₂ -yl-CH2

5-CH (CH ₃ ) ₂ -1. _{3,4-thiadiazol-2-yl-CH2}

5-C6H5-1,3,4-thiadiazol- ₂ -yl-CH2

1,2,4-thiadiazol-3-ylCH ₂

B.1316

5-CH ₃ -1,2,4-thiadiazol-3-yl-CH ₂

B.1317

5-CF ₃ -1,2,4-thiadiazol-3-ylCH ₂

B.1318

5-OCH ₃ -1,2,4-thiadiazol-3-ylCH ₂

B.1319

5-Cl 1, 2,4-thiadiazol-3-yl CH ₂

B.1320

5-CH (CH ₃ ) ₂ -1,2,4-thiadiazol-3-yl-CH ₂

B.1321

B.1322

B.1323

B.1324 _{pyrrol-2-yl-CH2}

4-C1-pyrrol- ₂ -yl-CH2

_{4-Br-pyrrol-2-y1-CH2 -CH3} roll pyrid - 2 yl 1 _CH2

B.1325

-C6H5-pyrrolidin - 2-yl 1 _CH2

B.1326

B.1327

B.1328

B.1329

B.1330

B.1331

B.1332 benzimidazol-2-yl-CH ₂ quinolin-2-yl-CH ₂ oxiranyl-CH ₂

_{2-CH3-oxiran-2} yľCH ₂

2-CH ₃ -oxiran-3-yl-CH ₂

2,2- (CH ₃ ) ₂ -oxiran-3-yl-CH ₂

2,3- (CH ₃ ) ₂ -oxiran-3-yl-CH ₂

B.1333

2,3,3- (CH ₃ ) ₃ -oxiran-2-yl-CH ₂

B.1334

B.1335

B.1336

B.1337

B.1338

B.1339

B.1340

B.1341

B.1342

B.1343

B.1344

B.1345

B.1346 oxiranyl-CH (CH ₃₎

_{2-CH3-oxiran-2-yl-CH (CH3)}

2-CH ₃ -oxiran-3-ylCH (CH ₃ )

2,2- _{(CH3) 2-oxiran-3-yl-CH (CH3)}

2,3- _{(CH3) 2-oxiran-3-yl-CH (CH3)}

2,3,3- _{(CH3) 3} oxirane-2-yl-CH _(CH3)

1,1-Cl ₂ -cyclopropan-2-yl-CH ₂

2-CH ₃ , 1,1-Cl ₂ -cyclopropan-2-yl-CH ₂

2-CH ₃ , 1,1-Cl ₂ -cyclopropan-3-yl-CH ₂

2,2- _{(CH3) 2,} 1, _{l-Cl2 -cyclopropan-3-yl-CH2}

2,3- _{(CH3) 2,} 1, _{l-Cl2 -cyclopropan-3-yl-CH2}

2,3,3- _{(CH3) 3,} 1, _{l-Cl2 -cyclopropan-2-yl-CH2}

1, _l-Cl2 -cyclopropan-2-yl-CH _(CH3)

Nr. R ³ B.1347 2-CH _3, 1, ₂ LCL -cyclopropan-2-yľCH (CH ₃₎ B.1348 2-CH 3, 1,1'Cl ₂ -cyclopropan-3-yl-CH (CH ₃ ) B.1349 2,2- _{(CH3) 2,} 1, _l-Cl2 -cyclopropan-3-yl-CH _(CH3) B.1350 2,3- _{(CH3) 2,} 1, l-Cl2-cyclopropan ~ 3-yl-CH _(CH3) B.1351 2,3,3- (CH ₃ ) 3,1,1-Cl ₂ -cyclopropan-2-yl-CH (CH ₃ ) B.1352 1,1-Br ₂ -cyclopropan-2-yl-CH ₂ B.1353 2-CH 3, 1,1-Br ₂ -cyclopropan-2-yl-CH ₂ B.1354 2-CH 3, 1,1-Br ₂ -cyclopropan-3-yl-CH ₂ B.1355 2,2- _{(CH3) 2,} 1, _{l-Br2 -cyclopropan-3-yl-CH2} B.1356 2,3- _{(CH3) 2,} 1, _{l-Br2 -cyclopropan-3-yl-CH2} B.1357 2,3,3- (CH 3) 3,1,1-Br ₂ -cyclopropan-2-yl-CH 2 B.1358 1, _l-Br2 -cyclopropan-2-yl-CH _(CH3) B.1359 2-CH 3, 1,1-Br ₂ -cyclopropan-2-yl-CH (CH ₃ ) B.1360 2-CH _3, 1, _l-Br2 -cyclopropan-3-yl-CH _(CH3) B.1361 2,2- _{(CH3) 2,} 1, _l-Br2 -cyclopropan-3-yl-CH _(CH3) B.1362 2,3- _{(CH3) 2,} 1, _l-Br2 -cyclopropan-3-yl-CH _(CH3) B.1363 2,3,3- _{(CH3) 3,} 1, _l-Br2 -cyclopropan-2-yl-CH _(CH3) B.1364 CH _(CH3) -O-phenyl B.1365 CH (CH ₃ ) CH ₂ -O-pheny1 B.1366 CH ₂ CH (CH ₃ ) -O-pheny 1 B.1367 CH _(CH3) CH _(CH3) -O-phenyl B.1368 CH (CH ₃ ) (CH ₂ ) 2 -O-phenyl B.1369 CH ₂ CH (CH ₃ ) CH ₂ -O-pheny 1 B.1370 (CH ₂ ) ₂ CH (CH ₃ ) -O-phenyl 1 B.1371 CH (CH ₃ ) CH (CH ₃ ) CH ₂ -O-phenyl 1 B.1372 CH (CH ₃ ) CH ₂ CH (CH ₃ ) -O-phenyl 1 B.1373 CH ₂ CH (CH ₃ ) CH (CH ₃ ) -O-phenyl B.1374 CH (CH ₃ ) CH (CH ₃ ) CH (CH ₃ ) -O-phenyl 1 B.1375 CH _{(CH3) (CH2) 3-O-phenyl} B.1376 2-FC ₆ H ₄ -CH ₂ B.1377 3-FC ₆ H ₄ -CH ₂ B.1378 4-FC ₆ H ₄ -OCH ₂ B.1379 2,3-F ₂ -C ₆ H ₃ -OCH ₂ B.1380 2,4-F ₂ -C ₆ H ₃ -OCH ₂ B.1381 2,5-F ₂ -C ₆ H ₃ -OCH ₂ B.1382 2,6-F ₂ -C ₆ H ₃ -OCH ₂ B.1383 3,4-F ₂ -C ₆ H ₃ -OCH ₂ B.1384 3,5-F ₂ -C ₆ H ₃ -OCH ₂ B.1385 2-Cl-C ₆ H ₄ OCH ₂

- 7W-

Nr. R ³ B.1386 3-Cl-C ₆ H ₄ OCH ₂ B.1387 4-Cl-C ₆ H 4 OCH _{2 5} B.1388 2,3-Cl ₂ -C ₈ H ₃ -OCH ₂ B.1389 2,4-Cl ₂ -C ₆ H ₃ -OCH ₂ B.1390 2,5-Cl ₂ -C ₆ H ₃ -OCH ₂ B.1391 2,6-Cl ₂ -C ₆ H ₃ -OCH ₂ B.1392 3 3,4-Cl ₂ -C ₆ H ₃ -OCH ₂ B.1393 3,5-Cl ₂ -C ₆ H ₃ -OCH ₂ B.1394 2,3,4-Cl ₃ -C ₆ H ₂ -OCH ₂ B.1395 2,3,5-Cl ₃ -C ₆ H ₂ -OCH ₂ B.1396 2.3,6-Cl ₃ -C ₆ H ₂ -OCH ₂ > B.1397 2,4,5-Cl ₃ -C ₆ H ₂ -OCH ₂ B.1398 2,4,6-Cl ₃ -C ₆ H ₂ -OCH ₂ B.1399 3,4,5-C ₃ -C _e H ₂ OCH ₂ B.1400 2-Br-C ₆ H ₄ -OCH ₂ B.1401 3-Br-C ₆ H ₄ -OCH ₂ B.1402 4-Br-C ₆ H ₄ -OCH ₂ B.1403 2,3-Br ₂ -C ₆ H ₃ -O-CH ₂ B.1404 2,4-Br ₂ -C ₆ H ₃ -O-CH ₂ B.1405 2.5 ^ -0 ^ 3-0-0¾ B.1406 2,6-Br ₂ -C ₆ H ₃ -O-CH ₂ B.1407 3,4-Br ₂ -C ₆ H ₃ -O-CH ₂ B.1408 3,5-Br ₂ -C ₆ H ₃ -O-CH ₂ B.1409 2-F, 3-Cl-C ₆ H ₃ -CH ₂ -O B.1410 2-F, 4-Cl-C ₆ H ₃ -CH ₂ -O B.1411 2-F, 5-Cl-C ₆ H ₃ -CH ₂ -O B.1412 2-F, 3-Br-C ₆ H ₃ -CH ₂ -O B.1413 2-F, 4-Br-C ₆ H ₃ -CH ₂ -O B.1414 2-F, 5-Br-C ₆ H ₃ -CH ₂ -O B.1415 2-Cl, 3-FC ₆ H ₃ -O-CH ₂ B.1416 2-Cl, 4-FC ₆ H ₃ -O-CH ₂ B.1417 2-Cl, 5-FC ₆ H ₃ -O-CH ₂ B.1418 2-Cl, 3-Br-C ₆ H ₃ -CH ₂ -O B.1419 2-Cl, 4-Br-C ₆ H ₃ -CH ₂ -O B.1420 2-Cl, 5-Br-C ₆ H ₃ -CH ₂ -O B.1421 2-Br, 3-FC ₆ H ₃ -O-CH ₂ B.1422 2-Br, 4-FC ₆ H ₃ -O-CH ₂ B.1423 2-Br, 5-FC ₆ H ₃ -O-CH ₂ B.1424 2-Br, 3-Cl-C 8 H ₃ -O-CH ₂

Nr. R ³ B.1425 2-Br, 4-Cl-C ₆ H ₃ -CH ₂ -O B.1426 2-Br, 5-Cl-C ₆ H ₃ -CH ₂ -O B.1427 4-Cl, 3,5-Br ₂ -C ₆ H ₂ -O-CH ₂ B.1428 2-CN-C ₆ H ₄ -O-CH ₂ B.1429 3-CN-C _with H ₄ -O-CH ₂ B.1430 4-CN-C ₆ H ₄ -O-CH ₂ B.1431 2-NO ₂ -C ₆ H ₄ -O-CH ₂ B.1432 3-NO ₂ -C ₆ H ₄ -O-CH 2 B.1433 4-NO ₂ -C ₆ H ₄ -O-CH ₂ B.1434 2-CH ₃ -C ₆ H ₄ -O-CH ₂ B.1435 3 -CH ₃ -C ₆ H ₄ -O-CH ₂ B.1436 4-CH ₃ -C ₆ H ₄ -O-CH ₂ B.1437 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1438 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1439 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1440 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1441 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1442 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1443 2 -CH ₂ CH ₃ -C ₆ H ₄ -O-CH ₂ B.1444 3 -CH ₂ CH ₃ -C ₆ H ₄ -O-CH ₂ B.1445 4 -CH ₂ CH ₃ -C ₆ H ₄ -O-CH ₂ B.1446 2-CH (CH ₃ ) ₂ -C ₆ H ₄ -O-CH ₂ B.1447 3-CH (CH ₃ ) ₂ -C ₆ H ₄ -O-CH ₂ B.1448 4-CH (CH ₃ ) ₂ -C ₆ H ₄ -O-CH ₂ B.1449 3-C (CH ₃ ) ₃ -C ₆ H ₄ -O-CH ₂ B.1450 4-C (CH ₃ ) ₃ -C ₆ H ₄ -O-CH ₂ B.1451 2-C ₆ H ₅ -C ₆ H ₄ -O-CH ₂ B.1452 3-C ₆ H ₅ -C ₆ H ₄ -O-CH ₂ B.1453 4-C ₆ H ₅ -C ₆ H ₄ -O-CH ₂ B.1454 2-OCH ₃ -C ₆ H ₄ -O-CH ₂ B.1455 3-OCH ₃ -C ₆ H ₄ -O-CH ₂ B.1456 4-OCH ₃ -C ₆ H ₄ -O-CH ₂ B.1457 2,3- (OCH ₃ ) 2 -C ₆ H ₃ -O-CH ₂ B.1458 2,4- (OCH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1459 2,5 - (OCH ₃ ) 2 -C ₆ H ₃ -O-CH ₂ B.1460 2,6- (OCH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1461 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1462 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -O-CH ₂ B.1463 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -O-CH ₂

^_ 3e & -

Nr. R ³ B.1464 2-OCH2CH3-C6H4-O-CH 2 B.1465 3-OCH 2 CH 3 -C ₆ H ₄ -O-CH ₂ B.1466 4-OCH ₂ CH ₃ -C ₆ H ₄ -O-CH ₂ B.1467 2-0 (CH ₂ ) ₂ ch ₃ -c ₆ h ₄ -och ₂ B.1468 3 -O (CH ₂ ) ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1469 4-0 (CH ₂ ) ₂ ch ₃ -c ₆ h ₄ -och ₂ B.1470 2-OCH (CH ₃₎ 2 -C ₆ H ₄ OCH ₂ B.1471 3-OCH (CH ₃ ) ₂ -C ₆ H ₄ -OCH ₂ B.1472 4-OCH (CH ₃ ) ₂ -C ₆ H ₄ -OCH ₂ B.1473 3-OC (CH ₃ ) ₃ -C ₆ H ₄ -OCH ₂ B.1474 4-OC (CH ₃ ) ₃ -C ₆ H ₄ -OCH ₂ B.1475 2-OCH ₂ CH = CH ₂ -C ₆ H ₄ -OCH ₂ B.1476 3 -OCH ₂ CH = CH ₂ -C ₆ H ₄ -OCH ₂ B.1477 4 -OCH ₂ CH = CH ₂ -C ₆ H ₄ -OCH ₂ B.1478 2-CF ₃ -C ₆ H ₄ -OCH ₂ B.1479 3-CF ₃ -C ₆ H ₄ -OCH ₂ B.1480 4-CF ₃ -C ₆ H ₄ -OCH ₂ B.1481 2-CO ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1482 3-CO ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1483 4 -CO ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1484 2-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1485 3 -CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1486 4-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1487 2-CONH ₂ -C ₆ H ₄ -OCH ₂ B.1488 3-CONH ₂ -C ₆ H ₄ -OCH ₂ B.1489 4-CONH ₂ -C ₆ H ₄ -OCH ₂ B.1490 2-CON (CH ₃ ) ₂ -c ₆ h ₄ -och ₂ B.1491 3-CON (CH ₃ ) ₂ -C ₆ H ₄ -OCH ₂ B.1492 4-CON (CH ₃ ) ₂ -c ₆ h ₄ -och ₂ B.1493 2 -CONHCH ₃ -C ₆ H ₄ OCH ₂ B.1494 3-conhch ₃ -c ₆ h ₄ -och ₂ B.1495 4 -CONHCH ₃ -C ₆ H ₄ OCH ₂ B.1496 2-NH ₂ -C ₆ H ₄ -OCH ₂ B.1497 3-NH ₂ -C ₆ H ₄ -OCH ₂ B.1498 4-NH ₂ -C ₆ H ₄ -OCH ₂ B.1499 2-N (CH ₃ ) ₂ -C ₆ H ₄ -OCH ₂ B.1500 3-N (CH ₃ ) 2 -C ₆ H ₄ -OCH ₂ B.1501 4-N (CH ₃ ) ₂ -C ₆ H ₄ -OCH ₂ B.1502 2-NHCH ₃ -C ₆ H ₄ -OCH ₂

Nr. R ³ B.1503 3-NHCH ₃ -C ₆ H ₄ -OCH 2 B.1504 4-NHCH ₃ -C ₆ H ₄ -OCH ₂ B.1505 2-CSNH ₂ -C ₆ H ₄ -OCH ₂ B.1506 3-CSNH ₂ -C ₆ H ₄ -OCH ₂ B.1507 4-CSNH ₂ -C ₆ H ₄ -OCH ₂ B.1508 2-SCH ₃ -C ₆ H ₄ -OCH ₂ B.1509 3-SCH ₃ -C ₆ H ₄ -OCH ₂ B.1510 4-SCH ₃ -C ₆ H ₄ -OCH ₂ B.1511 2-SOCH ₃ -C ₆ H ₄ -OCH ₂ B.1512 3-SOCH ₃ -C ₆ H ₄ -OCH ₂ B.1513 4-sculpture ₃ -c ₆ h _4- sc. ₂ B.1514 2-SO ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1515 3-SO ₂ CH ₃ -C ₆ H 4 -OCH ₂ B.1516 4-SO ₂ CH ₃ -C ₆ H ₄ -OCH ₂ B.1517 2-OCF ₃ -C ₆ H ₄ -OCH ₂ B.1518 3-OCF ₃ -C ₆ H ₄ -OCH ₂ B.1519 4-OCF ₃ -C ₆ H ₄ -OCH ₂ B.1520 2-OCHF ₂ -C ₆ H ₄ -OCH ₂ B.1521 3-OCHF ₂ -C ₆ H ₄ -OCH ₂ B.1522 4-OCHF ₂ -C ₆ H ₄ -OCH ₂ B.1523 3-CF ₃ , 4-OCF ₃ -C ₆ H ₃ -OCH ₂ Β.Τ524 2-CH ₂ CH ₂ F-C ₈ H ₄ -OCH ₂ B.1525 3-CH ₂ CH ₂ FC ₆ H ₄ -OCH ₂ B.1526 4-CH ₂ CH ₂ FC ₆ H ₄ -OCH ₂ B.1527 1 2-CH ₂ CF ₃ -C ₆ H ₄ -OCH ₂ B.í528 1 3 -CH ₂ CF ₃ -C ₆ H ₄ -OCH ₂ B.1529 1 4-CH ₂ CF ₃ -C ₆ H ₄ -OCH ₂ B.1530 2-cf ₂ chf ₂ -c ₆ h ₄ -och ₂ B.1531 3 -cf ₂ chf ₂ -c ₆ h ₄ -och ₂ B, 1532 4 -cf ₂ chf ₂ -c ₆ h ₄ -och ₂ B.1533 2-CHF ₂ -C ₆ H ₄ -OCH ₂ B.1534 3-CHF ₂ -C ₆ H ₄ -OCH ₂ B.1535 4-CHF ₂ -C ₆ H ₄ -OCH ₂ B.1536 naphthalin-1-yl-OCH ₂ B.1537 naphthalin-2-yl-OCH ₂ B.1538 pyridin-2-yl ₂ -CH ₂ B.1539 pyridin-3-yl-OCH ₂ b.1540 Pyridin-4-ylOCH ₂ B.1541 5-CH ₃ -pyridin-2-ylOCH ₂

-3νΖ-

Nr. R ³ B.1542 6-CH ₃ -pyridin-2-yl-OCH ₂ B.1543 5-CH 3 -pyridin-3-yl-OCH ₂ B.1544 6-CH 3 -pyridin-3-yl-OCH ₂ B.1545 5-OCH 3 -pyridin-2-yl 1 -OCH ₂ B.1546 6-OCH3-pyridin-2-yl-OCH 2 B.1547 5-OCH 3 -pyridin-3-yl-OCH 2 B.1548 6 -OCH 3 -pyridin-3-yl-OCH ₂ B.1549 4-Cl-pyridin-2-yl-OCH ₂ B.1550 _{5-C1-pyridin-2-2} y1-0CH B.1551 6-Cl-pyridin-2-yl-OCH ₂ B.1552 2-Cl-pyridin-3-yl-OCH 2 B.1553 5-Cl-pyridin-3-yl-OCH ₂ B.1554 6-Cl-pyridin-3-yl-OCH ₂ B.1555 2-Cl-pyridin-4-yl-OCH ₂ B.1556 3,5-Cl ₂ -pyridin-2-yl-OCH ₂ B.1557 pyrimidin-2-yl-OCH ₂ B.1558 4-C 1 -pyrimidin-2-yl-OCH ₂ B.1559 5-Cl-pyrimidin-2-yl-OCH ₂ B.1560 4-CH ₃ -pyrimidin-2-yl-OCH ₂ B.1561 5-CH ₃ -pyrimidin-2-yl-OCH ₂ B.1562 4-OCH 3 -pyrimidin-2-yl-OCH ₂ B.1563 5-OCH 3 -pyrimidin-2-yl-OCH ₂ B.1564 pyrimidin-4-yl-OCH ₂ B.1565 2-Cl-pyrimidin-4-yl-OCH ₂ B.1566 6-Cl-pyrimidin-4-yl-OCH ₂ B.1567 2,6-Cl ₂ -pyrimidin-4-yl-OCH ₂ B.1568 2-CH ₃ -pyrimidin-4-yl-OCH ₂ B.1569 6-CH ₃ -pyrimidin-4-yl-OCH ₂ B.1570 2-OCH 3 -pyrimidin-4-yl-OCH ₂ B.1571 6-OCH 3 -pyrimidin-4-yl-CH ₂ B.1572 pyridin imi DIN-5-yl 1 - OCH ₂ B.1573 2-C 1 -pyrimidin-5-yl-OCH ₂ B.1574 2-CH ₃ -pyrimidin-5-yl-OCH ₂ B.1575 2-OCH ₃ -pyrimidin-5-yl-OCH ₂ B.1576 furan-2-yl-OCH ₂ B.1577 4-Br-furan-2-yl-OCH ₂ B.1578 4-Cl-furan-2-yl-OCH ₂ B.1579 4-CN-furan-2-yl-OCH ₂ B.1580 _{4-CH3-furan-2-yl-OCH2}

Nr. R ³ B.1581 5-Br-furan-2-ylCH ₂ B.1582 5-Cl-furan-2-yl-OCH ₂ B.1583 5-CN-furan-2-yl-OCH ₂ B.1584 5-CH3-furan-2-yl-OCH 2 B.1585 f uran-3-ylCH ₂ B.1586 5-Br-furan-3-yl-OCH ₂ B.1587 5-Cl-furan-3-yl-OCH ₂ B.1588 5-CN-furan-3-yl-OCH ₂ B.1589 _{5-CH3-furan-3-yl-OCH2} B.1590 thien-2-ylCH ₂ B.1591 _{4-Br-thien-2-yl-2} 0CH B.1592 4-Cl-thien-2-yl-OCH ₂ B.1593 4-CN-thien-2-yl-OCH ₂ B.1594 4-CH ₃ -thien-2-yl-OCH ₂ B.1595 5-Br-thien-2-yl-OCH ₂ B.1596 5-Clthien-2-yl-OCH ₂ B.1597 5-CN-thien-2-yl-OCH ₂ B.1598 5-CH ₃ -thien-2-yl-OCH ₂ B.1599 thien-3-yl-OCH ₂ B.1600 5-Br-thien-3-yl-OCH ₂ B.1601 5-Cl-thien-3-yl-OCH ₂ B.1602 5 -CN _thien-3-2 yľOCH B.1603 5-CH ₃ -thien-3-yl-OCH ₂ B.1604 oxa-1-2-yl-OCH ₂ B.1605 4-Br-oxazol-2-yl-OCH ₂ B.1606 4-Cl-oxazol-2-yl-OCH ₂ B.1607 4-CN-oxazol-2-yl-OCH ₂ B.1608 4-CH ₃ -oxazol-2-yl-OCH ₂ B.1609 5-Br-oxazol-2-yl-OCH ₂ B.1610 5-Cl-oxazol-2-yl-OCH ₂ B.1611 5-CN-oxazol-2-yl-OCH ₂ B.1612 5-CH ₃ -oxazol-2-yl-OCH ₂ B.1613 oxa-4-yl-OCH ₂ B.1614 2-Br-oxazol-4-yl-OCH ₂ B.1615 2-Cl-oxazol-4-yl-OCH ₂ B.1616 2-CN-oxazol-4-yl-OCH ₂ B.1617 2-CH ₃ -oxazol-4-yl-OCH ₂ B.1618 2-C 6 H 5 -oxazol-4-yl-OCH ₂ B.1619 5-Br-oxazol-4-yl-OCH ₂

Nr. R ³ B.1620 5-Cl-oxazol-4-yl-OCH ₂ B.1621 5-CN-oxazol-4-yl-OCH 2 B.1622 5-CH 3 -oxazol-4-yl-OCH ₂ B.1623 oxazol-5-yl-OCH ₂ B.1624 4-Br-oxazol-5-yl-OCH ₂ B.1625 4-Cl-oxazol-5-yl-OCH ₂ B.1626 _{4-CN-oxazol-5-yl-O-CH2;} B.1627 4-CH 3 -oxazol-5-yl-OCH ₂ i B.1628 2-Br-oxazol-5-yl-OCH ₂ B.1629 2-Cl-oxazol-5-yl-OCH ₂ B.1630 2-CN-oxazol-5-yl-OCH ₂ B.1631 2-CH 3 -oxazol-5-yl-OCH ₂ ; B.1632 Isoxazol-3-yl-OCH ₂ 1 B.1633 4-Br-isoxazol-3-yl-OCH ₂ f B.1634 4-Cl-isoxazol-3-yl-OCH ₂ B.1635 4-CN-isoxazol-3-yl-OCH ₂ B.1636 4-CH 3 -isoxazol-3-yl-OCH ₂ j B.1637 5-Br-isoxazol-3-yl-OCH ₂ | B.1638 5-Cl-isoxazol-3-yl-OCH ₂ B.1639 5-CN-isoxazol-3-yl-OCH ₂ B.1640 5-CH ₃ -isoxazol-3-yl-OCH ₂ B.1641 isoxazol-4-yl-OCH ₂ B.1642 3-Br-isoxazol-4-yl-OCH ₂ B.1643 3-Cl-isoxazol-4-yl-OCH ₂ B.1644 3-CN-isoxazol-4-yl-OCH ₂ B.1645 3-CH ₃ -isoxazol-4-yl-OCH ₂ B.1646 5-Br-isoxazol-4-yl-OCH ₂ B.1647 5-Cl-isoxazol-4-yl-OCH ₂ B.1648 5-CN-isoxazol-4-yl-OCH ₂ B.1649 5-CH ₃ -isoxazol-4-yl-OCH ₂ B.1650 3,5- (CH ₃ ) ₂ -isoxazol-4-yl-OCH ₂ B. 1651 isoxazol-5-yl-OCH ₂ B. 1652 3-Br-isoxazol-5-yl-OCH ₂ B.1653 3-Cl-isoxazol-5-yl-OCH ₂ B.1654 3-CN-isoxazol-5-yl-OCH ₂ B.1655 3-CH ₃ -isoxazol-5-yl-OCH ₂ B.1656 _{3-C6H5-isoxazol-5-yl-OCH2} B.1657 4-C1, _{3-C6H5-isoxazol-5-yl-OCH2} B.1658 4-Br-C 6 H _{3-isoxazol-5-yl-OCH2}

-505 ~ -

Nr. R ³ B.1659 4-Br-isoxazol-5-yl-OCH 2 B.1660 4-Cl-isoxazol-5-yl-OCH ₂ B.1661 4-CN-isoxazol-5-yl-OCH 2 B.1662 4-CH ₃ -isoxazol-5-yl-OCH 2 B.1663 thiazol-2-yl-OCH ₂ B.1664 _{4-Br-thiazol-2-yl-OCH2} B.1665 4-Cl-thiazol-2-yl-OCH ₂ B.1666 4-CN-thiazol-2-yl-OCH ₂ B.1667 4 CH _3-thia-zo1-2 and _y1-OCH2 B.1668 5-Br-thiazol-2-yl-OCH ₂ B.1669 5-Cl-thiazol-2-yl-OCH ₂ B.1670 5-CN-thiazol-2-yl-OCH ₂ B.1671 5-CH ₃ -thiazol-2-yl-OCH ₂ B.1672 thiazol-4-yl-OCH ₂ B.1673 2-Br-thiazol-4-yl-OCH ₂ B.1674 2-Cl-thiazol-4-yl-OCH ₂ B.1675 2-CN-thiazol-4-yl-OCH ₂ B.1676 2-CH ₃ -thiazol-4-yl-OCH ₂ B.1677 5-Br-thiazol-4-yl-OCH ₂ B.1678 5-Cl-thiazol-4-yl-OCH ₂ B.1679 5-CN-thiazol-4-yl-OCH ₂ B.1680 5-CH ₃ -thiazol-4-yl-OCH ₂ B.1681 thiazol-5-yl-OCH ₂ B.1682 4-Br-thiazol-5-yl-OCH ₂ B.1683 _{4-Cl-thiazol-5-yl-OCH2} B.1684 4-CN-thiazol-5-yl-OCH ₂ B.1685 4-CH ₃ -thiazol-5-yl-OCH ₂ b.1686 2-Br-thiazol-5-yl-OCH ₂ B.1687 2-Cl-thiazol-5-yl-OCH ₂ B.1688 2-CN-thiazol-5-yl-OCH ₂ B.1689 2-CH ₃ -thiazol-5-yl-OCH ₂ B.1690 isothiazol-3-yl-OCH ₂ B.1691 4-Br-isothiazol-3-yl-OCH ₂ B.1692 4-Cl-isothiazol-3-yl-OCH ₂ B.1693 4-CN-isothiazol-3-yl-OCH ₂ B.1694 4-CH ₃ -isothiazol-3-yl-OCH ₂ B.1695 5-Br-isothiazol-3-yl-OCH ₂ B.1696 5-Cl-isothiazol-3-yl-OCH ₂ B.1697 3-CN-isothiazol-3-yl-OCH 2

~ 5%> -

Nr. R ³ B.1698 5-CH ₃ -isothiazol-3-yl-OCH ₂ B.1699 isothiazol-4-yl-OCH ₂ B.1700 3-Br-isothiazol-4-yl-OCH ₂ b.1701 3-Cl-isothiazol-4-yl-OCH ₂ B.1702 3-CN-isothiazol-4-yl-OCH ₂ B.1703 3-CH 3 -isothiazol-4-yl-OCH ₂ B.1704 5-Br-isothiazol-4-yl-OCH ₂ B.1705 5-Cl-isothiazol-4-yl-OCH ₂ B.1706 5-CN-isothiazol-4-yl-OCH ₂ B.1707 5-CH 3 -isothiazol-4-yl-OCH ₂ B.1708 3,5- (CH ₃ ) ₂ -isothiazol-4-yl-OCH ₂ B.1709 isothiazol-5-yl-OCH ₂ B.1710 3-Br-isothiazol-5-yl-OCH ₂ B.1711 3-Cl-isothiazol-5-yl-OCH ₂ B.1712 3-CN-isothiazol-5-yl-OCH ₂ B.1713 3-CH ₃ -isothiazol-5-yl-OCH ₂ B.1714 _{4-Br-isothiazol-5-yl-OCH2} B.1715 4-Cl-isothiazol-5-yl-OCH ₂ B.1716 4-CN-isothiazol-5-yl-OCH ₂ B.1717 4-CH 3 -isothiazol-5-yl-OCH ₂ B.1718 imidazol-2-yl-OCH ₂ B.1719 1-Cl-imidazol-2-yl-OCH ₂ B.1720 1-Br-imidazol-2-yl-OCH ₂ B.1721 1-CN-imidazol- ₂ -yl-OCH ₂ B.1722 1-CH ₃ -inidazol-2-yl-OCH ₂ B.1723 4-Cl-imidazol-2-yl-OCH ₂ B.1724 4-Br-imidazol-2-yl-OCH ₂ B.1725 4-CN-imidazol-2-yl-OCH ₂ B.1726 4-CH ₃ -imidazol-2-yl-OCH ₂ B.1727 1-CH ₃ , 5-Cl-imidazol-2-yl-OCH ₂ B.1728 1,4- (CH ₃ ) ₂ -imidazol-2-yl-OCH ₂ B.1729 1,5- (CH ₃ ) ₂ -imidazol-2-yl-OCH ₂ B.1730 imidazol-4-yl-OCH ₂ B.1731 2-Cl-imidazol-4-yl-OCH ₂ B.1732 2-Br-imidazol-4-yl-OCH ₂ B.1733 2-CN-imidazol-4-yl-OCH ₂ B.1734 1-CH ₃ -imidazol-4-yl-OCH ₂ B.1735 2-CH ₃ -imidazol-4-yl-OCH ₂ B.1736 5-Cl-imidazol-4-yl-OCH ₂

Nr. R ³ B.1737 5-Br-imidazol-4-yľOCH2 b.1738 5-CN-imidazol-4-yl-OCH 2 B.1739 5-CH3-imidazol-4-yl-OCH 2 B.1740 I-CH 3, _{5-Cľimidazol-4-yl-OCH2} B.1741 1,2- (CH ₃ ) ₂ -imidazol-4-ylCH ₂ B.1742 1,5- (CH ₃ ) ₂ -imidazol-4-yl-OCH ₂ B.1743 .. pyrazol-3-yl-OCH ₂ B.1744 5-Br-pyrazol-3-yl-OCH ₂ b.1745 5-Cl-pyrazol-3-yl-OCH ₂ B.1746 5-CN-pyrazol-3-yl-COH ₂ B.1747 5-CH ₃ -pyrazol-3-yl-OCH ₂ B.1748 l-C 6 H _{-pyrazol-3-yl-OCH2} B.1749 4-Br-pyrazol-3-yl-OCH ₂ B.1750 4 - C ips once 0 ¾ 3-y O OCH ₂ B.1751 4-CN-pyrazol-3-ylCH ₂ B.1752 4-CH ₃ -pyrazol 3 -yl -OCH ₂ B.1753 1-CH ₃ -pyrazol-3-yl-OCH 2 B.1754 1,4- (CH ₃ ) ₂ -pyrazol-3-yl-OCH ₂ B.1755 1,5- (CH ₃ ) ₂ -pyrazol-3-yl-OCH ₂ B.1756 1-CH ₃ , 4-C 1 -pyrazol-3-ylCH ₂ B.1757 I-CH 3, 5-Cl-pyrazol-3-yl-OCH ₂ B.1758 pyra from 01-4-y1-OCH ₂ B.1759 3-Br-pyrazol-4-yl-OCH ₂ B.1760 3-Cyclopyrazol-4-yl-OCH ₂ B.1761 3-CN-pyrazol-4-ylCH ₂ B.1762 3-CH ₃ -pyrazol-4-yl-OCH ₂ B.1763 1-CH ₃ -pyrazol-4-yl-OCH ₂ B.1764 1,5- (CH ₃ ) ₂ -pyrazol-4-yl-OCH ₂ b.1765 1,3- (CH ₃ ) ₂ -pyrazol-4-yl-OCH ₂ B.1766 1-CH ₃ , 3-Cl-pyrazol-4-yl-OCH ₂ B.1767 1-CH ₃ , 5-Cl-pyrazol-4-yl-OCH ₂ B.1768 pyra from 01-5-y1-OCH ₂ B.1769 3 -Br-pyrazol-5-ylCH ₂ B.1770 3-Cl-pyrazol-5-yl-OCH ₂ B.1771 3-CN-pyrazol-5-yl-OCH ₂ B.1772 3-CH ₃ -pyrazol-5-yl-OCH ₂ B.1773 1-CH ₃ -pyrazol-5-yl-OCH ₂ B.1774 _{4-Br-pyrazol-5-yl-OCH2} B.1775 -Cl-pyrazol-5-yl-OCH ₂

- $ w

Nr. R ³ B. 1776 4-CN-pyrazol-5-yl-OCH ₂ B.1777 4-CH ₃ -pyrazol-5-yl-OCH ₂ 5 B.1778 1,3- (CH ₃ ) ₂ -pyrazol-5-yl-OCH ₂ B.1779 1,4- (CH ₃ ) ₂ -pyrazol-5-yl-OCH ₂ B.1780 I-CH 3, 3-Cl-pyrazol-5-yl-OCH ₂ B.1781 1-CH ₃ , 4-Cl-pyrazol-5-yl-OCH ₂ 10 B.1782 1,3,4-Oxadiazol-5-yl-OCH ₂ B.1783 2-CH ₃ -1,3,4-oxadiazol-5-yl-OCH ₂ B.1784 2-CF ₃ -1,3,4-oxadiazol-5-yl-OCH ₂ B.1785 2-OCH 3 -1,3,4-oxadiazol-5-yl-OCH ₂ B.1786 2-Cl-1,3,4-oxadiazol-5-yl-OCH ₂ 15 B.1787 2-CH (CH ₃ ) 2-1,3,4-oxadiazol-5-yl-OCH ₂ B.1788 1,3,4-Oxadiazol-2-yl-OCH ₂ B.1789 5-CH ₃ -1,3,4-oxadiazol-2-yl-OCH ₂ B.1790 5-CF ₃ -1,3,4-oxadiazol-2-yl-OCH ₂ 20 B.1791 5-Cl-1,3,4-oxadiazol-2-yl-OCH ₂ B.1792 5-CH (CH ₃ ) ₂ -1,3,4-oxadiazol-2-yl-OCH ₂ b.1793 S-C 6 H 8 -1,3,4-oxadiazol-2-yl-OCH ₂ B.1794 1,2,4-Oxadiazol-3-yl-OCH ₂ 25 B.1795 5-CH ₃ -1,2,4-oxadiazol-3-yl-OCH ₂ B.1796 5-CF ₃ -1,2,4-oxadiazol-3-yl-OCH ₂ B.1797 5-Cl-1,2,4-oxadiazol-3-yl-OCH 2 B.1798 5-CH (CH ₃ ) 2 -1,2,4-oxadiazol-3-yl-OCH ₂ 30 B.1799 1,2,4-triazol-3-yl-OCH ₂ B.1800 1-CH ₃ -1,2,4-triazol-3-yl-OCH ₂ B.1801 5-CH 3 -1,2,4-triazol-3-yl-OCH ₂ B.1802 5-CF 3 -1,2,4-triazol-3-yl-OCH ₂ B.1803 5-OCH ₃ -1,2,4-triazol-3-yl-OCH ₂ 35 B.1804 5-Cl-1,2,4-triazol-3-yl-OCH ₂ B.1805 5-CH (CH ₃ ) ₂ -1,2,4-triazol-3-yl-OCH ₂ B.1806 1-C 5 H 5 -1,2,4-triazol-3-yl-OCH ₂ B.1807 1,3,4-thiadiazol-5-yl-OCH ₂ 40 B.1808 2-CH ₃ -1,3,4-thiadiazol-5-yl-OCH ₂ B.1809 2-CF ₃ -1,3,4-thiadiazol-5-yl 1 -CH ₂ B.1810 2-OCH ₃ -1,3,4-thiadiazol-5-yl-OCH ₂ B.1811 2-Cl-1,3,4-thiadiazol-5-yl-OCH ₂ 4ς. B.1812 2-CH (CH ₃ ) ₂ -1,3,4-thiadiazol-5-yl-OCH ₂ B.1813 1,3,4-thiadiazol-2-yl-OCH ₂ B.1814 5-CH ₃ -1,3,4-thiadiazol-2-yl-OCH 2

- ν $ $ -

Nr. R ³ B.1815 5-CF 3 -1,3,4-thiadiazol-2-yl-OCH ₂ B.1816 5-OCH 3 -1,3,4-thiadiazol-2-yl-OCH ₂ B.1817 5-Cl, 3,4-thiadiazol-2-yl-OCH 2 B.1818 5-CH (CH ₃ ) ₂ -1,3,4-thiadiazol-2-yl-OCH ₂ b.1819 5-C 8 H 5 -1,3,4-thiadiazol-2-ylCH ₂ B.1820 1,2,4-thiadiazol-3-yl-OCH ₂ B.1821 5-CH 3 -1,2,4-thiadiazol-3-yl-OCH ₂ B.1822 5-CF 3 -1,2,4-thiadiazol-3-yl-OCH ₂ B.1823 5-OCH 3 -1,2,4-thiadiazol-3-yl-OCH ₂ B.1824 5-Cl-1,2,4-thiadiazol-3-yl-OCH ₂ b.1825 5-CH (CH ₃ ) ₂ -1,2,4-thiadiazol-3-yl-OCH ₂ B.1826 pyrrol-2-yl-OCH ₂ B.1827 4-C1-pyrrole- ₂ -yl-OCH2 B.1828 4-Br-pyrrol-2-yl-OCH ₂ B.1829 4-CH ₃ -pyrrol-2-yl-OCH ₂ B.1830 _{4-C6H5-pyrrol-2-yl-OCH2} B.1831 benzimidazol-2-yl-OCH ₂ B.1832 quinolin-2-yl-OCH ₂ B.1833 1,1-Cl ₂ -cyclopropan-2-yl-OCH ₂ B.1834 2-CH ₃ , 1,1-Cl ₂ -cyclopropan-2-yl-OCH ₂ b.1835 2-CH ₃ , 1,1-Cl 2 -cyclopropan-3-yl-OCH 2 B.1836 2,2- _{(CH3) 2,} 1, _{l-Cl2 -cyclopropan-3-yl-OCH2} B.1837 2,3- _{(CH3) 2,} 1, _{l-Cl2 -cyclopropan-3-yl-OCH2} B.1838 2,3,3- _{(CH3) 3,} 1, _{l-Cl2 -cyclopropan-2-yl-OCH2} B.1839 1,1-Cl2 ^- cyclopropan-2-yl-O-CH (CH ₃ ) B.1840 2-CH ₃ , 1,1-Cl ₂ -cyclopropan-2-yl-O-CH (CH ₃ ) B.1841 2-CH _3, 1, _l-Cl2 -cyclopropan-3-yl-0-CH (CH ₃₎ B.1842 2,2- _{(CH3) 2,} 1, _l-Cl2 -cyclopropan-3-yl-0-CH (CH ₃₎ b.1843 2,3- _{(CH3) 2,} 1, ₂ LCL -cyclopropan-3-yl-0-CH (CH ₃₎ B.1844 2,3,3 - (CH _{3) 3,} 1, _l-Cl2 -cyclopropan-2-yl-0-CH (CH ₃₎ B.1845 1,1-Br 2 -cyclopropan-2-yl-OCH ₂ B.1846 2-CH _3, 1, _{l-Br2 -cyclopropan-2-yl-OCH2} b.1847 2-CH _3, 1, _{l-Br2 -cyclopropan-3-yl-OCH2} B.1848 2,2- _(CH3) 2, 1, _{l-Br2 -cyclopropan-3-yl-OCH2} B.1849 2,3- (CH ₃ ) 2 H 11 -Br ₂ -cyclopropan-3-yl-OCH ₂ b.1850 2,3,3- _{(CH3) 3,} 1, _{l-Br2 -cyclopropan-2-yl-OCH2} B.1851 1-Br ₂ -cyclopropan-2-yl-OCH (CH ₃ ) B.1852 2-CH ₃ , 1,1-Br ₂ -cyclopropan-2-yl-OCH (CH ₃ ) B.1853 2-CH ₃ , 1,1-Br ₂ -cyclopropan-3-yl-OCH (CH ₃ )

Nr. R ³ B.1854 2,2- _{(CH3) 2,} 1, _l-Br2 -cyclopropan-3-yl-OCH _(CH3) B.1855 2,3- _{(CH3) 2,} 1, _l-Br2 -cyclopropan-3-yl-OCH _(CH3) B.1856 2,3,3- (CH ₃ ) 3,1,1-Br ₂ -cyclopropan-2-yl-OCH (CH ₃ ) B.1857 2-F-C 8 H ₄ -CH (CH ₃ ) B.1858 3-FC ₆ H ₄ -CH (CH ₃ ) B.1859 4-FC ₆ H ₄ -CH <CH ₃ ) B.1860 2,3-F ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1861 2,4-F ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1862 2,5-F ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1863 2,6-F ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1864 3,4-F ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1865 3,5-F ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1866 2-Cl-C ₆ H ₄ -CH (CH ₃₎ B.1867 3-Cl-C ₆ H ₄ -CH (CH ₃₎ B.1868 4-Cl-C ₆ H ₄ -CH (CH ₃ ) B.1869 2,3-Cl ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1870 2,4-Cl ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1871 2,5-Cl ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1872 2,6-Cl ₂ -C ₆ H ₃ -CH (CH ₃ ) b.1873 3,4-Cl ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1874 3,5-Cl ₂ -C ₈ H ₃ -CH (CH ₃ ) b.1875 2,3,4-Cl ₃ -C ₈ H ₂ -CH (CH ₃ ) B.1876 2,3,5-Cl ₃ -C ₈ H ₂ -CH (CH ₃ ) B.1877 2,3,6-Cl ₃ -C ₈ H ₂ -CH (CH ₃ ) B.1878 2,4,5-Cl ₃ -C ₆ H ₂ -CH (CH ₃ ) B.1879 2,4,6-Cl ₃ -C ₈ H ₂ -CH (CH ₃ ) B.1880 3,4,5-Cl ₃ -C ₈ H ₂ -CH (CH ₃ ) B.1881 2-Br-C ₆ H ₄ -CH (CH ₃ ) B.1882 3-Br-C ₆ H ₄ -CH (CH ₃ ) B.1883 4-Br-C ₆ H ₄ -CH (CH ₃ ) B.1884 2,3-Br ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1885 2,4-Br ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1886 2,5-Br ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1887 2,6-Br ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1888 3,4-Br ₂ -C ₈ H ₃ -CH (CH ₃ ) B.1889 3,5-Br ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1890 2-F, 3-Cl-C 8 H ₃ -CH (CH ₃ ) B.1891 2-F, 4-Cl-C ₆ H ₃ CH (CH ₃₎ B.1892 2-F, 5-Cl _3-CGH -CH (CH ₃₎

~ 511-

Nr. R ³ B.1893 2-F, 3-Br-C ₆ H ₃ -CH (CH ₃ ) B. 1894 2-F, 4-Br-C ₆ H ₃ -CH (CH ₃ ) B.1895 2-F, 5-Br-C ₆ H ₃ -CH (CH ₃ ) b.1896 2-C1,3-FC ₆ H ₃ -CH (CH ₃ ) B.1897 2-C1,4-FC ₆ H ₃ -CH (CH ₃ ) B.1898 2-C1,5-FC ₆ H ₃ -CH (CH ₃ ) B.1899 2-C1, 3-Br-C ₆ H ₃ CH (CH ₃₎ B.1900 2-C1, 4-Br-C ₆ H ₃ CH (CH ₃₎ B.1901 2-C1, 5-Br-C ₆ H ₃ CH (CH ₃₎ B.1902 2-Br, 3-F-C ₅ H ₃ -CH (CH ₃ ) B.1903 2-Br, 4-FC ₆ H ₃ -CH (CH ₃ ) B.1904 2-Br, 5-FC ₆ H ₃ -CH (CH ₃ ) B.1905 2-Br, 3-Cl-C ₆ H ₃ CH (CH ₃₎ B.1906 2-Br, 4-Cl-C ₆ H ₃ CH (CH ₃₎ B.1907 2-Br, 5-Cl-C ₆ H ₃ CH (CH ₃₎ B.1908 4-Cl, 3,5-Br ₂ -C ₆ H ₂ CH (CH ₃₎ B.1909 2-CN-C ₆ H ₄ -CH (CH ₃₎ B.1910 3-CN-C ₆ H ₄ -CH (CH ₃ ) B.1911 4-0 ^ 06 ^ -011 (013) B.1912 2-NO ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1913 3-NO ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1914 4-NO ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1915 2-CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1916 3-CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1917 4-CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1918 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1919 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) b.1920 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) b.1921 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1922 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) b.1923 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1924 2-CH (CH ₃ ), CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1925 3-CH (CH ₃ ) CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1926 4-CH (CH ₃ ) CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1927 2-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1928 3-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1929 4-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH (CH ₃ ) b.1930 3-C (CH ₃ ) ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1931 4-C (CH ₃ ) ₃ -C ₆ H ₄ -CH (CH ₃ )

-í1i ~

Nr. R ³ b.1932 2-C ₆ H ₅ -C ₆ H ₄ -CH (CH ₃ ) B.1933 3-C ₆ H ₅ -C ₆ H ₄ -CH (CH ₃ ) b.1934 4-C ₆ H ₅ -C ₆ H ₄ -CH (CH ₃ ) b.1935 2-OCH ₃ -C ₆ H ₄ -CH (CH ₃ ) b.1936 3-OCH ₃ -C ₆ H ₄ -CH (CH ₃ ) b.1937 4-OCH ₃ -C ₆ H ₄ -CH (CH ₃ ) b.1938 2,3- (OCH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) B.1939 2,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) b.1940 2,5- (OCH ₃ ) 2-C ₅ H ₃ -CH (CH ₃ ) B.1941 2,6- (OCH ₃ ) ₂ -C ₆ H ₃ -CH (CH ₃ ) b.1942 3,4- (OCH ₃ ) 2 -C ₆ H ₃ -CH (CH ₃ ) b.1943 3,5 - _(OCH3) 2 -C ₆ H ₃ -CH (CH ₃₎ B.1944 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH (CH ₃ ) b.1945 2-OCH (CH ₃ ) CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1946 3-OCH (CH ₃ ) CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1947 4-OCH (CH ₃ ) CH ₃ -C ₆ H ₄ -CH (CH ₃ ) b.1948 2-O (CH (CH ₃ )) ₂ CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1949 3-O (CH (CH _{3)) 2} CH _{3 S} C H ₄ -CH (CH ₃₎ B.1950 4-O (CH (CH ₃ )) ₂ CH ₃ -C ₆ H ₄ -CH (CH ₃ ) b.1951 2-OCH (CH ₃ ) 2-C ₆ H ₄ -CH (CH ₃ ) B.1952 3-OCH (CH ₃₎ 2 -C ₆ H ₄ -CH (CH ₃₎ B.1953 4-OCH (CH ₃ ) ₂ -C ₆ H ₄ -CH (CH ₃ ) b.1954 3 -OC (CH ₃ ) ₃ -C ₈ H ₄ -CH (CH ₃ ) B.1955 4-OC (CH ₃ ) ₃ -C ₆ H ₄ -CH (CH ₃ ) b.1956 2-OCH (CH ₃ ) CH = CH (CH ₃ ) -C ₆ H ₄ -CH (CH ₃ ) b.1957 3-OCH (CH ₃ ) CH = CH (CH ₃ ) -C ₆ H ₄ -CH (CH ₃ ) B.1958 4-OCH (CH ₃ ) CH = CH (CH ₃ ) -C ₆ H ₄ -CH (CH ₃ ); B.1959 2-CF ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1960 3-CF ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1961 4-CF ₃ -C ₆ H ₄ -CH (CH ₃ ); B.1962 2-CO ₂ CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1963 3-co ₂ ch ₃ -c ₆ h ₄ -ch (ch ₃ ); b.1964 4-CO ₂ CH ₃ -C ₆ H ₄ -CH (CH ₃ ); B.1965 2 - CO ₂ CH ₂ CH ₃ - C ₄ H ₄ - CH (CH ₃ ) B.1966 3 - CO ₂ CH ₂ CH ₃ - C ₆ H ₄ - CH (CH ₃ ) B.1967 4 - CO ₂ CH ₂ CH ₃ - C ₆ H ₄ - CH (CH ₃ ) B.1968 2-CONH ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1969 3-CONH ₂ -C ₆ H ₄ -CH (CH ₃ ) - B.1970 4-CONH ₂ -C ₆ H ₄ -CH (CH ₃ )

Nr. R ³ B.1971 2-CON (CH ₃ ) ₂ -C _e H ₄ -CH (CH ₃ ) B.1972 3-CON (CH ₃ ) ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1973 4 -CON (CH ₃ ) ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1974 2-CONHCH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1975 3-CONHCH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1976 4-CONHCH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1977 2-NH ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1978 3-NH ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1979 4-NH ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1980 2-N (CH ₃ ) ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1981 3-n (ch ₃ ) _2- c _with h ₄ -ch (ch ₃ ) B.1982 4-N (CH ₃ ) 2 -C ₆ H ₄ -CH (CH ₃ ) B.1983 2-NHCH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1984 3-NHCH ₃ -C _e H ₄ -CH (CH ₃ ) B.1985 4-NHCH ₃ -C ₆ H ₄ -CH (ch ₃ ) B.1986 2-CSNH ₂ -C ₆ H ₄ -CH _(CH3) B.1987 3-ennh ₂ -c ₆ h ₄ -ch (CH ₃ ) B.1988 4-CSNH ₂ -C ₆ H ₄ -CH (CH ₃ ) B.1989 2-SCH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1990 3-SCH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1991 4-SCH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1992 2-SOCH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1993 3-sculpture _3- c ₆ h ₄ -ch (ch ₃ ) B.1994 4-sculpture _3- c ₆ h ₄ -ch (CH ₃ ) B.1995 2-Sat ₂ ch ₃ -c ₆ h ₄ -ch <ch ₃ ) B.1996 3-Sat ₂ ch ₃ -c ₆ h ₄ -ch (ch ₃ ) B.1997 4-SO ₂ CH ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1998 2-OCF ₃ -C ₆ H ₄ -CH (CH ₃ ) B.1999 3-OCF ₃ -C ₆ H ₄ -CH (CH ₃ ) B.2000 4 -OCF ₃ -C ₆ H ₄ -CH (CH ₃ ) B.2001 2-OCHF ₂ -C ₆ H ₄ -CH (CH ₃ ) B.2002 3 -OCHF ₂ -C ₆ H ₄ -CH (CH ₃ ) B.2003 4-OCHF ₂ -C ₆ H ₄ -CH (CH ₃ ) B.2004 3-CF ₃ , 4-OCF ₃ -C ₆ H ₃ -CH (CH ₃ ) B.2005 2-CH ₂ CH ₂ FC ₆ H ₄ -CH (CH ₃ ) B.2006 3-CH ₂ CH ₂ FC ₆ H ₄ -CH (CH ₃ ) B.2007 4 -CH ₂ CH ₂ F - C ₆ H ₄ - CH (CH ₃ ) B.2008 2-CH ₂ CF ₃ -C ₆ H ₄ -CH (ch ₃ ) B.2009 3 -CH ₂ CF ₃ -C ₆ H ₄ -CH (CH ₃ )

Ή ¹ / -

Nr. R ³ B.2010 4-CH 2 CF 3 -C 6 H 4 -CH (CH ₃ ) B.2011 2-CF ₂ CHF ₂ -C ₆ H ₄ -CH _(CH3) B.2012 3-CF ₂ CHF 2-C ₆ H ₄ -CH (CH ₃ ) B.2013 4-CHF ₂ CF ₂ -C ₆ H ₄ -CH _(CH3) B.2014 2-CHF _2- C ₆ H ₄ -CH (CH ₃ ) B.2015 3-CHF _2- C ₆ H ₄ -CH (CH ₃ ) B.2016 4-CHF _2- C ₆ H ₄ -CH (CH ₃ ) B.2017 naphthal in-1-ylCH (CH ₃ ) B.2018 naphthalin-2-y 1 -CH (CH ₃ ) B.2019 pyridin-2-yl-CH _(CH3) B.2020 pyridin-3-yl-CH _(CH3) B.2021 pyridin-4-yl-CH _(CH3) B.2022 _{5-CH3-pyridin-2-yľCH} (CH ₃₎ B.2023 _{6-CH3-pyridin-2-yľCH} (CH ₃₎ B.2024 _{5-CH3-pyridin-3-yľCH} (CH ₃₎ B.2025 _{6-CH3-pyridin-3-yľCH} (CH ₃₎ B.2026 _{5-OCH3-pyridin-2-yl-CH (CH3)} B.2027 6-OCH ₃ -pyridin-2-ylCH (CH ₃ ) B.2028 _{5-OCH3-pyridin-3-yl-CH (CH3)} B.2029 6-OCH ₃ -pyridin-3-ylCH (CH ₃ ) B.2030 4-C 1-pyridin-2-yl-CH _(CH3) B.2031 5-Cyclopyridin-2-ylCH (CH ₃ ) B.2032 6-Cl-pyridin-2-yľCH (CH ₃₎ B.2033 2-Cl-pyridin-3-yl-CH _(CH3) B.2034 5-Cl-pyridin-3-yl-CH _(CH3) B.2035 6-clpyridine-3-yl-CH _(CH3) B.2036 2-Cl-pyridin-4-yl-CH _(CH3) B.2037 3,5-Cl ₂ -pyridin-2-yľCH (CH ₃₎ B.2038 pyrimidin-2-yl-CH _(CH3) B.2039 4-Cl-pyrimidin-2-yl-CH _(CH3) B.2040 5-Cyclopyrimidin-2-ylCH (CH ₃ ) B.2041 _4-CH3 -pyrimidin-2-yl-CH _(CH3) B.2042 5-CH ₃ -pyrimidin-2-yl-CH _(CH3) B.2043 _4-OCH3 -pyrimidin-2-yl-CH _(CH3) B.2044 _5-OCH3 -pyrimidin-2-yl-CH _(CH3) B.2045 pyrimidin-4-yl-CH _(CH3) B.2046 2-Cl-pyrimidin-4-yl-CH _(CH3) B.2047 6-C 1 -pyrimidin-4-yl-CH (CH ₃ ) B.2048 _2,6-Cl2 -pyrimidin-4-yl-CH _(CH3)

Nr. R ³ B.2049 _2-CH3 -pyrimidin-4-yl-CH _(CH3) B.2050 6-CH ₃ -pyrimidin-4-yl-CH (CH ₃ ) B.2051 2-OCH ₃ -pyrimidin-4-yl-CH (CH ₃ ) B.2052 6-OCH ₃ -pyrimidin-4-yl-CH (CH ₃ ) B.2053 pyrimidin-5-yl-CH _(CH3) B.2054 2-Cl-pyrimidin-5-yl-CH _(CH3) B.2055 _2-CH3 -pyrimidin-5-yl-CH _(CH3) B.2056 _2-OCH3 -pyrimidin-5-yl-CH _(CH3) B.2057 2-OCH 2 CH ₃ -pyrimidin-5-yl-CH (CH ₃ ) B.2058 furan-2-yl-CH _(CH3) B.2059 4-Br-furan-2-yl-CH _(CH3) B.2060 4-Cl-furan-2-yl-CH _(CH3) B.2061 4-CN-furan-2-yl-CH _(CH3) B.2062 _{4-CH3-furan-2-yl-CH (CH3)} B.2063 5-Br-furan-2-yl-CH _(CH3) B.2064 5-Cl-furan-2-yl-CH _(CH3) B.2065 5-CN-furan-2-yl-CH _(CH3) B.2066 _{5-CH3-furan-2-yl-CH (CH3)} B.2067 furan-3-yl-CH _(CH3) B.2068 5-Br-furan-3-yl-CH _(CH3) B.2069 5-Cl-furan-3-yl-CH _(CH3) B.2070 5-CN-furan-3-yl-CH _(CH3) B.2071 _{5-CH3-furan-3-yl-CH (CH3)} B.2072 thien-2-yl-CH _(CH3) B.2073 4-Br-thien-2-yl-CH _(CH3) B.2074 4-Cl-thien-2-yl-CH _(CH3) B.2075 4-CN-thien-2-yl-CH _(CH3) B.2076 4-CH ₃ -thien-2-yl CH (CH ₃ ) B.2077 5-Br-thien-2-yl-CH _(CH3) B.2078 5-Cl-thien-2-yl-CH _(CH3) B.2079 5-CN-thien-2-yl-CH _(CH3) B.2080 5-CH ₃ -thien-2-yl CH (CH ₃ ) B.2081 thien-3-yl-CH _(CH3) B.2082 5-Br-thien-3-yl-CH _(CH3) B.2083 5-Cl-thien-3-yl-CH _(CH3) B.2084 5-CN-thien-3-yl-CH _(CH3) B.2085 5-CH ₃ -thien-3-yl CH (CH ₃ ) B.2086 □ oxazol-2-yl-CH _(CH3) B.2087 l-Br-oxazol-2-yl-CH _(CH3)

-3Η-

Nr. R ³ B.2088 4-Cl-oxazol-2-yl-CH _(CH3) B.2089 4-CN-oxazol-2-yl-CH _(CH3) B.2090 _{4-CH3-oxazol-2-yl-CH (CH3)} B.2091 5-Br-oxazol-2-yl-CH _(CH3) B.2092 5-Cl-oxazol-2-yl-CH _(CH3) B.2093 5-CN-oxazol-2-yl-CH _(CH3) B.2094 _{5-CH3-oxazol-2-yl-CH (CH3)} B.2095 oxazol-4-yl-CH _(CH3) B.2096 2-Br-oxazol-4-yl-CH _(CH3) B.2097 2-Cl-oxazol-4-yl-CH _(CH3) B.2098 2-CN-oxazol-4-yl-CH _(CH3) B.2099 _{2-CH3-oxazol-4-yl-CH (CH3)} B.2100 2-C ₆ H _{5-oxazol-4-yl-CH (CH3)} B.2101 5-Br-oxazol-4-yl-CH _(CH3) B.2102 5-Cl-oxazol-4-yl-CH _(CH3) B.2103 5-CN-oxazol-4-yl-CH _(CH3) B.2104 _{5-CH3-oxazol-4-yl-CH (CH3)} B.2105 oxazol-5-yl-CH _(CH3) B.2106 4-Br-oxazol-5-yl-CH _(CH3) B.2107 4-Cl-oxazol-5-yl-CH _(CH3) B.2108 4-CN-oxazol-5-yl-CH _(CH3) B.2109 _{4-CH3-oxazol-5-yl-CH (CH3)} B.2110 2-Br-oxazol-5-yl-CH _(CH3) B.2111 2-Cl-oxazol-5-yl-CH _(CH3) B.2112 2-CN-oxazol-5-yl-CH _(CH3) B.2113 _{2-CH3-oxazol-5-yl-CH (CH3)} B.2114 isoxazol-3-yl-CH _(CH3) B.2115 4-Br-isoxazol-3-yl-CH _(CH3) B.2116 4-Cl-isoxazol-3-yl-CH _(CH3) B.2117 4-CN-isoxazol-3-yl-CH _(CH3) B.2118 _4-CH3 isoxazol-3-yl-CH _(CH3) B.2119 5-Br-isoxazol-3-yl-CH _(CH3) B.2120 5-Cl-isoxazol-3-yl-CH _(CH3) B.2121 5-CN-isoxazol-3-yl-CH _(CH3) B.2122 _{5-CH3-isoxazol-3-yl-CH (CH3)} B.2123 isoxazol-4-yl-CH _(CH3) B.2124 3-Br-isoxazol-4-yl-CH _(CH3) B.2125 3-Cl-isoxazol-4-yl-CH _(CH3) B.2126 3-CN-isoxazol-4-yl-CH _(CH3)

Nr. R ³ B.2127 _{3-CH3-isoxazol-4-yl-CH (CH3)} B.2128 5-Br-isoxazol-4-yl-CH _(CH3) 5 B.2129 5-Cl-isoxazol-4-yl-CH _(CH3) B.2130 5-CN-isoxazol-4-yl-CH _(CH3) B.2131 _{5-CH3-isoxazol-4-yl-CH (CH3)} B.2132 3,5- _(CH3) 2 ^- isoxazol-4-yl-CH _(CH3) B.2133 isoxazol-5-yl-CH _(CH3) B.2134 3-Br-isoxazol-5-yl-CH _(CH3) B.2135 3-Cl-isoxazol-5-yl-CH _(CH3) B.2136 3-CN-i soxa zo1-5-yl-CH _(CH3) B.2137 _{3-CH3-isoxazol-5-yl-CH (CH3)} B.2138 3-C6H5-isoxazol-5-yl-CH _(CH3) B.2139 4-C1, 3-C6H5-isoxazol-5-yl-CH _(CH3) B.2140 4-Br, 3-C 6 H 5 -isoxazol-5-yl-CH (CH ₃ ) B.2141 4-Br-isoxazol-5-yl-CH _(CH3) B.2142 4-Cl-isoxazol-5-yl-CH _(CH3) B.2143 4-CN-isoxazol-5-yl-CH (CH ₃ ) B.2144 _{4-CH3-isoxazol-5-yl-CH (CH3)} B.2145 thiazol-2-yl-CH _(CH3) B.2146 4-Br-thiazol-2-yl-CH _(CH3) B.2147 4-C 1 -thiazol-2-yl-CH (CH ₃ ) B.2148 4-CN-thiazol-2-yl-CH _(CH3) B.2149 _{4-CH3-thiazol-2-yl-CH (CH3)} B.2150 5-Br-thiazol-2-yl-CH _(CH3) B.2151 5-Cl-thiazol-2-yl-CH _(CH3) B.2152 5-CN-thiazol-2-yl-CH _(CH3) B.2153 5-CH ₃ -thiazol-2-yl-CH (CH ₃ , B.2154 thiazol-4-yl-CH _(CH3) B.2155 2-Br-thiazol-4-yl-CH _(CH3) B.2156 2-Cl-thiazol-4-yl-CH _(CH3) B.2157 2-CN-thiazol-4-yl-CH _(CH3) B.2158 2-CH ₃ -thiazol-4-yl CH (CH ₃ ) B.2159 5-Br-thiazol-4-yl-CH _(CH3) B.2160 5-Cl-thiazol-4-yl-CH _(CH3) B.2161 5-CN-thiazol-4-yl-CH _(CH3) B.2162 _{5-CH3-thiazol-4-yl-CH (CH3)} B.2163 thiazol-5-yl-CH _(CH3) B.2164 1'-Br-thiazol-5-yl-CH (CH ₃ ) B.2165 i-Cl-thiazol-5-yl-CH _(CH3)

Nr. R ³ B.2166 4-CN-thiazol-5-yl-CH _(CH3) B.2167 4-CH ₃ -thiazol-5-yl CH (CH ₃ ) B.2168 2-Br-thiazol-5-yl-CH _(CH3) B.2169 2-Cl-thiazol-5-yl-CH _(CH3) B.2170 2-CN-thiazol-5-yl-CH _(CH3) B.2171 2-CH ₃ -thiazol-5-yl CH (CH ₃ ) B.2172 isothiazol-3-yl-CH _(CH3) B.2173 4-Br-isothiazol-3-yl-CH _(CH3) B.2174 4-Cl-isothiazol-3-yl-CH _(CH3) B.2175 4-CN-isothiazol- ₃ -ylCH (CH3) B.2176 4-CH ₃ -isothiazol-3-ylCH (CH ₃ ) B.2177 5-Br-isothiazol-3-yľCH (CH ₃₎ B.2178 5-Cl-isothiazol-3-yl-CH _(CH3) B.2179 5-CN-isothiazol-3-yl-CH (CH3 ₎ , B.2180 5-CH ₃ -isothiazol-3-yl CH (CH ₃ ) B.2181 isothiazol-4-yl-CH _(CH3) B.2182 3-Br-isothiazol-4-yl-CH _(CH3) B.2183 3-Cl-isothiazol-4-yl-CH _(CH3) B.2184 3-CN-isothiazol-4-yl-CH _(CH3) B.2185 3-CH ₃ -isothiazol-4-yl CH (CH ₃ ) B.2186 5-Br-isothiazol-4-yl-CH _(CH3) B.2187 5-Cl-isothiazol-4-yl-CH _(CH3) B.2188 5-CN--isothiazole-4-yl-CH _(CH3) B.2189 5-CH ₃ -isothiazol-4-yl CH (CH ₃ ) B.2190 3,5- _(CH3) 2 ^- isothiazole-4-yl-CH _(CH3) B.2191 isothiazol-5-yl-CH _(CH3) B.2192 3-Br-isothiazol-5-yľCH (CH ₃₎ B.2193 3-Cl-isothiazol-5-yl-CH _(CH3) B.2194 3-CN-isothiazol-5-yl-CH _(CH3) B.2195 3-CH ₃ -isothiazol-5-yl CH (CH ₃ ) B.2196 4-Br-isothiazoľ5-yl-CH (CFI ₃₎ B.2197 4-Cl-isothiazoľ5 yľCH (CH ₃₎ B.2198 4-CN-isothiazol-5-yľCH (CH ₃₎ B.2199 4-CH ₃ -isothiazol-5-yl CH (CH ₃ ) B.2200 imidazol-2-yl-CH _(CH3) B.2201 1'-imidazol-2-yl-CH (CH ₃ ) B.2202 l-Br-imidazol-2-yl-CH _(CH3) B.2203 L-CN-imidazol-2-yl-CH _(CH3) B.2204 L-CH ₃ -imidazol-2-yl-CH (CH ₃ )

-51? -

Nr. R ³ B.2205 4-Cl-imidazol-2-yl-CH _(CH3) B.2206 4-Br-imidazol-2-yl-CH _(CH3) B.2207 4-CN-imidazol-2-yl-CH _(CH3) B.2208 _{4-CH3-imidazol-2-yl-CH (CH3)} B.2209 _1-CH3, 5-Cl-imidazol-2-yl-CH _(CH3) B.2210 1,4- (CH ₃ ) ₂ -imidazol-2-yl-CH (CH ₃ ) B.2211 1,5- (CH ₃ ) ₂ -imidazol-2-yl-CH (CH ₃ ) B.2212 imidazol-4-yl-CH _(CH3) B.2213 2-Cl-imidazol-4-yl-CH _(CH3) B.2214 2-Br-imidazol-4-yl-CH _(CH3) B.2215 2-CN-imidazol-4-yl-CH _(CH3) B.2216 1-CH ₃ -imidazol-4-yl-CH (CH ₃ ) B.2217 _{2-CH3-imidazol-4-yl-CH (CH3)} B.2218 5-Cl-imidazol-4-yl-CH _(CH3) B.2219 5-Br-imidazol-4-yl-CH _(CH3) B.2220 5-CN-imidazol-4-yl-CH _(CH3) B.2221 _{5-CH3-imidazol-4-yl-CH (CH3)} B.2222 _1-CH3, 5-Cl-imidazol-4-yl-CH _(CH3) B.2223 1,2- (CH ₃ ) ₂ -imidazol-4-yl-CH (CH ₃ ) B.2224 1,5- (CH ₃ ) ₂ -imidazol-4-yl-CH (CH ₃ ) B.2225 pyrazol-3-yl-CH _(CH3) B.2226 5-Br-pyrazol-3-yl-CH _(CH3) B.2227 5-Cl-pyrazol-3-yl-CH _(CH3) B.2228 5-CN-pyrazol-3-yl-CH _(CH3) B.2229 _{5-CH3-pyrazol-3-yl-CH (CH3)} B.2230 1C ₆ H ₅ -pyrazol-3-yl-CH (CH ₃ ) B.2231 4-Br-pyrazol-3-yl-CH _(CH3) B.2232 4-Cl-pyrazol-3-yl-CH _(CH3) B.2233 4-CN-pyrazol-3-yl-CH _(CH3) B.2234 4-CH ₃ -pyrazol-3-yl CH (CH ₃ ) B.2235 1-CH ₃ -pyreo- _3- y 1-CH (CH ₃ ) B.2236 1,4- _{(CH3) 2-pyrazol-3-yl-CH (CH3)} B.2237 1,5- _{(CH3) 2-pyrazol-3-yl-CH (CH3)} B.2238 _1-CH3, 4-Cl-pyrazol-3-yl-CH _(CH3) B.2239 _1-CH3, 5-Cl-pyrazol-3-yl-CH _(CH3) B.2240 pyrazol-4-yl-CH _(CH3) B.2241 3-Br-pyrazol-4-yl-CH _(CH3) B.2242 3-Cl-pyrazol-4-yl-CH _(CH3) B.2243 3-CN-pyrazol-4-yl-CH _(CH3)

Nr. R ³ B.2244 3-CH ₃ -pyrazol-4-yl CH (CH ₃ ) B.2245 1-CH ₃ -pyrazol-4-yl-CH (CH ₃ ) - 5 B.2246 1,5- _{(CH3) 2-pyrazol-4-yl-CH (CH3)} B.2247 1,3- _{(CH3) 2-pyrazol-4-yl-CH (CH3)} B.2248 _1-CH3, 3-Cl-pyrazol-4-yl-CH _(CH3) B.2249 _1-CH3, 5-Cl-pyrazol-4-yl-CH _(CH3) η . B.2250 pyrazol-5-yl-CH _(CH3) B.2251 3-Br-pyrazol-5-yl-CH _(CH3) B.2252 3-Cl-pyrazol-5-yl-CH _(CH3) B.2253 3-CN-pyrazol-5-yl-CH _(CH3) B.2254 3-CH ₃ -pyrazol-5-yl-CH (CH ₃ ) 5 B.2255 1-CH ₃ -pyrazol-5-yl-CH (CH ₃ ) - B.2256 4-Br-pyrazol-5-yl-CH _(CH3) B.2257 4-Cl-pyrazol-5-yl-CH _(CH3) B.2258 4-CN-pyrazol-5-yl-CH _(CH3); 0 B.2259 _{4-CH3-pyrazol-5-yl-CH (CH3)} B.2260 1,3- (CH ₃ ) ₂ -pyrazol-5-yl-CH (CH ₃ ); B.2261 1,4- (CH ₃ ) ₂ -pyrazol-5-yl-CH (CH ₃ ) i B.2262 1-CH 3, 3-Cl-pyrazol-5-yl-CH (CH ₃ ) f B.2263 _1-CH3, 4-Cl-pyrazol-5-yl-CH _(CH3) B.2264 1,3,4-oxadiazol-5-yl-CH _(CH3) B.2265 2-CH ₃ -1,3,4-oxadiazol-5-yl-CH (CH ₃ ) B.2266 2-CF ₃ -1,3,4-oxadiazol-5-yl-CH (CH ₃ ) B.2267 2-OCH 3 -1,3,4-oxadiazol-5-yl-CH (CH ₃ ) B.2268 2-C1-1,3,4-oxadiazol-5-yl-CH _(CH3) B.2269 2-CH _(CH3) 2-1,3,4-oxadiazol-5-yl-CH _(CH3) B.2270 1,3,4-oxadiazol-2-yl-CH _(CH3) B.2271 5-CH ₃ -1,3,4-oxadiazol-2-yl-CH (CH ₃ ) B.2272 5-CF ₃ -1,3,4-oxadiazol-2-yl-CH (CH ₃ ) B.2273 5-OCH ₃ -1,3,4-oxadiazol-2-yl-CH (CH ₃ ) B.2274 5-C1-1,3,4-oxadiazol-2-yl-CH _(CH3) B.2275 5-CH _(CH3) 2-1,3,4-oxadiazol-2-yl-CH _(CH3) B.2276 S-C 8 H 8 -1,3,4-oxadiazol-2-yl-CH (CH ₃ ) B.2277 1,2,4-oxadiazol-3-yl-CH _(CH3) B.2278 5-CH ₃ -1,2,4-oxadiazol-3-yl-CH (CH ₃ ) B.2279 5-CF ₃ -1,2,4-oxadiazol-3-yl-CH (CH ₃ ) B.2280 5-OCH ₃ -1,2,4-oxadiazol-3-yl-CH (CH ₃ ) B.2281 5-C1-1,2,4-oxadiazol-3-yl-CH _(CH3) B.2282 5-CH (CH ₃ ) ₂ -1,2,4-oxadiazol-3-yl-CH (CH ₃ )

Nr. R ³ B.2283 1,2,4-triazol- ₃ -ylCH (CH ₃ ) B.2284 1-CH ₃ -1,2,4-triazol- ₃ -ylCH (CH ₃ ) B.2285 5-CH ₃ -1,2,4-triazol- ₃ -ylCH (CH ₃ ) B.2286 5-CF ₃ -1,2,4-triazol-3-yl-CH (CH ₃ ) B.2287 5-OCH ₃ -1,2,4-triazol-3-yl-CH (CH ₃ ) B.2288 5-Cl ', 2,4-triazol- ₃ -ylCH (CH ₃ ) B.2289 5-CH _(CH3) 2-1,2,4-triazole-3-yľCH (CH ₃₎ B.2290 1-C ₆ H ₅ -1,2,4-triazol- ₃ -ylCH (CH ₃ ) B.2291 1,3,4-thiadiazol-5-ylCH (CH ₃ ) B.2292 2-CH ₃ -1,3,4-thiadiazol-5-ylCH (CH ₃ ) B.2293 2-CF ₃ -1,3,4-thiadiazol-5-ylCH (CH ₃ ) B.2294 2-OCH ₃ -1,3,4-thiadiazol-5-yl-CH (CH ₃ ) B.2295 2-CH ₂ OCH ₃ -1,3,4-thiazol-5-yl-CH (CH ₃ ) B.2296 2-C1-1,3,4-thiadiazol-5-yľCH (CH ₃₎ B.2297 2-CH _(CH3) 2-1,3,4-thiadiazol-5-yl-CH _(CH3) B.2298 1,3,4-thiadiazol-2-ylCH (CH ₃ ) B.2299 5-CH ₃ -1,3,4-thiadiazol-2-ylCH (CH ₃ ) B.2300 5-CF ₃ -1,3,4-thiadiazol-2-yl-CH (CH ₃ ) B.2301 5-OCH ₃ -1,3,4-thiadiazol-2-yl-CH (CH ₃ ) B.2302 5-Cl ', 3,4-thiadiazol-2-ylCH (CH ₃ ) B.2303 5-CH _(CH3) 2-1,3,4-thiadiazol-2-yl-CH _(CH3) B.2304 5-C6H5-1,3,4-thiadiazol-2-yl-CH _(CH3) B.2305 1,2,4-thiadiazol- ₃ -ylCH (CH ₃ ) B.2306 5-CH ₃ -1,2,4-thiadiazol-3-yl-CH (CH ₃ ) B.2307 5-CF ₃ -1,2,4-thiadiazol-3-yl-CH (CH ₃ ) B.2308 5-OCH ₃ -1,2,4-thiadiazol- ₃ -ylCH (CH ₃ ) B.2309 5-C1-1,2,4-thiadiazol-3-yľCH (CH ₃₎ B.2310 5-CH _(CH3) 2-1,2,4-thiadiazole-3-yľCH (CH ₃₎ B.2311 pyrrol-2-yl-CH _(CH3) B.2312 4-Cl-pyrrol-2-yl-CH _(CH3) B.2313 4-Br-pyrrol-2-yl-CH _(CH3) B.2314 4-CH ₃ -pyrro-2-yl 1 -CH (CH ₃ ) B.2315 4-C 6 H 5 -pyrrole-2-yl 1 -CH (CH ₃ ) B.2316 benzimidazol-2-yl-CH _(CH3) B.2317 quinolin-2-ylCH (CH ₃ ) B.2318 2-F-C6H4-OCH _(CH3) B.2319 3-FC ₆ H ₄ -OCH (CH ₃₎ B.2320 4-FC ₆ H ₄ -OCH (CH ₃ ) B.2321 2,3-F ₂ -C ₆ H ₃ -OCH (CH ₃ )

-ÍÍ2-

Nr. R ³ B.2322 2,4-F ₂ -C ₆ H ₃ -OCH (CH ₃ ) 5 B.2323 2,5-F ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2324 2,6-F ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2325 3,4-F ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2326 3,5-F ₂ -C ₆ H ₃ -OCH (CH ₃ ) 10 B.2327 2-Cl-C ₆ H ₄ -OCH (CH ₃ ) B.2328 3-Cl-C ₆ H ₄ -OCH (CH ₃ ) B.2329 4-Cl-C ₆ H ₄ -OCH (CH ₃ ) B.2330 2,3-Cl ₂ -C ₆ H ₃ -OCH (CH ₃ ) 15 B.2331 2,4-Cl ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2332 2,5-Cl ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2333 2,6-Cl ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2334 3,4-Cl ₂ C _{fi 3} H OCH (CH ₃₎ 20 B.2335 3,5-Cl ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2336 2,3,4-Cl ₃ -C ₆ H ₂ -OCH (CH ₃ ) B.2337 2,3,5-Cl ₃ -C ₆ H ₂ -OCH (CH ₃ ) B.2338 2,3,6-Cl ₃ -C ₆ H ₂ -OCH (CH ₃ ) B.2339 2,4,5-Cl ₃ -C ₆ H ₂ -OCH (CH ₃ ) 25 B.2340 2,4,6-Cl ₃ -C ₆ H ₂ -OCH (CH ₃ ) B.2341 3,4,5-Cl ₃ -C ₆ H ₂ -OCH (CH ₃ ) B.2342 2-Br-C ₆ H ₄ -OCH (CH ₃ ) B.2343 3-Br-C ₆ H ₄ -OCH (CH ₃ ) 30 B.2344 4-Br-C ₆ H ₄ -OCH (CH ₃ ) B.2345 2,3-Br ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2346 2,4 -Br ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2347 2,5-Br ₂ -C ₆ H ₃ -OCH (CH ₃ ) qc B.2348 2,6-Br ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2349 3,4-Br ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2350 3,5-Br ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2351 2-F, 3-Cl-C ₆ H ₃ OCH (CH ₃₎ B.2352 2-F, 4-Cl-C ₅ H ₃ -OCH (CH ₃ ) 40 B.2353 2-F, 5-Cl-C ₆ H ₃ OCH (CH ₃₎ B.2354 2-F, 3-Br-C ₆ H ₃ -OCH (CH ₃ ) B.2355 2-F, 4-Br-C ₆ H ₃ -OCH (CH ₃ ) B.2356 2-F, 5-Br-C ₆ H ₃ -OCH (CH ₃ ) 45 B.2357 2-C1,3-FC ₆ H ₃ -OCH (CH ₃ ) B.2358 2-C1,4-FC ₆ H ₃ -OCH (CH ₃ ) B.2359 2-Cl, 5-FC ₆ H ₃ -OCH (CH ₃ ) ¹

-} 2i-

Nr. R ³ B.2360 2-Cl, 3-Br-C ₆ H ₃ -OCH (CH ₃ ) B.2361 2-C1, 4-Br-C ₆ H ₃ -OCH (CH ₃ ) ; B.2362 2-C1, 5-Br-C ₆ H ₃ -OCH (CH ₃ ) B.2363 2-Br, 3-FC ₆ H ₃ -OCH (CH ₃ ) B.2364 2-Br, 4-FC ₆ H ₃ -OCH (CH ₃ ) B.2365 2-Br, 5-FC ₆ H ₃ -OCH (CH ₃ ) B, 2366 2-Br, 3-Cl-C ₆ H ₃ -OCH (CH ₃ ) B.2367 2-Br, 4-Cl-C ₅ H ₃ -OCH (CH ₃ ) B.2368 2-Br, 5-Cl-C ₆ H ₃ -OCH (CH ₃ ) B.2369 4-C 1, 3,5-Br ₂ -C ₆ H ₂ OCH (CH ₃₎ B.2370 2-CN-C ₆ H ₄ -OCH (CH ₃ ) B.2371 3-CN-C ₆ H ₄ -OCH (CH ₃ ) B.2372 4-CN-C ₆ H ₄ -OCH (CH ₃ ) B.2373 2-NO ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2374 3-NO ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2375 4-NO ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2376 2-CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2377 3-CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2378 4-CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2379 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2380 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2381 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2382 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2383 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2384 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2385 2-CH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2386 3-CH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2387 4-CH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2388 2-CH (CH ₃ ) ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2389 3 -CH (CH ₃ ) ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2390 4-CH (CH ₃ ) ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2391 3-C (CH ₃ ) ₃ -c ₆ h ₄ -CH (CH ₃ ) B.2392 4-C (ch ₃ ) ₃ -c ₆ h _4- ch (CH ₃ ) B.2393 2-C ₆ H 5 -C ₆ H 4 OCH (CH ₃₎ B.2394 3-C ₆ H ₅ -C ₆ H ₄ -OCH (CH ₃ ) B.2395 4-C ₆ H ₅ -C ₆ H ₄ -OCH (CH ₃ ) B.2396 2-OCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2397 3- and _3- c ₆ h _4- ch (CH ₃ ) B.2398 4-OCH ₃ -C ₆ H ₄ -OCH (CH ₃ )

Nr. R ³ B.2399 2,3- (OCH ₃ , 2 ~ C ₆ H ₃ -OCH (CH ₃ ) B.2400 2,4- (OCH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2401 2,5- (OCH ₃ ) ₂ 'C 6 H ₃ -OCH (CH ₃ ) B.2402 2,6- (OCH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2403 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2404 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -OCH (CH ₃ ) B.2405 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -OCH (CH ₃ ) B.2406 2-OCH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2407 3-OCH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2408 4-OCH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2409 2-0 <ch ₂ ) ₂ ch _{3 -} c ₆ h _{4 -} (CH ₃ ) B.2410 3-0 (ch ₂ ) ₂ ch ₃ -c ₆ h _4- ch (ch ₃ ) B.2411 4-0 (ch ₂ ) ₂ ch ₃ -c ₆ h _4- ch (ch ₃ ) B.2412 2-OCH (CH ₃ ) 2-C ₆ H ₄ -OCH (CH ₃ ) B.2413 3-OCH (CH ₃ ) ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2414 4-OCH (CH ₃ ) 2 -C ₆ H ₄ -OCH (CH ₃ ) B.2415 3-OC (CH ₃ ) ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2416 4-OC (CH ₃ ) ₃ -c ₆ h _4- CH (CH ₃ ) B.2417 2-ch ₂ ch = ch ₂ -c ₆ h _4- ch (ch ₃ ) B.2418 3-ch ₂ ch = ch ₂ -c ₆ h _4- ch (ch ₃ ) B.2419 4-ch ₂ ch = ch ₂ -c ₆ h _4- ch (ch ₃ ) B.2420 2-CF ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2421 3-CF ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2422 4-CF ₃ -C ₆ H ₄ -OCH (CH ₃ ) 1 B.2423 2-CO ₂ CH ₃ -C ₆ H ₄ -OCH (ch ₃ ) B.2424 3-CO ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2425 4-CO ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2426 2 -CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2427 3 -CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2428 4-CO ₂ CH ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) J B.2429 2-CONH ₂ -C ₆ H ₄ -OCH (CH ₃ )! B.2430 3-CONH ₂ -C ₆ H ₄ -OCH (CH ₃ ) i B.2431 4-CONH ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2432 2-con (ch ₃ ) ₂ -c ₆ h ₄ -och (ch ₃ ); B.2433 3-con (ch ₃ ) ₂ -c ₆ h ₄ -och (ch ₃ ); B.2434 4-CON (CH ₃ ) ₂ -C _s H ₄ -OCH (CH ₃ ); B.2435 2-conhch ₃ -c ₆ h _4- ch (ch ₃ ) B.2436 3-conhch ₃ -c ₆ h _4- ch (ch ₃ ) B.2437 4 -CONHCH ₃ -C ₆ H ₄ -OCH (CH ₃₎

- & 5 ~ -

Nr. R ³ B.2438 2-NH ₂ -C ₈ H ₄ -OCH (CH ₃ ) B.2439 3-NH ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2440 4-NH ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2441 2 -N (CH ₃ ) ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2442 3 -N (CH ₃ ) ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2443 4-N (CH ₃ ) ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2444 2-NHCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2445 3-NHCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2446 4-NHCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2447 2-CSNH ₂ 'C ₆ H ₄ -OCH (CH ₃ ) B.2448 3-ennh ₂ -c ₆ h _4- ch (CH ₃ ) B.2449 4-CSNH ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2450 2-SCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2451 3-SCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2452 4-SCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2453 2-SOCH ₃ -C ₆ H ₄ -OCH (ch ₃ ) B.2454 3-SOCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2455 4-SOCH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2456 2-SO ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2457 3-SO ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2458 4-SO ₂ CH ₃ -C ₆ H ₄ -OCH (CH ₃₎ B.2459 2-OCF ₃ -C ₆ H ₄ -OCH (CH ₃ , B.2460 3-OCF ₃ -C ₆ H ₄ -OCH (ch ₃ ) B.2461 4-OCF ₃ -C ₆ H ₄ -OCH (CH ₃₎ B.2462 2-OCHF ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2463 3-OCHF ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2464 4-OCHF ₂ -C ₆ H ₄ -OCH (ch ₃ ) B.2465 3 — CF ₃ , 4-OCF ₃ -C ₆ H ₃ -OCH (CH ₃ ) B.2466 2-CH ₂ CH ₂ FC ₆ H ₄ -OCH (CH ₃ ) B.2467 3-CH ₂ CH ₂ FC ₆ H ₄ -OCH (CH ₃ ) B.2468 4-CH ₂ CH ₂ FC ₆ H ₄ -OCH (ch ₃ ) B.2469 2-CH ₂ CF ₃ , -C ₆ H ₄ -OCH (CH ₃ ) B.2470 3 -CH ₂ CF ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2471 4-CH ₂ CF ₃ -C ₆ H ₄ -OCH (CH ₃ ) B.2472 2-CF ₂ CHF ₂ -C ₈ H ₄ -OCH (CH ₃ ) B.2473 3-CF ₂ CHF _2- C ₆ H ₄ -OCH (CH ₃ ) B.2474 4-CF ₂ CHF ₂ -C ₆ H ₄ -OCH (CH ₃ ) B.2475 2-CHF _2- C ₆ H ₄ -OCH (CH ₃ ) B.2476 3-CHF _2- C ₆ H ₄ -OCH (CH ₃ )

-ΖΖ6-

Nr. p ' B.2477 4 -CHF ₂ -C ₆ H ₄ -OCH (ch ₃ ) B.2478 naphthalin-l-yl-OCH _(CH3) B.2479 naphthalin-2-yl-OCH _(CH3) B.2480 pyridin-2-yl-OCH _(CH3) B.2481 pyridin-3-yl-OCH _(CH3) B.2482 pyridin-4-yl-OCH _(CH3) B.2483 _{5-CH3-pyridin-2-yl-OCH (CH3)} B.2484 _{6-CH3-pyridin-2-yl-OCH (CH3)} B.2485 _{5-CH3-pyridin-3-yl-OCH (CH3)} B.2486 _{6-CH3-pyridin-3-yl-OCH (CH3)} B.2487 5-OCH ₃ -pyridin-2-yl-OCH (CH ₃ ) B.2488 _{6-OCH3-pyridin-2-yl-OCH (CH3)} B.2489 _{5-OCH3-pyridin-3-yl-OCH (CH3)} B.2490 _{6-OCH3-pyridin-3-yl-OCH (CH3)} B.2491 4-Cl-pyridin-2-yl-OCH _(CH3) B.2492 5-Cl-pyridin-2-yl-OCH _(CH3) B.2493 6-Cl-pyridin-2-yl-OCH _(CH3) B.2494 2-C 1 -pyridin-3-yl-OCH (CH ₃ ) B.2495 5-Cl-pyridin-3-yl-OCH _(CH3) B.2496 6-Cl-pyridin-3-yl-OCH _(CH3) B.2497 2-Cl-pyridin-4-yl-OCH _(CH3) B.2498 3,5-Cl ₂ -pyridin-2-yl-OCH _(CH3) B.2499 pyrimidin-2-yl-OCH _(CH3) B.2500 4-Cl-pyrimidin-2-yl-OCH _(CH3) B.2501 5-Cl-pyrimidin-2-yl-OCH _(CH3) B.2502 4-CH ₃ -pyrimidin-2-yl-OCH (CH ₃ ) B.2503 5-CH ₃ -pyrimidin-2-yl-OCH _(CH3) B.2504 4-OCH ₃ -pyrimidin-2-yl-OCH (CH ₃ ) B.2505 5-OCH ₃ -pyrimidin-2-yl-OCH (CH ₃ ) B.2506 4-OCH ₂ CH ₃ -pyrimidin-2-yl-OCH (CH ₃ ) B.2507 5-OCH ₂ CH ₃ -pyrimidin-2-yl-OCH (CH ₃ ) B.2508 pyrimidin-4-yl-OCH _(CH3) B.2509 2-C 1 -pyrimidin-4-yl-OCH (CH ₃ ) B.2510 6-Cl-pyrimidin-4-yl-OCH _(CH3) B.2511 2,6-Cl 2 -pyrimidin-4-yl-OCH (CH ₃ ) B.2512 _2-CH3 -pyrimidin-4-yl-OCH _(CH3) B.2513 6-CH ₃ -pyrimidin-4-yl-OCH (CH ₃ ) B.2514 2-OCH ₃ -pyrimidin-4-yl-OCH (CH ₃ ) B.2515 S-OCH ₃ -pyrimidin-4-yl-OCH (CH ₃ )

-521-

Nr. R ³ B.2516 2-OCH ₂ CH ₃ -pyrimidin-4-yl-OCH (CH ₃ ) B.2517 6-OCH ₂ CH ₃ -pyrimidin-4-yl-OCH (CH ₃ ) ; B.2518 pyrimidin-5-yl-OCH _(CH3) B.2519 2-Cl-pyrimidin-5-yl-OCH _(CH3) B.2520 _2-CH3 -pyrimidin-5-yl-OCH _(CH3) B.2521 2-OCH ₃ -pyrimidin-5-yl-OCH (CH ₃ ) B.2522 2-OCH ₂ CH ₃ -pyrimidin-5-yl 1 -OCH (CH ₃ ) B.2523 furan-2-yl-OCH _(CH3) B.2524 4-Br-furan-2-y1-OCH (CH ₃₎ B.2525 4-Cl-furan-2-yl-OCH _(CH3) B.2526 4-CN-furan-2-yl-OCH _(CH3) B.2527 _{4-CH3-furan-2-yl-OCH (CH3)} B.2528 5-Br-furan-2-yl-OCH _(CH3) B.2529 5-Cl-furan-2-yl-OCH _(CH3) B.2530 5-CN-furan-2-yl-OCH _(CH3) B.2531 _{5-CH3-furan-2-yl-OCH (CH3)} B.2532 furan-3-yl-OC H (CH ₃ ) B.2533 5-Br-furan-3-yl-OCH _(CH3) B.2534 5-Cl-furan-3-yl-OCH _(CH3) B.2535 5-CN-furan-3-y1-OCH (CH ₃₎ B.2536 _{5-CH3-furan-3-yl-OCH (CH3)} B.2537 thien-2-yl-OCH _(CH3) B.2538 4-Br-thien-2-yl-OCH _(CH3) B.2539 4-Cl-thien-2-yl-OCH _(CH3) B.2540 4-CN-thien-2-yl-OCH _(CH3) B.2541 _{4-CH3-thien-2-yl-OCH (CH3)} B.2542 5-Br-thien-2-yl-OCH _(CH3) B.2543 5-Cl-thien-2-yl-OCH _(CH3) B.2544 5-CN-thien-2-yl-OCH _(CH3) B.2545 5-CH ₃ -thien-2-yl-OCH (CH ₃ , B.2546 thien-3-yl-OCH _(CH3) B.2547 5-Br-thien-3-yl-OCH _(CH3) B.2548 5-C1-thien-3-y1-OCH (CH ₃₎ B.2549 5-CN-thien-3-y1-OCH (CH ₃₎ B.2550 5-CH ₃ -thien-3-yl-OCH (CH ₃ ) B.2551 □ xazol-2-yl-OCH (CH ₃ ) B.2552 l-Br-oxazol-2-yl-OCH _(CH3) B.2553 l-Cl-oxazol-2-yl-OCH _(CH3) B.2554 L-CN-oxazol-2-yl-OCH _(CH3)

-Hf-

Nr. R ³ B.2555 4-CH ₃ -oxazol-2-ylCH (CH ₃ ) B.2556 5-Br-oxazol-2-yl-OCH _(CH3) B.2557 5-Cl-oxazol-2-yl-OCH _(CH3) B.2558 5-CN-oxazol-2-yl-OCH _(CH3) B.2559 _{5-CH3-oxazol-2-yl-OCH (CH3)} B.2560 oxazol-4-yl-OCH _(CH3) B. 2561 2-Br-oxazol-4-yl-OCH _(CH3) B.2562 2-Coxazol-4-ylCH (CH ₃ ) B.2563 2-CN-oxazol-4-yl-OCH _(CH3) B.2564 2-CH ₃ -oxazol-4-ylCH (CH ₃ ) B.2565 2-C6H5-oxazol-4-yľOCH (CH ₃₎ B.2566 5-Br-oxazol-4-yľOCH (CH ₃₎ B.2567 5-Coxazol-4-ylCH (CH ₃ ) B.2568 5-CN-oxazol-4-yl-OCH _(CH3) B.2569 _{5-CH3-oxazol-4-yľOCH} (CH ₃₎ B.2570 oxazol-5-yl-OCH _(CH3) B.2571 4-Br-oxazol-5-yľOCH (CH ₃₎ B.2572 4-Coxazol-5-ylCH (CH ₃ ) B.2573 4-CN-oxazol-5-yl-OCH _(CH3) B.2574 _{4-CH3-oxazol-5-yl-OCH (CH3)} B.2575 2-Br-oxazol-5-ylCH (CH ₃ ) B.2576 2-C 1-oxazol-5-yl-OCH (CH ₃ ) B.2577 2-CN-oxazol-5-yl-OCH _(CH3) B.2578 _{2-CH3-oxazol-5-yl-OCH (CH3)} B.2579 isoxazol-3-yl-OCH _(CH3) B.2580 4-Br-isoxazol-3-yl-OCH _(CH3) B.2581 4-Cl-isoxazol-3-yl-OCH _(CH3) B.2582 4-CN-isoxazol-3-yl-OCH _(CH3) B.2583 4-CH ₃ -isoxazol-3-yl-OCH (CH ₃ ) B.2584 5-Br-isoxazol-3-yl-OCH _(CH3) B.2585 5-Cl-isoxazol-3-yl-OCH _(CH3) B.2586 5-CN-isoxazol-3-ylCH (CH ₃ ) B.2587 5-CH ₃ -isoxazol-3-yl-OCH (CH ₃ ) B.2588 isoxazol-4-yl-OCH _(CH3) B.2589 3-Br-isoxazol-4-yl-OCH _(CH3) B.2590 3-Cl-isoxazol-4-yl-OCH _(CH3) B.2591 3-CN-isoxazol-4-yl-OCH _(CH3) B.2592 3-CH ₃ -isoxazol-4-yl-OCH (CH ₃ ) B.2593 5-Br-isoxazol-4-yl-OCH _(CH3)

- Μί-

Nr. R ³ B.2594 5-Cl-isoxazol-4-yl-OCH _(CH3) B.2595 5-CN-isoxazol-4-yl-OCH _(CH3) B.2596 _{5-CH3-isoxazol-4-yl-OCH (CH3)} B.2597 3,5- _{(CH3) 2-isoxazol-4-yl-OCH (CH3)} B.2598 isoxazol-5-yl-OCH _(CH3) B.2599 3-Br-isoxazol-5-yl-OCH _(CH3) B.2600 3-Cl-isoxazol-5-yl-OCH _(CH3) B.2601 3-CN-isoxazol-5-yl-OCH _(CH3) B.2602 3-CH ₃ -isoxazol-5-yl-OCH (CH ₃ ) B.2603 3-C 6 H-isoxazol-5-yl-OCH _(CH3) B.2604 4-C1-C 6 H 3-isoxazol-5-yl-OCH _(CH3) B.2605 4-Br, 3-C6H5-isoxazol-5-yl-OCH _(CH3) B.2606 4-Br-isoxazol-5-yl-OCH _(CH3) B.2607 4-Cl-isoxazol-5-yl-OCH _(CH3) B.2608 4-CN-isoxazol-5-yl-OCH _(CH3) B.2609 _{4-CH3-isoxazol-5-yl-OCH (CH3)} B.2610 thiazol-2-yl-OCH _(CH3) B.2611 4-Br-thiazol-2-yl-OCH _(CH3) B.2612 4-Cl-thiazol-2-yl-OCH _(CH3) B.2613 4-CN-thiazol-2-yl-0CH (CH ₃₎ B.2614 _{4-CH3-thiazol-2-yl-OCH (CH3)} B.2615 5-Br-thiazol-2-yl-OCH _(CH3) B.2616 5-Cl-thiazol-2-yl-OCH _(CH3) B.2617 5-CN-thiazol-2-yl-OCH _(CH3) B.2618 5-CH ₃ -thiazol-2-yl-OCH (CH ₃ ) B.2619 thiazol-4-yl-OCH _(CH3) B.2620 2-Br-thiazol-4-yl-OCH _(CH3) B.2621 2-Cl-thiazol-4-yl-OCH _(CH3) B.2622 2-CN-thiazol-4-yl-0CH (CH ₃₎ B.2623 _{2-CH3-thiazol-4-yl-OCH (CH3)} B.2624 5-Br-thiazol-4-yl-OCH _(CH3) B.2625 5-Cl-thiazol-4-yl-OCH _(CH3) B.2626 5-CN-thiazol-4-yl-OCH _(CH3) B.2627 5 -CH ₃ -thi and zo-4-yl-OCH (CH ₃ ) B.2628 thiazol-5-yl-OCH _(CH3) B.2629 l-Br-thiazol-5-yl-OCH _(CH3) B.2630 l-Cl-thiazol-5-yl-OCH _(CH3) B.2631 L-CN-thiazol-5-yl-OCH _(CH3) B.2632 1-CH ₃ -thiazol-5-yl-OCH (CH ₃ )

-35ο-

Nr. R ³ B.2633 2-Br-thiazol-5-yl-OCH _(CH3) B.2634 2-Cl-thiazol-5-yl-OCH _(CH3) j B.2635 2-CN-thiazol-5-yl-OCH _(CH3) B.2636 _{2-CH3-thiazol-5-yl-OCH (CH3)} B.2637 isothiazol-3-yl-OCH _(CH3) B.2638 4-Br-isothiazol-3-yl-OCH _(CH3) B.2639 4-Cl-isothiazol-3-yl-OCH _(CH3) B.2640 4-CN-isothiazol-3-yl-OCH _(CH3) B.2641 4-CH ₃ -isothiazol-3-yl-OCH (CH ₃ ) B.2642 5-Br-isothiazol-3-yl-OCH _(CH3) B.2643 5-Cl-isothiazol-3-yl-OCH _(CH3) B.2644 5-CN-isothiazol-3-yl-OCH _(CH3) B.2645 5-CH ₃ -isothiazol-3-yl-OCH (CH ₃ ) B.2646 isothiazol-4-yl-OCH _(CH3) B.2647 3-Br-isothiazol-4-yl-OCH _(CH3) B.2648 3-Cl-isothiazol-4-yl-OCH _(CH3) B.2649 3-CN-isothiazol-4-yl-OCH _(CH3) B.2650 3-CH ₃ -isothiazol-4-yl-OCH (CH ₃ ) B.2651 5-Br-isothiazol-4-yl-OCH _(CH3) B.2652 5-Cl-isothiazol-4-yl-OCH _(CH3) B.2653 5-CN-isothiazol-4-yl-OCH _(CH3) B.2654 5-CH ₃ -isothiazol-4-yl-OCH (CH ₃ ) B.2655 3,5- (CH ₃ ) ₂ -isothiazol-4-yl-OCH (CH ₃ ) B.2656 isothiazol-5-yl-OCH _(CH3) B.2657 3-Br-isothiazol-5-yl-OCH _(CH3) B.2658 3-Cl-isothiazol-5-yl-OCH _(CH3) B.2659 3-CN-isothiazol-5-yl-OCH _(CH3) B.2660 3-CH ₃ -isothiazol-5-yl-OCH (CH ₃ ) B.2661 4-Br-isothiazol-5-yl-OCH _(CH3) B.2662 4-Cl-isothiazol-5-yl-0CH (CH ₃₎ B.2663 4-CN-isothiazol-5-yl-OCH _(CH3) B.2664 4-CH ₃ -isothiazol-5-yl-OCH (CH ₃ ) B.2665 imidazol-2-yl-OCH _(CH3) B.2666 l-Cl-imidazol-2-yl-0CH (CH ₃₎ B.2667 l-Br-imidazol-2-yl-OCH _(CH3) B.2668 L-CN-imidazol-2-yl-OCH _(CH3) B.2669 1-CH ₃ -irtiidazol-2-yl-OCH (CH ₃ ) B.2670 I-Cl-imidazol-2-yl-0CH (CH ₃₎ ¹ B.2671 l-Br-imidazol-2-ethyl-OCH (CH ₃₎

- /// -

Nr. R ³ B.2672 4-CN-imidazol-2-yl-OCH _(CH3) B.2673 4-CH ₃ -imidazol-2-yl-OCH (CH ₃ ) B.2674 _1-CH3, 5-Cl-imidazol-2-yl-OCH _(CH3) B.2675 1,4- (CH ₃ ) ₂ -imidazol-2-yl-OCH (CH ₃ ) B.2676 1,5- (CH ₃ ) ₂ -imidazol-2-yl-OCH (CH ₃ ) B.2677 imidazol-4-yl-OCH _(CH3) B.2678 2-Cl-imidazol-4-ylCH (CH ₃ ) B.2679 2-Br-imidazol-4-yl-OCH _(CH3) B.2680 2-CN-imidazol-4-yl-OCH _(CH3) B.2681 1-CH ₃ -imidazol-4-yl-OCH (CH ₃ ) B.2682 2-CH ₃ -imidazol-4-yl-OCH (CH ₃ ) B.2683 5-Cl-imidazol-4-yl-OCH _(CH3) B.2684 5-Br-imidazol-4-yl-OCH _(CH3) B.2685 5-CN-imidazol-4-yl-OCH _(CH3) B.2686 5-CH ₃ -imidazol-4-yl-OCH (CH ₃ ) B.2687 _1-CH3, 5-Cl-imidazol-4-yl-OCH _(CH3) B.2688 1,2- _(CH3) 2 ^- imidazol-4-yl-OCH _(CH3) B.2689 1,5- (CH ₃ ) ₂ -imidazol-4-yl-OCH (CH ₃ ) B.2690 pyrazol-3-yl-OCH _(CH3) B.2691 5-Br-pyrazol-3-y1-OCH (CH ₃₎ B.2692 5-Cl-pyrazol-3-ylCH (CH ₃ ) B.2693 5-CN-pyrazol-3-yl-OCH _(CH3) B.2694 5-CH ₃ -pyrazol-3-yl-OCH (CH ₃ ) B.2695 1-C 6 H 5 -pyrazol-3-yl-OCH (CH ₃ ) B.2696 4-Br-pyrazol-3-yl-OCH _(CH3) B.2697 4-Cl-pyrazol-3-yl-OCH _(CH3) B.2698 4-CN-pyrazol-3-yl-OCH _(CH3) B.2699 4-CH ₃ -pyrazol-3-yl-OCH (CH ₃ ) B.2700 1-CH ₃ -pyrazol-3-yl-OCH (CH ₃ ) B.2701 1, 4- _{(CH3) 2-pyrazol-3-yl-OCH (CH3)} B.2702 1,5- _{(CH3) 2-pyrazol-3-yl-OCH (CH3)} B.2703 1-CH ₃ , 4-Cl-pyrazol-3-yl-OCH (CH ₃ ) B.2704 1-CH ₃ , 5-Cl-pyrazol-3-yl-OCH (CH ₃ ) B.2705 pyrazol-4-yl-OCH _(CH3) B.2706 3-Br-pyrazol-4-yl-OCH _(CH3) B.2707 3-Cl-pyrazol-4-yl-OCH _(CH3) B.2708 3-CN-pyrazol-4-yl-OCH _(CH3) B.2709 _{3-CH3-pyrazol-4-yl-OCH (CH3)} B.2710 1-CH ₃ -pyrazol-4-yl-OCH (CH ₃ )

-Ž52-

Nr. R ³ B.2711 1,5- _{(CH3) 2-pyrazol-4-yl-OCH (CH3)} B.2712 1, 3 - _(CH3) 2-pyrazol-1-4 from 1-yl OCH (CH ₃₎ ; B.2713 1-CH ₃ , 3-Cl-pyrazol-4-yl-OCH (CH ₃ ) B.2714 1-CH ₃ , 5-Cl-pyrazol-4-yl-OCH (CH ₃ ) B.2715 pyrazol-5-yl-OCH _(CH3) B.2716 3-Br-pyrazol-5-yl-OCH _(CH3) B.2717 3-Cl-pyrazol-5-yl-OCH _(CH3) B.2718 3-CN-pyrazol-5-yl-OCH _(CH3) B.2719 3-CH ₃ -pyrazol-5-yl-OCH (CH ₃ ) B.2720 1-CH ₃ -pyrazol-5-yl-OCH (CH ₃ ) B.2721 4-Br-pyrazol-5-yl-OCH _(CH3) B.2722 4-Cl-pyrazol-5-yl-OCH _(CH3) B.2723 4-CN-pyrazol-5-yl-0CH (CH ₃₎ B.2724 4-CH ₃ -pyrazol-5-yl-OCH (CH ₃ ) B.2725 1,3- _{(CH3) 2-pyrazol-5-yl-OCH (CH3)} B.2726 1,4- _{(CH3) 2-pyrazol-5-yl-OCH (CH3)} B.2727 1-CH ₃ , 3-Cl-pyrazol-5-yl-OCH (CH ₃ ) B.2728 1-CH ₃ . 4-Cl-pyrazol-5-yl-OCH _(CH3) B.2729 1,3,4-oxadiazol-5-yl-0CH (CH ₃₎ B.2730 2-CH ₃ -1,3,4-oxadiazol-5-yl-OCH (CH ₃ ) B.2731 2-CF 3 -1,3,4-oxadiazol-5-yl-OCH (CH ₃ ) B.2732 2-OCH ₃ -1,3,4-oxadiazol-5-yl-OCH (CH ₃ ) B.2733 2-C1-1,3,4-oxadiazol-5-yl-OCH _(CH3) B.2734 2-CH _(CH3) 2-I / 3,4-oxadiazol-5-yl-OCH _(CH3) B.2735 1,3,4-oxadiazol-2-yl-0CH (CH ₃₎ B.2736 5-CH ₃ -1,3,4-oxadiazol-2-yl-OCH (CH ₃ ) B.2737 5-CF 3 -1,3,4-oxadiazol-2-yl-OCH (CH ₃ ) B.2738 5-OCH ₃ -1,3,4-oxadiazol-2-yl-OCH (CH ₃ ) B.2739 5-C1-1,3,4-oxadiazol-2-yl-OCH _(CH3) B.2740 5-CH _(CH3) 2-1,3,4-oxadiazol-2-yl-OCH _(CH3) B.2741 5-C ₆ H ₅ -1,3,4-oxadiazol-2-yl-OCH (CH ₃ ) B.2742 1,2,4-oxadiazol-3-yl-OCH _(CH3) B.2743 5-CH ₃ -1,2,4-oxadiazol-3-yl-OCH (CH ₃ ) B.2744 5-CF ₃ -1,2,4-oxadiazol-3-yl-OCH (CH ₃ ) B.2745 5-OCH ₃ -1,2,4-oxadiazol-3-yl-OCH (CH ₃ ) B.2746 5-C1-1,2,4-oxadiazol-3-yl-OCH _(CH3) B.2747 5-CH _(CH3) 2-I, 2,4-oxadiazol-3-yl-OCH _(CH3) B.2748 1,2,4-triazol-3-yl-OCH _(CH3) B.2749 L-CH ₃ -1,2,4-triazol-3-yl-OCH (CH ₃ )

Nr. R ³ B.2750 5-CH3-I, 2,4-triazol-3-yl-OCH _(CH3) B.2751 5-CF ₃ -1,2,4-triazol-3-yl-OCH (CH ₃ ) B.2752 5-OCH ₃ -1,2,4-triazol-3-yl-OCH (CH ₃ ) B.2753 5-C1-1,2,4-triazol-3-yl-OCH _(CH3) B.2754 5-CH _(CH3) 2-1,2,4-triazol-3-yl-OCH _(CH3) B.2755 1C ₆ H ₅ -1,2,4-triazol-3-yl-OCH (CH ₃ ) B.2756 1,3,4-thiadiazol-5-yl-OCH _(CH3) B.2757 2-CH ₃ -1,3,4-thiadiazol-5-yl-OCH (CH ₃ ) B.2758 2-CF ₃ -1,3,4-thiadiazol-5-yl-OCH (CH ₃ ) B.2759 2-OCH ₃ -1,3,4-thiadiazol-5-yl-OCH (CH ₃ ) B.2760 2-CH ₂ OCH ₃ -1,3,4-thiadiazol-5-yl-OCH (CH ₃ ) B.2761 2-C1-1,3,4-thiadiazol-5-yl-OCH _(CH3) B.2762 2-CH (CH ₃ ) ₂ -1,3,4-thiadiazol-5-yl-OCH (CH ₃ ) B.2763 1,3,4-thiadiazol-2-yl-OCH _(CH3) B.2764 5-CH ₃ -1,3,4-thiadiazol-2-yl-OCH (CH ₃ ) B.2765 5-CF ₃ -1,3,4-thiadiazol-2-yl-OCH (CH ₃ ) B.2766 _5-OCH3 -1,3,4-thiadiazol-2-yl-OCH _(CH3) B.2767 5-C1-1,3,4-thiadiazol-2-yl-OCH _(CH3) B.2768 5-CH (CH ₃ ) ₂ -1,3,4-thiadiazol-2-yl-OCH (CH ₃ ) B.2769 5-C ₆ H ₅ -1,3,4-thiadiazol-2-yl-OCH (CH ₃ ) B.2770 1,2,4-thiadiazol-3-yl-OCH _(CH3) B.2771 5-CH ₃ -1,2,4-thiadiazol-3-yl-OCH (CH ₃ ) B.2772 5-CF ₃ -1,2,4-thiadiazol-3-yl-OCH (CH ₃ ) B.2773 5-OCH ₃ -1,2,4-thi adi az 01-3 -y 1 -OCH (CH ₃ ) B.2774 5-C1-1,2,4-thiadiazol-3-yl-OCH _(CH3) B.2775 5-CH (CH ₃ ) ₂ -1,2,4-thiadiazol-3-yl-OCH (CH ₃ ) B.2776 pyrrol-2-yl-OCH _(CH3) B.2777 4-C1-Y1-pyrro1-2-OCH (CH ₃₎ B.2778 4-Br-pyrrol-2-yl-OCH _(CH3) B.2779 4-CH ₃ -pyrrol-2-yl-OCH (CH ₃ ) B.2780 4-C ₆ H ₅ -pyrrol-2-yl-OCH (CH ₃ ) B.2781 □ benzimidazole-2-yl-OCH _(CH3) B.2782 quinolin-2-yl-0CH (CH ₃₎ B.2783 ch = ch ₂ B.2784 C (CH ₃ ) = CH ₂ B.2785 CH-CH _(CH3) (E) B.2786 CH-CH _(CH3) (Z) B.2787 ch ₂ ch = ch ₂ B.2788 3 (CH ₂ CH ₃ ) = CH ₂

Nr. R ³ B.2789 C (CH ₃ ) = CH (CH ₃ ) (E) B.2790 C _(CH3) CH _(CH3) (Z) 5 B.2791 C (CH ₃ ) = C (CH ₃ ) ₂ B.2792 CH _(CH3) CH = CH ₂ B.2793 CH = C _{(CH3) 2} B.2794 CH ₂ -C (CH ₃ ) = CH ₂ B.2795 CH (CH ₃ ) -ch ₂ -ch = ch ₂ B.2796 ch ₂ -ch (ch ₃ ) -ch = ch ₂ B.2797 ch ₂ ccl = ch ₂ B.2798 CH ₂ CH = CHCl (E) B.2799 CH ₂ CH = CHCl (Z) B.2800 CH ₂ CC 1 = CHCl 1 (E) B.2801 CH ₂ CC 1 = CHCl 1 (Z) B.2802 CH ₂ CH = CC _{1 2} B.2803 ch ₂ cci = cci ₂ B.2804 CH ₂ CBr = CH ₂ B.2805 CH ₂ CH = CHBr (E) B.2806 CH ₂ CH = CHBr (Z) B.2807 CH ₂ CBr = CHBr (E) B.2808 CH ₂ CBr = CHBr (Z) B.2809 CH ₂ CH = CBr ₂ B.2810 CH ₂ CBr = CBr ₂ B.2811 CH ₂ CH = CHCH ₃ (E) B.2812 CH ₂ CH = CHCH ₃ (Z) B.2813 CH ₂ C (CH ₃ ) = CHCH ₃ (E) B.2814 CH ₂ C (CH ₃ ) = CHCH ₃ (Z) B.2815 CH ₂ CH = C (CH ₃ ) ₂ B.2816 ch ₂ ch ₂ ch = ch ₂ B.2817 CH ₂ CC 1 = CHCH ₃ (E) B.2818 CH ₂ CC 1 = CHCH ₃ (Z) B.2819 CH ₂ CH = CC ₁ CH ₃ (E) B.2820 CH ₂ CH = CC ₁ CH ₃ (Z) B.2821 CH ₂ C (CH ₃ ) = C (CH ₃ ) ₂ B.2822 CH ₂ CBr = CHCH ₃ (E) B.2823 CH ₂ CBr = CHCH ₃ (Z) B.2824 2H ₂ = CH ₃ CBrCH (E) B.2825 2H ₂ = CH ₃ CBrCH (Z) B.2826 3 H ₂ CH = CHCH ₂ C 1 (E) B.2827 h ₂ ch = chch ₂ ci (z)

-535--

Nr. R ³ B.2828 CH ₂ CH = CH ₂ CH ₃ (E) B.2829 CH ₂ CH = CH ₂ CH ₃ (Z) 5 B.2830 CH ₂ CH = CHCH ₂ Br (E) B.2831 CH ₂ CH = CHCH ₂ Br (Z) B.2832 CH ₂ CC 1 = CC 1 CH ₂ C1 (E) B.2833 CH ₂ CC 1 = CC 1 CH ₂ C1 (Z) B.2834 J ch ₂ cf = ch ₂ B.2835 CH ₂ CH = CHF B.2836 CH ₂ CH = CHF (C) B.2837 ch ₂ ch = cf ₂ B.2838 ch ₂ cf = chf B.2839 ch ₂ cf = chf B.2840 CH (CH ₃ ) CH = CH ₂ B.2841 CH (CH ₃ ) CC 1 = CH ₂ B.2842 CH _(CH3) CH = CHC1 (E) B.2843 CH _(CH3) CH = CHC1 (z) B.2844 CH (CH ₃ ) CC 1 = CHCl 1 (E) B.2845 CH (CH ₃ ) CC 1 = CHCl 1 (Z) B.2846 CH _(CH3) CH = CC1 ₂ B.2847 CH (CH ₃ ) CC 1 = CC _{1 2} B.2848 CH _(CH3) CBr = CH ₂ B.2849 CH _(CH3) CH = CHBr (E) B.2850 CH _(CH3) CH = CHBr (Z) B.2851 CH _(CH3) CBr = CHBr (E) B.2852 CH _(CH3) CBr = CHBr (Z) B.2853 CH (CH ₃ ) CH = CBr ₂ B.2854 CH _(CH3) CBr = CBr ₂ B.2855 CH (CH ₃ ) C (CH ₃ ) = CH ₂ B.2856 CH _(CH3) CH = CHCH ₃ (E) B.2857 CH _(CH3) CH = CHCH ₃ (Z) B.2858 CH _(CH3) C (CH ₃₎ = CHCH ₃ (E) B.2859 CH _(CH3) C (CH ₃₎ = CHCH ₃ (Z) B.2860 CH (CH ₃ ) CH = C (CH ₃ ) ₂ B.2861 CH (CH ₃ ) CC 1 = CHCH ₃ (E) B.2862 CH (CH ₃ ) CC 1 = CHCH ₃ (Z) B.2863 CH _(CH3) CH = CC1CH ₃ (E) B.2864 ( : h (ch ₃ ) ch = cca ₃ (z) B.2865 ( CH _(CH3) CBr = CHCH ₃ (E) B.2866 C 1 H (CH ₃ ) CBr = CHCH ₃ (Z)

Nr. I ^r3 B.2867 J CH _(CH3) CH = CBrCH ₃ (E) B.2868 | CH (CH _{3) 3} CH = CBrCH (Z) B.2869 | ch (ch ₃ ) ch = chch ₂ or (E) B.2870 | ch (ch ₃ ) ch = chch ₂ or (Z) B.2871 1 CH (CH ₃ ) CH = CHCH ₂ CH ₃ (E) B.2872 j CH (CH ₃ ) CH = CHCH ₂ CH ₃ (Z) B.2873 j CH (CH ₃₎ CH = CHCH ₂ Br (E) B.2874 j CH (CH ₃ ) CH = CHCH ₂ Br (Z) B.2875 Jch (ch ₃ ) cci = cca ₂ ci (E) B.2876 | ch (ch ₃ ) cci = cca ₂ ci (Z) B.2877 | CH _(CH3) CF = CH ₂ B.2878 , CH (CH ₃₎ CH = CHF (E) B.2879 | CH _(CH3) CH = CHF (Z) B.2880 | CH _(CH3) CH = CF ₂ B.2881 JCH _(CH3) CF = CHF (E) B.2882 | CH _(CH3) CF = CHF (Z) B.2883 Jch ₂ want = ch ₂ B.2884 1CH ₂ CH ₂ CH = C (CH ₃ ) 2 B.2885 | ch ₂ ch _{2 c 3} ) = ch ₃ (E) B.2886 1 ch ₂ ch ₂ c (ch ₃ ) = ch ₃ (Z) B.2887 [2-FC ₆ H ₄ CH = CH B.2888 3-fc ₆ h ₄ -ch = ch B.2889 14-FC ₆ H ₄ -CH = CH B.2890 12,3-F ₂ -C ₆ H ₃ -CH = CH B.2891 1,2,4-F ₂ -C ₆ H ₃ -CH = CH B.2892 1 2,5-F ₂ -C ₆ H ₃ -CH = CH B.2893 J 2 _R 6 F ₂ -C ₆ H 3 -CH-CH B.2894 J 3,4-F ₂ -C ₆ H ₃ -CH = CH B.2895 J 3,5-F ₂ -C ₆ H ₃ -CH = CH B.2896 2-ci-c _with h ₄ -ch = ch B.2897 | 3-C 1-C ₆ H ₄ CH = CH B.2898 1 4-Cl-C ₆ H ₄ CH = CH B.2899 J 2.3-Cl ₂ -C ₆ H ₃ -CH = CH B.2900 12,4-Cl ₂ -C ₆ H ₃ -CH = CH B.2901 12,5-Cl ₂ -C ₆ H ₃ -CH = CH B.2902 | 2,6-Cl ₂ -C ₆ H ₃ -CH = CH B.2903 13,4-Cl ₂ -C ₆ H ₃ -CH = CH B.2904 J 3,5-Cl ₂ -C ₆ H ₃ -CH = CH B.2905 1,2,3,4-Cl ₃ -C ₆ H ₂ -CH = CH

-3sy-

Nr. R ³ B.2906 2,3,5-Cl ₃ -C ₆ H ₂ -CH = CH B.2907 2,3,6-Cl ₃ -C ₆ H ₂ -CH = CH _; B.2908 2,4,5-Cl ₃ -C ₆ H ₂ -CH = CH B.2909 2,4,6-Cl ₃ -C ₆ H ₂ -CH = CH B.2910 3,4,5-Cl ₃ -C ₆ H ₂ -CH = CH B.2911 2-Br-C ₆ H ₄ CH = CH B.2912 3-Br-C ₆ H ₄ CH = CH B.2913 4-Br-C ₆ H ₄ CH = CH B.2914 2,3-Br ₂ -C ₆ H ₃ -CH = CH B.2915 2,4-Br ₂ -C ₆ H ₃ -CH = CH B.2916 2,5-Br ₂ -C ₆ H ₃ -CH = CH B.2917 2,6-Br ₂ -C ₆ H ₃ -CH = CH B.2918 3,4-Br ₂ -C ₆ H ₃ -CH = CH B.2919 3,5-Br ₂ -C ₆ H ₃ -CH = CH B.2920 2-F, 3-Cl-C ₆ H ₃ CH = CH B.2921 2-F, 4-Cl-C ₆ H ₃ CH = CH B.2922 2-F, 5-Cl-C ₆ H ₃ CH = CH B.2923 2-F, 3-Br-C ₆ H ₃ CH = CH B.2924 2-F, 4-Br-C ₆ H ₃ CH = CH B.2925 2-F, 5-Br-C ₆ H ₃ CH = CH B.2926 2-Cl, 3-FC ₆ H ₃ -CH = CH B.2927 2-Cl, 4-FC ₆ H ₃ -CH = CH B.2928 2-Cl, 5-FC ₆ H ₃ -CH = CH B.2929 2-C1, 3-Br-C ₆ H ₃ CH = CH B.2930 2-C1, 4-Br-C ₆ H ₃ CH = CH B.2931 2-C1, 5-Br-C ₆ H ₃ CH = CH B.2932 2-Br, 3-FC ₆ H ₃ -CH = CH B.2933 2-Br, 4-FC ₆ H ₃ -CH = CH B.2934 2-Br, 5-FC ₆ H ₃ -CH = CH B.2935 2-Br, 3-Cl-C ₆ H ₃ CH = CH B.2936 2-Br, 4-Cl-C ₆ H ₃ CH = CH B.2937 2-Br, 5-Cl-C ₆ H ₃ CH = CH B.2938 4-Cl, 3,5-Br ₂ -C ₆ H ₂ -CH = CH B.2939 2-CN-C ₆ H ₄ CH = CH B.2940 3-CN-C ₆ H ₄ CH = CH B.2941 4-CN-C ₆ H ₄ CH = CH B.2942 2-NO ₂ -C ₆ H ₄ -CH = CH B.2943 3-NO ₂ -C ₆ H ₄ -CH = CH B.2944 i-no _{2 -} c ₆ h ₄ - ch = ch

Nr. R ³ B.2945 2-CH ₃ -C ₆ H ₄ -CH = CH B.2946 3-CH ₃ -C ₆ H ₄ -CH = CH . B.2947 4-CH ₃ -C ₆ H ₄ -CH = CH B.2948 2,3- (CH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2949 2,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2950 2,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2951 2,6- (CH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2952 3,4- (CH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2953 3,5- (CH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2954 2-CH ₂ CH ₃ -C ₆ H ₄ -CH = CH B.2955 3 -ch ₂ ch ₃ -c ₆ h ₄ -ch = ch B.2956 4 -CH ₂ CH ₃ -C ₆ H ₄ -ch = ch B.2957 2-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH B.2958 3-CH (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH B.2959 4-CH (CH ₃ ) ₂ -C ₈ H ₄ -CH = CH B.2960 3-C (CH ₃ ) ₃ -C ₆ H ₄ -CH = CH B.2961 4-C (CH ₃ ) ₃ -C ₆ H ₄ -CH = CH B.2962 2-C ₆ H ₅ -C ₆ H ₄ CH = CH B.2963 3-C ₆ H ₅ -C ₆ H ₄ CH = CH B.2964 4-C ₆ H ₅ -C ₆ H ₄ CH = CH B.2965 2-OCH ₃ -C ₆ H ₄ -CH = CH B.2966 3-OCH ₃ -C ₆ H ₄ -CH = CH B.2967 4-OCH ₃ -C ₆ H ₄ -CH = CH B.2968 2,3- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2969 2,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2970 2,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2971 2,6- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2972 3,4- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2973 3,5- (OCH ₃ ) ₂ -C ₆ H ₃ -CH = CH B.2974 3,4,5- (OCH ₃ ) ₃ -C ₆ H ₂ -CH = CH B.2975 2-OCH ₂ CH ₃ -C ₆ H ₄ -CH = CH B.2976 3-a ₂ ch ₃ -c ₆ h ₄ -ch = ch B.2977 4 -och ₂ ch ₃ -c ₆ h ₄ -ch = ch B.2978 2-O (CH ₂ ) ₂ CH ₃ -C ₆ H ₄ -CH = CH B.2979 3-0 (CH ₂ ) ₂ ch ₃ -c ₆ h ₄ -ch = ch B.2980 4-0 (CH ₂ ) ₂ CH ₃ -C ₆ H ₄ -CH = CH B.2981 2-OCH (CH ₃ ) ₂ -c ₆ h ₄ -ch = ch B.2982 _3- CH (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH B.2983 4-OCH (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH

-Z Zq -

1 Nr. R ³ j B.2984 3-OC (CH ₃ ) ₃ -c ₆ h ₄ -ch = ch j B.2985 4-OC (CH ₃ ) ₃ -c ₆ h ₄ -ch = ch ₅ B.2986 2-ch ₂ ch = ch ₂ -c ₆ h ₄ -ch = ch | B.2987 3-ch ₂ ch = ch ₂ -c ₆ h ₄ -ch = ch 1 B.2988 4-ch _2- ch = ch ₂ -c ₆ h ₄ -ch = ch j B.2989 2-CF ₃ -C ₆ H ₄ -CH = CH B.2990 3-CF ₃ -C ₆ H ₄ -CH = CH | B.2991 4-CF ₃ -C ₆ H ₄ -CH = CH J B.2992 2-co ₂ ch ₃ -c ₆ h ₄ -ch = ch J B.2993 3 -co ₂ ch ₃ -c ₆ h ₄ -ch = ch 1 B.2994 4-co ₂ ch ₃ -c ₆ h ₄ -ch = ch ⁵ B.2995 2 -co ₂ ch ₂ ch ₃ -c ₆ h ₄ -ch = ch j B.2996 3 -co ₂ ch ₂ ch ₃ -c ₆ h ₄ -ch = ch 1 B.2997 4 -co ₂ ch ₂ ch ₃ -c ₆ h ₄ -ch = ch | B.2998 2-conh ₂ -c ₆ h ₄ -ch = ch ) B.2999 3-CONH ₂ -C ₆ H ₄ -CH = CH j B.3000 4 -CONH ₂ -C ₆ H ₄ CH = CH J B.3001 2 -CON (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH 1 B.3002 3-CON (CH ₃ ) ₂ -c ₆ h ₄ -ch = ch B.3003 4-CON (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH | B.3004 _{2-CONHCH3-C 6} H ₄ CH = CH | B.3005 _{3-CONHCH3-C 6} H ₄ CH = CH 1 B.3006 _{4-CONHCH3-C 6} H ₄ CH = CH J B.3007 2-NH ₂ -C ₆ H ₄ -CH = CH j B.3008 3-NH ₂ -C ₆ H ₄ -CH = CH 1 B.3009 _{4-NH2-C s} H ₄ CH = CH j B.3010 2-N (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH 1 B.3011 3 -N (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH j B.3012 4-N (CH ₃ ) ₂ -C ₆ H ₄ -CH = CH j B.3013 2-NH-CH ₃ -C ₆ H ₄ CH = CH | B.3014 3-NH-CH ₃ -C ₆ H ₄ CH = CH 1 B.3015 4-NHCH ₃ -C ₆ H ₄ -CH = CH 1 B.3016 2-CSNH ₂ -C ₆ H ₄ -CH = CH 1 B.3017 3-csnh ₂ -c ₆ h ₄ -ch = ch B.3018 4-csnh ₂ -c ₆ h ₄ -ch = ch B.3019 2-SCH ₃ -C ₆ H ₄ -CH = CH B.3020 3-SCH ₃ -C ₆ H ₄ -CH = CH B.3021 4-SCH ₃ -C ₆ H ₄ -CH = CH B.3022 2-sculpture ₃ -c ₆ h ₄ -ch = ch

Nr. R ³ B.3023 3-SOCH ₃ -C ₆ H ₄ -CH = CH B.3024 4-sculpture ₃ -c ₆ h ₄ -ch = ch B.3025 2 -so ₂ ch ₃ -c ₆ h ₄ -ch = ch B.3026 3-SO ₂ CH ₃ -C ₆ H 4 -CH = CH B.3027 4-SO ₂ CH ₃ -C ₆ H ₄ -CH = CH B.3028 2-OCF ₃ -C ₆ H ₄ -CH = CH B.3029 3-OCF ₃ -C ₆ H ₄ -CH = CH B.3030 4-OCF ₃ -C ₆ H ₄ -CH = CH B.3031 2 -OCHF ₂ -C ₆ H ₄ -CH = CH B.3032 3 -OCHF ₂ -C ₆ H ₄ CH = CH B.3033 4-ochf ₂ -c ₆ h ₄ -ch = ch B.3034 3-CF ₃ , 4-OCF ₃ -C ₆ H ₃ -CH = CH B.3035 2-ch ₂ ch ₂ fc ₆ h ₄ -ch = ch B.3036 3-ch ₂ ch ₂ fc ₆ h ₄ -ch = ch B.3037 4-ch ₂ ch ₂ fc ₆ h ₄ -ch = ch B.3038 2-CH ₂ CF ₃ -C ₆ H ₄ -CH = CH B.3039 3 -CH ₂ CF ₃ -C ₆ H ₄ -CH = CH B.3040 4-CH ₂ CF ₃ -C ₆ H ₄ -CH = CH B.3041 2 - cf ₂ chf _{2 -} c ₆ h ₄ - ch = ch B.3042 3-CF ₂ CHF ₂ -C ₆ H ₄ CH = CH B.3043 4-CF ₂ CHF ₂ -C ₆ H ₄ -CH = CH B.3044 2-CHF ₂ -C ₆ H ₄ -CH = CH B.3045 3-CHF ₂ -C ₆ H ₄ -CH = CH B.3046 4-CHF ₂ -C ₆ H ₄ -CH = CH B.3047 naphthalin-1-y1-CH = CH B.3048 naphthalin-2-yl-CH = CH B.3049 pyridin-2-yl-CH = CH B.3050 pyridin-3-yl-CH = CH B.3051 pyridin-4-yl-CH = CH B.3052 _{5-CH3-pyridin-2-yl-CH} = CH B.3053 6-CH ₃ -pyridin-2-yl-CH = CH B.3054 _{5-CH3-pyridin-3-yl-CH} = CH B.3055 _{6-CH3-pyridin-3-yl-CH} = CH B.3056 _{5-OCH3-pyridin-2-yl-CH} = CH B.3057 6-OCH- _3- pyridin-2-yl-CH = CH B.3058 5-OCH ₃ -pyridin-3-yl-CH = CH B.3059 6-OCH ₃ -pyridin-3-yl-CH = CH B.3060 4-Cl-pyridin-2-yl-CH = CH B.3061 5-Cl-pyridin-2-yl-CH = CH

s-TL

Nr. R ³ B.3062 6-clpyridine-2-yľCH CH B.3063 2-C1-pyridin-3-yl-CH = CH _; B.3064 5-Cl-pyridin-3-yl-CH = CH B.3065 6-clpyridine-3-yľCH CH B.3066 2-clpyridine-4-yľCH CH B.3067 3,5-Cl ₂ -pyridin-2-yl-CH = CH B.3068 pyrimidin-2-yľCH CH B.3069 4-C-pyrimidin-2-yl-CH = CH B.3070 5-Cl-pyrimidin-2-yl-CH = CH B.3071 4-CH ₃ -pyrimidin-2-yl-CH = CH B.3072 5-CH ₃ -pyrimidin-2-yl-CH = CH B.3073 4-OCH ₃ -pyrimidin-2-yl-CH = CH B.3074 5-OCH ₃ -pyrimidin-2-ylCH = CH B.3075 pyrimidin-4-yl-CH = CH B.3076 2 -C 1 -pyrimidin-4-yl-CH = CH B.3077 6-C1-pyrimidin-4-y1-CH = CH B.3078 _2,6-Cl2 -pyrimidin-4-yl-CH = CH B.3079 2-CH ₃ -pyrimidin-4-yl-CH = CH B.3080 6-CH ₃ -pyrimidin-4-yl-CH = CH B.3081 2-OCH ₃ -pyrimidin-4-yl-CH = CH B.3082 6-OCH ₃ -pyrimidin-4-yl-CH = CH B.3083 2-OCH ₂ CH ₃ -pyrimidin-4-yl -CH = CH B.3084 6-OCH ₂ CH ₃ -pyrimidin-4-yl-CH = CH B.3085 pyrimidin-5-yl-CH = CH B.3086 2-C1-pyrimidin-5-y1-CH = CH B.3087 2-CH ₃ -pyrimidin-5-yl-CH = CH B.3088 2-OCH ₃ -pyrimidin-5-ylCH = CH B.3089 furan-2-yl-CH = CH B.3090 4-Br-furan-2-yl-CH = CH B.3091 4-Cl-furan-2-yl-CH = CH B.3092 4-CN-furan-2-y1-CH = CH B.3093 _{4-CH3-furan-2-yl-CH} = CH B.3094 5-Br-furan-2-yl-CH = CH B.3095 5-Cl-furan-2-yl-CH = CH B.3096 5-CN-furan-2-yl-CH = CH B.3097 _{5-CH3-furan-2-yľCH} CH B.3098 E uran-3-yl-CH = CH B.3099 5-Br-furan-3-yl-CH = CH B.3100 5-Cl-furan-3-yl-CH = CH

- // 2

Nr. R ³ B.3101 5-CN-furan-3-yľCH CH B.3102 _{5-CH3-furan-3-yľCH} CH ₃ B.3103 thien-2-yl-CH = CH B.3104 4-Br-thien-2-yl-CH = CH B.3105 4-Cľthien-2-yľCH CH B.3106 4-CN-thien-2-yl-CH = CH B.3107 J 4-CH- _3- thien-2-yl-CH = CH B.3108 5-Br-thien-2-yl-CH = CH B.3109 5-C1-thien-2-yl-CH = CH B.3110 5-CN-thien-2-yl-CH-CH B.3111 5-CH ₃ - thien-2-yl-CH = CH B.3112 thien-3-yl-CH = CH B.3113 5-Br-thien-3-yl-CH = CH B.3114 5-Cl-thien-3-yl-CH = CH B.3115 5-CN-thien-3-yl-CH = CH B.3116 5-CH ₃ -thien-3-yl-CH = CH B.3117 oxazol-2-yl-CH = CH B.3118 4-Br-oxazol-2-yl-CH = CH B.3119 4-Cl-oxazol-2-yl-CH = CH B.3120 4-CN-oxazol-2-yľCH CH B.3121 4-CH ₃ -oxazol-2-yl-CH = CH B.3122 5-Br-oxazol-2-yl-CH = CH B.3123 5-Cl-oxazol-2-yl-CH = CH B.3124 5-CN-oxazol-2-yl-CH = CH B.3125 5-CH ₃ -oxazol-2-yl-CH = CH B.3126 oxazol-4-yl-CH = CH B.3127 2-Br-oxazol-4-yl-CH = CH B.3128 2-Cl-oxazol-4-yl-CH = CH B.3129 2-CN-oxazol-4-yl-CH = CH B.3130 2 -CH ₃ -oxazol-4-ylCH = CH B.3131 2-C ₆ H _{5-oxazol-4-yl-CH} = CH B.3132 5-Br-oxazol-4-yl-CH = CH B.3133 5-Cľoxazoľ4 yľCH-CH B.3134 5-CN-oxazol-4-yl-CH = CH B.3135 5-CH ₃ -oxazol-4-yl-CH = CH B.3136 oxazol-5-yl-CH = CH B.3137 4-Br-oxazol-5-yl-CH = CH B.3138 -Cľoxazoľ5 yľCH-CH B.3139 1 -CN-oxazol-5-y 1 CH = CH

Nr. R ³ B.3140 4-CH ₃ -oxazol-5-yl-CH = CH B.3141 2-Br-oxazol-5-yl-CH = CH ₃ B.3142 2-Cl-oxazol-5-yl-CH = CH B.3143 2-CN-oxazol-5-yl-CH = CH B.3144 _{2-CH3-oxazol-5-yl-CH} = CH B.3145 isoxazol-3-yl-CH = CH B.3146 4-Br-isoxazol-3-yl-CH = CH B.3147 4-Cl-isoxazol-3-yl-CH = CH B.3148 4-CN-isoxazol-3-yl-CH = CH B.3149 4-CH ₃ -isoxazol-3-yl-CH = CH B.3150 5-Br-isoxazol-3-yl-CH = CH B.3151 5-Cl-isoxazol-3-yl-CH = CH B.3152 5-CN-isoxazol-3-yl-CH = CH B.3153 5-CH ₃ -isoxazol-3-yl-CH = CH B.3154 isoxazol-4-yl-CH = CH B.3155 3-Br-isoxazol-4-yl-CH = CH B.3156 3-Cl-isoxazol-4-yl-CH = CH B.3157 3-CN-isoxazol-4-y1-CH = CH B.3158 3-CH ₃ -isoxazol-4-yl-CH = CH B.3159 5-Br-isoxazol-4-yl-CH = CH B.3160 5-Cl-1-oxazol-4-yl-CH = CH B.3161 5-CN-isoxazol-4-yl-CH = CH B.3162 5-CH ₃ -isoxazol-4-yl-CH = CH B.3163 3,5- (CH ₃ ) 2 -isoxazol-4-yl-CH = CH B.3164 with oxa-1-5-yl-CH = CH B.3165 3-Br-isoxazol-5-yl-CH = CH B.3166 3-Cl-isoxazol-5-yl-CH = CH B.3167 3-CN-isoxazol-5-yl-CH = CH B.3168 3-CH ₃ -is oxazol-5-yl-CH = CH B.3169 3-C 6 H-isoxazol-5-yl-CH = CH B.3170 4-Cl, 3-C6H5-isoxazol-5-yl-CH-CH B.3171 4-Br, 3-C6H5-isoxazol-5-yl-CH = CH B.3172 4-Br-isoxazol-5-yl-CH = CH B.3173 4-Cl-isoxazol-5-yl-CH = CH B.3174 4-CN-isoxazol-5-yl-CH = CH B.3175 -CH ₃ -isoxazol-5-yl-CH = CH B.3176 Ľhiazol-2-yl-CH = CH B.3177 1-Br-thiazol-2-yl-CH = CH B.3178 -C1-thiazol-2-yl-CH = CH

Nr. R ³ B.3179 4-CN-thiazol-2-CH yľCH B.3180 4-CH ₃ -thiazol-2-yl-CH = CH 5 B.3181 5-Br-thiazol-2-CH yľCH B.3182 5-Cl-thiazol-2-CH yľCH B.3183 5-CN-thiazol-2-yl-CH = CH B.3184 5-CH ₃ -thiazol-2-yl-CH = CH B.3185 thiazol-4-yl-CH = CH B.3186 2-Br-thiazol-4-yl-CH = CH B.3187 2-Cl-thiazoľ4-yl-CH = CH B.3188 2-CN-thiazol-4-yl-CH = CH B.3189 _{2-CH3-thiazol-4-yl-CH} = CH B.3190 5-Br-thiazoľ4 yľCH-CH B.3191 5-C-thiazoľ4 yľCH CH B.3192 5-CN-thiazoľ4-yl-CH = CH B.3193 5-CH ₃ -thiazol-4-ylCH = CH B.3194 thiazole-5-yľCH CH B.3195 4-Br-thiazole-5-yl-CH = CH B.3196 4-C1-thiazol-5-yl-CH = CH B.3197 4-CN-thiazol-5-yl-CH = CH B.3198 _{4-CH3-thiazol-5-yl-CH} = CH B.3199 2-Br-thiazol-5-yl-CH = CH B.3200 2-Cl-thiazol-5-yl-CH = CH B.3201 2-CN-thiazol-5-yl-CH = CH B.3202 2-CH- _3- thiazol-5-yl-CH = CH B.3203 isothiazol-3-yl-CH = CH B.3204 4-Br-isothiazol-3-yl-CH = CH B.3205 4-Cl-isothiazol-3-yl-CH = CH v; B.3206 4-CN-isothiazol-3-yl-CH = CH B.3207 4-CH ₃ -isothiazol-3-yl-CH = CH B.3208 5-Br-isothiazol-3-yl-CH = CH B.3209 5-Cl-isothiazol-3-yl-CH = CH B.3210 5-CN-isothiazol-3-yl-CH = CH B.3211 5-CH ₃ -isothiazol-3-yl-CH = CH B.3212 isothiazol-4-yl-CH = CH B.3213 3-Br-isothiazol-4-yl-CH = CH B.3214 3-Cl-isothiazol-4-yl-CH = CH B.3215 3-CN-isothiazol-4-yl-CH = CH B.3216 3-CH ₃ -isothiazol-4-yl-CH = CH B.3217 5-Br-isothiazol-4-yl-CH = CH

Nr. R ³ B.3218 5-Cl-isothiazol-4-yl-CH = CH B.3219 5-CN-isothiazol-4-yl-CH = CH ; B.3220 5-CH3-isothiazol-4-yl-CH = CH B.3221 3,5- (CH ₃ ) ₂ -isothiazol-4-yl-CH = CH B.3222 isothiazol-5-yl-CH = CH B.3223 3-Br-isothiazol-5-yl-CH = CH B.3224 J 3-Cl-isothiazol-5-yl-CH = CH B.3225 3-CN-isothiazol-5-yl-CH = CH B.3226 3-CH ₃ -isothiazol-5-yl-CH = CH B.3227 4-Br-isothiazol-5-yl-CH = CH B.3228 4-Cl-isothiazol-5-yl-CH = CH B.3229 4-CN-isothiazol-5-yl-CH = CH B.3230 4-CH ₃ -isothiazol-5-yl-CH = CH B.3231 imide of ol-2-yl-CH = CH B.3232 l-Cl-imidazol-2-yl-CH = CH B.3233 l-Br-imidazol-2-yl-CH = CH B.3234 L-CN-imidazol-2-yl-CH = CH B.3235 1-CH- _3- imidazol-2-yl-CH = CH B.3236 4-Cl-imidazol-2-yl-CH = CH B.3237 4-Br-imidazol-2-yl-CH = CH B.3238 4-CN-imidazol-2-yl-CH = CH B.3239 4-CH- _3- imidazol-2-yl-CH = CH B.3240 _1-CH3, 5-Cl-imidazol-2-yl-CH = CH B.3241 1,4- (CH ₃ ) ₂ -imidazol-2-yl-CH = CH B.3242 1,5- (CH ₃ ) ₂ -imidazol-2-yl-CH = CH B.3243 imidazol-4-yl-CH = CH B.3244 2-C1-imidazol-4-yl-CH = CH B.3245 2-Br-imidazol-4-yl-CH = CH B.3246 2-CN-imidazol-4-yl-CH = CH B.3247 1-CH- _3- imidazol-4-yl-CH = CH B.3248 2-CH- _3- imidazol-4-yl-CH = CH B.3249 5-Cl-imidazol-4-yl-CH = CH B.3250 5-Br-imidazol-4-yl-CH = CH B.3251 5-CN-imidazol-4-yl-CH = CH B.3252 5-CH- _3- imidazol-4-yl-CH = CH B.3253 _1-CH3, 5-Cl-imidazol-4-yl-CH = CH B.3254 1,2- (CH ₃ ) ₂ -imidazol-4-yl-CH = CH B.3255 1,5- (CH ₃ ) 2 -imidazol-4-yl-CH = CH B.3256] oyrazol-3-yl-CH = CH

Nr. R ³ B.3257 5-Br-pyrazol-3-yľCH CH B.3258 5 -C 1 -pyrazol-3-yl-CH = CH ₅ B.3259 5-CN-pyrazol-3-yľCH CH B.3260 5-CH ₃ -pyrazol- ₃ -yl-CH = CH B.3261 1-C 6 H ₅ -pyrazol-3-yl-CH = CH B.3262 4-Br-pyrazol-3-yl-CH = CH B.3263 4-Cypyrazo 1-3-yl-CH = CH B.3264 4-CN-pyrazol-3-yl-CH = CH B.3265 4-CH ₃ -pyrazol-3-yl-CH = CH B.3266 _{1-CH3-pyrazol-3-yl-CH} = CH B.3267 1,4- (CH ₃ ) 2 -pyrazol-3-yl-CH = CH B.3268 1,5- (CH ₃ ) ₂ -pyrazol-3-yl-CH = CH B.3269 _1-CH3, 4-Cl-pyrazol-3-yl-CH = CH B.3270 1-CH _3,5 -C ₁ -pyrazol-3-ylCH = CH B.3271 pyrazol-4-yl-CH = CH B.3272 3-Br-pyrazol-4-yľCH CH B.3273 3-Cľpyrazoľ4 yľCH-CH B.3274 3-CN-pyrazol-4-yl-CH = CH B.3275 _{3-CH3-pyrazol-4-yl-CH} = CH " B.3276 1-CH ₃ -pyrazol-4-yl-CH = CH B.3277 1,5- (CH ₃ ) ₂ -pyrazol-4-yl-CH = CH B.3278 1,3- (CH ₃ ) 2 -pyrazol-4-yl-CH = CH B.3279 1-CH ₃ , 3-C 1 -pyrazol-4-ylCH = CH B.3280 1-CH _3,5 -C ₁ -pyrazol-4-ylCH = CH B.3281 pyrazol-5-yl-CH = CH B.3282 3-Br-pyrazol-5-yl-CH = CH B.3283 3-Cľpyrazoľ5 yľCH-CH B.3284 3-CN-pyrazol-5-yl-CH = CH B.3285 3-CH ₃ -pyrazol-5-ylCH = CH B.3286 1-CH ₃ -pyrazol-5-yl-CH = CH B.3287 4-Br-pyrazol-5-yl-CH = CH B.3288 4-C1-pyrazol-5-yl-CH = CH B.3289 4-CN-pyrazol-5-yl-CH = CH B.3290 _{4-CH3-pyrazol-5-yl-CH} = CH B.3291 1,3- (CH ₃ ) ₂ -pyrazol-5-yl-CH = CH B.3292 1,4- (CH ₃ ) ₂ -pyrazol-5-yl-CH = CH B.3293 L-CH ₃ , 3-C 1 -pyrazol-5-ylCH = CH B.3294 1-CH ₃ , 4-C 1 -pyrazol-5-ylCH = CH B.3295 ., 3,4-oxadiazol-5-yl-CH = CH

5 0 5 0 Nr. R ³ B.3296 2-CH3-I, 3,4-oxadiazol-5-yl-CH = CH B.3297 2-CF3-l, 3,4-oxadiazol-5-yl-CH = CH B.3298 2-OCH 3-I, 3,4-oxadiazol-5-yl-CH = CH B.3299 2-C1-1,3,4-oxadiazol-5-yl-CH = CH B.3300 2-CH (CH ₃ ) 2-1,3,4-oxadiazol-5-yl-CH = CH B.3301 1,3,4-oxadiazol-2-yl-CH = CH B.3302 5-CH3-I, 3,4-oxadiazol-2-yl-CH = CH B.3303 5-CF ₃ -1,3,4-oxadiazol-2-yl-CH = CH B.3304 5-OCH ₃ -1,3,4-oxadiazol-2-yl-CH = CH B.3305 5-C1-1,3,4-oxadiazol-2-yl-CH = CH B.3306 5-CH (CH ₃ ) 2 -1,3,4-oxadiazol-2-yl-CH = CH B.3307 5-C6H5-I, 3,4-oxadiazol-2-yl-CH = CH B.3308 1,2,4-oxadiazol-3-yl-CH = CH B.3309 5-CH ₃ -1,2,4-oxadiazol-3-yl-CH = CH B.3310 5-CF ₃ -1,2,4-oxadiazol-3-yl-CH = CH B.3311 5-C1-1,2,4-oxadiazol-3-yl-CH = CH B.3312 5-CH _(CH3) 2 ^_1 '2,4-oxadiazol-3-yl-CH = CH B.3313 1,2,4-triazol-3-yl-CH = CH B.3314 1-CH ₃ -1,2,4-triazol-3-yl-CH = CH B.3315 5-CH ₃ -1,2,4-triazol-3-yl-CH = CH B.3316 5-CF3-l, 2,4-triazol-3-yl-CH = CH B.3317 5-OCH ₃ -1,2,4-triazol-3-yl-CH = CH B.3318 5-C1-1,2,4-triazol-3-yl-CH = CH B.3319 5-CH (CH ₃ ) 2-1,2,4-triazol-3-yl-CH = CH B.3320 1-C ₆ H ₅ 1,2,4-triazol-3-yl-CH = CH B.3321 1,3,4-thiadiazol-5-yl-CH = CH B.3322 2-CH3-I, 3,4-thiadiazol-5-yl-CH = CH B.3323 2-CF3-I, 3,4-thiadiazol-5-yl-CH = CH B.3324 2-OCH ₃ -1,3,4-thiadiazol-5-yl-CH = CH B.3325 2-Cl-1,3,4-thiadiazol-5-yl-CH = CH B.3326 2-CH (CH ₃ ) 2 -1,3,4-thiadiazol-5-yl-CH = CH B.3327 1,3,4-thiadiazol-2-yl-CH = CH B.3328 5-CH ₃ -1,3,4-thiadiazol-2-yl-CH = CH B.3329 5-CF ₃ -1,3,4-thiadiazol-2-yl-CH = CH B.3330 5-OCH ₃ -1,3,4-thiadiazol-2-yl-CH = CH B.3331 5-C1-1,3,4-thiadiazol-2-yl-CH = CH B.3332 5-CH (CH ₃ ) 2-1,3,4-thiadiazol-2-yl-CH = CH B.3333 5-C ₆ H ₅ -1,3,4-thiadiazol-2-yl-CH = CH B.3334 L, 2,4-thiadiazol-3-yl-CH = CH

348

The compounds of formula I are useful as fungicides.

The compounds of the formula I are distinguished by their excellent activity against a broad spectrum of pathogenic fungi, in particular of the class Ascomycetes, Phycomycetes and Bsidiomycetes. They are partially systemically effective and can be used as foliar and soil fungicides.

They are of particular importance for protection against numerous fungi in various crop plants such as wheat, rye, barley, oats, rice, corn, grass, cotton, soybeans, coffee, sugar cane, vine, fruit and ornamental plants and vegetables such as cucumbers , pea and pumpkin plants, as well as the seeds of such plants.

Especially suitable for protection against the following plant diseases: Erysiphe graminis (powdery mildew) for grain, Erisiphe cichoracearum and Sphaerotheca fuliginae on pumpkin plants, Podosphera leucotricha on apples, Unicula necator on vines, Puccinia species on cereals and grass, Ustilago species on grain and sugar cane, Venturia inaequalis on apples, Helminthosporium grain, Sptoria nodorum on wheat, Botrytis cinerea (gray mold) on strawberries, vegetables, ornamental plants and vines, Cercospora arachidicola on groundnut, Pella on wheat, barley, Pyricularia oryzae on rice, Phytophthora infestans on potatoes and tomatoes, Fusarium and Verticilium species on

Plasmopara viticola nine and fruits.

different plants, Alternaria green vines, species

The compounds of the formula I are furthermore suitable for destroying malignant fungi in the protection of material (for example, wood, paper, fibers and possibly fabrics) and in the protection of stocks.

The compounds of the formula I are used by treating fungi or plants, seeds, materials or soil to be protected against fungal attack by a fungicidally effective compound.

49 amount of substances. The use takes place before or after fungal attack of the materials, plants or seeds.

They can be used in the form of customary formulations such as solutions, emulsions, suspensions, dust, powder, paste or granulate. The form of use depends on the intended use and in any case is intended to ensure a fine and uniform distribution of the compounds according to the invention. The formulations are prepared in a known manner, for example by mixing the active ingredient with a solvent and / or excipients as desired, using emulsifying and dispersing agents, and in the case of water as a diluent, other organic solvents such as co-solvents may be used. Basically, excipients which may be used are: diluents such as aromatics (e.g. xylol), chlorinated aromatics (e.g. chlorophenols), paraffins (e.g. petroleum fractions), alcohols (e.g. methanol, butanol), ketones (e.g. cyclohexanone), amines (e.g. ethanolamine) dimethylformamide) and water; carriers such as natural stone meal (e.g. kaolin, alumina, talc, chalk) and synthetic stone meal (e.g. high disperse silicic acid, silicates); emulsifying agents such as non-ionic and anionic emulsifiers (e.g. polyoxyethylene fatty alcohol ether, alkylsulfonates and arylsulfonates) and dispersing agents such as lignosulfite lyes and methylcellulose.

The fungicidal compositions generally contain between 0.1 and 95, preferably between 0.5 and 90% by weight of active ingredient.

The amounts used for plant protection vary between 0.01 and 2.0 kg of active substance per ha, depending on the type of effect desired.

In the treatment of seed, generally 0.001 to 0.1 g of t, preferably 0.01 to 0.05 g of active ingredient per kilogram of seed, is required.

When used for the protection of materials or stocks, the amount of active substance applied depends on the type of territorial use and the desired effect. Usual quantities for protection

The 350 of the material is, for example, 0.001 g to 2 kg, preferably 0.005 g to 1 kg of active ingredient per meter of cubic material.

The compositions according to the invention can be used as fungicides together with other active substances, for example with herbicides, insecticides, growth regulators, fungicides or even fertilizers.

When mixed with fungicides, in many cases the fungicidal effective spectrum is increased.

The following overview of fungicides with which the compounds of the invention can be used together explains but does not limit the possibilities of combination:

Sulfur, dithiocarbamates and their derivatives, such as iron dimethyldithiocarbamate, zinc dimethyldithiocarbamate, zinc ethylenebisdithiocarbamate, magnesium ethylenebisdithiocarbamate, magnesium zinc ethylenediamine-bis-dithiocarbamate, tetramethylthiurodisulfamate complex, Zinc Ν, Ν-propylene-bis-dithiocarbamate, zinc N, N-propylene-bis-dithiocarbamate, N, N-propylpropylene bis (thiocarbamoyl) disulfide;

nitro derivatives, such as dinitro (1-methylheptyl) -phenyl crotonate, 2-sec-butyl-4,6-dinitrophenyl-3,3-dimethylacrylate, 2-sec-butyl-4,6-dinitrophenyl-isopropyl carbonate, diisopropyl ester of 5- nitro-isophthalic acid;

heterocyclic compounds such as 2-heptadecyl-2-imidazoline acetate, 2,4-dichloro-6- (o-chloroanilino) -s-triazine, O, O-diethylphthalimidophosphonothioate, 5-amino-1- [bis- (dimethylamino)) phosphonyl] -3-phenyl-1,2,4-triazole, 2,3-dicyano-1,4-dithioanthraquinone, 2-thio-1,3-dithiolo [4,5-b] quinoxaline, methyl 1- ester (butylcarbamoyl) -2-benzimidazolecarbamic, 2-methoxycarbonylaminobenzimidazole, 2- (furyl- (2)) - benzimidazole, 2- (thiazolyl- (4)) - benzimidazole, N- (1,1,2,3-tetrachloroethylthio) - tetrahydrophthalimide, N-trichloromethylthio-tetrahydrophthalimide, N-trichloromethyl351 thiophthalimide, N-dichlorofluoromethylthi-N, N-dimethyl-N-phenyl-diamide sulfuric acid, 5-ethoxy-3-trichloromethyl-1,2,3-thiadiazole, 2-rodanomethylthiobenzene 1,4-dichloro-2,5-dimethoxybenzole, 4- (2-chlorophenylhydrazono) -3-methyl-5-isoxazolone, pyridine-2-thio-1-oxide, 8-hydroxyquinoline or its copper salt, 2,3-dihydro-5-carboxanilido-6-methyl-1,4-oxathiin, salt, 2,3-dihydro-5-carboxanilido-6-methyl-1,4-oxathiin-4,4-dioxide, 2- methyl-5,6-dihydro r-4H-pyran-3-carboxylic acid anilide, 2,5-dimethylfuran-3-carboxylic acid anilide, 2,4,5-trimethylfuran-3-carboxylic acid anilide, 2,5-dimethylfuran-3-cyclohexylamide carboxylic acid, N-Cyclohexyl-N-methoxy-2,5-dimethylfuran-3-carboxylic acid amide, 2-methylanilide of benoic acid, 2-iodoanilide of benzoic acid, N-formyl-N-morpholino-2,2,2-trichloroacetal piperazine-1m4 -dyilbis- (1- (2,2,2-trichloroethyl) formamide, 1- (3,4-dichloroanilino) -1-formylamino-2,2,2-trichloroethane, 2,6-dimethyl-N-tridecylmorpholine, optionally its salts,

2,6-dimethyl-N-cyclododecylmorpholine or its salts, N- [3- (p-tert-butylphenyl) -2-methylpropyl] -cis-2,6-dimethylmorpholine, N- (p-tert-butylphenyl) - 2-methylpropyl] -piperidine, 1- [2- (2,4-dichlorophenyl) -4-ethyl-1,3-dioxolan-2-yl-ethyl] -1H-1,2,4-triazole, 1- [ 2- (2,4-Dichlorophenyl) -4-n-propyl-1,3-dioxolan-2-yl-ethyl] -1H-1,2,4-triazole, N- (n-propyl) -N- ( 2,4,6-Trichlorophenoxyethyl) -N-imidazolylurea, 1- (4-chlorophenoxy) -3,3-dimethyl-1- (1H-1,2,4-triazol-1-yl) -2-butanone 1- (4-chlorophenoxy) -3,3-dimethyl-1- (1H-1,2,4-triazol-1-yl) -2-butanol, α- (2-chlorophenyl) -a- (4- chlorophenyl) -5-pyrimidinomethylene, 5-butyl-2-dimethylamino-4-hydroxy-6-methylpyrimidine, bis- (p-chlorophenyl) -3-pyridinemethanol, 1,2-bis- (3-ethoxycarbonyl-2-thioureudo) benzol, 1,2-bis- (3-methoxycarbonyl-2-thioureudo) benzole, as well as various fungicides such as dodecylguanidine acetate, 3- [3- (3,5-dimethyl-2-oxycyclohexyl) -2-hydroxyethyl] glutarimide, hexachlorobenzole, DL-methyl-N- (2,6-dimethylpheynl) -N-furoyl, (2) -alaninate, DL-N- (2,6-dimethylphenyl) -N- (2-methoxyacetyl) -alanínmetyl ester,

N- (2,6-dimethylphenyl) -N-chloroacetyl-DL-2-aminobutyrolactone, DL-N- (2,6-dimethylphenyl) -N- (phenylacetyl) -alanine methyl ester, 5-methyl-5-vinyl-3- (3,5-Dichlorophenyl) -2,4-dioxo-1,3-oxazolidine, 3- [3,5-dichlorophenyl- (5-methyl-5-methoxymethyl) -1,3-oxazolidine-2,4352

-dione, 3- (3,5-dichlorophenyl) -1-isopropylcarbamoylhydantoin, N- (3,5-dichlorophenyl) -1,2-dimethylcyclopropane-1,2-diimide carboxylic acid, 2-cyano- [N- (ethylaminocarbonyl) -2-Methoxyimino] acetamide, 1- [2- (2,4-dichlorophenyl) pentyl] -1H-1,2,4-triazole, 2,4-difluoro-α- (1H-1,2,4-trioazoles) -1-methyl) benzhydryl alcohol, N- (3-chloro-2,6-dinitro-4-trifluoromethylphenyl) -5-trifluoromethyl-3-chloro-2-aminopyridine, 1 - ((bis- (4-fluorophenyl) methylsilyl) - methyl) -lH-1,2,4-triazole.

Strobilurines such as methyl-E-methoxyimino- [α- (o-tolyloxy) -o-tolyl] acetate, methyl-E-2- [2- [6- (2-cyanophenoxy) pyrimidin-4-yloxy] -phenyl] 3-methoxyacrylate, methyl E-methoxyimino- [α- (2-phenoxyphenyl)] acetamide, methyl E-methoxyimino- [α- (2,5-dimethylphenoxy) -otolyl] acetamide.

Anilinopyridines such as N- (4,6-dimethylpyrimidin-2-yl) aniline, N- [4-methyl-5- (1-propynyl) -pyrimidin-2-yl] aniline, N- (4-methyl-6- cyclopropyl-pyrimidin-2-yl) aniline.

Phenylpyrrole such as 4- (2,2-difluoro-1,3-benzodioxol-4-yl) -pyrrole-3-carbonitrile.

Cinnamic acid amides such as 3- (4-chlorophenyl) -3- (3,4-dimethoxyphenyl) acrylic acid morpholide.

The compounds of the formula I are furthermore suitable as effective protection against pests of the insect, arachnid and nematode class. They can be used in plant protection as well as in the field of hygiene, stock protection and in the veterinary field as preparations for pests.

The harmful insects include, for example, Lepidoptera, such as Agrotis ypsilon, Agrotis segetum, Alabama argillacea, Anticarsia gemmatalis, Argyresthia conjugella, Autographa gamma, Bupalus piniarius, Cacoecia murinan, Ciracunisura fila, Cheimatobistura brumata, Cheimatobia brumata, Cheimatobia brumata, Cyndia pomonella, Dendrolimus pini, Diaphania nitidalis, Diatraea grandiosella, Earias insulana, Elasmopalpus lignosellus, Eupoecilia ambiquella, Fatteria subterranea, Galleria mellonella, Hilibellia heli, Graphilithis armis, Hilisella, Graphilitha molis, , Hyphantria cunea, Hyponomeuta malinellus, Keiferia lycopersicella, Lamvdina fiscellaria, Laphygma exigua, Leucoptera coffeella, Leucoptera scitella, Lithocolletis blancadella, Lobesia botrana, Loxistege sticticalis, Lymantria monarcicae, Lymantria, and pseudotsugate, Ostrinia nubilalis, Panolis flammea, Pectinophora gyssypiella, Peridroma saucia, Phalea bucephala, Phthorimaea operculella, Phyllocnistis citrella, Pieris brassicae, Spotted scorpionfish, Plutella xylostella, Plutipella pliaspia, Pseudopia Spodoptera littoralis, Spodoptera litura, Traumatopoea pityocampa, Tortrix viridina, Trichopulsia ni, Zeiraphera canadensis.

Among the beetles (Coleoptera, for example, Agrilus sinuatus, Agriotes lineatus, Agriotes ovscurus, Amphimallus solstitialis, Anisandrus dispar, Anthonomus grandis, Anthonomus pomorum, Atomaria linearis, Blastophagus piniperda, Blitophaga undata, Bruchus rufimanisis, Bruchus, Bruchus, Bruchus, Bruchus, Bruchus) , Cerotoma trifurcata, Ceuthorrynchus assimilis, Ceutrhorrynchus napi, Chaetocnema tibialis, Conoderus, vespertinus, Crioceris asparagi, Diabrotica 12-punctat, Diabrotica virgifera, Epilachna varivestis, Epilachna varivestis, Ips typographus, Lema bilineata, Lema malonopus, Leptinotarsa decemlibeata, Limonius califoricus, Lessorhoptrus oryzophilus, Melanotus communis, Meligontes aeneus, Melolontha hippocastini, Phololothha melolontha, Oulema oryzaeus, Oriorrhynchuschiaus, orcorrhnus sp., Phyllopertha horticola, Phyllotreta nemorum, Phyllotreta striolata, Popillia japica, Sitona lineatus, Sitophilus granaria.

354

Among the double-winged species, for example, Aedes aegypti, Aedes vexans, Anastrepha ludens, Anopheles maculipennis, Ceratitis capitata, Crysomya bezziana, Chrysomya hominivorax, Crysomya macellaria, Cordylobia anthropucus, Clexus, Clexus, Clexus, Clexus, Intestinalis, Glossina morsitans, Haematobia irritans, Haplodiplosis equestris, Hylemyia platura, Hypoderma lineata, Liriomyza sativae, Liriomyza trifolii, Lucilia caprina, Lucilia cuprina, Lucilia sericata. Lycoria pectoralis, Mayetiola destrucktor, Musca domestica, Muscina stabulans, Oestrus ovis, Oscinella frit, Pegomya hysocyami, Phorbia antiqua, Phorbia brassicae, Kc coarcata, Rhagoletis cerasi, Rhagoletis pomonella, Tipula oludosa, Tipula.

From the order of the tufts (Thysanoptera), for example, Frankliniella fusca, Frankliniella occidentalis, Frankliniella tritici, Scirtothrips citri, Thrips oryzae, Thrips palmi, Thrips tabaci.

From the order of the Hymenoptera, for example, Athalia rosae, Atta cephalotes, Atta sexdens, Atta texana, Hoplocampa minuta, Hoplocampa testudinea, Monomorium pharaonis, Solenopsis geminata, Solenopsis invicta.

From the range of Heteroptera, for example, Acrosternum hilare, Blissus leucopterus, Cyrtopeltis notarus, Dysdercus cingulatus, Dysdercus intermedius, Eurusgaster intergriceps, Leptoglossus phyllopus, Lygus guineagrassis, Lygus praestisis, Lygus praestisis, Lygus praetisis, Lygus praesis.

In the family of homoptera (Homoptera), for example, Acyrhosiphon onobrychis, Adelges laricis, Aphidula nasturtii, Aphis fabae, Aphis pomi, Aphis sambuci, Brachycaudus cardui, Brevicoryne brassicae, Cerosipha gossypii, Dreyfusia nismaneolae, avenae, Macrosiphum euphor355 biae, Macrosiphon rosae, Megoura viciae, Metopolophium lugens, Pemphigus bursarius, Perkinsiella saccharidica, Phorodon humuli, Psylla Mali, Psylla piri, Rhopalomyzus ascalonicus ,. Rhopalosiphum maidis, Sappaphis mala, Sappaphis mali, Schizaphis graminum, Schizoneura lanuginosa, Trialeurodes vaporariorum, Viteus vitifolii.

From the series of termites (Isoptera), for example, Calotermes flavicollis, Leucotermes flavipes, Reticulitermes lucifugus, Termes natalensis.

In the range of Orthoptera, for example, Acheta domestica, Blatta orientalis, Blattella germanica, Forticula auricularia, Gryllotalpa gryllotalpa, Locusta migratoria, Melanoplus femur rubrum, Melanoplus mexicanus, Melanoplus spp. Schistocerca peregrina, Stauronotus maroccanus, Tachycines asynamorus.

Among the triads of Arachnoides, for example, arachnids (Acarina) such as Amblyomma americanum, Amblyomma variegatum, Argas persicus Boophilus annulatus, Boophilus decoloratus, Boophilus microplus, Brevipalpus phoenicis, Rbyobia praetiosa, Dermacentor silvarum, Eotetranyusesus carpodes, Ornithodorus Moubata, Otobius megnini, Paratetranychus pilosus, Dermanyssus gallinae, Phyllocoptruta oleivora, Polyphagotarsonemus latus, Psoroptes ovis, Rhipicephalus appendiculatus, Tetraweed, Tetranususus, Tetranyususus, Tetranyususus, Tetranyususus, Tetranyususus, Tetranyususus, Tetranyususus

From the nematode class, for example, root nematodes, for example Meloidogyne hapla, Meloidogyne incognita, Meloidogyne javanica, cyst nematodes such as Globodera rostochiensis, Heterodera avenae, Heterodera glycines, Heterodera schachtat,

356

Belonolaimus longicaudatus, Ditylenchus destructor, Ditylenchus dipsaci, Heliocotylenchus multicinctus, Longidorus elongatus, Radopholus similis, Rotylôenchus robustus, Trichodorus primitivus, Tylenchorhynchus claytoni, Tylenchorhynchus dubus, Pratylen, pratylenetus, Pratylenetus, Pratylen.

The active compounds can be applied alone, in the form of their formulations or their application forms, for example in the form of directly sprayable solutions, powders, suspensions or dispersions, emulsions, oil dispersions, pastes, dusts, spreading agents, granules, by spraying, fogging, dusting, sprinkling or watering. The dosage forms depend on the intended use; in any case, the application of the active compounds according to the invention should be as fine as possible.

The concentrations of the active ingredients in ready-to-use preparations are highly variable.

They are generally between 0.0001 and 10%, preferably between 0.01 and 1%.

The active compounds can also be applied with good results by the Ultra Low Volumetric Method (ULV), with formulations of more than 95% by weight. or even an active substance without additives.

The application rates of the active ingredients for pest control are 0.1 to 2.0 kg, preferably 0.2 to 1.0 kg ha, under outdoor conditions.

For the production of directly sprayable solutions, emulsions, pastes or oil dispersions, suitable fractions of medium or high boiling mineral oils, such as kerosene or diesel fuel, coal tar oils such as vegetable or animal oils, aliphatic, cyclic or aromatic hydrocarbons, for example d benzene, toluene, xylene ,.

357 paraffin, tetrahydronaphthalene, alkylated naphthalenes and derivatives thereof, methanol, ethanol, propanol, butanol, chloroform, carbon tetrachloride, cyclohexanol, cyclohexanone, chlorobenzene, isophorone, strong polar solvents such as dimethylformamide, dimethylsulfoxide, N-methylpyrrolidone, water.

Suitable dosage forms can be prepared from emulsion concentrates, pastes or wettable powders (dusting agents, oil dispersions) by adding water. For the production of emulsions, pastes or oil dispersions, substances alone or dissolved in an oil or solvent, homogenized with wetting agents, adhesives, dispersing or emulsifying agents in water may be used. However, concentrates consisting of the active ingredient, wetting agents, adhesives, dispersing or emulsifying agents and optionally solvents or oils which are suitable for dilution with water can also be prepared.

Suitable surfactants are alkali metal salts, alkaline earth metal salts, ammonium salts of lignminesulfonic acid, naphthalenesulfonic acid, phenolsulfonic acid, dibutylnaphthalenesulfonic acid, alkylarylsulfonates, alkylsulfates, alkylsulfonates, sulfonates of fatty alcohols and their fatty acids, and their fatty acids, alkaline earth metal salts, salts of sulfated fatty alcohol glycol ether, condensates of sulfonated naphthalene and naphthalene derivatives with formaldehyde, condensates of naphthalene or of naphthalenesulfonic acid with phenol and formaldehyde, polyoxyethylene octylphenol ether, ethoxylated isooctylphenol, octylphenol, nonylphenol, alkylphenyl polyglycol ethers, tributylphenyl, alkylaryl polyether alcohols, isotridecyl alcohol, kondezáty ethylene oxide fatty alcohol, ethoxylated castor oil, polyoxyethylene alkyl ether, ethoxylated polyoxypropylene, lauryl alcoholpolyglycol teracetal, sorbitester, lignosulfite waste liquors and methylcellulose.

Powder, dusting and spreading agents are prepared by mixing or grinding the active ingredients with a solid

358 carrier.

The formulations generally comprise between 0.01 and 95% by weight, preferably between 0.1 and 90% by weight. of the active substance. The active compounds are employed in a purity of 90% to 100%, preferably 95% to 100% (according to NMR spectrum).

Formulation examples:

1.5 parts by weight of the compound of the invention are intimately mixed with 95 parts by weight of fine kaolin. In this way, a dusting composition is obtained which contains 5% by weight of active ingredient.

II. 30 parts by weight of the compound of the invention are intimately mixed with a mixture of 92 parts by weight of a silica gel powder and 8 parts by weight of paraffin oil sprayed onto the surface of the silica gel. This produces a modified active substance with good adhesion (23% by weight of active substance).

III. 10 parts by weight of a compound of the invention are dissolved in a mixture consisting of 90 parts by weight of xylene, 6 parts by weight of a composite product consisting of 8 to 10 moles of ethylene oxide per mole of N-monoethanolamide oleic acid, 2 parts by weight of calcium dodecylbenzenesulfonic acid and 2 parts by weight. a product consisting of 40 moles of ethylene oxide per mole of castor oil (9% active ingredient content).

IV. 20 parts by weight of the compound are released in a mixture consisting of cyclohexanone, 30 parts by weight of the compound of the invention are 60 parts by weight of isobutanol, 5 parts by weight of ethylene oxide per mole of isooctylphenol, 5 parts by weight of composite product per mole of castor oil (16% active ingredient content).

V. 80 parts by weight of the compound of the invention are intimately mixed with 3 parts by weight of diisobutylnaphthalenesulfonic acid sodium salt, 10 parts by weight of lignin sulphonic acid sodium salt from sulphite waste liquors and 7 parts by weight of silica gel powder and ground in an 80% hammer mill. active substance).

VI. 90 parts by weight of the compound of the invention are mixed with 10 parts by weight of N-methyl-pyrrolidone to form a solution suitable for application in tiny drops (90% by weight of active ingredient).

VII. 20 parts by weight of a compound of the invention are dissolved in a mixture consisting of 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight of a product composed of 7 moles of ethylene oxide per mole of isooctylphenol and 10 parts by weight of a product composed of 40 moles of ethylene oxide per mole. castor oil. Pouring and thoroughly mixing the solution in 100,000 parts by weight of water produces an aqueous dispersion containing 0.02% by weight of the active ingredient.

VIII. 20 parts by weight of the compound of the invention are intimately mixed with 3 parts by weight of diisobutylnaphthalenesulphonic acid sodium salt, 17 parts by weight of lignin sulphonic acid sodium salt from sulphite waste liquors and 60 parts by weight of a silica gel powder and ground in a hammer mill. Mixing the mixture in 20,000 parts by weight of water gives a spray solution containing 0.1% by weight of the active ingredient.

60

Granules, for example, shell, impregnation or homogeneous granules, may be prepared by binding the active ingredients to solid carriers. Solid carriers are, for example, mineral soils such as silica, silicic acid, silica gel, silicates, talc, kaolin, aluminous, limestone, lime, chalk, ore, loess, clay, dolomite, diatomaceous earth, calcium sulphate, magnesium sulphate, magnesium oxide , ground plastics, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas and plant products such as cereal flour, tree bark flour, wood and walnut shells, cellulose powder and other solid carriers.

The active ingredients may optionally be added immediately prior to application of oils of various types, herbicides, fungicides, other pest control agents, bactericides. These compositions may be admixed with the compositions of the invention in a weight ratio of 1: 10 to 10: 1.

DETAILED DESCRIPTION OF THE INVENTION

The procedures outlined in the following Synthesis Examples were used in the appropriate treatment of the starting compounds to give additional compounds of Formula I. The compounds thus prepared are listed in the following tables with physical data.

Example 1

Phenylacetic acid 2 - [[[[2- (isopropyl) -1- (methyl) -2- (oxo) ethylidene] amino] oxy] methyl] -α- (methoxymethylene) methyl ester

O c = choch _{3 and 2} ch ₃

To a mixture of 8 g (62 mmol) of 1-isopropyl-1,2-propanedione-2-oxime in 50 ml of N, N-dimethylformamide is added 11 g of a 30% methanolic sodium trimethylate solution. The mixture is allowed to stir at room temperature for 30 minutes, then a solution of 18.6 g (68 mmol) of 2- (bromomethyl) -a- (methoxymethylene) methyl phenylacetic ester in 50 ml of N, N-dimethylformamide is added dropwise and the mixture is stirred for about 1 hour at 40 ° C. Finally, the reaction solution is diluted with water and extracted with methyl tert-butyl ether. Drying of the organic extracts over sodium sulfate and concentration on a rotary evaporator gave 18 g of a yellow solid. Recrystallization from hexane and suction and drying in a vacuum dryer gave 15 g (73%) of the title compound as a slightly yellowish solid (mp 67-69%).

IR [cm ^-1 ] (KBr): 768, 997, 1009, 1109, 1127, 1210, 1254, 1630, 1683, 1699, 2950.

Example 2

2 - [[[[2- (Allyloxy) imino-2- (isopropyl) -1- (methyl) ethylidene] amino] oxy] methyl] -α- (methoxymethylene) methyl phenylacetic ester

co ₂ ch ₃

To a mixture consisting of 1.5 g (62 mmol) of 2 - [[[[2- (isopropyl) -1- (methyl) -2- (oxo) ethylidene] amino] oxy] methyl] -a- (methoxymethylene) methyl Phenylacetic acid ester in 60 ml of methanol was added 0.7 g (9 mmol) of o-allylhydroxylamine and 0.9 g (4.5 mmol) of p-toluenesulfonic acid. The reaction mixture is allowed to stand for 4 days at room temperature, then diluted with water and extracted with methyl tert-butyl ether. The purified organic extracts were dried over sodium sulfate and concentrated. After column chromatography on silica gel, the title compound is obtained in the form of two isomers [side chain isomerism, (Z, E) or (E, E)].

1. Isomer (0.3 g; slightly yellowish oil) ¹ H-NMR (CDCl ₃ ):

δ = 1.16 (d, 6H), 1.99 (s, 3H), 3.50 (m, 1H), 3.67 (s, 3H), 3.81 (s, 3H), 4.60 (d, 2H), 5.08 (s, 2H), 5.25 (m, 2H), 5.97 (m, 1H), 7.12 - 7.46 (m, 4H), 7.56 ( s, 1H) ppm.

2. Isomer (0.6 g; white solid; mp 58-60 ° C) .delta. = 1.08 (d, 6H), 2.00 (s, 3H), 2.71 (m, 1H), 3.67 (s, 3H), 3.81 (s, 3H), 4.53 (d, 2H), 5.06 (s, 2H), 5.21 (m, 2H), 5.96 (m 1H, 7.12-7.46 (m, 4H), 7.56 (s, 1H) ppm.

Example 3

Phenylacetic acid 2 - [[[[2- (isopropyl) -1- (methyl) -2-oxoethylidene] amino] oxy] methyl] - (ethylidene) methyl ester

^CO 2 ^CH 3

A mixture of 9 g (33 mmol) of 2- (bromomethyl) -α-ethylidene-methyl phenylacetic ester in 50 ml of N, N-dimethylformamide is mixed with 9.2 g (67 mmol) of sodium carbonate and after addition of 4.3 g The 1-isopropyl-1,2-propanedione-2-oxime is stirred at

JOJ temperature 50 ⁼ C for 2 hours. Finally, the reaction solution is diluted with water and extracted with methyl tert-butyl ether. The purified organic extracts are washed with water, dried over sodium sulfate and concentrated. Column chromatography on silica gel (cyclohehane / ethyl acetate) afforded 7.8 g of the title compound as a yellowish oil.

1 H-NMR (CDCl ₃ ):

δ = 1.06 (d, 6H), 1.62 (s, 3H), 1.90 (s, 3H), 3.86 (m, 1H), 3.70 (s, 3H), 5.13 (s, 2H), 7.08-7.50 (m, 4H) ppm.

Example 4

Phenylacetic acid 2 - [[[[2- (isopropyl) -2- (methoxyimino) -1 '(methyl) ethylidene] amino] oxy] methyl] - (ethylidene) methyl ester

To a mixture of 2 g (6.3 mmol) of 2 - [[[[2- (isopropyl) -1- (methyl) -2- (oxo) ethylidene] amino] oxy] methyl] - and - (ethylidene) - of methyl phenylacetic acid ester in 50 ml of methanol are added 7.9 g of a 20% solution of O-methylhydroxylamine hydrochloride in methanol and 2-3 g of molecular sieve (3A). The reaction mixture is allowed to stand for three days at room temperature and then stirred for 4 hours at 40 ° C. After filtering off the molecular sieve, the solution is placed on ice water and extracted with methyl tert-butyl ether. The purified organic extracts were washed with water, dried over sodium sulfate and concentrated. Column chromatography on silica gel (cyclohexane / ethyl acetate) afforded 1.7 g (78%) of the title compound as a mixture of isomers (side chain isomerism, isomers 1: 2) as a yellowish oil.

IR [cm ^-1 ] (film): 761, 907, 1013, 1038, 1208, 1252, 1435, 1719,

2937, 2963.

Example 5 (E, E, E) -2 - [[[[2- (Isopropyl) -2- (methoxyimino) -1- (methyl) ethylidene] amino] oxy] methyl] -a- (methoxyimino) methyl ester phenylacetic acid

ch (ch ₃ ) ₂

CO ₂ ^ch 3

To a mixture of 49.7 g (315 mmol) of (E, E) -1- (isopropyl) -1- (methoxyiminopropan-2-one-2-oxime in 400 ml of N, N-dimethylformamide) is added 1 eq of sodium methylate ( 30% methanol solution) and the mixture is stirred for 30 minutes at room temperature, then a solution of 8 2.8 g (2 90 mmol) of 2- (bromomethyl) -α-methoxyimino-methyl-phenylacetic ester in 200 ml Ν is added dropwise. After stirring for one hour at room temperature, the reaction solution was poured onto ice water, and the solid formed was filtered off with suction and washed several times with water and pentane to give 94.5 g of crystalline solid, m.p. up to 94 ° C.

¹ H-NMR (CDCl ₃ ):

.delta. = 1.12 (d, 6H), 1.96 (s, 3H), 3.45 (m, 1H), 3.84 (s, 3H), 3.39 (s, 3H), 4.04 (s, 3H), 5.05 (s, 2H), 7.15-7.48 (m, 4H) ppm.

Example 6 (E, E, E) -2 - [[[[2- (Isopropyl) -2- (methoxyimino) -1- (methyl) ethylidene] amino] oxy] methyl] -α- (methoxyimino) -methylamide fenyloctove j

ch (ch ₃ ) ₂ conhch ₃ g (138 mmol) of (E, E, E) -2 - [[[[2- (isopropyl) -2- (methoxyimino) -1- (methyl) ethylidene] amino] oxy] The methyl] -? - (methoxyimino) methyl ester of phenylacetic acid is dissolved in 500 ml of tetrahydrofuran, mixed with 107 g of a 40% aqueous monomethylamine solution and stirred for 30 to 60 minutes at 50 ° C. Water is then added and extracted with methyl tert-butyl ether. The organic phase was washed with water, dried over Na ₂ SO ₄ and concentrated. 41 g of a brown solid are obtained, which is purified by slurrying in pentane. After aspiration, washing of the residue and drying, 37 g of the title compound is isolated as colorless crystals. Melting point 78-79 ° C.

¹ H-NMR (CDCl ₃ ):

.delta. = 1.13 (d, 6H), 1.95 (s, 3H), 2.88 (d, 3H), 3.46 (m,

1H), 3.89 (s, 3H), 3.94 (s, 3H), 5.06 (s, 2H), 6.72 (s, broad, 1H), 7.15-7.46 (m) (4H) ppm.

Example 7

Phenylacetic acid 2 - [[[[2- (methoxyimino) -1- (methyl) -2- (phenoxymethyl) ethylidene] amino] oxy] methyl] -a- (methoxyimino) methyl ester

^co 2 ^CH 3

To a solution consisting of 2 g of phenylacetic acid 2 - [[[[1- (methyl) -2- (oxo) -2- (phenoxymethyl) ethylidene] amino] oxy] methyl] -α- (methoxyimino) methyl ester in 5 0.4 ml of O-methylhydroxylamine hydrochloride and 1.2 g of pyridine are added in ml of methanol. The reaction solution is allowed to stir for 60 minutes at room temperature, then the residue is taken up in dichloromethane and the organic phase is washed with dilute hydrochloric acid and water. The organic phase is dried over sodium sulphate and concentrated. Crystallization of the residue from pentane gave 0.7 g of the title compound as slightly reddish crystals (flash point 81-83 ° C).

Example 8

Phenylacetic acid 2 - [[[[2- (methoxyimino) -1- (methyl) -2- (phenoxymethyl) ethylidene] amino] oxy] methyl] -a- (methoxyimino) -methylamide

CONHCH ₃

Dissolve 0,5 g of phenylacetic acid 2 - [[[[2- (methoxyimino) -1- (methyl) -2- (phenoxymethyl) ethylidene] amino] oxy] methyl] -a- (methoxyimino) methyl ester in 5 ml tetrahydrofuran, 0.5 g of aqueous monomethylamine solution is added and stirred at room temperature. The reaction solution is concentrated and the residue is triturated with pentane. Filtration of the precipitate and washing with pentane gave 0.5 g of the title compound as pink crystals (flash point 136-138 ° C).

Example 9

Phenylacetic acid 2 - [[[[2- (bromomethyl) -1- (methyl) -2- (oxo) ethylidene] amino] oxy] methyl] -a- (methoxyimino) methyl ester

To a solution consisting of 39,8 g of 2 - [[([1,2- (dimethyl) -2- (oxo) ethylidene] amino] oxy] methyl] -a- (methoxyimino) methyl ester of phenylacetic acid in 200 ml of chloroform is first added 5 ml of a solution of 20.8 g of bromine in 20 ml of chloroform are added dropwise at 40 DEG C. After the start of the reaction, the remainder of the bromine solution is added dropwise so that the temperature remains at 40-50 DEG C. If the starting material is present, additional bromine solution is added dropwise until the reaction is complete (40 ° C, control by TLC) and the reaction mixture is allowed to cool to room temperature. The organic phase was separated, washed with sodium bicarbonate solution and water, dried over sodium sulfate and concentrated to give the title compound as a dark solid. oil (50 g) The crude product may be reacted further without prior purification.

¹ H-NMR (CDCl ₃ ):

.delta. = 1.94 (s, 3H),

2H), 5.18 (s, 2H), 7.15

3.86 (s, 3H), 4.04

7.0 (m, 4H) ppm.

(s, 3H), 4.35 (s,

Example 10

Phenylacetic acid 2 - [[[[2- (chlorophenoxymethyl) -1- (methyl) -2-oxoethylidene] amino] oxy] methyl] - (methoxyimino) methyl ester

Solution consisting of 21,9 g of phenylacetic acid 2 - [[[[2- (bromomethyl) -1 (methyl) -2- (oxo) ethylidene] amino] oxy] methyl] - and - (methoxyimino) methyl ester in 150 ml of acetone is mixed with 15.7 g of potassium carbonate and 11 g of 4-chlorophenol and stirred for 24 hours at room temperature. The reaction mixture is concentrated on a rotary evaporator and the residue is bound with acetate. The organic phase was washed with water, dried over Na ₂ SO ₄ and concentrated. Purification by silica gel column chromatography affords the title compound as a crystalline solid (10.8 g). Flash point 110-114 ° C.

Example II

Phenylacetic acid 2 - [[[[2- (chlorophenoxymethyl) -2- (ethoxyimino) -1- (methyl) ethylidene] amino] oxy] methyl] - α (methoxyimino) methyl ester: NOCH.

H ₅ C ₂ ON:

noch c = ₃ [4-Cl-C ₆ H _{4] -O-CH2 CO2 CH3}

A solution consisting of 2,5 g of 2 - [[[[2- (4-chlorophenoxymethyl) -1- (methyl) -2- (oxo) ethylidene] amino] oxy] methyl] -a- (methoxyimino) methyl phenylacetic ester in 5 ml of methanol is mixed with 0.6 g of O-ethylhydroxyamine hydrochloride and 1.4 g of pyridine. The reaction solution is allowed to stir for 18 hours at room temperature, the mixture is bound to dichloromethane, washed with dilute hydrochloric acid and water. Concentration on a rotary evaporator gave 2.7 g of the title compound as a crystalline solid, flash point 84-87 ° C.

Example 12

3- (methoxyimino) -1- (phenyl) pent-l-yn-4-one-4-oxime

A solution consisting of 1.6 g of 1- (phenyl) -pent-1-yne-3,4-dione-4-oxime in 20 ml of methanol is mixed with 2 g of pyridine and 4.9 g of an 18% methanolic solution of O-methylhydroxylamine. of hydrochloride and at room temperature (about 25 ° C) is bound to tert-butyl methyl ether and mixed with 10% hydrochloric acid. water

The phase 70 is extracted with tert. butylmetyléter'om. Subsequently, 10% hydrochloric acid and washed out with water the organic phases, dry over Na ₂ SO ₄ and the solvent was distilled off under reduced pressure. 1.4 g of the title compound is obtained as a colorless solid (yield 76%). Flash point 140-144 ° C.

Example 13

2 - [[[[2- (Methoxyimino-1 '(methyl) -2- (phenyletter-yl) ethylidene] amino] oxy] methyl] -a- (methoxyimino) methyl phenylacetic ester

A solution consisting of 1.4 g of 1- (methoxyimino) -1- (phenyletter-1-yl) -propan-2-one-2-oxime in 20 ml of Ν, Ν-dimethylformaid is mixed with 1.4 g of 30% methanol. solution of sodium methylate and stirred for 10 minutes at room temperature. Subsequently, a solution of 2.1 g of 2- (bromomethyl) -? - methoxyimino-methyl phenylacetic ester in 20 ml of N, N-dimethylformamide is added dropwise. The reaction mixture is stirred for 1 hour at room temperature, poured into water and extracted with tert-butyl methyl ether. The organic phase was washed with water, dried over Na ₂ SO _4, filtered at reduced pressure and concentrated. Crystallization of the oily residue from methanol gave 1.9 g of the title compound (yield 60%). Melting point: 100-104 ° C.

Example 14

Phenylacetic acid 2-1 '[[[2- (methoxyimino-1- (methyl) -2- (phenylog-1-yl) ethylidene] amino] oxy] methyl] -α- (methoxyimino) -methylamide

HgCO

NOCHi c = noch ₃

The CONHCHg g of the ester of Example 13 is dissolved in 50 ml of tetrahydrofuran, mixed with 1.4 g of a 40% aqueous monomethylamine solution and stirred for 20 hours at room temperature. Subsequently, the reaction mixture is poured into water and extracted with tert-butyl methyl ether. The organic phase was washed with water, dried over Na ₂ SO _4, filtered at reduced pressure and concentrated. Crystallization of the oily residue from methanol gave 0.8 g of the title compound as a solid (yield 79%). Melting point: 131-133 ° C.

- 372 Table I.A

co ₂ ch ₃

no. R ² R ³ R ⁴ Data 1 ch ₃ ^C 2 ^H 5 ch ₃ oil, IR (film) 877, 893, 956, 1017 1208, 1252, 1435,173 2939 2 ch ₃ ^C 2 ^H 5 ^C 2 ^H 5 oil, IR (film) 877, 918, 956, 1038 1208, 1252, 1435, 17l 2975

3 ch ₃ ^C 2 ^H 5 nC ₃ ^H 7 oil, IR (film) 881, 907, 959, 988, 1037 1252, 1453, 1720, 2939, 2968 4 ch ₃ ch (ch ₃ ) ₂ ch ₃ oil, IR (film) 761, 907, 1013, 1038, 1208, 1252, 1435, 1719, 2937, 2963 5 ch ₃ ch (ch ₃ ) ₂ ^C 2 ^H 5 oil, IR (film) 761, 902, 922, 1039, 1208, 1252, 1435, 1719, 2934, 2972 6 ch ₃ ch (ch ₃ ) ₂ Oil, IR (film) 924, 984, 1017, 1037, 1208, 1252, 1435, 1719, 2934, 2964 7 ^C 2 ^H 5 ^{n C} 3 ^H Jt ch ₃ oil, IR (film) 873, 956, 1018, 1050, 1207, 1252, 1436, 1719, 2938, 2963 8 ^C 2 ^H 5 ⁿ “ ^C 3 ^H ? ^C 2 ^H 5 oil, IR (film)

897, 914, 959, 1019, 1049,

1252, 1435, 1720, 2937,

2.971 ^C 2 ^H 5 ^nc 3 ^H 7 CH ₂ C = CH oil, IR (film)

870, 956, 1009, 1040, 120;

1254, 1435, 1717, 2120,

2937, 2962

CH ₃ C = CC ₆ H ₅ CH ₃ ¹ H-NMR (CDCl ₃ ): 1.61 (d, 3H); 2.09 (s, 3H); 3.69 (s, 3H); 4.09 (s, 3H); 5.13 (s, 2 H); 7.05-7.56 (m, 10H) ppm

Table I.B

^CO 2 ^CH 3

375

no. R ² R ³

R ⁴

Data ₃ ch ₂ h ₅ nC ₃ H _? oil, IR (film)

958, 989, 1021, 1047

1069, 1218, 1437, 1729,

2939, 2968

CH ₃ C ₂ H ₅ iC

3 ^ 7

- 60 ° C flash point

CH ₃ C ₂ H ₅ nC ₄ H _g oil, IR (film)

880 959 1021 1070

1219 1437 1730 2939

2957

CH ₃ C ₂ H _5- prop-1-en-3-yl IR (KBr)

774, 895, 958, 1011,

1028, 1068, 1303, 1739,

2925 ^{5 c} h ₃ c ₂ h ₅ prop-1-yn-3-yl, 85-88 ° C flash point

CH ₃ C ₂ H ₅

3-methyl-but-oil, IR (film) 2-en-1-yl 883, 958, 1020, 1070,

1219, 1438, 1729, 2939

CH ₃ CH (CH ₃ ) ₂ CH ₃

- 95 ° C flash point

J / ύ

WITH ch ₃ CH _{(CH3) 2} ^C 2 ^H 5 68 - 7 ° C flash point 9 ch ₃ ch (ch ₃ ) ₂ nC ₃ H _{7 n} . 48 - 49 ° C flash point 10 ch ₃ ch (ch ₃ ) ₂ t-c ₃ h ₇ Mp: 4-40 ° C. 58-61 ° C flash point 11 ch ₃ ch (ch ₃ ) ₂ N-C ^ Hg 4- - 4- 4- 4- ⁵⁸ ° ⁶¹ ° ^C flash point 12 ch ₃ CH _(CH3) 2 prop-ene 3-yl 59-61 [deg.] flash point 13 ^C 2 ^H 5 ch (ch ₃ ) ₂ ch ₃ _,. Mp 62-64 ° C flash point 14 ^C 2 ^H 5 ch (ch ₃ ) ₂ ^C 2 ^H 5 -4- 4- ° -71-71 ° C flash point 15 ^C 2 ^H 5 ^{n C} 3 ^H 7 ch ₃ oil; IR (film) 872, 957, 1020, 1052 1070, 1219, 1438, 1730, 2940 (1962) 16 ^C 2 ^H 5 ^C 2 ^H 5 oil; IR (film) 914, 959, 1020, 1070, 1219, 1437, 1730, 2939, 2972 17 C ₂ ^H 5 H ,,. 102-104 ° flash point 18 ^C 2 ^H 5 nC ₃ H ₇ prop-en-3 -yl oil; IR (film)

914, 959, 1020, 1070

3, 1219, 1321, 1437, 1730

2939, 2961

C ₂ H ₅ n C ₃ H ₇ prop-1-in-3-yl oil; IR (film)

958, 1010, 1044, 1070,

1219, 1321, 1438, 1729,

2940, 2962

C ₂ H ₅ nC ₃ H ₇ CH ₂ - oil; IR (film) [3-CF ₃ -C ₄ H ₄ ] 958, 1019, 1050, 1072,

1127, 1166, 1201, 1219,

1330, 1729, 2940, 2960

2i ch ₃ -ch ₂ oc ₆ h ₅ ch ₃

- 83 ° C flash point

CH ₃ -CH ₂ C ₆ H ₅ CH ₂ CH ₃ = 79-81 ° C flash point

CH ₃ -CH ₂ OC ₆ H ₅ CH ₂ C = CH ¹ H-NMR (CDCl ₃ ):

delta tPP > m] = 2.04 (WITH, 3H) 2.45 (M, 1H), 3.81 (with, 3H) 3.99 (with, 3H), 4.78 (with, 2H) 4.92 (with, 2H), 5.03 (with, 2H) 6,85- 7.45 > (m, 9H)

CH ₃ 4-FC ₆ H ₄ -CH ₃ o-ch ₂

80 ° C flash point

25 ch ₃ 4-F-Cg ^H 4 -O-ch ₂ ^CH 2 ^CH 3 flash point 85 · 26 ch ₃ 4-FC _with H ₄ - ch ₃ c = ch ¹ H-NMR (CDCl ₃ ) o-ch ₂ .delta. [ppm] = 2, by: 2.47 (m, IH), 3,8: 4.01 (s, 3H); 4,7 ' 4.87 (s, 2H). 5 on: 6.75-7.40 (m, 8H) 27 ch ₃ 4-Ck-C ₆ H ₄ -o-ch ₂ ch ₃ 112 · flash point 28 ch ₃ 4-Cl-C ₆ H ₄ - _-O-CH2 ch ₂ ch ₃ flash point 84 ·

29 ch ₃ 4-Cl-C ₆ H ₄ - _O-CH2 ch ₃ c = ch ¹ H-NMR (CDC1 ₃₎ d [ppm] = 2.0, 2.47 (m, 1H), 3.8 3.99 (s, 3H), 4.7 4.88 (s, 2H); 5.0 6.75-7.45 (m, 8H) 30 ch ₃ ch ₂ -cn ch ₃ flash point 143

CH ₃ CH ₂ -CN C ₂ H ₅ Flash point

32 ch ₃ ch ₂ -cn ch ₂ c = ch oil 33 ch ₃ ch ₂ -o- [2-CN- ch ₃ 100 ° C flash point 34 ch ₃ ch ₂ -o- [2-CN- C ₆ ^H 4] ^C 2 ^H 5 84 ° C flash point 35 ch ₃ ch ₂ -o- [2-CN- c ₆ h ₄ ] ch ₂ c ^ ch 120 - 124 ° <flash point 36 ch ₃ ch ₂ scn ch ₃ oil 37 ch ₃ ch ₂ -scn ^C 2 ^H 5 oil 38 ch ₃ ch ₂ scn ch ₂ c = ch oil 39 ch ₃ ch ₂ -o- [4-CN-C ₆ H ₄ ] ch ₂ c = ch oil 40 ch ₃ ch ₂ -o- [4-CN-C ₆ H ₄ ] ^C 2 ^H 5 85 ° C flash point

ό ϋ

CH, CH ₉ -0- CH ₉ , 88-92 ° C ^S - ⁵ flash point [4-CN-C ₆ H ₄ ]

42 ch ₃ ch ₂ -o- [i-ch _3- (3-CF ₃ -pyrazol-5-yl)] ch ₂ c ^ ch oil 43 ch ₃ ch ₂ -o- [i-ch _3- (3-CF ₃ -pyrazol-5-yl)] ^C 2 ^H 5 oil 44 ch ₃ CH ₂ O- [CH _{i-3-3-CF3-tetrazol} -py- 5-yl] ch ₃ oil 45 ch ₃ ch ₂ sc 0- nhch ₃ ^C 2 ^H 5 oil 46 ch ₃ ch ₂ sc 0- nhch ₃ ch ₃ oil 47 ch ₃ c _of cc ₆ h ₅ ch ₃ 100 - 104 ° flash point

3S1

Table I.C

no. R ² R ³ R ⁴ Data 1 ch ₃ ^C 2 ^H 5 ⁿ ~ ^c 3 ^H 7 62-63 ° C flash point 2 ch ₃ ^C 2 ^H 5 t-c ₃ h ₇ oil, IR (film 883, 960, 980, 1038, 1121 1369, 1526, 1668, 2938, 2974, 3340 3 ch ₃ ^C 2 ^H 5 Π ^ Hg-C oil, IR (film) 880, 962, 979, 1038, 1526 1668, 2875 2937 2960 3340 4 ch ₃ ^C 2 ^H 5 prop-ene 3-yl 53 - 67 ° C flash point

J Ο -

5 ch ₃ ^C 2 ^H 5 prop-in- 3-yl oil, IR (film) 870, 884, 980, 1008,103 1526, 1670, 2115, 3280 2939, 6 ch ₃ ^C 2 ^H 5 3-methyl-but-oil, IR (film) 2-en-1-yl 884,956,980,108,103 1448, 1525, 1671, 2938, 2972, 3340 7 ch ₃ ch (ch ₃ ) ₂ ch ₃ 78 flash point - 79 ° C 8 ch ₃ ch (ch ₃ ) ₂ ^C 2 ^H 5 64 flash point - 67 ° C 9 ch ₃ ch (ch ₃ ) ₂ 72 flash point - 74 ° C 10 ch ₃ ch (ch ₃ ) ₂ I-C3H7 . 74 flash point -77 ° C 11 ch ₃ ch (ch ₃ ) ₂ N-C ^ Hg 68 flash point - 70 ° C 12 ch ₃ ch (ch ₃ ) ₂ prop-ene 3-yl 59 flash point - 62 ° C 13 ^C 2 ^H 5 ch (ch ₃ ) ₂ prop-in- 3-yl 55 flash point - 57 ° C 14 ^C 2 ^H 5 n-C ^ H? ch ₃ 94 flash point - 96 ° C

38:

^C 2 ^H 5 ^{n C} 3 ^H 7

IR (KBr)

767 890 913 983

1023, 1035, 1523, 1659,

2940, 2970,3408

16 ch ₃ ch ^ chch ₃ ch ₃ ¹ H-NMR (CDCl ₃ ): δ [ppm] 1.8 (d, 3H), 2.03 (s, 3H), 2.90 (d, 3H), 3.96 (s, 6H), 5 10.08 (s, 2H), 6.2 5-6.50 (m, 2H), 6.73 (s 1H), 7.10-7.50 (m, 4H) 17 ch ₃ ch ₂ oc ₆ ch ₅ ch ₃ 136 - 138 ° C flash point 18 ch ₃ CH ₂ ° ^C 6 ^H 5 ch ₂ ch ₃ 108 - 110'C flash point 19 ch ₃ ch ₂ oc ₆ h ₅ ch ₂ -c> ch ¹ H-NMR (CDCl ₃ ):

.delta. [ppm] = 2.02 (s, 3H), 2.46 (m, 1H), 2.81 (d, 3H), 3.86 (s, 3H), 4.78 (s, 2H), 4.9 (s, 2H), 5.05 (s, 2H), 6.69 (s, 1H), 6.80-7.45 (m, 9H)

CH ₃ CH ₂ -O- · CH ₂ -C ₂ CH oil [4-Cl-C ₆ H ₄ ]

384

21 ch ₃ ch ₂ -o- [4-Cl-C ₅ H ₄ ] ch ₂ ch ₃ 105 ° C flash point 22 ch ₃ ch ₂ -o- [4-Cl-C ₆ H ₄ ] ch ₃ 155 ° C flash point 23 ch ₃ ch ₂ -o [4-FC ₆ H ₄ ] ch _{2 -} c = ch . 09 - 90 ° C flash point 24 ch ₃ ch ₂ -o [4-FC ₆ H ₄ ] ch ₂ ch ₃ . 108 ° C flash point 25 ch ₃ ch ₂ -o [4-FC ₆ H ₄ ] ch ₃ . 153 - 156 ° flash point 26 ch ₃ ch ₂ cn ch ₃ . 114 - 116 ° flash point 27 ch ₃ ch ₂ cn ^C 2 ^H 5 . 100 ° C flash point 28 ch ₃ ch ₂ cn ch ₂ c = ch oil 29 ch ₃ ch ₂ -o- [2-CN-C ₆ H ₄ ] ch ₃ .. 103 - 106 ° flash point 30 ch ₃ ch ₂ -o- [2-CN-C ₆ H ₄ ] ^C 2 ^H 5 oil 31 ch ₃ ch ₂ -o- ch ₂ -c _from ch 108 - 112 ° flash point

385 [2-CN-C ₆ H ₅ ]

32 ch ₃ CH ₂ -OCH ₂ -CH [4-CN-C ₆ H ₄ ] Mp 97-100 ° C flash point 33 ch ₃ ch ₂ -o c ₂ h ₅ [4-CN-C ₆ H ₄ ] . 118 - 120 ° <flash point 34 ch ₃ ch ₂ -o c ₂ h ₅ [4-CN-C ₆ H ₄ ] 150 ° C flash point 35 ch ₃ ch ₂ -o- CH ₂ C> CH [1-CH ₃ -3-CF ₃ -pyrazol-5-yl] oil 36 ch ₃ ch ₂ -o- c ₂ h ₅ [1-CH ₃ -3-CF ₃ -pyrazol-5-yl] oil 37 ch ₃ ch ₂ -o-ch ₃ [1-CH ₃ -3-CF ₃ -pyrazol-5-yl] oil 38 ch ₃ c = cc ₆ h ₅ ch ₃ 131-133 ° ( flash point

j bo Table I.D

CO ₂ CH ₃

No R ² R ³ R ⁴ Data 1 ch ₃ ch (ch ₃ ) ₂ prop-ene 3-yl Mp 58-60 ° C flash point 2 ch ₃ ch (ch ₃ ) ₂ but-in- 3-yl oil, IR (film) 925, 950, 1038, 1057, 11

1130, 1256, 1284, 1634, 1710, 2940, 2970, 3290

3 ch ₃ ch (ch ₃ ) ₂ 3-methyl but-2-ene 1-yl . 57-59 ° C flash point 4 ch ₃ ch (ch ₃ ) ₂ prop-in- 3-yl . 51-54 ° C flash point

5 C ₂ H ₅ Ng ₃ H ₇ ch ₃ oil; 1019 ,. IR (film) 1055 1111 1130, 1256 1284 1635 1711, 2939, 2963

C ₂ H ₅ nC ₃ H ₇ CH ₂ CH = CH ₂ oil; IR (film)

957, 1017, 1036, 1111,

1130

1256, 1236, 1436, 1635,

1711, 2940, 2960

C ₂ H ₅ n C ₃ H _?

C ₂ H ₅ n C ₃ H ₇

CH ₂ CH = CH oil; IR (film)

956, 1088, 1043,

1130, 1256, 1284, 1436, 1635,

1710, 2120, 2940, 2960

_CH2 - oil; IR (film) [3-CF 3 -C 6 H 4] 1016, 1074, 1128, 1166,

1192, 1201, 1257, 1330,

1636, 1711, 2940, 2960

CH ₃ C = CC ₆ H ₅ CH ₃ 1 H-NMR (CDCl ₃ ):

2.10 (with, 3H); 3.67 (with , 3H) 3.79 (WITH, 3H); 4.09 (with , 3H) 5.20 (with, 2H); 7,13 -7. 60 (M, 10H) PPm

388 ch ₃ C 4 -C 8 H ₅ ch ₂ c = ch

¹ H-NMR (CDCl ₃ ; ): 2.10 (s. 3H); 2.50 (s, 11 3.67 (s, 3H); 3.77 (S, 31 4.85 (s, 2H); 5.19 (S, 21 7.13-7.58 (m, 10H) ppm

Table I. E

no. R ² R ³ R ⁴ Data 1 ch ₃ ch (ch ₃ ) ₂ ch ₃ 99-100 ° C flash point 2 ch ₃ ^C 2 ^H 5 ch ₃ 85-90 ° C flash point

Tabulks τ.

^{1 CH} 3 ^C 2 ^H 5 ^C 2 ^H 5 78 - 92'C Flash point (β.β)

Examples of effects on harmful fungi

The fungicidal activity of the compounds of formula I can be demonstrated by the following experiments:

The active ingredients were formulated as a 20% emulsion in a mixture of 70% cyclohexanone, 20% Nekanil ^R LN (Lutensol ^R AP6, ethoxylated alkylphenol based wetting agent) and 10% Emulphor ^R EL (Emulan ^R EL, emulsifier based on ethoxylated fatty alcohols) and diluted to the desired concentration with water.

Action against Botrytis cinerea (Gray mold)

Slices of green pepper were sprayed intensively with the treated active ingredient. After drying, the paprika slices were sprayed with a spore suspension of Botrytis cinerea (1.7.10 &lt; 10 &gt;) spores per ml of 2% biological malt solution) and stored for 4 days at 18 [deg.] C. and high humidity. Evaluation was performed visually.

390

In this test, plants treated with 250 ppm of the compounds of the invention showed IC numbers: IC / 7, IC / 8, IC / 10, IC / 11, IC / 13, IB / 7, IB / 8, IB / 10 and IB / 11. (number) infestation of 40% or less, while untreated (control) plants were infested up to 100%.

In the respective test, the plants treated with 250 ppm of the compounds of the invention showed the number IA / 1, IA / 4, IA / 8, IB / 3, IB / 7, IB / 8, IB / 10, IB / 11, IB / 12, IB / 15, IB / 16, IB / 18, IB / 21, IB / 22, IB / 23, IC / 1, IC / 4, IC / 5, IC / 7 IC / 12, IC / 13, IC / 16, IC / 17, IC / 18, IC / 19, ID / 1, ID / 2, ID / 3, ID / 5 and ID / 6 (table / number) 40% or less, while untreated (control) plants were infected up to 100%.

Effect against Erysiphe graminis var. tritici (powdery mildew of wheat)

Wheat germ leaves (Fruhgold species) were first treated with an aqueous solution of the active ingredients. After approximately 24 hours, the plants were dusted with spores of Erysiphe graminis vyr. tritici. The treated plants were then incubated for 7 days at 20-22 ° C and 75-80% relative humidity. Subsequently, the content of fungal development was examined.

In this test, the plants treated with 16 ppm of the compounds of the invention showed IC numbers: IC / 7, IC / 8, IC / 10, IC / 11, IC / 13, IB / 7, IB / 8, IB / 10 and IB / 11. (number) infestation of 25% or less, while untreated (control) plants were infested up to 80%.

In the respective test, plants treated with 16 ppm of the compounds of the invention showed the number IA / 1, IA / 2, IA / 3, IA / 4, IA / 5, IA / 7, IA / 8, IA / 9, IB / 1, IB IB / 3, IB / 5, IB / 6, IB / 9, IB / 12, IB / 13, IB / 14, IB / 15, IB / 16, IB / 17, IB / 18, IC / 1 IC / 2 IC / 3 IC / 4 IC / 5 IC / 9 IC / 12 IC / 14 IC / 15 IC / 16 IC / 35 IC / 38 ID / 1 ID / 2, ID / 3, ID / 4

391

I.D / 5, I.D / 6, I.D / 7, I.D / 8 and I.F / 1 (table / number) infestation of 15% or less, while untreated (control) plants were infested up to 80%.

Effect against Puccinia recondita (Wheat Rust)

Wheat seedlings (Kanzler species) were dusted with spores of Puccinia recondita. The plants so treated were then incubated for 24 hours at a temperature of 20 to 22 ° C and a relative air humidity of 90 to 95% and subsequently treated with an aqueous solution of the active ingredients. After a further 8 days at 20-22 ° C and 65-70% relative humidity, the extent of fungal development was determined. The evaluation was performed visually.

In this test, the plants treated with 63 ppm of the compounds of the invention showed IC / 7, IC / 8, IC / 10, IC / 11, IC / 13, IB / 8, IB / 10 and IB / 11 (table / number) challenge 15% or less, while untreated (control) plants were infected up to 70%.

In the respective test, plants treated with 63 ppm of the compounds of the invention showed IA / 1, IA / 2, IA / 3, IA / 4, IA / 5, IA / 6, IA / 8, IA / 9, IB IB / 2, IB / 3, IB / 9, IB / 12, IB / 13, IB / 14, IB / 15, IB / 16, IB / 19, IB / 22, IB / 24, IC / 1 IC / 2 IC / 3 IC / 4 IC / 5 IC / 6 IC / 9 IC / 12 IC / 13 IC / 16 IC / 24 IC / 27 IC / 28 ID / 2, ID / 5, ID / 6, ID / 7 and ID / 8 (table / number) infestation of 15% or less, while untreated (control) plants were infested up to 70%.

Effect against Pyricularia oryzae

Rice sprouts (Tai Nong 67) were sprayed intensively with the modified active ingredients. After 24 hours, the plants were sprayed with an aqueous spore suspension of Pyricularia oryzae and allowed to stand for 6 days at 20-24 ° C and 95-99% relative humidity. The evaluation was performed visually.

392

In this test, plants treated with 63 ppm of the compounds of the invention showed IC / 7, IC / 8, IC / 10, IC / 11, IC / 13, IB / 7, IB / 8, IB / 10 and IB / 11 (number) infestation of 15% or less, while untreated (control) plants were infested up to 80%.

In the respective test, plants treated with 63 ppm of the compounds of the invention showed the number I.A / 1, I.A / 2, I.A / 4, I.A / 5,

IA / 6, IA / 7, IA / 8, IA / 9, IB / 1, IB / 2, IB / 3, IB / 4, IB / 5, IB / 6, IB / 9 13, IB / 14, IB / 15, IB / 16, IB / 17

I.B / 18, I.B / 19, I.B / 20, I.B / 24, I.B / 26, I.B / 30, I.B / 31,

I.B / 36, I.B / 37, I.B / 38, I C / 1, I C / 2, I C / 3, I C / 4, I C / 5,

I.C / 6, I.C / 9, I.C / 12, I.C / 13, I.C / 14, I.C / 15, I.C / 16, - I.C / 20,

I.C / 21, I.C / 23, I.C / 27, I.C / 28, I.C / 28, I.C / 35, I.C / 36,

IC / 37, ID / 1, ID / 2, ID / 3, ID / 5, ID / 6 and ID / 7 (table / number) infestation of 15% or less, while untreated (control) plants were infested up to 80 %.

Examples of effects against animal pests

The effect of the compounds of formula I on animal pests has been demonstrated by the following experiments:

The active substances were treated as

(a) 0,1% acetone solution; or

(b) 10% emulsion in a mixture consisting of 70% by weight of cyclohexanone, 20% by weight of Nekanil ^R LN (Lutensol ^R AP6, wetting agent with emulsifying and dispersing effect based on ethoxylated alkylphenols) and 10% by weight of Emulphor ^R EL (Emulan ^R EL, emulsifier for base of ethoxylated fatty alcohols) and diluted to the desired concentration with acetone in case a) or water in case b).

393

At the end of the experiments, the lowest concentration was always found, at which the compounds induce 80-100% of the attack or mortality (efficiency threshold or minimum concentration) in comparison with the control experiments on untreated plants.

Nephotettix cincticeps (green cicada), contact effect

Round filters were treated with an aqueous solution of the active ingredients. 5 adult cicadas were then introduced. Mortality was evaluated after 24 hours.

In this experiment, an activity threshold for compounds I.B / 7 and I.B / 10 of less than 0.4 mg was determined.

In the respective test, the compounds of the invention showed the number I.A / 1, I.A / 2, I.A / 4, I.A / 5, I.A / 6, I.A / 9, I.B / 12,

I.B / 13, I.B / 14, I.B / 15, I.B / 29, I.B / 32, IC / 3, IC / 20, IC / 21,

I.C / 22, I.C / 23, I.C / 24, I.C / 25, I.C / 27, I.C / 28 and I.C / 30 Threshold of efficacy 0.4 mg or less.

Nephotettix cincticeps (green cicada), contact effect, spray test

Approximately 8 cm long rice plants were treated with an aqueous solution of the active ingredients, and after drying 10 adult cicadas were introduced. Mortality was assessed after 48 hours.

In this experiment, the activity threshold for compounds I.A / 1, I.A / 2, I.A / 3, I.A / 5, I.A / 6 and I.B / 12 was determined to be 400 ppm or less.

Prodenia litura, contact effect

The bottom of the test vessel was sprayed with acetone solution of the active substance and after evaporation of the solvent, 5 larvae were introduced into the larvae in the 4th stage of larvae development. Mortality was determined after 4 hours.

394

In this experiment, the activity threshold for the compound was determined

1.C / 13 0.4 mg and less.

In the respective assay, the compounds of the invention showed I.A / 8, I.B / 18, I.D / 5, I.D / 6 and I.D / 7 activity thresholds of 0.4 mg or less.

Aphis fabae (system aphid), systemic effect

The heavily attacked cervix (Vicia faba) was treated with an aqueous solution of the active ingredients. After 48 hours, the mortality rate was determined.

In this experiment, compounds I.B / 8, I.B / 10 and I.C / 8 showed activity thresholds of 100-400 ppm.

In the respective test, the compounds of the invention showed I.A / 1, I.A / 2, I.A / 5, I.A / 6, I.B / 25 and I.E / 1 activity thresholds of 400 ppm or less.

Tetranychus urticae (mite) contact effect

The strongly attacked potato bean with two developed leaves was treated with an aqueous solution of the active ingredients. After 5 days in the greenhouse, the result of the intervention was evaluated with a binocular.

In this experiment, compound I.C / 13 showed an activity threshold of less than 100 ppm.

In the respective test, the compounds of the invention showed IA / 7, IA / 8, IA / 9, IB / 15, IB / 16, IB / 18, IB / 19, IB / 20, IC / 20, IC / 23, ID / 4 , ID / 5, ID / 6, ID / 7 and ID / 8 efficiency thresholds of 400 ppm or less.

Claims (7)

1. Phenylacetic acid derivatives of the general formula I rv wz-9 & (I) c = x in which the substituents and the index have the following meanings: X NOCH ₃ , CHOCH ₃ and CHCH ₃ ; Y NR and oxygen; R 1, R ^{1 is} hydrogen or C ₁ -C ₄ -alkyl; R ^{2 is} hydrogen, C ₁ -C 8 -alkyl, C 1 -C 8 -haloalkyl and C ₃ -C 8 -cycloalkyl; R ₄ C ³ -C ₆ -cycloalkyl, C ₂ -C alkyl or C -C alkyl which is partially or fully halogenated and / or carries one to three of the following radicals: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C - ^ - Cg-alkylaminocarbonyl, di-C ^^ - Cg-alkylaminocarbonyl, C _L -C-alkylaminothiocarbonyl, di-C ^ -C-alkylaminothiocarbonyl, C - ^ - Cg-alkylsulfonyl , C 1 -C 8 -alkylsulfoxyl, C 1 -C 8 -alkoxy, C ₁ -C 8 -haloalkoxy, C ₁ -C 8 -alkoxycarbonyl, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylamino, di-C 1 -C 8 -alkylamino, C ₂ -C 8 -alkenyloxy, C ₃ -C 8 -cycloalkyl, C -C _{3-cycloalkoxy,} heterocyclyl, heterocyclyloxy, aryl, aryloxy, aryl C ~ ^- _C4-alkoxy, arylthio, aryl-C, -C ₄ -alkylthio, hetaryl, 396 hetaryloxy, _{hetaryl-C1-C4-alkoxy,} hetarylthio, _{hetaryl-Ci-C4-alkylthio,} wherein the cyclic radicals to be partially or fully halogenated and / or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl, C 1 -C 8 -alkylsulfonyl, C ₁ -C 8 -alkylsulfoxyl, C ₃ -C 8 -cycloalkyl, C 1 -C 8 -alkoxy , C 1 -C 8 -haloalkoxy, C 1 -C 8 -alkoxycarbonyl, C ₁ -C 8 -alkylthio, C 1 -C 8 -alkylamino, di-C 1 -C 8 -alkylamino, C 1 -C 8 -alkylaminocarbonyl, di -C 1 -C 8 -alkylaminocarbonyl, C 1 -C 8 -alkylaminothiocarbonyl, di-C 1 -C 8 -alkylaminothiocarbonyl, C ₂ -C 8 -alkenyl, C ₂ -C 8 -alkenyl, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy , hetarylthio and C (= NOR ^a ) -A _n -R ^b ; C ₂ -C 8 -alkynyl or C ₂ -C 8 -alkenyl, which may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1-4 alkyl; -C-alkylaminocarbonyl, di-C - ^ - Cg-alkylaminocarbonyl, C - ^ - C-alkylaminothiocarbonyl, di-C - ^ - C-alkylaminothiocarbonyl, C - ^ - Cg-alkylsulfonyl, C ₁ -C -alkylsulfoxyl, CJ -C alkoxy, C -C haloalkoxy, C - ^ - C alkoxycarbonyl, C ^ -C alkylthio, C -C -alkylamino, di-C - ^ - C-amino, C ₂ -C alkenyloxy, C ₃ ~ Cg cycloalkyl, C ₃ -C cycloalkoxy, heterocyclyl, heterocyclyloxy, aryl, aryloxy, aryl-C ₁ -C ₄ -alkoxy, arylthio, _{aryl-C1-C4-alkylthio,} hetaryl, hetaryloxy, hetaryl-C ₁ -C ₄ -alkoxy, hetarylthio, hetaryl-aryl-C ₁ -C ₄ -alkylthio, wherein the cyclic radicals may be partially or fully halogenated and / or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino , carboxyl, aminocarbonyl, aminothiocarbonyl, C 1-4 -C 8 -alkyl, C ₁ -C 8 -haloalkyl, C 1 -C 8 -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C ₃ -C 8 -cycloalkyl, C 1 -C 8 -alkoxy, C ₁ -C 8 -haloalkoxy, C 8 -C 8 -alkoxy C ₁ -C 8 -alkoxycarbonyl, C 1 -C 8 -alkylthio, C ₁ -C 8 -alkylamino, di-C ₁ -C 8 -alkylamino, C 1 -C 8 -alkylaminocarbonyl, di-C 1 -C 8 -alkylaminocarbonyl, 397 C ₁ -C -alkylaminothiocarbonyl, di-C - ^ - -alkylaminothiocarbonyl, C ₂ -C alkenyl, C ₂ -C alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarylthio C (= NOR ^a ) -A _n -R ^b ; R ⁴ hydrogen, C 1 -C 10 -alkyl;₃-C₆-cycloalkyl, C₂-C₁₀-alkenyl, C₂-C₁₀-alkynyl, C₂-C₁₀alkylcarbonyl;₃-C₁₀-alkynylcarbonyl or C₁"C._{1 (}-₎alkylsulfonyl, which radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C1-C6-alkyl, C1-C6 -haloalkyl, C1-C6-alkylsulfonyl, C1-C6-alkylsulfoxyl, C1-C6-alkoxy, C1-C6-haloalkoxy, C1-C6-alkoxycarbonyl, C1-C6-alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, C1-C6-alkylaminocarbonyl, di-C1-C6-alkylaminocarbonyl,^Cand^-C6 -alkylaminothiocarbonyl, di-C 1 -C 8 -alkylaminothiocarbonyl, C 2 -C 6 -alkenyl, C 2 -C 8 -alkenyloxy, C 3 -C 8 -cycloalkyl, C 3 -C 8 -cycloalkoxy, heterocyclyl, heterocyclyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, wherein the cyclic radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1 -C 8 -alkyl, C 1 -C 8 - haloalkyl, C 1 -C 8 -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C 3 -C 8 -cycloalkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C 1 -C 8 -alkoxycarbonyl, C 1 -C 8 -alkoxy alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, C1-C6-alkylaminocarbonyl, di-C1-C6-alkylaminocarbonyl, C1-C6-alkylaminothiocarbonyl, di-C1-C6-alkylaminothiocarbonyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarythio or C (= NOR^and) -An ~ R^b; aryl, arylcarbonyl, arylsulfonyl, hetaryl, hetarylcarbonyl wherein these radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carbonyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1 -C 8 - alkyl,^Cand^-c6^-haloalkyl,^Cand^-c6 -alkylsulfonyl, C1-C6-alkylsulfoxyl, C3-C6-cycloalkyl, C1-C6-alkoxy, C1-C6-haloalkoxy, C1-C6-alkoxycarbonyl, C1-C6-alkylthio, C1-C6-alkylamino, di-C 1 -C 6 -alkylamino, C 1 -C 6 -alkylaminocarbonyl, di C 1 -C 6 -alkylaminocarbonyl, C 1 -C 6 -alkylaminothiocarbonyl, di C 1 -C 6 -alkylaminothiocarbonyl, C 2 -C 6 -alkenyl, C 2 -C 8 -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, hetaryl, hetaryloxy, or C (= NOR^and) -An-R k; where A represents oxygen, sulfur or nitrogen, the nitrogen bearing hydrogen or C1-C6-alkyl; n is 0 or 1; R ^a is hydrogen or C 1 -C 6 -alkyl and VR ^d is hydrogen or C 1 -C 6 -alkyl, and salts thereof, with the exception of compounds in which R ¹ and R ² are methyl, R ³ ethyl, R ⁴ methyl or ethyl, X NOCH ₃ and Y NH or O, as well as with the exception of compounds of formula I wherein R ³ is tert-butyl. 2. Phenylacetic acid derivatives of the general formula I C = X 399 in which the substituents and the index have the following meanings: X NOCH ₃ , CHOCH ₃ and CHCH ₃ ; Y NR and oxygen; R 1, R ^{1 is} hydrogen or C ₁ -C ₄ -alkyl; R ² is hydrogen ,. C ₁ -C 8 -alkyl and C ₃ -C 8 -cycloalkyl; R ₄ C ³ -C ₆ cycloalkyl, C ₂ -C -alkyl, C ₂ -C-alkynyl, and C ₂ -C alkenyl; R ⁴ hydrogen, C-C-LQ-alkyl, C ₃ -C cycloalkyl, ^C 2 -C ₁₀ -alkenyl, C ₂ -Cio-alkynyl, C ₂ -C ₁₀ -alkylcarbonyl, C ₂ -C ₁₀ alkenylcarbonyl ~, C ₃ -C _10- alkynylcarbonyl or C 1 -C 6 -alkylsulfonyl, which radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl, C ₁ -C 8 -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C 1 -C 8 -alkoxycarbonyl, C -C alkylthio, C ^ -C-alkylamino, di-C ^ -C-alkyl amino, C -C -alkyl aminocarbonyl, di-C - ^ - Cg-alkylaminocarbonyl, ^C I ^C 6 "-alkylaminotiokarbonyl, di-C _{C 1} -C 8 -alkylaminothiocarbonyl, C ₂ -C 8 -alkenyl, C ₂ -C 8 -alkenyloxy, C ₃ -C 8 -cycloalkyl, C ₃ -C 8 -cycloalkoxy, heterocyclyl, heterocyclyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, wherein the cyclic radicals may be partially or fully halogenated or carry one to three from the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl, C 1 -C 8 -alkyl sulfonyl, C 1 -C 8 -alkylsulfoxyl C ₃ -C-cycloalkyl, C ^ -C alkoxy, C -C haloalkoxy, C - ^ - C-alkoxykarbo400 phenyl, C ₁ -C ₆ -alkylthio, C Cg-alkylamino, di-C ₁ -C alkylamino, C - ^ - Cg-alkylaminocarbonyl, di-C ^ -C-alkylaminocarbonyl, C - ^ - C-alkylaminothiocarbonyl, di-C by lower alkyl aminocarbonyl, C ₂ -C alkenyl, C ₂ -CG- alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarythio or C (= NOR ^a ) -A _n -R ^b ; aryl, arylcarbonyl, arylsulfonyl, hetaryl, hetarylcarbonyl wherein these radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carbonyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1 -C 8 - alkyl, C1-C6-haloalkyl,^CI '^C6 -alkylsulfonyl, C 1 -C 6 -alkylsulfoxyl, C 3 -C 8 -cycloalkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C 1 -C 8 -alkoxycarbonyl, C 1 -C 8 -alkylthio, C 1 -C 8 -alkyloxy; alkylamino, di-C 1 -C 8 -alkylamino, C 1 -C 8 -alkylaminocarbonyl, di-C 1 -C 8 -alkylaminocarbonyl, C 1 -C 8 -alkylaminothiocarbonyl, di-C 1 -C 8 -alkylaminothiocarbonyl, C 2 -C 8- alkenyl, C 2 -C 8 -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, hetaryl, hetaryloxy, or C (= NOR^and) -An-R^b; where A is oxygen, sulfur or nitrogen, the nitrogen having attached to it hydrogen or C ₁ -C alkyl; n is 0 or 1; R ^a is hydrogen or C ₁ -C 8 -alkyl and R ^b is hydrogen or C 1 -C 6 -alkyl and salts thereof, with the exception of compounds in which R ¹ and R ² are methyl, R ³ ethyl, R ⁴ methyl or ethyl, X NOCH ₃ and Y NH or O as well as with the exception of compounds of formula I in which R ³ is tert-butyl. 3. Phenylacetic acid derivatives of the general formula I (I) ON R-C (R · ⁵⁾ -C (R ²⁾ = NOCH ₂ C = X O = C — Y — R ¹ wherein the substituents and the index have the following meanings: noch _3, CKD ₃ and CHCH _3; NR and oxygen; R ^{1 is} hydrogen or C ₁ -C ₄ -alkyl; hydrogen, by lower alkyl, C ^^ - C ^^ - haloalkyl and C ₃ -C cycloalkyl; C 1 -C 6 -alkyl which is partially or fully halogenated and / or carries one to three of the following radicals: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1 -C 6 -alkylaminocarbonyl, di-C ₁ -C 8 -alkylaminocarbonyl, C ₁ -C 8 -alkylaminothiocarbonyl, di C 1 -C 8 -alkylaminothiocarbonyl, C 1 -C 8 -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C 1 -C 8 -alkoxy, C 1 -C 8 -alkoxy cg-haloalkoxy, C - ^ - C alkoxycarbonyl, C ^ -C alkylthio, C ^ -C-alkylamino, di-Cl-cg-alkylamino, C ₂ -C alkenyloxy, C ₃ -C -cycloalkyl, C ₃ -C 8 -cycloalkoxy, heterocyclyl, heterocyclyloxy, aryl, aryloxy, aryl-C 1 -C 4 -alkoxy, arylthio, aryl-C ₁ -C ₄ -alkylthio, hetaryl, hetaryloxy, hetaryl-C ₁ -C ₄ - alkoxy, hetarylthio, hetaryl-C ₁ -C ₄ -alkylthio, wherein the cyclic radicals may be partially or fully halogenated and / or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, C ₁ -C 8 -alkyl, C 1 -C 8 -halo-402 genoalkyl, C 1 -C 8 -alkyl; -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C ₃ -C 8 -cycloalkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C 1 -C 8 -alkoxycarbonyl, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylamino , di-C 1 -C ₈ -alkylamino, C 1 -C 8 -alkylaminocarbonyl, di-C ₁ -C ₆ -alkylaminocarbonyl, C 1 -C 8 -alkylaminothiocarbonyl, di-C ₁ -C 8 -alkylaminothiocarbonyl, C ₂ -C 8 -alkenyl, C ₂ - C 8 -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarythio and C (= NOR ^a ) -A _n -R ^b ; C ₂ -C 8 -alkynyl or C ₂ -C 8 -alkenyl, which may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1-4 alkyl; -C-alkylaminocarbonyl, di-C ₁ -C alkylaminocarbonyl, C -alkylaminothiocarbonyl, di-C ^ -C-alkylaminothiocarbonyl, C ^ -C alkylsulfonyl, C -C-alkylsulfoxyl, C -C alkoxy, C ^ -C -haloalkoxy, C ^ -C alkoxycarbonyl, C ^^ - Cg-alkylthio, C ₁ -C -alkylamino, di-C-Cg-alkylamino, C ₂ -C alkenyloxy, C ₃ -C -cycloalkyl, C ₃ -C 8 -cycloalkyloxy, heterocyclyl, heterocyclyloxy, aryl, aryloxy, aryl-C ₁ -C ₄ -alkoxy, arylthio, aryl-C ₁ -C ₄ -alkylthio, hetaryl, hetaryloxy, hetaryl-C ₁ -C ₄ -alkoxy , hetarylthio, hetaryl-aryl-C 1 -C 4 -alkylthio, wherein the cyclic moieties may be partially or fully halogenated and / or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, C ^ -C-a alkyl, C 1 -C 8 -haloalkyl, C 1 -C 8 -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C ₃ -C 8 -cycloalkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C 1 -C 8 -cycloalkyl alkoxycarbonyl, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylamino, di-C ₁ -C 8 -alkylamino, C ₁ -C 8 -alkylaminocarbonyl, di-C ₁ -C 8 -alkylaminocarbonyl, C 1 -C 8 -alkylaminothiocarbonyl, di-C 1 -C 8 -alkylaminothiocarbonyl, C ₂ -C 8 -alkenyl, C ₂ -C 8 -alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarythio and C (= NO R ^a ) -A _n -R ^b ; R ⁴ hydrogen, 403 C ₁ -C ₁₀ -alkyl, C ₃ -C ₆ cycloalkyl, C ₂ -C ₁₀ -alkenyl, C ₂ -C ₁₀ -alkynyl, ^C 2 -C ₁₀ -alkylcarbonyl, C ₂ -C ₁₀ -alkenylkarbonyl, C ₃ -C ₁₀ -alkynylcarbonyl or C ₁ -C ₁₀ -alkylsulfonyl, which radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C -C alkyl, C ^ -C haloalkyl, C - ^ - C alkylsulfonyl, C -C-alkylsulfoxyl, C ^ -C alkoxy, ^{C -} Cg-haloalkoxy, C ^ -C alkoxycarbonyl, CJ C1-C6-alkylthio, C1-C6-alkylamino, di-C1-C6-alkylamino, C1-C6-alkylaminocarbonyl, di-C1-C6-alkylaminocarbonyl, C1-C6-alkylaminothiocarbonyl, di-C1-C6 -alkylaminothiocarbonyl, C2-C6-alkenyl, C2-C6-alkenyloxy, C3-C6-cycloalkyl, C3-C6-cycloalkoxy, heterocyclyl, heterocyclyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, wherein the cyclic radicals may be partially or wholly halogenated or carrying one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carboxyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1 -C 8 -alkyl, C 1 -C 8 -haloalkyl, C 1 -C 8 -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C 8 -C 8 -cycloalkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C 1 -C 8 -alkoxycarbonyl, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylamino, di-C 1 -C 8 -alkylamino, C 1 -C 8 -alkyloxy; C8-alkylaminocarbonyl, di-C1-C6-alkylaminocarbonyl, C1-C6-alkylaminothiocarbonyl, di-C1-C6-alkylaminothiocarbonyl, C2-C6-alkenyl, C2-C6-alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, arylthio, hetaryl, hetaryloxy, hetarylthio or C (= N0R ^a) -An-R ^b; aryl, arylcarbonyl, arylsulfonyl, hetaryl, hetarylcarbonyl wherein these radicals may be partially or fully halogenated or carry one to three of the following groups: cyano, nitro, hydroxy, mercapto, amino, carbonyl, aminocarbonyl, aminothiocarbonyl, halogen, C 1 -C 6 -alkyl , C 1 -C 8 -haloalkyl, C 1 -C 8 -alkylsulfonyl, C 1 -C 8 -alkylsulfoxyl, C ₃ -C 8 -cycloalkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -haloalkoxy, C 1 -C 8 -haloalkoxy C 1 -C 8 -alkoxycarbonyl, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylamino, di C 1 -C 8 -alkylamino, C 1 -C 8 -alkylaminocarbonyl, di C 1 -C 8 -alkylaminocarbonyl, C ₁ -C 8 -alkylaminocarbonyl alkylaminothiocarbonyl, di-C. ^ - -alkylaminothiocarbonyl, C ₂ -C alkenyl, C ₂ ~ Cg-alkenyloxy, benzyl, benzyloxy, aryl, aryloxy, hetaryl, hetaryloxy or C (= NOR ^a) R ~ n _n ^b ; where A represents oxygen, sulfur or nitrogen, the nitrogen bearing hydrogen or C1-C6-alkyl; n is 0 or 1; R ^a is hydrogen or C 1 -C 6 -alkyl and R ^b is hydrogen or C 1 -C 8 -alkyl, and salts thereof. 4. A compound as claimed in claim 1, wherein X is NOCH ^, Y-NH, R ¹ and R ² methyl, isopropyl, ^R3 and ^R4 is methyl or ethyl Compounds of formula I according to claim 1, wherein R ¹ is methyl. A process for the preparation of compounds of the formula I according to claim 1, characterized in that the benzyl derivative of the formula II is reacted. C = X O = CYR ¹ (II) in which L ¹ represents a nucleophilic exchangeable starting group, in a known manner, with a nydroxyimine of formula III R ⁴ ON = C (R ³ ) -C (R ² ) = NOH (III) A process for the preparation of compounds of formula I according to claim 1, characterized in that the benzyl derivative of formula II according to claim 6 is reacted in a known manner with a dihydroxyimine of formula IV HON = C (R ³ ) -C (R ² ) = NOH to the compound of formula V HON = C (R ³ ) -C (R ² ) = NOCH ₂ c = x OC-YR ¹ (V)