SI2552930T1 - Kristalni (s)-izopropil 2-(((s) - (((2r,3r,4r,5r)-5-(2,4-diokso-3,4-dihidropirimidin-1-(2h)-il)-4- fluoro-3-hidroksi-4-metiltetrahidrofuran-2-il)metoksi)(fenoksi) fosforil)amino)propanoat - Google Patents

Kristalni (s)-izopropil 2-(((s) - (((2r,3r,4r,5r)-5-(2,4-diokso-3,4-dihidropirimidin-1-(2h)-il)-4- fluoro-3-hidroksi-4-metiltetrahidrofuran-2-il)metoksi)(fenoksi) fosforil)amino)propanoat

Info

Publication number
SI2552930T1
SI2552930T1 SI201130617T SI201130617T SI2552930T1 SI 2552930 T1 SI2552930 T1 SI 2552930T1 SI 201130617 T SI201130617 T SI 201130617T SI 201130617 T SI201130617 T SI 201130617T SI 2552930 T1 SI2552930 T1 SI 2552930T1
Authority
SI
Slovenia
Prior art keywords
dihydropyrimidin
propanoate
methyltetrahydrofuran
phosphoryl
dioxo
Prior art date
Application number
SI201130617T
Other languages
English (en)
Inventor
Bruce S. Ross
Michael Joseph Sofia
Ganapati Reddy Pamulapati
Suguna Rachakonda
Hai-Ren Zhang
Byoung-Kwon Chun
Peiyuan Wang
Original Assignee
Gilead Pharmasset Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US12/783,680 external-priority patent/US8642756B2/en
Application filed by Gilead Pharmasset Llc filed Critical Gilead Pharmasset Llc
Priority claimed from EP11714465.9A external-priority patent/EP2552930B1/en
Publication of SI2552930T1 publication Critical patent/SI2552930T1/sl

Links

Classifications

    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
SI201130617T 2010-03-31 2011-03-31 Kristalni (s)-izopropil 2-(((s) - (((2r,3r,4r,5r)-5-(2,4-diokso-3,4-dihidropirimidin-1-(2h)-il)-4- fluoro-3-hidroksi-4-metiltetrahidrofuran-2-il)metoksi)(fenoksi) fosforil)amino)propanoat SI2552930T1 (sl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US31951310P 2010-03-31 2010-03-31
US31954810P 2010-03-31 2010-03-31
US12/783,680 US8642756B2 (en) 2009-05-20 2010-05-20 Nucleoside phosphoramidates
EP11714465.9A EP2552930B1 (en) 2010-03-31 2011-03-31 Crystalline (s)-isopropyl 2-(((s)-(((2r,3r,4r,5r)-5-(2,4-dioxo-3,4-dihydropyrimidin-1-(2h)-yl)-4-fluoro-3-hydroxy-4-methyltetrahydrofuran-2-yl)methoxy)(phenoxy)phosphoryl)amino)propanoate
PCT/US2011/030725 WO2011123645A2 (en) 2010-03-31 2011-03-31 Nucleoside phosphoramidates

Publications (1)

Publication Number Publication Date
SI2552930T1 true SI2552930T1 (sl) 2016-02-29

Family

ID=55359000

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201130617T SI2552930T1 (sl) 2010-03-31 2011-03-31 Kristalni (s)-izopropil 2-(((s) - (((2r,3r,4r,5r)-5-(2,4-diokso-3,4-dihidropirimidin-1-(2h)-il)-4- fluoro-3-hidroksi-4-metiltetrahidrofuran-2-il)metoksi)(fenoksi) fosforil)amino)propanoat

Country Status (4)

Country Link
BR (1) BR122013004621A2 (sl)
ME (2) ME02294B (sl)
RS (1) RS56229B1 (sl)
SI (1) SI2552930T1 (sl)

Also Published As

Publication number Publication date
BR122013004621A2 (pt) 2016-11-22
ME02294B (me) 2016-02-20
ME02846B (me) 2018-01-20
RS56229B1 (sr) 2017-11-30

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