SI1032386T1 - Use of oxazolidinone derivatives for treating arthritis - Google Patents

Use of oxazolidinone derivatives for treating arthritis

Info

Publication number
SI1032386T1
SI1032386T1 SI9830387T SI9830387T SI1032386T1 SI 1032386 T1 SI1032386 T1 SI 1032386T1 SI 9830387 T SI9830387 T SI 9830387T SI 9830387 T SI9830387 T SI 9830387T SI 1032386 T1 SI1032386 T1 SI 1032386T1
Authority
SI
Slovenia
Prior art keywords
treating arthritis
oxazolidinone derivatives
oxazolidinone
psoriasis
arthritis
Prior art date
Application number
SI9830387T
Other languages
English (en)
Slovenian (sl)
Inventor
Donald H. Batts
Roger G. Ulrich
Original Assignee
Pharmacia & Upjohn Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Company filed Critical Pharmacia & Upjohn Company
Publication of SI1032386T1 publication Critical patent/SI1032386T1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
SI9830387T 1997-11-18 1998-11-10 Use of oxazolidinone derivatives for treating arthritis SI1032386T1 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US6568997P 1997-11-18 1997-11-18
US7129798P 1998-01-16 1998-01-16
US7366298P 1998-02-04 1998-02-04
US7524798P 1998-02-19 1998-02-19
US7767298P 1998-03-12 1998-03-12
EP98960157A EP1032386B1 (en) 1997-11-18 1998-11-10 Use of oxazolidinone derivatives for treating arthritis
PCT/US1998/023233 WO1999025344A1 (en) 1997-11-18 1998-11-10 Use of oxazolidinone derivatives for treating psoriasis, arthritis and reducing the toxicity of cancer chemotherapy

Publications (1)

Publication Number Publication Date
SI1032386T1 true SI1032386T1 (en) 2003-06-30

Family

ID=27535698

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9830387T SI1032386T1 (en) 1997-11-18 1998-11-10 Use of oxazolidinone derivatives for treating arthritis

Country Status (16)

Country Link
EP (1) EP1032386B1 (es)
JP (1) JP2001522886A (es)
KR (2) KR100574307B1 (es)
CN (2) CN1546030A (es)
AT (1) ATE233092T1 (es)
AU (1) AU743941B2 (es)
BR (1) BR9815615A (es)
CA (1) CA2303961A1 (es)
DE (1) DE69811717T2 (es)
DK (1) DK1032386T3 (es)
ES (1) ES2193592T3 (es)
HK (1) HK1036591A1 (es)
NZ (1) NZ504612A (es)
PT (1) PT1032386E (es)
SI (1) SI1032386T1 (es)
WO (1) WO1999025344A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP0103082A3 (en) 1998-06-05 2002-12-28 Astrazeneca Ab Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
JP2003529544A (ja) * 1999-09-13 2003-10-07 インサイト・ビジョン・インコーポレイテッド 眼感染症の予防たのための局所処置
US6451345B1 (en) * 2000-01-20 2002-09-17 Eurand Pharmaceuticals Ltd. Functional coating of linezolid microcapsules for taste-masking and associated formulation for oral administration
IL139975A0 (en) * 2000-11-29 2002-02-10 Univ Ramot Anti proliferative drugs
US20050250709A1 (en) * 2003-12-19 2005-11-10 Bionaut Pharmaceuticals Anti-neoplastic agents, combination therapies and related methods
CN107456442A (zh) * 2016-06-03 2017-12-12 四川赛卓药业股份有限公司 一种噁唑烷酮化合物的亚微乳注射剂及其制备方法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2119556C (en) * 1991-11-01 2004-07-06 Michael Robert Barbachyn Substituted aryl- and heteroaryl-phenyloxazolidinones
SK283420B6 (sk) * 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
US5688792A (en) * 1994-08-16 1997-11-18 Pharmacia & Upjohn Company Substituted oxazine and thiazine oxazolidinone antimicrobials
ATE182142T1 (de) * 1993-11-22 1999-07-15 Upjohn Co Substituierte hydroxyacetyl piperazine phenyl oxazolidinonsäureester

Also Published As

Publication number Publication date
DK1032386T3 (da) 2003-05-26
CN1142777C (zh) 2004-03-24
DE69811717T2 (de) 2003-10-16
EP1032386B1 (en) 2003-02-26
KR20050100009A (ko) 2005-10-17
CA2303961A1 (en) 1999-05-27
CN1546030A (zh) 2004-11-17
DE69811717D1 (de) 2003-04-03
HK1036591A1 (en) 2002-01-11
WO1999025344A1 (en) 1999-05-27
BR9815615A (pt) 2000-10-24
ES2193592T3 (es) 2003-11-01
AU1582399A (en) 1999-06-07
NZ504612A (en) 2002-08-28
CN1299281A (zh) 2001-06-13
KR20010032178A (ko) 2001-04-16
EP1032386A1 (en) 2000-09-06
JP2001522886A (ja) 2001-11-20
AU743941B2 (en) 2002-02-07
PT1032386E (pt) 2003-07-31
KR100589545B1 (ko) 2006-06-19
ATE233092T1 (de) 2003-03-15
KR100574307B1 (ko) 2006-04-27

Similar Documents

Publication Publication Date Title
NZ307509A (en) Use of 1L agonists in the treatment of incontinence
IL123142A0 (en) The use of adamantan-derivatives for the treatment of the inner ear
DE50214206D1 (de) Kombinationstherapie substituierter oxazolidinone
MX9707453A (es) Derivados de quinazolina.
UA39936C2 (uk) 2-(2,6-дифторфеніл)-4-(2-етокси-4-трет-бутилфеніл)-2-оксазолін, спосіб мiтицидної обробки та мiтицидна композиція
ES2164040T1 (es) Uso de agonistas del sitio de union de la glicina o de inhibidores de la absorcion de la glicina para el tratamiento de trastornos neuropsiquiatricos.
BR0107667A (pt) Composto de linezolida em forma de cristal que e farmaceuticamente útil como agente antibacteriano e método de preparação do mesmo
DE60016460D1 (de) Verwendungen und zusammenstellungen von nitratestern als sedativa
PL346876A1 (en) Mglur5 antagonists for the treatment of pain and anxiety
IL129748A0 (en) Novel compounds useful as neuro-protective agents
DE69818294D1 (de) Oxazolidinone derivate und pharmazeutische zusammensetzungen
SI1032386T1 (en) Use of oxazolidinone derivatives for treating arthritis
NZ320355A (en) Use of 1-(2-naphth-2-ylethyl)-4-(3-trifluoromethylphenyl)-1,2,3,6- tetrahydropyridine for preparing drugs for treating amyotrophic lateral sclerosis
BR0009380A (pt) Tratamento de câncer melhorado comtemozolomida
MY137595A (en) N-(3-methoxy-5-methylpyrazin-2-yl)-2-(4-[1,3,4-oxadiazol-2-yl]phenyl)pyridine-3-sulphonamide for the treatment of cancer
AU655958B2 (en) Use of quisqualate-receptor antagonists for treating Parkinson's disease
PT75728A (en) 6-fluoro-3-<3-(1-heterocyclo)propyl>-1,2-benzisoxazoles a process for their preparation pharmaceutical compositions thereof and their use as medicaments
ES2187156T3 (es) Terapia antidepresiva.
PH24609A (en) 5-(3-alkyl-5-tert, butyl-s-hydroxyphenyl)-2-amino-6h-1,3,4-thiadiazines, medicaments containing same and the use thereof
MY111623A (en) Neuroprotective compounds
EP1304107A3 (en) Use of oxazolidinines derivatives for treating psoriasis
EA199800085A1 (ru) Способ лечения боли висцерального происхождения, способ лечения воспалительного колита
TW362097B (en) 3-Phenyl-1, 4-dialkyl-1,2,4-triazolium salts and their use as antidepressants
AR035986A1 (es) Uso de derivados anti-convulsivos para la manufactura de un medicamento util para el tratamiento del temblor esencial
ZA966775B (en) Use of prostane derivatives and the combination thereof with antibiotics in the treatment of bacterial infections.