SG11202112354SA - Crystal form of pyridone derivative, and preparation method and use thereof - Google Patents

Crystal form of pyridone derivative, and preparation method and use thereof

Info

Publication number
SG11202112354SA
SG11202112354SA SG11202112354SA SG11202112354SA SG11202112354SA SG 11202112354S A SG11202112354S A SG 11202112354SA SG 11202112354S A SG11202112354S A SG 11202112354SA SG 11202112354S A SG11202112354S A SG 11202112354SA SG 11202112354S A SG11202112354S A SG 11202112354SA
Authority
SG
Singapore
Prior art keywords
preparation
crystal form
pyridone derivative
pyridone
derivative
Prior art date
Application number
SG11202112354SA
Other languages
English (en)
Inventor
Qing Shao
Libin Gan
Li Chen
Original Assignee
Jiangxi Caishi Pharmaceutical Technology Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jiangxi Caishi Pharmaceutical Technology Co Ltd filed Critical Jiangxi Caishi Pharmaceutical Technology Co Ltd
Publication of SG11202112354SA publication Critical patent/SG11202112354SA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53831,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/20Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SG11202112354SA 2019-05-08 2019-11-05 Crystal form of pyridone derivative, and preparation method and use thereof SG11202112354SA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN201910381020.0A CN111909174B (zh) 2019-05-08 2019-05-08 吡啶酮衍生物的晶型及制备方法和应用
PCT/CN2019/115641 WO2020224208A1 (fr) 2019-05-08 2019-11-05 Forme cristalline d'un dérivé de pyridone, procédé de préparation correspondant et utilisation associée

Publications (1)

Publication Number Publication Date
SG11202112354SA true SG11202112354SA (en) 2021-12-30

Family

ID=73050743

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202112354SA SG11202112354SA (en) 2019-05-08 2019-11-05 Crystal form of pyridone derivative, and preparation method and use thereof

Country Status (8)

Country Link
US (1) US20230144122A1 (fr)
EP (1) EP3967697A4 (fr)
CN (2) CN111909174B (fr)
AU (1) AU2019444375B2 (fr)
CA (1) CA3139343A1 (fr)
SG (1) SG11202112354SA (fr)
WO (1) WO2020224208A1 (fr)
ZA (1) ZA202108765B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115385932A (zh) * 2021-05-22 2022-11-25 江西彩石医药科技有限公司 吡啶酮衍生物的中间体及其制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT2444400T (lt) * 2009-06-15 2018-06-11 Shionogi & Co., Ltd. Pakeistasis policiklinis karbamoilpiridono darinys
AU2011307087B2 (en) * 2010-09-24 2016-11-10 Shionogi & Co., Ltd. Substituted polycyclic carbamoyl pyridone derivative prodrug
MX2017013809A (es) * 2015-04-28 2018-03-15 Shionogi & Co Derivados de piridona policiclica sustituida y profarmaco de los mismos.
KR20190014086A (ko) * 2016-08-10 2019-02-11 시오노기세야쿠 가부시키가이샤 치환된 다환성 피리돈 유도체 및 그의 프로드러그를 함유하는 의약 조성물
WO2019141179A1 (fr) * 2018-01-17 2019-07-25 银杏树药业(苏州)有限公司 Dérivé de pyridone, composition de celui-ci et son utilisation en tant que médicament contre la grippe

Also Published As

Publication number Publication date
CA3139343A1 (fr) 2020-11-12
CN111670191B (zh) 2021-07-13
CN111909174B (zh) 2022-01-21
WO2020224208A1 (fr) 2020-11-12
EP3967697A1 (fr) 2022-03-16
CN111909174A (zh) 2020-11-10
CN111670191A (zh) 2020-09-15
EP3967697A4 (fr) 2023-07-05
AU2019444375A1 (en) 2021-12-02
AU2019444375B2 (en) 2023-04-20
US20230144122A1 (en) 2023-05-11
ZA202108765B (en) 2023-07-26

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