SG11202112354SA - Crystal form of pyridone derivative, and preparation method and use thereof - Google Patents

Crystal form of pyridone derivative, and preparation method and use thereof

Info

Publication number
SG11202112354SA
SG11202112354SA SG11202112354SA SG11202112354SA SG11202112354SA SG 11202112354S A SG11202112354S A SG 11202112354SA SG 11202112354S A SG11202112354S A SG 11202112354SA SG 11202112354S A SG11202112354S A SG 11202112354SA SG 11202112354S A SG11202112354S A SG 11202112354SA
Authority
SG
Singapore
Prior art keywords
preparation
crystal form
pyridone derivative
pyridone
derivative
Prior art date
Application number
SG11202112354SA
Inventor
Qing Shao
Libin Gan
Li Chen
Original Assignee
Jiangxi Caishi Pharmaceutical Technology Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jiangxi Caishi Pharmaceutical Technology Co Ltd filed Critical Jiangxi Caishi Pharmaceutical Technology Co Ltd
Publication of SG11202112354SA publication Critical patent/SG11202112354SA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53831,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/20Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SG11202112354SA 2019-05-08 2019-11-05 Crystal form of pyridone derivative, and preparation method and use thereof SG11202112354SA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN201910381020.0A CN111909174B (en) 2019-05-08 2019-05-08 Crystal form of pyridone derivative, preparation method and application
PCT/CN2019/115641 WO2020224208A1 (en) 2019-05-08 2019-11-05 Pyridone derivative crystal form and preparation method and application therefor

Publications (1)

Publication Number Publication Date
SG11202112354SA true SG11202112354SA (en) 2021-12-30

Family

ID=73050743

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202112354SA SG11202112354SA (en) 2019-05-08 2019-11-05 Crystal form of pyridone derivative, and preparation method and use thereof

Country Status (8)

Country Link
US (1) US20230144122A1 (en)
EP (1) EP3967697A4 (en)
CN (2) CN111909174B (en)
AU (1) AU2019444375B2 (en)
CA (1) CA3139343A1 (en)
SG (1) SG11202112354SA (en)
WO (1) WO2020224208A1 (en)
ZA (1) ZA202108765B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022247759A1 (en) * 2021-05-22 2022-12-01 江西彩石医药科技有限公司 Intermediate of pyridone derivative and preparation method therefor

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT2444400T (en) * 2009-06-15 2018-06-11 Shionogi & Co., Ltd. Substituted polycyclic carbamoylpyridone derivative
TR201810736T4 (en) * 2010-09-24 2018-08-27 Shionogi & Co Substituted polycyclic carbamoyl pyridone derivative prodrug.
EP4219508B1 (en) * 2015-04-28 2024-06-05 Shionogi & Co., Ltd Substituted polycyclic pyridone derivative and prodrug thereof
CN110494141A (en) * 2016-08-10 2019-11-22 盐野义制药株式会社 Pharmaceutical composition containing substituted polycyclic Pyridione derivatives and its prodrug
KR102477187B1 (en) * 2018-01-17 2022-12-12 장시 카이시 파마슈티컬 테크놀로지 컴퍼니 리미티드 Pyridone derivatives, their stereoisomers and their applications as anti-influenza virus drugs

Also Published As

Publication number Publication date
AU2019444375B2 (en) 2023-04-20
EP3967697A4 (en) 2023-07-05
CN111670191A (en) 2020-09-15
CN111670191B (en) 2021-07-13
ZA202108765B (en) 2023-07-26
CN111909174B (en) 2022-01-21
CA3139343A1 (en) 2020-11-12
AU2019444375A1 (en) 2021-12-02
CN111909174A (en) 2020-11-10
WO2020224208A1 (en) 2020-11-12
EP3967697A1 (en) 2022-03-16
US20230144122A1 (en) 2023-05-11

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