SG11201604954YA - Novel tetrahydropyridopyrimidine compound or salt thereof - Google Patents
Novel tetrahydropyridopyrimidine compound or salt thereofInfo
- Publication number
- SG11201604954YA SG11201604954YA SG11201604954YA SG11201604954YA SG11201604954YA SG 11201604954Y A SG11201604954Y A SG 11201604954YA SG 11201604954Y A SG11201604954Y A SG 11201604954YA SG 11201604954Y A SG11201604954Y A SG 11201604954YA SG 11201604954Y A SG11201604954Y A SG 11201604954YA
- Authority
- SG
- Singapore
- Prior art keywords
- salt
- tetrahydropyridopyrimidine compound
- novel
- novel tetrahydropyridopyrimidine
- compound
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2014111147 | 2014-05-29 | ||
| PCT/JP2015/065425 WO2015182712A1 (en) | 2014-05-29 | 2015-05-28 | Novel tetrahydropyridopyrimidine compound or salt thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG11201604954YA true SG11201604954YA (en) | 2016-07-28 |
Family
ID=54699035
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG11201604954YA SG11201604954YA (en) | 2014-05-29 | 2015-05-28 | Novel tetrahydropyridopyrimidine compound or salt thereof |
Country Status (21)
| Country | Link |
|---|---|
| US (3) | US9662333B2 (en) |
| EP (1) | EP3150599B1 (en) |
| JP (1) | JP5851663B1 (en) |
| KR (1) | KR101708604B1 (en) |
| CN (1) | CN106103434B (en) |
| AU (2) | AU2015268494B2 (en) |
| BR (1) | BR112016027691B1 (en) |
| CA (1) | CA2941668C (en) |
| DK (1) | DK3150599T3 (en) |
| ES (1) | ES2703168T3 (en) |
| HU (1) | HUE041645T2 (en) |
| MX (1) | MX360496B (en) |
| MY (1) | MY162886A (en) |
| PH (1) | PH12016501252A1 (en) |
| PL (1) | PL3150599T3 (en) |
| PT (1) | PT3150599T (en) |
| RU (1) | RU2636310C1 (en) |
| SG (1) | SG11201604954YA (en) |
| TR (1) | TR201819419T4 (en) |
| TW (1) | TWI585087B (en) |
| WO (1) | WO2015182712A1 (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112016027691B1 (en) | 2014-05-29 | 2019-07-02 | Taiho Pharmaceutical Co., Ltd. | TETRAHYDROPYRYPYRYRIMIDINE COMPOSITE AND ITS USES |
| CN108431001B (en) * | 2015-11-27 | 2021-09-17 | 大鹏药品工业株式会社 | Fused ring pyrimidine compound or salt thereof |
| TWI726969B (en) | 2016-01-11 | 2021-05-11 | 比利時商健生藥品公司 | Substituted thiohydantoin derivatives as androgen receptor antagonists |
| BR112019009448A2 (en) * | 2016-11-28 | 2019-07-30 | Teijin Pharma Ltd | crystal of a compound, its use and pharmaceutical composition |
| CN106727588A (en) * | 2016-11-30 | 2017-05-31 | 顾克斌 | A kind of pharmaceutical composition for treating ALI |
| CN108484594B (en) * | 2018-02-09 | 2020-08-04 | 福建医科大学 | Alkoxy substituted tetrahydropyridopyrimidine compound or available salt thereof, and preparation method and application thereof |
| KR20210095659A (en) | 2018-11-26 | 2021-08-02 | 다이호야쿠힌고교 가부시키가이샤 | A method for treating and preventing tumors to which endocrine therapy is applied by using a combination of a fibroblast growth factor receptor inhibitor and endocrine therapy |
| WO2021058017A1 (en) * | 2019-09-29 | 2021-04-01 | Beigene, Ltd. | Degradation of androgen receptor (ar) by conjugation of ar antagonists with e3 ligase ligand and methods of use |
| WO2022212631A1 (en) * | 2021-03-31 | 2022-10-06 | Taiho Pharmaceutical Co., Ltd. | Treatment of patients metastatic castration-resistant prostate cancer with an androgen receptor antagonist |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002088073A (en) * | 2000-09-08 | 2002-03-27 | Yamanouchi Pharmaceut Co Ltd | Anti-androgenic agent |
| TW200530235A (en) | 2003-12-24 | 2005-09-16 | Renovis Inc | Bicycloheteroarylamine compounds as ion channel ligands and uses thereof |
| US7312330B2 (en) | 2003-12-24 | 2007-12-25 | Renovis, Inc. | Bicycloheteroarylamine compounds as ion channel ligands and uses thereof |
| US20060128710A1 (en) | 2004-12-09 | 2006-06-15 | Chih-Hung Lee | Antagonists to the vanilloid receptor subtype 1 (VR1) and uses thereof |
| NZ555974A (en) * | 2005-01-10 | 2010-11-26 | Acadia Pharm Inc | Aminophenyl derivatives as selective androgen receptor modulators |
| BRPI0614397A2 (en) * | 2005-08-04 | 2011-03-29 | Janssen Pharmaceutica Nv | pyrimidine compounds as serotonin receptor modulators |
| US7598255B2 (en) | 2005-08-04 | 2009-10-06 | Janssen Pharmaceutica Nv | Pyrimidine compounds as serotonin receptor modulators |
| EP2328871B1 (en) | 2008-08-25 | 2020-04-01 | Novartis AG | Hedgehog pathway modulators |
| BR112016027691B1 (en) * | 2014-05-29 | 2019-07-02 | Taiho Pharmaceutical Co., Ltd. | TETRAHYDROPYRYPYRYRIMIDINE COMPOSITE AND ITS USES |
-
2015
- 2015-05-28 BR BR112016027691-4A patent/BR112016027691B1/en active IP Right Grant
- 2015-05-28 SG SG11201604954YA patent/SG11201604954YA/en unknown
- 2015-05-28 KR KR1020167020993A patent/KR101708604B1/en active IP Right Grant
- 2015-05-28 WO PCT/JP2015/065425 patent/WO2015182712A1/en active Application Filing
- 2015-05-28 JP JP2015543973A patent/JP5851663B1/en active Active
- 2015-05-28 DK DK15799768.5T patent/DK3150599T3/en active
- 2015-05-28 RU RU2016125885A patent/RU2636310C1/en active
- 2015-05-28 PL PL15799768T patent/PL3150599T3/en unknown
- 2015-05-28 ES ES15799768T patent/ES2703168T3/en active Active
- 2015-05-28 EP EP15799768.5A patent/EP3150599B1/en active Active
- 2015-05-28 PT PT15799768T patent/PT3150599T/en unknown
- 2015-05-28 MX MX2016010427A patent/MX360496B/en active IP Right Grant
- 2015-05-28 TR TR2018/19419T patent/TR201819419T4/en unknown
- 2015-05-28 HU HUE15799768A patent/HUE041645T2/en unknown
- 2015-05-28 CN CN201580012484.4A patent/CN106103434B/en active Active
- 2015-05-28 AU AU2015268494A patent/AU2015268494B2/en active Active
- 2015-05-28 US US15/023,894 patent/US9662333B2/en active Active
- 2015-05-28 MY MYPI2016702470A patent/MY162886A/en unknown
- 2015-05-28 TW TW104117335A patent/TWI585087B/en active
- 2015-05-28 CA CA2941668A patent/CA2941668C/en active Active
-
2016
- 2016-06-24 PH PH12016501252A patent/PH12016501252A1/en unknown
- 2016-07-06 US US15/203,059 patent/US9889136B2/en active Active
-
2017
- 2017-08-24 AU AU2017219032A patent/AU2017219032B2/en active Active
-
2018
- 2018-02-12 US US15/893,804 patent/US10300067B2/en active Active
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