SG10201400420PA - Therapeutic applications in the cardiovascular field of quinazolinedione derivatives - Google Patents

Therapeutic applications in the cardiovascular field of quinazolinedione derivatives

Info

Publication number
SG10201400420PA
SG10201400420PA SG10201400420PA SG10201400420PA SG10201400420PA SG 10201400420P A SG10201400420P A SG 10201400420PA SG 10201400420P A SG10201400420P A SG 10201400420PA SG 10201400420P A SG10201400420P A SG 10201400420PA SG 10201400420P A SG10201400420P A SG 10201400420PA
Authority
SG
Singapore
Prior art keywords
therapeutic applications
cardiovascular field
quinazolinedione derivatives
quinazolinedione
derivatives
Prior art date
Application number
SG10201400420PA
Inventor
Philip Janiak
Gilbert Marciniak
Jean-Francois Nave
Fabrice Viviani
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of SG10201400420PA publication Critical patent/SG10201400420PA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
SG10201400420PA 2009-04-09 2010-04-07 Therapeutic applications in the cardiovascular field of quinazolinedione derivatives SG10201400420PA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0901755A FR2944206B1 (en) 2009-04-09 2009-04-09 THERAPEUTIC APPLICATIONS IN THE CARDIOVASCULAR FIELD OF QUINAZOLINEDIONE DERIVATIVES

Publications (1)

Publication Number Publication Date
SG10201400420PA true SG10201400420PA (en) 2014-05-29

Family

ID=41181038

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10201400420PA SG10201400420PA (en) 2009-04-09 2010-04-07 Therapeutic applications in the cardiovascular field of quinazolinedione derivatives
SG2011073459A SG175131A1 (en) 2009-04-09 2010-04-07 Therapeutic applications in the cardiovascular field of quinazolinedione derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG2011073459A SG175131A1 (en) 2009-04-09 2010-04-07 Therapeutic applications in the cardiovascular field of quinazolinedione derivatives

Country Status (35)

Country Link
US (1) US8846654B2 (en)
EP (1) EP2416777B1 (en)
JP (1) JP5685578B2 (en)
KR (1) KR101686267B1 (en)
CN (1) CN102458409B (en)
AR (1) AR076232A1 (en)
AU (1) AU2010233596B2 (en)
BR (1) BRPI1010256A2 (en)
CA (1) CA2758234A1 (en)
CL (1) CL2011002525A1 (en)
CO (1) CO6440577A2 (en)
CR (1) CR20110527A (en)
CY (1) CY1115987T1 (en)
DK (1) DK2416777T3 (en)
DO (1) DOP2011000306A (en)
EA (1) EA020984B1 (en)
EC (1) ECSP11011377A (en)
ES (1) ES2528633T3 (en)
FR (1) FR2944206B1 (en)
HK (1) HK1165997A1 (en)
HR (1) HRP20150106T1 (en)
HU (1) HUE024161T2 (en)
IL (1) IL215610A (en)
MA (1) MA33254B1 (en)
MX (1) MX2011010645A (en)
NI (1) NI201100180A (en)
NZ (1) NZ595660A (en)
PL (1) PL2416777T3 (en)
PT (1) PT2416777E (en)
SG (2) SG10201400420PA (en)
SI (1) SI2416777T1 (en)
TN (1) TN2011000506A1 (en)
TW (1) TWI457330B (en)
UY (1) UY32555A (en)
WO (1) WO2010116090A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2944282B1 (en) * 2009-04-09 2013-05-03 Sanofi Aventis QUINAZOLINEDIONE DERIVATIVES, THEIR PREPARATION AND THEIR VARIOUS THERAPEUTIC APPLICATIONS
WO2013184806A1 (en) 2012-06-05 2013-12-12 University Of Kansas Inhibitors of respiratory syncytial virus
US9951038B2 (en) 2012-12-27 2018-04-24 Purdue Pharma L.P. Quinazolin-4(3H)-one-type piperidine compounds and uses thereof
WO2024038089A1 (en) 2022-08-18 2024-02-22 Mitodicure Gmbh Use of a therapeutic agent with phosphodiesterase-7 inhibitory activity for the treatment and prevention of diseases associated with chronic fatigue, exhaustion and/or exertional intolerance

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3879393A (en) * 1973-06-18 1975-04-22 Miles Lab Derivatives of 1,3-disubstituted 2,4(1h,3h)-quinazolinediones
JPS56164172A (en) * 1980-05-22 1981-12-17 Masayuki Ishikawa Novel 2,4 1h,3h -quinazolinedione derivative
EP0040793B1 (en) * 1980-05-22 1985-08-28 Masayuki Ishikawa Novel quinazoline-dione compounds, process for production thereof and pharmaceutical use thereof
US5624926A (en) 1993-02-18 1997-04-29 Kyowa Hakko Kogyo Co., Ltd. Piperidinyl-dioxoquinazolines as adenosine reuptake inhibitors
BR9909781A (en) 1998-04-20 2000-12-19 Fujisawa Pharmaceutical Co Compound of formula (i), process for its preparation, pharmaceutical composition comprising said compound, its use and method.
AU2525701A (en) 1999-12-14 2001-06-25 Sanofi-Synthelabo Derivatives of quinazolinedione phthalimide, preparations thereof and their therapeutic uses
WO2006092692A1 (en) 2005-03-01 2006-09-08 Pfizer Limited Use of combinations of pde7 inhibitors and alpha-2-delty ligands for the treatment of neuropathic pain
AU2006219643A1 (en) 2005-03-01 2006-09-08 Pfizer Limited Use of PDE7 inhibitors for the treatment of neuropathic pain
WO2007067946A2 (en) 2005-12-07 2007-06-14 The Regents Of The University Of California Diagnosis and treatment of chronic lymphocytic leukemia (cll)
BRPI0809244A2 (en) 2007-03-27 2014-09-23 Omeros Corp METHODS OF TREATMENT OF A MOVEMENT ABNORMALITY, AND FOR IDENTIFYING AN AGENT INHIBITING PDE7 ACTIVITY.
TW200911755A (en) 2007-04-19 2009-03-16 Astellas Pharma Inc Bicyclic heterocyclic compounds
FR2921926B1 (en) * 2007-10-03 2009-12-04 Sanofi Aventis QUINAZOLINEDIONE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC APPLICATIONS THEREOF.
FR2943673B1 (en) * 2009-03-27 2013-03-29 Sanofi Aventis THERAPEUTIC APPLICATIONS OF QUINAZOLINEDIONE DERIVATIVES

Also Published As

Publication number Publication date
US8846654B2 (en) 2014-09-30
IL215610A (en) 2013-07-31
ECSP11011377A (en) 2011-11-30
CY1115987T1 (en) 2017-01-25
NZ595660A (en) 2013-03-28
DK2416777T3 (en) 2015-02-09
MA33254B1 (en) 2012-05-02
FR2944206A1 (en) 2010-10-15
PL2416777T3 (en) 2015-05-29
AU2010233596B2 (en) 2016-06-23
SG175131A1 (en) 2011-11-28
US20120184522A1 (en) 2012-07-19
SI2416777T1 (en) 2015-02-27
UY32555A (en) 2010-11-30
CA2758234A1 (en) 2010-10-14
AU2010233596A1 (en) 2011-11-03
CN102458409B (en) 2014-06-18
KR101686267B1 (en) 2016-12-13
NI201100180A (en) 2012-01-11
CL2011002525A1 (en) 2012-02-17
EP2416777A1 (en) 2012-02-15
HK1165997A1 (en) 2012-10-19
BRPI1010256A2 (en) 2016-03-22
AR076232A1 (en) 2011-05-26
PT2416777E (en) 2015-02-04
EA201171229A1 (en) 2012-12-28
KR20120005499A (en) 2012-01-16
EP2416777B1 (en) 2014-11-12
EA020984B1 (en) 2015-03-31
TN2011000506A1 (en) 2013-05-24
WO2010116090A1 (en) 2010-10-14
TW201040155A (en) 2010-11-16
TWI457330B (en) 2014-10-21
JP5685578B2 (en) 2015-03-18
CO6440577A2 (en) 2012-05-15
HUE024161T2 (en) 2016-02-29
CR20110527A (en) 2014-05-12
IL215610A0 (en) 2011-12-29
FR2944206B1 (en) 2012-12-28
HRP20150106T1 (en) 2015-05-08
DOP2011000306A (en) 2011-10-31
ES2528633T3 (en) 2015-02-11
CN102458409A (en) 2012-05-16
MX2011010645A (en) 2012-01-19
JP2012523398A (en) 2012-10-04

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