SE8401321D0 - NEW AZOLES, PROCESSES FOR THEIR PREPARATION AND THEIR USE - Google Patents

NEW AZOLES, PROCESSES FOR THEIR PREPARATION AND THEIR USE

Info

Publication number
SE8401321D0
SE8401321D0 SE8401321A SE8401321A SE8401321D0 SE 8401321 D0 SE8401321 D0 SE 8401321D0 SE 8401321 A SE8401321 A SE 8401321A SE 8401321 A SE8401321 A SE 8401321A SE 8401321 D0 SE8401321 D0 SE 8401321D0
Authority
SE
Sweden
Prior art keywords
optionally substituted
processes
preparation
represent hydrogen
substituted aliphatic
Prior art date
Application number
SE8401321A
Other languages
Swedish (sv)
Other versions
SE8401321L (en
Inventor
A Stutz
H Egger
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of SE8401321D0 publication Critical patent/SE8401321D0/en
Publication of SE8401321L publication Critical patent/SE8401321L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/215—Radicals derived from nitrogen analogues of carbonic acid

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Compounds of formula I <IMAGE> wherein R1 and R2 represent independently an optionally substituted aliphatic, heteroaryl or aryl group or R1 may also represent hydrogen, R3 and R4 represent hydrogen, halogen, nitro, an optionally substituted aliphatic group which is optionally attached via S, O, SO or SO2, or optionally substituted phenyl or phenoxy and X represents N or Ch; in free form or in the form of an acid addition salt, are indicated for use as pharmaceuticals in particular as anti mycotics, and as agrochemicals e.g. as fungicides.
SE8401321A 1983-03-11 1984-03-09 NEW AZOLES, THE PROCEDURES FOR THEIR PRODUCTION AND THEIR USE SE8401321L (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1332/83A CH655103A5 (en) 1983-03-11 1983-03-11 AZOLE DERIVATIVES, METHOD FOR THEIR PRODUCTION AND THEIR USE.

Publications (2)

Publication Number Publication Date
SE8401321D0 true SE8401321D0 (en) 1984-03-09
SE8401321L SE8401321L (en) 1984-09-12

Family

ID=4207992

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8401321A SE8401321L (en) 1983-03-11 1984-03-09 NEW AZOLES, THE PROCEDURES FOR THEIR PRODUCTION AND THEIR USE

Country Status (24)

Country Link
JP (1) JPS59175472A (en)
KR (1) KR890000377B1 (en)
AU (1) AU571494B2 (en)
BE (1) BE899073A (en)
CA (1) CA1242723A (en)
CH (1) CH655103A5 (en)
DE (1) DE3408127A1 (en)
DK (1) DK149784A (en)
ES (1) ES530461A0 (en)
FI (1) FI840968A (en)
FR (1) FR2542315B1 (en)
GB (1) GB2136801B (en)
GR (1) GR81869B (en)
HU (1) HUT36098A (en)
IL (1) IL71203A (en)
IT (1) IT1199085B (en)
LU (1) LU85245A1 (en)
NL (1) NL8400730A (en)
NZ (1) NZ207453A (en)
PH (1) PH24667A (en)
PL (1) PL146072B1 (en)
PT (1) PT78226B (en)
SE (1) SE8401321L (en)
ZA (1) ZA841782B (en)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8618188D0 (en) * 1986-07-25 1986-09-03 Ici Plc Diamine compounds
DE3644616A1 (en) * 1986-12-29 1988-07-07 Lentia Gmbh IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION AND USE THEREOF
DE3644615A1 (en) * 1986-12-29 1988-07-07 Lentia Gmbh IMIDAZOLE AND TRIAZOLE DERIVATIVES FOR USE AS AN ANTIMYCOTIC AGENTS
US5252594A (en) * 1992-06-17 1993-10-12 Rohm And Haas Company Fungicidal (2-aryl-2-substituted)ethyl-1,2,4-triazoles
US5358939A (en) * 1992-06-25 1994-10-25 Rohm And Haas Company Fungicidal 2-aryl-2,2-disubstituted ethyl-1,2,4-triazoles
DE4412358A1 (en) * 1994-04-11 1995-10-12 Bayer Ag Cyclopropyl ethyl azoles
GB9409882D0 (en) * 1994-05-18 1994-07-06 Sandoz Ltd Organic compounds
JP3214987B2 (en) * 1994-09-05 2001-10-02 日本碍子株式会社 Semiconductor device and method of manufacturing the same
AU2003299750A1 (en) * 2002-12-20 2004-07-22 Irm Llc Differential tumor cytotoxocity compounds and compositions
WO2004056744A1 (en) 2002-12-23 2004-07-08 Janssen Pharmaceutica N.V. Adamantyl acetamides as hydroxysteroid dehydrogenase inhibitors
NZ551077A (en) 2004-05-07 2009-05-31 Janssen Pharmaceutica Nv Pyrrolidin-2-one and piperidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors
JP5137574B2 (en) 2004-08-30 2013-02-06 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Tricyclic lactam derivatives as 11-beta hydroxy steroid hydrogenase inhibitors
ES2338441T3 (en) 2004-08-30 2010-05-07 Janssen Pharmaceutica Nv N-2-ADAMANTIL-2-PHENOXY-ACETAMIDE DERIVATIVES AS INHIBITORS OF 11-BETAHYDROXIESTEROID-DEHYDROGENASE.
DE602005017159D1 (en) 2004-08-30 2009-11-26 Janssen Pharmaceutica Nv OXYSTEROID DEHYDROGENASE INHIBITORS
MX2007003319A (en) 2004-09-20 2007-06-05 Xenon Pharmaceuticals Inc Pyridazine derivatives for inhibiting human stearoyl-coa- desaturase.
WO2006101521A2 (en) 2004-09-20 2006-09-28 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
AU2005286846A1 (en) 2004-09-20 2006-03-30 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as therapeutic agents
MX2007003318A (en) 2004-09-20 2007-05-18 Xenon Pharmaceuticals Inc Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes.
JP4958786B2 (en) 2004-09-20 2012-06-20 ゼノン・ファーマシューティカルズ・インコーポレイテッド Heterocyclic derivatives and their use as therapeutic agents
TW200626572A (en) 2004-09-20 2006-08-01 Xenon Pharmaceuticals Inc Heterocyclic derivatives and their use as therapeutic agents
WO2006034441A1 (en) * 2004-09-20 2006-03-30 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
WO2007130075A1 (en) 2005-06-03 2007-11-15 Xenon Pharmaceuticals Inc. Aminothiazole derivatives as human stearoyl-coa desaturase inhibitors
CN104530038A (en) * 2014-12-10 2015-04-22 沈阳药科大学 Amide imidazole derivative and application thereof
CN112142673B (en) * 2020-09-18 2023-06-30 聊城大学 Aryl alkene azole derivative and preparation method and application thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU557755A3 (en) * 1968-08-19 1977-05-05 Янссен Фармасьютика Н.В. (Фирма) Method for preparing imidazole derivatives
CA1189857A (en) * 1981-03-27 1985-07-02 Janssen Pharmaceutica Naamloze Vennootschap Antimicrobial triazole derivatives
AU8314482A (en) * 1981-05-19 1982-11-25 Imperial Chemical Industries Plc 3-triazolyl(imidazolyl)-2,2 bis phenyl-propionamides
EP0117462A3 (en) * 1983-02-28 1986-08-20 American Cyanamid Company N-(2-4-(1h-imidazol-1-yl)alkyl)arylamides

Also Published As

Publication number Publication date
PL246600A1 (en) 1985-03-12
IL71203A0 (en) 1984-06-29
NL8400730A (en) 1984-10-01
CA1242723A (en) 1988-10-04
FI840968A0 (en) 1984-03-09
ZA841782B (en) 1985-10-30
LU85245A1 (en) 1984-11-14
GR81869B (en) 1984-12-12
ES8506639A1 (en) 1985-07-16
IT1199085B (en) 1988-12-30
JPS59175472A (en) 1984-10-04
PL146072B1 (en) 1988-12-31
FI840968A (en) 1984-09-12
KR890000377B1 (en) 1989-03-15
GB2136801B (en) 1987-03-04
GB2136801A (en) 1984-09-26
DE3408127A1 (en) 1984-09-13
NZ207453A (en) 1987-09-30
AU571494B2 (en) 1988-04-21
DK149784D0 (en) 1984-02-29
FR2542315A1 (en) 1984-09-14
PT78226B (en) 1986-07-15
AU2547584A (en) 1984-09-13
ES530461A0 (en) 1985-07-16
DK149784A (en) 1984-09-12
GB8405900D0 (en) 1984-04-11
HUT36098A (en) 1985-08-28
SE8401321L (en) 1984-09-12
FR2542315B1 (en) 1986-02-07
PH24667A (en) 1990-09-07
PT78226A (en) 1984-04-01
CH655103A5 (en) 1986-03-27
IT8447817A0 (en) 1984-03-08
IL71203A (en) 1988-10-31
BE899073A (en) 1984-09-05
KR850006386A (en) 1985-10-05

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