SE7700705L - 1-legre-alkyl-4,5-dihydro-5-fenyl-2-legre-alkoxikarbonylaminoimidazoler och substituerade fenylderivat derav samt sett att framstella dessa foreningar - Google Patents

1-legre-alkyl-4,5-dihydro-5-fenyl-2-legre-alkoxikarbonylaminoimidazoler och substituerade fenylderivat derav samt sett att framstella dessa foreningar

Info

Publication number
SE7700705L
SE7700705L SE7700705A SE7700705A SE7700705L SE 7700705 L SE7700705 L SE 7700705L SE 7700705 A SE7700705 A SE 7700705A SE 7700705 A SE7700705 A SE 7700705A SE 7700705 L SE7700705 L SE 7700705L
Authority
SE
Sweden
Prior art keywords
legre
phenyl
alcoxicarbonylaminoimidazoles
dihydro
alkyl
Prior art date
Application number
SE7700705A
Other languages
English (en)
Inventor
A P Roszkowski
C C Beard
C Dvorak
K Weinhardt
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of SE7700705L publication Critical patent/SE7700705L/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44Nitrogen atoms not forming part of a nitro radical
    • C07D233/46Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms attached to said nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44Nitrogen atoms not forming part of a nitro radical
    • C07D233/48Nitrogen atoms not forming part of a nitro radical with acyclic hydrocarbon or substituted acyclic hydrocarbon radicals, attached to said nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SE7700705A 1976-07-26 1977-01-24 1-legre-alkyl-4,5-dihydro-5-fenyl-2-legre-alkoxikarbonylaminoimidazoler och substituerade fenylderivat derav samt sett att framstella dessa foreningar SE7700705L (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/708,651 US4088771A (en) 1976-07-26 1976-07-26 1-Lower alkyl-4,5-dihydro-5-phenyl-2-lower alkoxy carbonylaminoimidazoles and substituted phenyl derivatives thereof

Publications (1)

Publication Number Publication Date
SE7700705L true SE7700705L (sv) 1978-01-27

Family

ID=24846651

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7700705A SE7700705L (sv) 1976-07-26 1977-01-24 1-legre-alkyl-4,5-dihydro-5-fenyl-2-legre-alkoxikarbonylaminoimidazoler och substituerade fenylderivat derav samt sett att framstella dessa foreningar

Country Status (14)

Country Link
US (1) US4088771A (sv)
JP (1) JPS5315376A (sv)
AU (1) AU2734977A (sv)
BE (1) BE857112R (sv)
DE (1) DE2733698A1 (sv)
DK (1) DK21177A (sv)
ES (2) ES461036A2 (sv)
FI (1) FI770159A (sv)
FR (1) FR2359828A1 (sv)
GB (1) GB1569386A (sv)
NL (1) NL7708084A (sv)
NZ (1) NZ184714A (sv)
SE (1) SE7700705L (sv)
ZA (1) ZA774527B (sv)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4172204A (en) * 1977-10-07 1979-10-23 Syntex (U.S.A.) Inc. Method for preparing 4,5-dihydro-2-alkoxycarbonylamino-5-carbocyclic aryl imidazoles and intermediates thereof
US4198422A (en) * 1979-05-17 1980-04-15 E. R. Squibb & Sons, Inc. Substituted 2,3-naphthimidazole carbamates and method
US4294844A (en) * 1979-06-04 1981-10-13 Syntex (U.S.A.) Inc. Use of 4,5-dihydro-2-lower alkoxycarbonylamino-4-phenyl imidazoles and substituted phenyl derivatives thereof as anti-hypertensive agents
YU204680A (en) * 1979-08-31 1983-10-31 Syntex Inc Process for obtaining 4-phenyl-and 5-phenyl-1,4,5,6-tetrahydro pyrimidine derivatives
US4322421A (en) * 1979-08-31 1982-03-30 Syntex (U.S.A.) Inc. 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydro-pyrimidine derivatives
US4261995A (en) * 1979-08-31 1981-04-14 Syntex (U.S.A.) Inc. 4-Phenyl-and 5-phenyl-1,4,5,6-tetrahydropyrimidine derivatives

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4080335A (en) * 1975-07-28 1978-03-21 Beecham Group Limited Anorexic chromans

Also Published As

Publication number Publication date
US4088771A (en) 1978-05-09
NZ184714A (en) 1979-10-25
DK21177A (da) 1978-01-27
NL7708084A (nl) 1978-01-30
ES463139A2 (es) 1978-10-16
BE857112R (fr) 1978-01-25
FR2359828B1 (sv) 1979-07-20
ZA774527B (en) 1979-02-28
AU2734977A (en) 1979-02-01
FI770159A (sv) 1978-01-27
GB1569386A (en) 1980-06-11
ES461036A2 (es) 1978-06-01
FR2359828A1 (fr) 1978-02-24
DE2733698A1 (de) 1978-02-02
JPS5315376A (en) 1978-02-13

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