RU2017115188A3 - - Google Patents

Download PDF

Info

Publication number
RU2017115188A3
RU2017115188A3 RU2017115188A RU2017115188A RU2017115188A3 RU 2017115188 A3 RU2017115188 A3 RU 2017115188A3 RU 2017115188 A RU2017115188 A RU 2017115188A RU 2017115188 A RU2017115188 A RU 2017115188A RU 2017115188 A3 RU2017115188 A3 RU 2017115188A3
Authority
RU
Russia
Application number
RU2017115188A
Other languages
Russian (ru)
Other versions
RU2017115188A (ru
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of RU2017115188A publication Critical patent/RU2017115188A/ru
Publication of RU2017115188A3 publication Critical patent/RU2017115188A3/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
RU2017115188A 2014-10-01 2015-10-01 Производные бороновой кислоты RU2017115188A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14003392 2014-10-01
EP14003392.9 2014-10-01
PCT/EP2015/002008 WO2016050359A1 (en) 2014-10-01 2015-10-01 Boronic acid derivatives

Publications (2)

Publication Number Publication Date
RU2017115188A RU2017115188A (ru) 2018-11-06
RU2017115188A3 true RU2017115188A3 (cg-RX-API-DMAC7.html) 2019-03-29

Family

ID=51690789

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2017115188A RU2017115188A (ru) 2014-10-01 2015-10-01 Производные бороновой кислоты

Country Status (14)

Country Link
US (1) US10294246B2 (cg-RX-API-DMAC7.html)
EP (1) EP3201207B1 (cg-RX-API-DMAC7.html)
JP (1) JP6835711B2 (cg-RX-API-DMAC7.html)
KR (1) KR102450583B1 (cg-RX-API-DMAC7.html)
CN (1) CN107001390B (cg-RX-API-DMAC7.html)
AU (1) AU2015327346B2 (cg-RX-API-DMAC7.html)
BR (1) BR112017006420A2 (cg-RX-API-DMAC7.html)
CA (1) CA2963205A1 (cg-RX-API-DMAC7.html)
ES (1) ES2873000T3 (cg-RX-API-DMAC7.html)
IL (1) IL251301B (cg-RX-API-DMAC7.html)
MX (1) MX370336B (cg-RX-API-DMAC7.html)
RU (1) RU2017115188A (cg-RX-API-DMAC7.html)
SG (1) SG11201702623TA (cg-RX-API-DMAC7.html)
WO (1) WO2016050359A1 (cg-RX-API-DMAC7.html)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2717558C2 (ru) 2014-10-01 2020-03-24 Мерк Патент Гмбх Производные бороновой кислоты
KR20170062518A (ko) 2014-10-01 2017-06-07 메르크 파텐트 게엠베하 보론산 유도체
RU2017115193A (ru) 2014-10-01 2018-11-06 Мерк Патент Гмбх Производные бороновой кислоты
DK3672977T3 (da) 2017-08-24 2022-09-26 Merck Patent Gmbh Boronsyrederivater
BR112021001359A2 (pt) * 2018-07-26 2021-04-20 Merck Patent Gmbh derivados de ácido borônico
CN113135944A (zh) * 2020-01-19 2021-07-20 首药控股(北京)有限公司 硼酸衍生物
CN113135943A (zh) * 2020-01-19 2021-07-20 首药控股(北京)有限公司 硼酸衍生物
US20250340577A1 (en) * 2021-03-02 2025-11-06 Case Western Reserve University Beta-lactomase inhibitors and uses thereof
CA3217594A1 (en) * 2021-05-19 2022-11-24 William Guy Whittingham Weed control method
JP2024529468A (ja) 2021-07-29 2024-08-06 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規の[(1r)-2-(1-ベンゾフラン-3-イル)-1-{[(1s,2r,4r)-7-オキサビシクロ[2.2.1]ヘプタン-2-イル]ホルムアミド}エチル]ボロン酸の結晶性形態、その付加物、および得るためのプロセス
JP7734276B2 (ja) * 2021-10-14 2025-09-04 ショウヤオ ホールディングス(ベイジン) カンパニー, リミテッド ボロン酸誘導体
WO2023232830A1 (en) 2022-06-02 2023-12-07 Merck Patent Gmbh Boronic acid adducts

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL111175A0 (en) * 1993-10-07 1994-12-29 Du Pont Merck Pharma Electrophilic peptide analogs as inhibitors of trypsin-like serine proteases and pharmaceutical compositions containing them
CA2376965A1 (en) * 1999-07-07 2001-01-11 Timothy Patrick Forsyth Peptide boronic acid inhibitors of hepatitis c virus protease
US7271186B1 (en) * 2002-12-09 2007-09-18 Northwestern University Nanomolar β-lactamase inhibitors
MX2010005252A (es) * 2007-11-13 2011-04-11 Novartis Int Pharm Ltd Inhibidores de beta-lactamasa.
AR075090A1 (es) * 2008-09-29 2011-03-09 Millennium Pharm Inc Derivados de acido 1-amino-2-ciclobutiletilboronico inhibidores de proteosoma,utiles como agentes anticancerigenos, y composiciones farmaceuticas que los comprenden.
JP6129203B2 (ja) * 2011-12-22 2017-05-17 アレス トレーディング ソシエテ アノニム α−アミノボロン酸誘導体、選択性免疫プロテアソーム阻害剤
RU2717558C2 (ru) 2014-10-01 2020-03-24 Мерк Патент Гмбх Производные бороновой кислоты
KR20170062518A (ko) 2014-10-01 2017-06-07 메르크 파텐트 게엠베하 보론산 유도체
RU2017115193A (ru) 2014-10-01 2018-11-06 Мерк Патент Гмбх Производные бороновой кислоты

Also Published As

Publication number Publication date
MX2017004046A (es) 2017-06-19
KR20170062517A (ko) 2017-06-07
IL251301B (en) 2022-02-01
CN107001390A (zh) 2017-08-01
AU2015327346B2 (en) 2019-12-05
JP2017536335A (ja) 2017-12-07
MX370336B (es) 2019-12-10
US10294246B2 (en) 2019-05-21
IL251301A0 (en) 2017-05-29
CN107001390B (zh) 2020-11-27
RU2017115188A (ru) 2018-11-06
SG11201702623TA (en) 2017-04-27
EP3201207A1 (en) 2017-08-09
EP3201207B1 (en) 2021-02-24
AU2015327346A1 (en) 2017-05-18
US20180105539A1 (en) 2018-04-19
ES2873000T3 (es) 2021-11-03
JP6835711B2 (ja) 2021-02-24
BR112017006420A2 (pt) 2017-12-19
KR102450583B1 (ko) 2022-10-04
WO2016050359A1 (en) 2016-04-07
CA2963205A1 (en) 2016-04-07

Similar Documents

Publication Publication Date Title
BR112016017659A2 (cg-RX-API-DMAC7.html)
BR112016018076A2 (cg-RX-API-DMAC7.html)
BR112016018374A2 (cg-RX-API-DMAC7.html)
BR112016019234A2 (cg-RX-API-DMAC7.html)
BR112016019490A2 (cg-RX-API-DMAC7.html)
BR112016016432A2 (cg-RX-API-DMAC7.html)
BR112016015813A2 (cg-RX-API-DMAC7.html)
BR112016016705A2 (cg-RX-API-DMAC7.html)
BR112016017278A2 (cg-RX-API-DMAC7.html)
BR112016016602A2 (cg-RX-API-DMAC7.html)
BR112016015971A2 (cg-RX-API-DMAC7.html)
BR112016017767A2 (cg-RX-API-DMAC7.html)
BR112016017265A2 (cg-RX-API-DMAC7.html)
BR112016015311A2 (cg-RX-API-DMAC7.html)
BR112016018384A2 (cg-RX-API-DMAC7.html)
BR112016019276A2 (cg-RX-API-DMAC7.html)
BR112016016770A2 (cg-RX-API-DMAC7.html)
BR112016016451A2 (cg-RX-API-DMAC7.html)
BR112016015385A2 (cg-RX-API-DMAC7.html)
BR112016018865A2 (cg-RX-API-DMAC7.html)
BR112016017226A2 (cg-RX-API-DMAC7.html)
BR112016019248A2 (cg-RX-API-DMAC7.html)
BR112016016823A2 (cg-RX-API-DMAC7.html)
BR112016014434A2 (cg-RX-API-DMAC7.html)
BR112016000228A2 (cg-RX-API-DMAC7.html)

Legal Events

Date Code Title Description
FA92 Acknowledgement of application withdrawn (lack of supplementary materials submitted)

Effective date: 20190919