RU2010142826A - HEPATIC ACTION MEANS AND METHOD FOR PRODUCING IT - Google Patents
HEPATIC ACTION MEANS AND METHOD FOR PRODUCING IT Download PDFInfo
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- RU2010142826A RU2010142826A RU2010142826/15A RU2010142826A RU2010142826A RU 2010142826 A RU2010142826 A RU 2010142826A RU 2010142826/15 A RU2010142826/15 A RU 2010142826/15A RU 2010142826 A RU2010142826 A RU 2010142826A RU 2010142826 A RU2010142826 A RU 2010142826A
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- RU
- Russia
- Prior art keywords
- surfactant
- maksar
- cremophor
- melt
- hepatoprotective
- Prior art date
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- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
1. Средство, обладающее гепатозащитным действием, на основе экстракта растительных полифенолов из ядровой древесины маакии амурской (Максар), отличающееся тем, что оно представляет собой водный раствор Максара в молекулярно-капсулированной форме в виде водорастворимого ассоциата. ! 2. Способ получения средства, обладающего гепатозащитным действием, на основе Максара, отличающийся тем, что процесс осуществляют путем гомогенизации Максара в расплаве поверхностно-активного вещества, имеющего гидрофильно-липофильный баланс в диапазоне 12-18, при соотношении поверхностно-активного вещества к Максару 4-5:1 в диапазоне температур 40-60°С с образованием молекулярно капсулированной формы целевого продукта. ! 3. Способ по п.2, отличающийся тем, что в расплав поверхностно-активного вещества дополнительно вводят структурно-дифильную добавку - аскорбилпальмитат, стабилизирующий Максар после перевода ассоциата в водную фазу. ! 4. Способ по п.2, отличающийся тем, что в качестве поверхностно-активного вещества используют Cremophor РН 40. ! 5. Способ по п.2, отличающийся тем, что в качестве поверхностно-активного вещества используют Cremophor EL. ! 6. Способ по п.2, отличающийся тем, что в качестве поверхностно-активного вещества используют Cremophor А25. ! 7. Способ по п.2, отличающийся тем, что в качестве поверхностно-активного вещества используют Cremophor® А6. ! 8. Способ по п.2, отличающийся тем, что в качестве поверхностно-активного вещества используют Soluplus. ! 9. Способ по п.2, отличающийся тем, что в качестве поверхностно-активного вещества используют Твин-80. ! 10. Способ получения средства, обладающего гепатозащитным действием, на основе Максара по п.2, отли 1. An agent with a hepatoprotective effect based on an extract of plant polyphenols from the kernel wood of maakia Amur (Maksar), characterized in that it is an aqueous solution of Maksar in molecular capsule form in the form of a water-soluble associate. ! 2. A method of producing a hepatoprotective agent based on Maksar, characterized in that the process is carried out by homogenizing Maksar in a melt of a surfactant having a hydrophilic-lipophilic balance in the range of 12-18, with a ratio of surfactant to Maksar 4 -5: 1 in the temperature range 40-60 ° C with the formation of a molecularly encapsulated form of the target product. ! 3. The method according to claim 2, characterized in that the structurally diphilic additive, ascorbyl palmitate stabilizing Maksar, is additionally added to the surfactant melt after the associate is transferred to the aqueous phase. ! 4. The method according to claim 2, characterized in that as a surfactant using Cremophor PH 40.! 5. The method according to claim 2, characterized in that as a surfactant using Cremophor EL. ! 6. The method according to claim 2, characterized in that as a surfactant using Cremophor A25. ! 7. The method according to claim 2, characterized in that as the surfactant use Cremophor® A6. ! 8. The method according to claim 2, characterized in that Soluplus is used as a surfactant. ! 9. The method according to claim 2, characterized in that Tween-80 is used as a surfactant. ! 10. The method of obtaining funds with hepatoprotective action, based on Maksar according to claim 2,
Claims (10)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
RU2010142826/15A RU2462259C2 (en) | 2010-10-20 | 2010-10-20 | Agent showing hepatoprotective action, and method for preparing it |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
RU2010142826/15A RU2462259C2 (en) | 2010-10-20 | 2010-10-20 | Agent showing hepatoprotective action, and method for preparing it |
Publications (2)
Publication Number | Publication Date |
---|---|
RU2010142826A true RU2010142826A (en) | 2012-04-27 |
RU2462259C2 RU2462259C2 (en) | 2012-09-27 |
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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RU2010142826/15A RU2462259C2 (en) | 2010-10-20 | 2010-10-20 | Agent showing hepatoprotective action, and method for preparing it |
Country Status (1)
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RU (1) | RU2462259C2 (en) |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2104027C1 (en) * | 1996-09-04 | 1998-02-10 | Тихоокеанский институт биоорганической химии ДВО РАН | Method of preparing vegetable polyphenols showing hepatoprotective effect |
RU2175237C2 (en) * | 1998-06-02 | 2001-10-27 | Гайсаев Руфат Омарович | Method of treating chronic hepatitis |
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2010
- 2010-10-20 RU RU2010142826/15A patent/RU2462259C2/en active
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RU2462259C2 (en) | 2012-09-27 |
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