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Application filed by Institutul De Cercetari Chimico-FarmaceuticefiledCriticalInstitutul De Cercetari Chimico-Farmaceutice
Priority to RO131494ApriorityCriticalpatent/RO99883B1/ro
Publication of RO99883B1publicationCriticalpatent/RO99883B1/ro
Organic Low-Molecular-Weight Compounds And Preparation Thereof
(AREA)
Abstract
Procedeul, conform inventiei, se refera la sinteza 3-(orto-aliloxifenoxi)-1-izopropilamino-propan-2-olului (Oxprenolul baza), intermediar în sinteza medicamentului Oxprenolol clorhidrat, prin deschiderea ciclului epoxidic cu exces mic de izopropilamina în metanol la 60 degree C.
RO131494A1987-12-301987-12-30Procedeu de obtinere a 3-(o-aliloxifenoxi)-1-izopropilamino-propan-2-olului
RO99883B1
(ro)
S-N-éthyl-3-[(1-diméthyl-amino)éthyl]-N-méthyl-phénylcarbamate ou un sel pharmaceutiquement acceptable de celui-ci en particulier le tartrate hydrogène
Procedimiento para la preparacion de trihidrato del (2r,3s)-3-terc-butoxicarbonilamino-2-hidroxi-3-fenilpropionato de 4-acetoxi-2alfa-benzoiloxi-5beta,20-epoxi-1,7beta,10beta-trihidroxi-9-oxo-tax-11-en-13alfa-ilo.
Substituted 1,2,3,4-tetrahydrocyclopent(b)indoles, 1,2,3,3a,4,8a-hexahydrocyclopent(b)indoles and related compounds, intermediates and a process for the preparation thereof and their use as medicaments