PT91895A - PROCESS FOR THE PREPARATION OF REPLACED 9H-PURINS - Google Patents
PROCESS FOR THE PREPARATION OF REPLACED 9H-PURINSInfo
- Publication number
- PT91895A PT91895A PT91895A PT9189589A PT91895A PT 91895 A PT91895 A PT 91895A PT 91895 A PT91895 A PT 91895A PT 9189589 A PT9189589 A PT 9189589A PT 91895 A PT91895 A PT 91895A
- Authority
- PT
- Portugal
- Prior art keywords
- purins
- replaced
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH373188 | 1988-10-06 |
Publications (2)
Publication Number | Publication Date |
---|---|
PT91895A true PT91895A (en) | 1990-04-30 |
PT91895B PT91895B (en) | 1995-05-31 |
Family
ID=4262288
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT91895A PT91895B (en) | 1988-10-06 | 1989-10-04 | PROCESS FOR THE PREPARATION OF REPLACED 9H-PURINS |
Country Status (17)
Country | Link |
---|---|
US (1) | US5110818A (en) |
EP (1) | EP0363320A3 (en) |
JP (1) | JPH02157279A (en) |
KR (1) | KR900006337A (en) |
AU (1) | AU632763B2 (en) |
CA (1) | CA2000154A1 (en) |
DD (1) | DD297820A5 (en) |
DK (1) | DK491389A (en) |
FI (1) | FI894707A (en) |
HU (1) | HUT52502A (en) |
IL (1) | IL91818A (en) |
MX (1) | MX17846A (en) |
NO (1) | NO172986C (en) |
NZ (1) | NZ230898A (en) |
PH (1) | PH27154A (en) |
PT (1) | PT91895B (en) |
ZA (1) | ZA897587B (en) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5391739A (en) * | 1989-03-29 | 1995-02-21 | Merrell Dow Pharmaceuticals Inc. | Selective adenosine receptor agents |
US5387684A (en) * | 1992-03-25 | 1995-02-07 | The Green Cross Corporation | Isoindazole compound |
FR2699176B1 (en) * | 1992-12-11 | 1995-03-03 | Adir | New bicyclic pyrimidine compounds, process for their preparation and pharmaceutical compositions containing them. |
GB9312853D0 (en) * | 1993-06-22 | 1993-08-04 | Euro Celtique Sa | Chemical compounds |
US5994361A (en) * | 1994-06-22 | 1999-11-30 | Biochem Pharma | Substituted purinyl derivatives with immunomodulating activity |
US5922751A (en) * | 1994-06-24 | 1999-07-13 | Euro-Celtique, S.A. | Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same |
US5591776A (en) * | 1994-06-24 | 1997-01-07 | Euro-Celtique, S.A. | Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV |
DE19535504A1 (en) * | 1995-09-25 | 1997-03-27 | Bayer Ag | Substituted xanthines |
US6166041A (en) * | 1995-10-11 | 2000-12-26 | Euro-Celtique, S.A. | 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma |
FR2741881B1 (en) * | 1995-12-01 | 1999-07-30 | Centre Nat Rech Scient | NOVEL PURINE DERIVATIVES HAVING IN PARTICULAR ANTI-PROLIFERATIVE PRORIETES AND THEIR BIOLOGICAL APPLICATIONS |
US6075016A (en) * | 1996-04-10 | 2000-06-13 | Euro-Celtique S.A. | 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity |
US5864037A (en) | 1996-06-06 | 1999-01-26 | Euro-Celtique, S.A. | Methods for the synthesis of chemical compounds having PDE-IV inhibitory activity |
US6294541B1 (en) | 1996-06-06 | 2001-09-25 | Euro-Celtique S.A. | Purine derivatives having phosphodiesterase IV inhibition activity |
CN1294590A (en) | 1997-12-12 | 2001-05-09 | 欧罗赛铁克股份有限公司 | Method of 3-substituted adenines via 2-thioxanthines |
US6319928B1 (en) | 1998-11-30 | 2001-11-20 | Euro-Celtique, S.A. | Purine derivatives having phosphodiesterase IV inhibition activity |
AR029347A1 (en) | 1999-04-02 | 2003-06-25 | Euro Celtique Sa | ADENINE COMPOUND, ISOGNANINE COMPOUND AND 2,6-DITIOXANTINE AS A PRECURSOR OF THE SAME, USE OF SUCH COMPOUNDS TO PREPARE A PHARMACEUTICAL COMPOSITION AND SUCH PHARMACEUTICAL COMPOSITION |
US7439359B2 (en) * | 2000-11-02 | 2008-10-21 | Sloan-Kettering Institute For Cancer Research | Small molecule compositions for binding to hsp90 |
EP1440072A4 (en) * | 2001-10-30 | 2005-02-02 | Conforma Therapeutic Corp | Purine analogs having hsp90-inhibiting activity |
US20070129334A1 (en) * | 2001-10-30 | 2007-06-07 | Conforma Therapeutics Corporation | Orally Active Purine-Based Inhibitors of Heat Shock Protein 90 |
JP2007505933A (en) | 2003-09-18 | 2007-03-15 | コンフォーマ・セラピューティクス・コーポレイション | Novel heterocyclic compounds as HSP90 inhibitors |
JP2008534609A (en) * | 2005-03-30 | 2008-08-28 | コンフォーマ・セラピューティクス・コーポレイション | Alkynylpyrrolopyrimidines and related analogs as HSP90 inhibitors |
EP1937258A2 (en) * | 2005-09-23 | 2008-07-02 | Conforma Therapeutics Corporation | Anti-tumor methods using multi drug resistance independent synthetic hsp90 inhibitors |
WO2009034386A1 (en) * | 2007-09-13 | 2009-03-19 | Astrazeneca Ab | Derivatives of adenine and 8-aza-adenine and uses thereof-796 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3846426A (en) * | 1971-03-03 | 1974-11-05 | Int Minerals & Chem Corp | 6-amino-9-(substituted benzyl) purines and their n{11 oxides |
GB1534163A (en) * | 1976-07-28 | 1978-11-29 | Merck & Co Inc | Adenine derivatives |
USRE31429E (en) * | 1977-02-14 | 1983-10-25 | Merck & Co., Inc. | Process for preparation of 9-(dihalobenzyl)adenines |
GB1547214A (en) * | 1977-08-09 | 1979-06-06 | Merck & Co Inc | Purine derivatives |
US4189485A (en) * | 1977-08-23 | 1980-02-19 | Takeda Chemical Industries, Ltd. | Purine derivatives |
US4361699A (en) * | 1981-09-28 | 1982-11-30 | Merck & Co., Inc. | Novel process for the preparation of N6 -alkyl-arprinocid |
ZW22283A1 (en) * | 1982-10-14 | 1985-05-22 | Wellcome Found | Antiviral compounds |
US4748177A (en) * | 1984-03-26 | 1988-05-31 | Warner-Lambert Company | Guanine derivatives |
GB8408615D0 (en) * | 1984-04-04 | 1984-05-16 | Wellcome Found | Heterocyclic compounds |
AU626983B2 (en) * | 1989-01-31 | 1992-08-13 | Whitby Research, Inc. | N6-substituted 9-methyladenines |
-
1989
- 1989-09-26 EP EP19890810731 patent/EP0363320A3/en not_active Withdrawn
- 1989-09-28 IL IL9181889A patent/IL91818A/en not_active IP Right Cessation
- 1989-10-04 DD DD89333303A patent/DD297820A5/en not_active IP Right Cessation
- 1989-10-04 CA CA002000154A patent/CA2000154A1/en not_active Abandoned
- 1989-10-04 NZ NZ230898A patent/NZ230898A/en unknown
- 1989-10-04 PT PT91895A patent/PT91895B/en not_active IP Right Cessation
- 1989-10-04 PH PH39332A patent/PH27154A/en unknown
- 1989-10-04 FI FI894707A patent/FI894707A/en not_active IP Right Cessation
- 1989-10-05 NO NO893965A patent/NO172986C/en unknown
- 1989-10-05 JP JP1258944A patent/JPH02157279A/en active Pending
- 1989-10-05 AU AU42612/89A patent/AU632763B2/en not_active Ceased
- 1989-10-05 MX MX17846A patent/MX17846A/en unknown
- 1989-10-05 HU HU895224A patent/HUT52502A/en unknown
- 1989-10-05 DK DK491389A patent/DK491389A/en not_active Application Discontinuation
- 1989-10-05 ZA ZA897587A patent/ZA897587B/en unknown
- 1989-10-06 KR KR1019890014356A patent/KR900006337A/en not_active Application Discontinuation
-
1990
- 1990-12-19 US US07/630,401 patent/US5110818A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP0363320A2 (en) | 1990-04-11 |
NO172986C (en) | 1993-10-06 |
KR900006337A (en) | 1990-05-07 |
HUT52502A (en) | 1990-07-28 |
NO893965D0 (en) | 1989-10-05 |
AU632763B2 (en) | 1993-01-14 |
AU4261289A (en) | 1990-04-12 |
DK491389D0 (en) | 1989-10-05 |
CA2000154A1 (en) | 1990-04-06 |
MX17846A (en) | 1994-03-31 |
JPH02157279A (en) | 1990-06-18 |
NO893965L (en) | 1990-04-09 |
US5110818A (en) | 1992-05-05 |
NZ230898A (en) | 1992-12-23 |
FI894707A (en) | 1990-04-07 |
IL91818A0 (en) | 1990-06-10 |
DD297820A5 (en) | 1992-01-23 |
EP0363320A3 (en) | 1991-11-21 |
NO172986B (en) | 1993-06-28 |
PT91895B (en) | 1995-05-31 |
ZA897587B (en) | 1990-05-30 |
DK491389A (en) | 1990-04-07 |
PH27154A (en) | 1993-04-02 |
IL91818A (en) | 1994-08-26 |
FI894707A0 (en) | 1989-10-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG3A | Patent granted, date of granting |
Effective date: 19941121 |
|
MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19960531 |