PT88699A - Processo para a preparacao de composicoes farmaceuticas diminuidoras da pressao intraocular compreendendo combinacoes sinergeticas de fenilefrina e certos derivados de labdano - Google Patents

Processo para a preparacao de composicoes farmaceuticas diminuidoras da pressao intraocular compreendendo combinacoes sinergeticas de fenilefrina e certos derivados de labdano

Info

Publication number
PT88699A
PT88699A PT88699A PT8869988A PT88699A PT 88699 A PT88699 A PT 88699A PT 88699 A PT88699 A PT 88699A PT 8869988 A PT8869988 A PT 8869988A PT 88699 A PT88699 A PT 88699A
Authority
PT
Portugal
Prior art keywords
fenilefrine
labdano
derivatives
understanding
certain
Prior art date
Application number
PT88699A
Other languages
English (en)
Inventor
Grover Cleveland Helsley
Paul Gary Conway
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of PT88699A publication Critical patent/PT88699A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT88699A 1987-10-08 1988-10-07 Processo para a preparacao de composicoes farmaceuticas diminuidoras da pressao intraocular compreendendo combinacoes sinergeticas de fenilefrina e certos derivados de labdano PT88699A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/105,850 US4902696A (en) 1987-10-08 1987-10-08 Synergistic intraocular pressure lowering combinations

Publications (1)

Publication Number Publication Date
PT88699A true PT88699A (pt) 1989-07-31

Family

ID=22308129

Family Applications (1)

Application Number Title Priority Date Filing Date
PT88699A PT88699A (pt) 1987-10-08 1988-10-07 Processo para a preparacao de composicoes farmaceuticas diminuidoras da pressao intraocular compreendendo combinacoes sinergeticas de fenilefrina e certos derivados de labdano

Country Status (8)

Country Link
US (1) US4902696A (pt)
EP (1) EP0311032A1 (pt)
JP (1) JPH01128920A (pt)
KR (1) KR890006231A (pt)
AU (1) AU2352988A (pt)
DK (1) DK563088A (pt)
PT (1) PT88699A (pt)
ZA (1) ZA887500B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5846992A (en) * 1987-10-08 1998-12-08 Hoechst Marion Roussel, Inc. Synergistic intraocular pressure lowering combinations
FR2650953B1 (fr) * 1989-08-17 1991-12-06 Lvmh Rech Composition a base de phases lamellaires lipidiques hydratees ou de liposomes contenant au moins un derive de labdane, ou un extrait de plante en contenant; composition cosmetique ou pharmaceutique, notamment dermatologique l'incorporant
US5629345A (en) * 1993-07-23 1997-05-13 Vide Pharmaceuticals Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US5965620A (en) * 1993-07-23 1999-10-12 Vide Pharmaceuticals Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure
US7005446B1 (en) * 1999-04-20 2006-02-28 Alcon Manufacturing, Ltd. Use of AP-1 activators to treat glaucoma and ocular hypertension
US10507245B2 (en) * 2012-07-19 2019-12-17 Luis Felipe Vejarano Restrepo Ophthalmic formulation and method for ameliorating presbyopia

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2557784C2 (de) * 1975-12-22 1986-04-17 Hoechst Ag, 6230 Frankfurt Forskolin, Verfahren zu dessen Gewinnung und diese Verbindung enthaltende pharmazeutische Präparate
DE2640275A1 (de) * 1976-09-08 1978-03-09 Hoechst Ag Pharmakologisch wirksame substanz aus labiaten
DE2654796A1 (de) * 1976-12-03 1978-06-08 Hoechst Ag Polyoxygenierte labdan-derivate
US4476140A (en) * 1983-05-16 1984-10-09 Yale University Composition and method for treatment of glaucoma
US4490379A (en) * 1984-04-04 1984-12-25 Steven Podos Method of reducing intraocular pressure and treating glaucoma using corynanthine
US4666904A (en) * 1984-12-14 1987-05-19 Hoechst-Roussel Pharmaceuticals Inc. Aminoacyllabdanes, pharmacuetical compositions and use
ATE60767T1 (de) * 1984-12-14 1991-02-15 Hoechst Roussel Pharma Aminoacyllabdane, verfahren und zwischenprodukte zu ihrer herstellung und ihre verwendung als arzneimittel.
US4639446A (en) * 1984-12-14 1987-01-27 Hoechst-Roussel Pharmaceuticals Inc. Aminoacyllabdanes, pharmaceutical compositions and use
US4771049A (en) * 1985-03-01 1988-09-13 Hoechst-Roussel Pharmaceuticals Labdanes, pharmaceutical compositions and use
US4639443A (en) * 1985-03-01 1987-01-27 Hoechst-Roussel Pharmaceuticals Inc. Labdane compounds, pharmaceutical compositions and use
DE3678736D1 (de) * 1985-03-01 1991-05-23 Hoechst Roussel Pharma Labdanderivate, verfahren zu deren herstellung und deren verwendung als arzneimittel.
US4677103A (en) * 1985-03-01 1987-06-30 Hoechst-Roussel Pharmaceuticals Inc. Labdane compounds, pharmaceutical compositions and use
IN163242B (pt) * 1985-05-03 1988-08-27 Hoechst India
CA1307530C (en) * 1986-12-29 1992-09-15 Hoechst-Roussel Pharmaceuticals Inc. Carbamoyloxylabdanes, intermediates and a process for the preparation thereof and their use as medicaments

Also Published As

Publication number Publication date
JPH01128920A (ja) 1989-05-22
US4902696A (en) 1990-02-20
EP0311032A1 (en) 1989-04-12
KR890006231A (ko) 1989-06-12
DK563088D0 (da) 1988-10-07
AU2352988A (en) 1989-06-08
DK563088A (da) 1989-04-09
ZA887500B (en) 1989-07-26

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Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19921027