PT86903A - Heterocyclic compounds - Google Patents

Heterocyclic compounds

Info

Publication number
PT86903A
PT86903A PT86903A PT8690388A PT86903A PT 86903 A PT86903 A PT 86903A PT 86903 A PT86903 A PT 86903A PT 8690388 A PT8690388 A PT 8690388A PT 86903 A PT86903 A PT 86903A
Authority
PT
Portugal
Prior art keywords
radical
alkyl
carbamoyl
halogenoalkyl
amino
Prior art date
Application number
PT86903A
Other languages
English (en)
Other versions
PT86903B (pt
Inventor
Francis Thomas Boyle
Zbigniew Stanley Matusiak
Brian Steele Tait
Original Assignee
Ici Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Plc filed Critical Ici Plc
Publication of PT86903A publication Critical patent/PT86903A/pt
Publication of PT86903B publication Critical patent/PT86903B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Separation Using Semi-Permeable Membranes (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Air Bags (AREA)
  • Detergent Compositions (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
PT86903A 1987-03-05 1988-03-04 Processo para a preparacao de compostos heterociclicos inibidores do enzima aromatase e de composicoes farmaceuticas ou veterinarias que os contem PT86903B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB878705174A GB8705174D0 (en) 1987-03-05 1987-03-05 Heterocyclic compounds

Publications (2)

Publication Number Publication Date
PT86903A true PT86903A (pt) 1988-04-01
PT86903B PT86903B (pt) 1992-05-29

Family

ID=10613373

Family Applications (1)

Application Number Title Priority Date Filing Date
PT86903A PT86903B (pt) 1987-03-05 1988-03-04 Processo para a preparacao de compostos heterociclicos inibidores do enzima aromatase e de composicoes farmaceuticas ou veterinarias que os contem

Country Status (15)

Country Link
US (1) US4910212A (pt)
EP (1) EP0281283B1 (pt)
JP (1) JPS63238070A (pt)
AT (1) ATE85613T1 (pt)
AU (1) AU612623B2 (pt)
CA (1) CA1304741C (pt)
DE (1) DE3878268T2 (pt)
DK (1) DK112688A (pt)
FI (1) FI881018A (pt)
GB (1) GB8705174D0 (pt)
IE (1) IE62827B1 (pt)
NO (1) NO169894C (pt)
NZ (1) NZ223752A (pt)
PT (1) PT86903B (pt)
ZA (1) ZA881008B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH683151A5 (de) * 1991-04-24 1994-01-31 Ciba Geigy Ag Antikonzeption bei weiblichen Primaten ohne Beeinflussung des menstruellen Zyklus.
US5998441A (en) * 1995-02-28 1999-12-07 Eli Lilly And Company Benzothiophene compounds, intermediates, compositions, and methods
US5856340A (en) * 1995-02-28 1999-01-05 Eli Lilly And Company Method of treating estrogen dependent cancers
US5856339A (en) * 1995-02-28 1999-01-05 Eli Lilly And Company Benzothiophene compounds, intermediates, compositions, and methods
US5919800A (en) * 1995-02-28 1999-07-06 Eli Lilly And Company Benzothiophene compounds, intermediates, compositions, and methods
US5977093A (en) * 1995-02-28 1999-11-02 Eli Lilly And Company Benzothiophene compounds, intermediates, compositions, and methods
US5510357A (en) * 1995-02-28 1996-04-23 Eli Lilly And Company Benzothiophene compounds as anti-estrogenic agents
US5998401A (en) 1995-02-28 1999-12-07 Eli Lilly And Company Naphthyl compounds, intermediates, compositions, and methods
US5811421A (en) * 1995-07-31 1998-09-22 Eli Lilly And Company Naphthyl and dihydronaphthyl intermediates, compounds, compositions, and methods
ID19392A (id) * 1996-08-29 1998-07-09 Lilly Co Eli Senyawa naftil dan bahan pertengahan serta komposisi dan metode penggunaan
US5916916A (en) * 1996-10-10 1999-06-29 Eli Lilly And Company 1-aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods
US5958969A (en) * 1996-10-10 1999-09-28 Eli Lilly And Company Benzo b!thiophene compounds, intermediates, formulations, and methods
ZA982877B (en) * 1997-04-09 1999-10-04 Lilly Co Eli Treatment of central nervous system disorders with selective estrogen receptor modulators.
US5929090A (en) * 1997-09-12 1999-07-27 Eli Lilly And Company 2-aryl-3-aminoaryloxynaphthy1 compounds, intermediates, compositions and methods
AR121486A1 (es) * 2020-03-06 2022-06-08 Kureha Corp Derivado de azol, metodo para producir derivado de azol, químico agrícola u hortícola, y protector de material industrial

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3369131D1 (en) * 1982-04-22 1987-02-19 Ici Plc Antifungal azolyl phenyl substituted alicyclic alcohols
GB8311678D0 (en) * 1983-04-28 1983-06-02 Ici Plc Phenol derivatives
GB8410899D0 (en) * 1984-04-27 1984-06-06 Ici Plc Phenol derivatives
GB8410901D0 (en) * 1984-04-27 1984-06-06 Ici Plc Phenol derivatives
IE58417B1 (en) * 1984-04-27 1993-09-22 Ici Plc Chemical derivatives
US4757082A (en) * 1984-06-18 1988-07-12 Eli Lilly And Company Method of inhibiting aromatase
US4659730A (en) * 1984-06-18 1987-04-21 Eli Lilly And Company Aromatase inhibiting imidazole derivatives
US4755526A (en) * 1984-06-18 1988-07-05 Eli Lilly And Company Method of inhibiting aromatase
US4737508A (en) * 1985-02-01 1988-04-12 Schering Corporation 1-aryl-1-(1H-azol-1-ylalkyl)-1,3-dihydroisobenzofurans, related derivatives and pharmaceutical compositions thereof useful as antifungals
DE3608144A1 (de) * 1986-03-12 1987-09-24 Hoechst Ag Aryl-azolylmethyl-benzocycloalken-derivate, verfahren zu ihrer herstellung und ihre verwendung
IL91542A0 (en) * 1988-10-06 1990-04-29 Erba Carlo Spa N-imidazolyl-and n-imidazolyl-methyl derivatives of substituted bicyclic compounds,their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
JPS63238070A (ja) 1988-10-04
NO880987D0 (no) 1988-03-04
PT86903B (pt) 1992-05-29
EP0281283B1 (en) 1993-02-10
IE880377L (en) 1988-09-05
NZ223752A (en) 1991-09-25
EP0281283A1 (en) 1988-09-07
FI881018A (fi) 1988-09-06
DK112688A (da) 1988-09-06
ATE85613T1 (de) 1993-02-15
DK112688D0 (da) 1988-03-02
DE3878268T2 (de) 1993-05-27
GB8705174D0 (en) 1987-04-08
NO169894C (no) 1992-08-19
NO169894B (no) 1992-05-11
ZA881008B (en) 1988-09-05
US4910212A (en) 1990-03-20
NO880987L (no) 1988-09-06
CA1304741C (en) 1992-07-07
AU1193488A (en) 1988-09-08
AU612623B2 (en) 1991-07-18
DE3878268D1 (de) 1993-03-25
IE62827B1 (en) 1995-03-08
FI881018A0 (fi) 1988-03-04

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Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19911127

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20030531