PT83977B - Processo para a preparacao de derivados piperazinicos de teofilina e teobromina - Google Patents

Processo para a preparacao de derivados piperazinicos de teofilina e teobromina

Info

Publication number
PT83977B
PT83977B PT83977A PT8397786A PT83977B PT 83977 B PT83977 B PT 83977B PT 83977 A PT83977 A PT 83977A PT 8397786 A PT8397786 A PT 8397786A PT 83977 B PT83977 B PT 83977B
Authority
PT
Portugal
Prior art keywords
teobromine
piperazinic
theophiline
derivatives
preparation
Prior art date
Application number
PT83977A
Other languages
English (en)
Other versions
PT83977A (en
Inventor
Jean-Claude Pascal
Serge Beranger
Henri Pinhas
Original Assignee
Syntex Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Lab filed Critical Syntex Lab
Publication of PT83977A publication Critical patent/PT83977A/pt
Publication of PT83977B publication Critical patent/PT83977B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/08Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/10Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 3 and 7, e.g. theobromine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT83977A 1985-12-20 1986-12-19 Processo para a preparacao de derivados piperazinicos de teofilina e teobromina PT83977B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/811,568 US4810706A (en) 1985-12-20 1985-12-20 Piperazine derivatives of theophylline and theobromine

Publications (2)

Publication Number Publication Date
PT83977A PT83977A (en) 1987-01-01
PT83977B true PT83977B (pt) 1989-01-17

Family

ID=25206910

Family Applications (1)

Application Number Title Priority Date Filing Date
PT83977A PT83977B (pt) 1985-12-20 1986-12-19 Processo para a preparacao de derivados piperazinicos de teofilina e teobromina

Country Status (14)

Country Link
US (1) US4810706A (pt)
EP (1) EP0227077A1 (pt)
JP (1) JPS62289580A (pt)
KR (1) KR870006050A (pt)
AU (1) AU589724B2 (pt)
CA (1) CA1274517A (pt)
DK (1) DK620586A (pt)
FI (1) FI865225A (pt)
HU (1) HU197902B (pt)
NO (1) NO865177L (pt)
NZ (1) NZ218716A (pt)
PH (1) PH23910A (pt)
PT (1) PT83977B (pt)
ZA (1) ZA869584B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117582353B (zh) * 2023-12-21 2024-05-03 湖北工业大学 一种主动引导宠物的雾化吸氧一体机

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55118488A (en) * 1979-03-05 1980-09-11 Eisai Co Ltd Theobromine derivative and its preparation
JPS5677278A (en) * 1979-09-11 1981-06-25 Maruko Seiyaku Kk Theobromine derivative
US4374835A (en) * 1980-01-31 1983-02-22 Laroche-Navarron, S.A. Piperazine derivatives of theophylline
CH648559A5 (de) * 1981-07-20 1985-03-29 Siegfried Ag Theophyllinderivate und verfahren zu deren herstellung.
US4374837A (en) * 1981-07-31 1983-02-22 Laroche Navarron, S.A. Piperazine derivatives of theobromine
US4400381A (en) * 1981-07-31 1983-08-23 Laroche-Navarron, S.A. Piperazine derivatives of theophylline
FR2531085A1 (fr) * 1982-07-28 1984-02-03 Adir Nouveaux derives de la xanthine, leur procede de preparation et les compositions pharmaceutiques les renfermant

Also Published As

Publication number Publication date
CA1274517A (en) 1990-09-25
HU197902B (en) 1989-06-28
US4810706A (en) 1989-03-07
HUT44031A (en) 1988-01-28
ZA869584B (en) 1988-07-27
FI865225A0 (fi) 1986-12-19
FI865225A (fi) 1987-06-21
PT83977A (en) 1987-01-01
DK620586D0 (da) 1986-12-19
NO865177D0 (no) 1986-12-19
AU589724B2 (en) 1989-10-19
KR870006050A (ko) 1987-07-08
JPS62289580A (ja) 1987-12-16
EP0227077A1 (en) 1987-07-01
AU6676486A (en) 1987-06-25
PH23910A (en) 1990-01-23
DK620586A (da) 1987-06-21
NO865177L (no) 1987-06-22
NZ218716A (en) 1990-01-29

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Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19911223