PT83048B - Processo de preparacao de derivados da beta-lactama e de seus intermediarios - Google Patents

Processo de preparacao de derivados da beta-lactama e de seus intermediarios

Info

Publication number
PT83048B
PT83048B PT83048A PT8304886A PT83048B PT 83048 B PT83048 B PT 83048B PT 83048 A PT83048 A PT 83048A PT 8304886 A PT8304886 A PT 8304886A PT 83048 B PT83048 B PT 83048B
Authority
PT
Portugal
Prior art keywords
lactama
intermediaries
beta
derivatives
preparation
Prior art date
Application number
PT83048A
Other languages
English (en)
Other versions
PT83048A (en
Original Assignee
Beecham Group Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB858518869A external-priority patent/GB8518869D0/en
Priority claimed from GB868610910A external-priority patent/GB8610910D0/en
Application filed by Beecham Group Plc filed Critical Beecham Group Plc
Publication of PT83048A publication Critical patent/PT83048A/pt
Publication of PT83048B publication Critical patent/PT83048B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT83048A 1985-07-25 1986-07-23 Processo de preparacao de derivados da beta-lactama e de seus intermediarios PT83048B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB858518869A GB8518869D0 (en) 1985-07-25 1985-07-25 Compounds
GB868610910A GB8610910D0 (en) 1986-05-03 1986-05-03 Compounds

Publications (2)

Publication Number Publication Date
PT83048A PT83048A (en) 1986-08-01
PT83048B true PT83048B (pt) 1988-10-14

Family

ID=26289559

Family Applications (1)

Application Number Title Priority Date Filing Date
PT83048A PT83048B (pt) 1985-07-25 1986-07-23 Processo de preparacao de derivados da beta-lactama e de seus intermediarios

Country Status (9)

Country Link
US (1) US4816452A (pt)
EP (1) EP0210815A3 (pt)
AU (1) AU598199B2 (pt)
CA (1) CA1283097C (pt)
DK (1) DK353286A (pt)
ES (1) ES2001031A6 (pt)
GR (1) GR861966B (pt)
NZ (1) NZ216946A (pt)
PT (1) PT83048B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0867676A (ja) * 1994-03-30 1996-03-12 Eisai Kagaku Kk 保護アミノチアゾリル酢酸誘導体
HUP9601096A2 (hu) * 1996-04-26 1998-01-28 János Aradi Anti-HIV-aktivitással rendelkező gyógynövényalapú gyógyászati és gyógyhatású készítmény,és vegyületek
IT1295935B1 (it) * 1997-10-30 1999-05-28 Acs Dobfar Spa Derivati aminotiazolici utili nella preparazione di antibiotici b -lattamici
US20050245498A1 (en) * 2002-05-14 2005-11-03 Shoichet Brian K Sterically-awkward beta-lactamase inhibitors
ES2422603T3 (es) * 2007-05-31 2013-09-12 Shionogi & Co Compuestos oxiimino y el uso de estos

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1399087A (en) * 1971-05-14 1975-06-25 Glaxo Lab Ltd Penicillin compounds
US3936443A (en) * 1974-05-03 1976-02-03 Glaxo Laboratories Limited Penicillin antibiotics
GB1536281A (en) * 1975-06-09 1978-12-20 Takeda Chemical Industries Ltd Cephem compounds
US4376203A (en) * 1976-01-23 1983-03-08 Roussell Uclaf Novel 3-acetoxymethyl-7-(iminoacetamido)-cephalosporanic acid derivatives
US4284631A (en) * 1978-07-31 1981-08-18 Fujisawa Pharmaceutical Co., Ltd. 7-Substituted cephem compounds and pharmaceutical antibacterial compositions containing them
DE2923339A1 (de) * 1979-06-08 1980-12-18 Bayer Ag Penicillin-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel
US4443444A (en) * 1980-08-11 1984-04-17 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
US4507487A (en) * 1982-09-23 1985-03-26 Bristol-Myers Company Chemical compounds
EP0189287B1 (en) * 1985-01-21 1992-12-16 Nippon Pharmaceutical Development Institute Company Limited Novel b-lactam antibiotics

Also Published As

Publication number Publication date
CA1283097C (en) 1991-04-16
PT83048A (en) 1986-08-01
DK353286D0 (da) 1986-07-24
AU6046686A (en) 1987-01-29
GR861966B (en) 1986-11-26
NZ216946A (en) 1990-03-27
EP0210815A2 (en) 1987-02-04
DK353286A (da) 1987-01-26
ES2001031A6 (es) 1988-04-16
AU598199B2 (en) 1990-06-21
US4816452A (en) 1989-03-28
EP0210815A3 (en) 1988-04-20

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Legal Events

Date Code Title Description
MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19920930