PT2945702T - Derivados de éter aminoalquil fenílico substituídos por hidroxi alifáticos - Google Patents

Derivados de éter aminoalquil fenílico substituídos por hidroxi alifáticos

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Publication number
PT2945702T
PT2945702T PT138115696T PT13811569T PT2945702T PT 2945702 T PT2945702 T PT 2945702T PT 138115696 T PT138115696 T PT 138115696T PT 13811569 T PT13811569 T PT 13811569T PT 2945702 T PT2945702 T PT 2945702T
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PT
Portugal
Prior art keywords
phenyl ether
ether derivatives
derivatives substituted
aliphatic hydroxy
aminoalkyl phenyl
Prior art date
Application number
PT138115696T
Other languages
English (en)
Portuguese (pt)
Inventor
R Prous Josep
Serradell Neus
Flores Ramón
García-Delgado Noemí
Carbò Banùs Marcel­Lì
Original Assignee
Prous Inst For Biomedical Res S A
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Application filed by Prous Inst For Biomedical Res S A filed Critical Prous Inst For Biomedical Res S A
Publication of PT2945702T publication Critical patent/PT2945702T/pt

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    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/18—Acyclic radicals, substituted by carbocyclic rings
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    • C07—ORGANIC CHEMISTRY
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    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

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PT138115696T 2012-12-21 2013-12-20 Derivados de éter aminoalquil fenílico substituídos por hidroxi alifáticos PT2945702T (pt)

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EP3043799A1 (en) * 2013-09-09 2016-07-20 Sanofi An h3 receptor antagonist combined with a cholinesterase inhibitor for use in the treatment of alzheimer's disease
CN106349211B (zh) * 2016-08-26 2020-10-16 江苏恩华药业股份有限公司 2-甲基-3-芳氧基-3-杂芳基丙胺类化合物及应用
KR101864085B1 (ko) * 2017-09-22 2018-06-01 동아대학교 산학협력단 발프로산 유도체, 이의 제조방법 및 이를 포함하는 항경련제
EP3697754A1 (en) * 2017-10-16 2020-08-26 Esteve Pharmaceuticals, S.A. Propanamine derivatives for treating pain and pain related conditions
WO2019208693A1 (en) 2018-04-27 2019-10-31 Shionogi & Co., Ltd. Tetrahydropyranooxazine derivatives having selective bace1 inhibitory activity
EP3838899A4 (en) 2018-08-17 2022-02-16 Shanghai Leado Pharmatech Co. Ltd. 3-aryloxyl-3-five-membered heteroaryl propylamine compound and use thereof
EP3989957A1 (en) * 2019-06-28 2022-05-04 University of Copenhagen Treatment of cns disorders with sleep disturbances
KR20250030127A (ko) * 2023-08-24 2025-03-05 경희대학교 산학협력단 피니톨을 함유한 감각 운동 관문 장애 예방 또는 치료용 조성물

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US20120004310A1 (en) * 2010-05-28 2012-01-05 Longo Frank M Non-peptide bdnf neurotrophin mimetics
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HRP20170539T1 (hr) 2017-06-16
US9624158B2 (en) 2017-04-18
ES2621960T3 (es) 2017-07-05
CA2895592A1 (en) 2014-06-26
AU2013366502A1 (en) 2015-07-09
US9980928B2 (en) 2018-05-29
EP2745876A1 (en) 2014-06-25
EP2945702A1 (en) 2015-11-25
US20150344408A1 (en) 2015-12-03
AU2013366502B2 (en) 2017-12-14
JP6302929B2 (ja) 2018-03-28
WO2014096377A1 (en) 2014-06-26
HUE032461T2 (en) 2017-09-28
EP2945702B1 (en) 2017-01-11
US20170239197A1 (en) 2017-08-24
DK2945702T3 (en) 2017-04-18

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