PT1315731E - Derivados de 2-piridinil-6,7,8,9-tetra-hidropirimido [1,2-a] pirimidin-4-ona e 7-piridinil-2,3-di-hidroimidazol [1,2-a]pirimidin-5 (1h) ona - Google Patents

Derivados de 2-piridinil-6,7,8,9-tetra-hidropirimido [1,2-a] pirimidin-4-ona e 7-piridinil-2,3-di-hidroimidazol [1,2-a]pirimidin-5 (1h) ona

Info

Publication number
PT1315731E
PT1315731E PT01980397T PT01980397T PT1315731E PT 1315731 E PT1315731 E PT 1315731E PT 01980397 T PT01980397 T PT 01980397T PT 01980397 T PT01980397 T PT 01980397T PT 1315731 E PT1315731 E PT 1315731E
Authority
PT
Portugal
Prior art keywords
group
ring
optionally substituted
alkyl group
naphthyl
Prior art date
Application number
PT01980397T
Other languages
English (en)
Inventor
Alistair Lochead
Thierry Gallet
Antonio Almario Garcia
Adrien Tak Li
Severine Marguerie
Mourad Saady
Philippe Yaiche
Alain Nedelec
Original Assignee
Sanofi Synthelabo
Mitsubishi Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo, Mitsubishi Pharma Corp filed Critical Sanofi Synthelabo
Priority claimed from PCT/EP2001/010726 external-priority patent/WO2002018386A1/en
Publication of PT1315731E publication Critical patent/PT1315731E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT01980397T 2000-09-01 2001-08-31 Derivados de 2-piridinil-6,7,8,9-tetra-hidropirimido [1,2-a] pirimidin-4-ona e 7-piridinil-2,3-di-hidroimidazol [1,2-a]pirimidin-5 (1h) ona PT1315731E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00402412A EP1184385A1 (en) 2000-09-01 2000-09-01 1-[Alkyl], 1-[(heteroaryl)alkyl] and 1-[(aryl)alkyl]-7-pyridin-4-yl-2,3-dihydroimidazo[1,2-a]pyrimidin-5(1H)-one derivatives
PCT/EP2001/010726 WO2002018386A1 (en) 2000-09-01 2001-08-31 2-PYRIDINYL-6,7,8,9-TETRAHYDROPYRIMIDO[1,2-a]PYRIMIDIN-4-ONE AND 7-PYRIDINYL-2,3-DIHYDROIMIDAZO[1,2-a]PYRIMIDIN-5(1H)ONE DERIVATI VES

Publications (1)

Publication Number Publication Date
PT1315731E true PT1315731E (pt) 2004-10-29

Family

ID=8173839

Family Applications (1)

Application Number Title Priority Date Filing Date
PT01980397T PT1315731E (pt) 2000-09-01 2001-08-31 Derivados de 2-piridinil-6,7,8,9-tetra-hidropirimido [1,2-a] pirimidin-4-ona e 7-piridinil-2,3-di-hidroimidazol [1,2-a]pirimidin-5 (1h) ona

Country Status (2)

Country Link
EP (1) EP1184385A1 (pt)
PT (1) PT1315731E (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1454909B1 (en) * 2003-03-07 2008-08-20 Sanofi Aventis 8'-pyridinyl-dihydrospiro (cycloalkyl) -pyrimido (1,2-a) pyrimidin-6-one and 8'-pyrimidinyl-dihydrospiro (cycloalkyl) pyrimido (1,2-a) pyrimidin-6 derivatives -one and their use against neurodegenerative diseases
WO2014053568A1 (en) * 2012-10-02 2014-04-10 Sanofi Indolyldihydroimidazopyrimidinone derivatives, preparation thereof and therapeutic use thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI241298B (en) * 1998-09-25 2005-10-11 Mitsubishi Chem Corp Pyrimidone derivatives

Also Published As

Publication number Publication date
EP1184385A1 (en) 2002-03-06

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