PL4138807T3 - Kokryształ gabapentyny, ketoprofenu i lizyny, kompozycje farmaceutyczne i ich zastosowanie medyczne - Google Patents

Kokryształ gabapentyny, ketoprofenu i lizyny, kompozycje farmaceutyczne i ich zastosowanie medyczne

Info

Publication number
PL4138807T3
PL4138807T3 PL21720272.0T PL21720272T PL4138807T3 PL 4138807 T3 PL4138807 T3 PL 4138807T3 PL 21720272 T PL21720272 T PL 21720272T PL 4138807 T3 PL4138807 T3 PL 4138807T3
Authority
PL
Poland
Prior art keywords
gabapentin
ketoprofen
lysine
crystal
pharmaceutical compositions
Prior art date
Application number
PL21720272.0T
Other languages
English (en)
Inventor
Andrea Aramini
Marcello Allegretti
Gianluca Bianchini
Samuele Lillini
Mara TOMASSETTI
Original Assignee
Dompé Farmaceutici Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dompé Farmaceutici Spa filed Critical Dompé Farmaceutici Spa
Publication of PL4138807T3 publication Critical patent/PL4138807T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PL21720272.0T 2020-04-21 2021-04-21 Kokryształ gabapentyny, ketoprofenu i lizyny, kompozycje farmaceutyczne i ich zastosowanie medyczne PL4138807T3 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20170740.3A EP3900716A1 (en) 2020-04-21 2020-04-21 Co-crystal of gabapentin, ketoprofen and lysine, pharmaceutical compositions and their medical use
PCT/EP2021/060421 WO2021214158A1 (en) 2020-04-21 2021-04-21 Co-crystal of gabapentin, ketoprofen and lysine, pharmaceutical compositions and their medical use

Publications (1)

Publication Number Publication Date
PL4138807T3 true PL4138807T3 (pl) 2026-01-12

Family

ID=70390939

Family Applications (1)

Application Number Title Priority Date Filing Date
PL21720272.0T PL4138807T3 (pl) 2020-04-21 2021-04-21 Kokryształ gabapentyny, ketoprofenu i lizyny, kompozycje farmaceutyczne i ich zastosowanie medyczne

Country Status (17)

Country Link
US (1) US12582624B2 (pl)
EP (2) EP3900716A1 (pl)
CN (1) CN115697315B (pl)
BR (1) BR112022019493A2 (pl)
CA (1) CA3176958A1 (pl)
DK (1) DK4138807T3 (pl)
ES (1) ES3049312T3 (pl)
FI (1) FI4138807T3 (pl)
HR (1) HRP20251314T1 (pl)
IL (1) IL296856A (pl)
LT (1) LT4138807T (pl)
PL (1) PL4138807T3 (pl)
PT (1) PT4138807T (pl)
RS (1) RS67340B1 (pl)
SI (1) SI4138807T1 (pl)
SM (1) SMT202500410T1 (pl)
WO (1) WO2021214158A1 (pl)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3907214A1 (en) * 2020-05-04 2021-11-10 Dompe' Farmaceutici S.P.A. Co-crystal of ketoprofen, lysine and gabapentin, pharmaceutical compositions and their medical use
EP4169903A1 (en) * 2021-10-25 2023-04-26 Dompe' Farmaceutici S.P.A. Co-crystals of nonsteroidal anti-inflammatory drugs, lysine and gabapentin, pharmaceutical compositions and their medical use

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1497044A (en) 1974-03-07 1978-01-05 Prodotti Antibiotici Spa Salts of phenyl-alkanoic acids
IT1104556B (it) 1977-05-12 1985-10-21 Medea Res Srl Sale di lisina dell'acido meta-benzoil-idratropico,processo per la sua preparazione e composizione farmaceutiche che lo contengono
EP1696959A2 (en) * 2003-12-24 2006-09-06 Sepracor, Inc. Melatonin combination therapy for improving sleep quality
CA2680792A1 (en) 2007-03-15 2008-09-18 Biogen Idec Ma Inc. Treatment of autoimmune disorders
JP5580345B2 (ja) 2009-03-06 2014-08-27 ゼノポート,インコーポレイティド 高充填量のガバペンチンプロドラッグを有する経口剤形
US9169279B2 (en) * 2009-07-31 2015-10-27 Thar Pharmaceuticals, Inc. Crystallization method and bioavailability
US20130109674A1 (en) * 2009-12-18 2013-05-02 Achelios Therapeutics Llc Methods and compositions for treating and preventing trigeminal autonomic cephalgias, migraine, and vascular conditions
CN110015955A (zh) * 2010-07-23 2019-07-16 格吕伦塔尔有限公司 3-(3-二甲基氨基-1-乙基-2-甲基-丙基)-苯酚的盐或共晶体
KR102298676B1 (ko) 2014-05-09 2021-09-07 테크니메데 소시에다데 테크니코-메디시날 에스.에이. 의약으로서 사용되기 위한 (s)-펄린돌 및 약학적으로 허용 가능한 그의 염
WO2017048702A1 (en) * 2015-09-14 2017-03-23 Infinity Pharmaceuticals, Inc. Solid forms of isoquinolinone derivatives, process of making, compositions comprising, and methods of using the same
EP3670489A1 (en) 2018-12-21 2020-06-24 Dompé farmaceutici S.p.A. Co-crystal of ketoprofen, compositions comprising the same, process of producing the same, and uses thereof
GB201820936D0 (en) 2018-12-21 2019-02-06 Rolls Royce Plc Low noise gas turbine engine
EP3842408A1 (en) 2019-12-23 2021-06-30 Dompé farmaceutici S.p.A. Co-crystal of ketoprofen and its preparation, pharmaceutical compositions comprising the same and uses thereof

Also Published As

Publication number Publication date
DK4138807T3 (da) 2025-10-20
CN115697315B (zh) 2024-05-24
EP4138807A1 (en) 2023-03-01
CA3176958A1 (en) 2021-10-28
RS67340B1 (sr) 2025-11-28
PT4138807T (pt) 2025-11-05
BR112022019493A2 (pt) 2023-01-10
IL296856A (en) 2022-11-01
LT4138807T (lt) 2025-11-25
HRP20251314T1 (hr) 2025-12-05
SMT202500410T1 (it) 2025-11-10
WO2021214158A1 (en) 2021-10-28
US12582624B2 (en) 2026-03-24
CN115697315A (zh) 2023-02-03
ES3049312T3 (en) 2025-12-16
EP4138807B1 (en) 2025-10-08
SI4138807T1 (sl) 2026-01-30
US20230181507A1 (en) 2023-06-15
FI4138807T3 (fi) 2025-11-19
EP3900716A1 (en) 2021-10-27

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