PL397662A1 - Terapia skojarzona niedrobnokomórkowego raka pluc - Google Patents
Terapia skojarzona niedrobnokomórkowego raka plucInfo
- Publication number
- PL397662A1 PL397662A1 PL397662A PL39766211A PL397662A1 PL 397662 A1 PL397662 A1 PL 397662A1 PL 397662 A PL397662 A PL 397662A PL 39766211 A PL39766211 A PL 39766211A PL 397662 A1 PL397662 A1 PL 397662A1
- Authority
- PL
- Poland
- Prior art keywords
- cell lung
- small
- combination therapy
- lung carcinoma
- combination
- Prior art date
Links
- 208000002154 non-small cell lung carcinoma Diseases 0.000 title abstract 2
- 238000002648 combination therapy Methods 0.000 title 1
- 150000003710 vitamin D derivatives Chemical class 0.000 abstract 2
- 239000005517 L01XE01 - Imatinib Substances 0.000 abstract 1
- 229930003316 Vitamin D Natural products 0.000 abstract 1
- QYSXJUFSXHHAJI-XFEUOLMDSA-N Vitamin D3 Natural products C1(/[C@@H]2CC[C@@H]([C@]2(CCC1)C)[C@H](C)CCCC(C)C)=C/C=C1\C[C@@H](O)CCC1=C QYSXJUFSXHHAJI-XFEUOLMDSA-N 0.000 abstract 1
- 229960002882 calcipotriol Drugs 0.000 abstract 1
- LWQQLNNNIPYSNX-UROSTWAQSA-N calcipotriol Chemical compound C1([C@H](O)/C=C/[C@@H](C)[C@@H]2[C@]3(CCCC(/[C@@H]3CC2)=C\C=C\2C([C@@H](O)C[C@H](O)C/2)=C)C)CC1 LWQQLNNNIPYSNX-UROSTWAQSA-N 0.000 abstract 1
- KTUFNOKKBVMGRW-UHFFFAOYSA-N imatinib Chemical compound C1CN(C)CCN1CC1=CC=C(C(=O)NC=2C=C(NC=3N=C(C=CN=3)C=3C=NC=CC=3)C(C)=CC=2)C=C1 KTUFNOKKBVMGRW-UHFFFAOYSA-N 0.000 abstract 1
- 229960002411 imatinib Drugs 0.000 abstract 1
- 239000004615 ingredient Substances 0.000 abstract 1
- BJYLYJCXYAMOFT-RSFVBTMBSA-N tacalcitol Chemical compound C1(/[C@@H]2CC[C@@H]([C@]2(CCC1)C)[C@H](C)CC[C@@H](O)C(C)C)=C\C=C1\C[C@@H](O)C[C@H](O)C1=C BJYLYJCXYAMOFT-RSFVBTMBSA-N 0.000 abstract 1
- 229960004907 tacalcitol Drugs 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
- 208000029729 tumor suppressor gene on chromosome 11 Diseases 0.000 abstract 1
- 229940121358 tyrosine kinase inhibitor Drugs 0.000 abstract 1
- 239000005483 tyrosine kinase inhibitor Substances 0.000 abstract 1
- 150000004917 tyrosine kinase inhibitor derivatives Chemical class 0.000 abstract 1
- 235000019166 vitamin D Nutrition 0.000 abstract 1
- 239000011710 vitamin D Substances 0.000 abstract 1
- 229940046008 vitamin d Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/59—Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
- A61K31/593—9,10-Secocholestane derivatives, e.g. cholecalciferol, i.e. vitamin D3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Wynalazek dotyczy terapii niedrobnokomórkowego raka pluc, w której skojarzenie z pochodnymi witamin D wzmaga dzialanie terapeutyczne inhibitora kinaz tyrozynowych imatinibu. Skladniki kombinacji - analogi witaminy D, korzystnie wybrane sa z grupy obejmujacej takalcytol i izomer 5,6-trans kalcypotriolu.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL397662A PL226174B1 (pl) | 2011-12-30 | 2011-12-30 | Polaczenie analogu witaminy D z imatinibem do stosowania w leczeniu skojarzonym niedrobnokomorkowego raka pluc |
| PCT/PL2012/000134 WO2013100772A1 (en) | 2011-12-30 | 2012-12-30 | The use of vitamin d analogues in combination with imatinib in therapy of non-small cell lung cancer |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PL397662A PL226174B1 (pl) | 2011-12-30 | 2011-12-30 | Polaczenie analogu witaminy D z imatinibem do stosowania w leczeniu skojarzonym niedrobnokomorkowego raka pluc |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL397662A1 true PL397662A1 (pl) | 2013-07-08 |
| PL226174B1 PL226174B1 (pl) | 2017-06-30 |
Family
ID=47666456
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL397662A PL226174B1 (pl) | 2011-12-30 | 2011-12-30 | Polaczenie analogu witaminy D z imatinibem do stosowania w leczeniu skojarzonym niedrobnokomorkowego raka pluc |
Country Status (2)
| Country | Link |
|---|---|
| PL (1) | PL226174B1 (pl) |
| WO (1) | WO2013100772A1 (pl) |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW225528B (pl) | 1992-04-03 | 1994-06-21 | Ciba Geigy Ag | |
| CO4940418A1 (es) | 1997-07-18 | 2000-07-24 | Novartis Ag | Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso |
| WO2004098612A2 (en) * | 2003-05-07 | 2004-11-18 | Ab Science | Calcitriol analogs of uses thereof |
| EP1631543A1 (en) * | 2003-06-11 | 2006-03-08 | Novacea, Inc. | Treatment of lung cancer with active vitamin d compounds in combination with other treatments |
-
2011
- 2011-12-30 PL PL397662A patent/PL226174B1/pl unknown
-
2012
- 2012-12-30 WO PCT/PL2012/000134 patent/WO2013100772A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| PL226174B1 (pl) | 2017-06-30 |
| WO2013100772A1 (en) | 2013-07-04 |
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