PH21372A - Beta-lactamase inhibiting 6-(alkoxy-aminoethyl) penicillanic acid 1,1-dioxide and derivatives - Google Patents

Beta-lactamase inhibiting 6-(alkoxy-aminoethyl) penicillanic acid 1,1-dioxide and derivatives

Info

Publication number
PH21372A
PH21372A PH30780A PH30780A PH21372A PH 21372 A PH21372 A PH 21372A PH 30780 A PH30780 A PH 30780A PH 30780 A PH30780 A PH 30780A PH 21372 A PH21372 A PH 21372A
Authority
PH
Philippines
Prior art keywords
beta
penicillanic acid
derivatives
aminoethyl
alkoxy
Prior art date
Application number
PH30780A
Other languages
English (en)
Inventor
Pirie Donald Klein
Volkmann Robert Alfred
Kleinman Edward Fox
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PH21372A publication Critical patent/PH21372A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
PH30780A 1983-06-06 1984-06-06 Beta-lactamase inhibiting 6-(alkoxy-aminoethyl) penicillanic acid 1,1-dioxide and derivatives PH21372A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/501,475 US4499017A (en) 1983-06-06 1983-06-06 Beta-lactamase inhibiting 6-(alkoxyamino-methyl) penicillanic acid 1,1-dioxide and derivatives

Publications (1)

Publication Number Publication Date
PH21372A true PH21372A (en) 1987-10-15

Family

ID=23993709

Family Applications (2)

Application Number Title Priority Date Filing Date
PH30780A PH21372A (en) 1983-06-06 1984-06-06 Beta-lactamase inhibiting 6-(alkoxy-aminoethyl) penicillanic acid 1,1-dioxide and derivatives
PH33521A PH22842A (en) 1983-06-06 1986-03-13 Process for the preparation of 6-alpha and 6-beta-(aminomethyl)penicillanic acid 1,1-dioxide beta-lactamase inhibiting-6 alkoxyaminomethyl

Family Applications After (1)

Application Number Title Priority Date Filing Date
PH33521A PH22842A (en) 1983-06-06 1986-03-13 Process for the preparation of 6-alpha and 6-beta-(aminomethyl)penicillanic acid 1,1-dioxide beta-lactamase inhibiting-6 alkoxyaminomethyl

Country Status (21)

Country Link
US (1) US4499017A (no)
EP (1) EP0128037B1 (no)
JP (1) JPS606693A (no)
KR (1) KR870000312B1 (no)
AT (1) ATE24512T1 (no)
AU (1) AU545467B2 (no)
CA (1) CA1247597A (no)
DE (1) DE3461800D1 (no)
DK (1) DK275884A (no)
ES (1) ES8506720A1 (no)
FI (1) FI842255A (no)
GR (1) GR82214B (no)
HU (1) HU193573B (no)
IL (1) IL72003A (no)
NO (1) NO842248L (no)
NZ (1) NZ208381A (no)
PH (2) PH21372A (no)
PL (1) PL144040B1 (no)
PT (1) PT78689A (no)
YU (1) YU97084A (no)
ZA (1) ZA844184B (no)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8928373D0 (en) * 1989-12-15 1990-02-21 Erba Carlo Spa Beta-lactam derivatives
RU2275363C2 (ru) 2000-07-19 2006-04-27 Новартис Аг Соли валсартана, фармацевтическая композиция на их основе и способ получения солей

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
RO84910B (ro) * 1982-01-11 1984-09-30 Pfizer Inc. Procedeu pentru prepararea unor derivati 1, 1-dioxizi ai acidului 6-aminoalchilpenicilanic

Also Published As

Publication number Publication date
PH22842A (en) 1989-01-19
EP0128037A1 (en) 1984-12-12
GR82214B (no) 1984-12-13
PL144040B1 (en) 1988-04-30
ZA844184B (en) 1986-01-29
DK275884D0 (da) 1984-06-04
PL248043A1 (en) 1985-07-30
CA1247597A (en) 1988-12-28
JPS606693A (ja) 1985-01-14
FI842255A0 (fi) 1984-06-05
HU193573B (en) 1987-10-28
HUT35266A (en) 1985-06-28
KR850000446A (ko) 1985-02-27
IL72003A (en) 1988-02-29
AU2907684A (en) 1984-12-13
DE3461800D1 (en) 1987-02-05
DK275884A (da) 1985-01-09
IL72003A0 (en) 1984-10-31
ES533147A0 (es) 1985-08-01
FI842255A (fi) 1984-12-07
AU545467B2 (en) 1985-07-18
NZ208381A (en) 1987-05-29
ATE24512T1 (de) 1987-01-15
KR870000312B1 (ko) 1987-02-26
NO842248L (no) 1984-12-07
YU97084A (en) 1986-10-31
US4499017A (en) 1985-02-12
EP0128037B1 (en) 1986-12-30
ES8506720A1 (es) 1985-08-01
PT78689A (en) 1984-07-01

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