PE296A1 - DERIVATIVES OF 2-IMIDAZOLINE-5-ONAS FUNGICIDES - Google Patents

DERIVATIVES OF 2-IMIDAZOLINE-5-ONAS FUNGICIDES

Info

Publication number
PE296A1
PE296A1 PE1995262006A PE26200695A PE296A1 PE 296 A1 PE296 A1 PE 296A1 PE 1995262006 A PE1995262006 A PE 1995262006A PE 26200695 A PE26200695 A PE 26200695A PE 296 A1 PE296 A1 PE 296A1
Authority
PE
Peru
Prior art keywords
group
radical
alkyl
heteroaril
attacked
Prior art date
Application number
PE1995262006A
Other languages
Spanish (es)
Inventor
Joseph Perez
Alain Gadras
Guy Lacroix
Christine Veyrat
Jean Philippe Bascou
Philippe Desbordes
Gilbert Emeric
Original Assignee
Rhone Poulenc Agrochimie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Agrochimie filed Critical Rhone Poulenc Agrochimie
Publication of PE296A1 publication Critical patent/PE296A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/70—One oxygen atom
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C331/00—Derivatives of thiocyanic acid or of isothiocyanic acid
    • C07C331/16—Isothiocyanates
    • C07C331/18—Isothiocyanates having isothiocyanate groups bound to acyclic carbon atoms
    • C07C331/22—Isothiocyanates having isothiocyanate groups bound to acyclic carbon atoms of an unsaturated carbon skeleton
    • C07C331/24—Isothiocyanates having isothiocyanate groups bound to acyclic carbon atoms of an unsaturated carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • C07D233/74—Two oxygen atoms, e.g. hydantoin with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to other ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • C07D233/76—Two oxygen atoms, e.g. hydantoin with substituted hydrocarbon radicals attached to the third ring carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/84—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/86—Oxygen and sulfur atoms, e.g. thiohydantoin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

CARACTERIZADOS PORQUE TIENEN LA FORMULA GENERAL (I); DONDE: R1 ES UN ATOMO DE CARBONO O GRUPO VINILO O ALILO, O UN RADICAL ALQUILO O HALOALQUILO; N = 0 o 1; Y ES O o S; R2 UN GRUPO ALQUILO O HALOALQUILO O EL GRUPO CICLOPROPILO; R3 ES UN RADICAL ARILO O HETEROARILO, PARTICULARMENTE FENILO, NAFTILO EVENTUALMENTE SUSTITUIDOS CON 1 A 3 GRUPOS SELECCIONADOS ENTRE LOS SIGNIFICADOS EN R5; R4 ES UN ATOMO DE HIDROGENO, UN RADICAL FORMILO O AROILO; R5 ES UN ATOMO DE HALOGENO O EL GRUPO HIDROXI, NITRO O UN RADICAL ALQUILO O CICLOALQUILO O AMINO; W ES O, S o SO; Ar1 ES UN RADICAL DIVALENTE DERIVADO DE UN RADICAL ARILO O HETEROARILO QUE COMPRENDE UN GRUPO FENILO, PIRIDILO; Ar2 ES UN SISTEMA MONO O BICICLICO DE 5 A 10 ATOMOS, QUE ES AROMATICO, SATURADO O INSATURADO QUE ES UN SISTEMA CARBOCICLICO O HETEROCICLICO CON 1 A 4 HETEROATOMOS; X ES UN ENCADENAMIENTO DE FORMULA -(R")j-A-(R`)k, DONDE k Y j = 0 o 1, R" Y R' SON UN HALOGENO, UN GRUPO CIANO, TIOCIANO DONDE UNO O VARIOS ATOMOS DE CARBONO PUEDEN SER REEMPLAZADOS POR O,S; A ES O, S, SO, CO Y OTROS. COMPOSICIONES FUNGICIDAS CON 0,05% A 95% EN PESO DE MATERIAS ACTIVAS, SON UTILES EN EL TRATAMIENTO DE PLANTAS CULTIVADAS, ATACADAS O SUSCEPTIBLES A SER ATACADAS POR ENFERMEDADES FUNGICAS, SIENDO APLICADAS A LAS PARTES AEREAS DE LAS PLANTAS CON UNA DOSIS COMPRENDIDA ENTRE 0,005 kg/ha Y 1 kg/haCHARACTERIZED BECAUSE THEY HAVE THE GENERAL FORMULA (I); WHERE: R1 IS A VINYL OR ALYL CARBON ATOMO OR GROUP, OR A RADICAL ALKYL OR HALOALKYL; N = 0 or 1; Y IS O or S; R2 AN ALKYL OR HALOALKYL GROUP OR THE CYCLOPROPYL GROUP; R3 IS A RADICAL ARYL OR HETEROARIL, PARTICULARLY PHENYL, NAPHTHYL EVENTUALLY SUBSTITUTED WITH 1 TO 3 GROUPS SELECTED FROM THE MEANINGS IN R5; R4 IS A HYDROGEN ATOM, A RADICAL FORMYL OR AROYL; R5 IS AN ATOM OF HALOGEN OR THE HYDROXY GROUP, NITRO OR A RADICAL ALKYL OR CYCLLOALKYL OR AMINO; W ES O, S or SO; Ar1 IS A DIVALENT RADICAL DERIVED FROM A RADICAL ARYL OR HETEROARIL WHICH INCLUDES A PHENYL, PIRIDILE GROUP; Ar2 IS A MONO OR BICYCLE SYSTEM OF 5 TO 10 ATOMS, WHICH IS AROMATIC, SATURATED OR UNSATURATED, WHICH IS A CARBOCICLIC OR HETERO-CYCLE SYSTEM WITH 1 TO 4 HETEROATOMES; X IS A FORMULA CHAIN - (R ") jA- (R`) k, WHERE k AND j = 0 or 1, R" YR 'ARE A HALOGEN, A CYAN GROUP, A TIOCIAN WHERE ONE OR MULTIPLE ATOMS OF CARBON CAN BE REPLACED BY O, S; A ES O, S, SO, CO AND OTHERS. FUNGICIDAL COMPOSITIONS WITH 0.05% TO 95% BY WEIGHT OF ACTIVE MATERIALS, ARE USEFUL IN THE TREATMENT OF CULTIVATED, ATTACKED, OR SUSCEPTIBLE PLANTS TO BE ATTACKED BY FUNGAL DISEASES, BEING APPLIED TO THE AERIAL PARTS OF PLANTS WITH A COMPREHENSIVE DOSE kg / ha AND 1 kg / ha

PE1995262006A 1994-02-17 1995-02-16 DERIVATIVES OF 2-IMIDAZOLINE-5-ONAS FUNGICIDES PE296A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9402135A FR2716192B1 (en) 1994-02-17 1994-02-17 2-Imidazoline-5-ones fungicidal derivatives.

Publications (1)

Publication Number Publication Date
PE296A1 true PE296A1 (en) 1996-01-19

Family

ID=9460402

Family Applications (1)

Application Number Title Priority Date Filing Date
PE1995262006A PE296A1 (en) 1994-02-17 1995-02-16 DERIVATIVES OF 2-IMIDAZOLINE-5-ONAS FUNGICIDES

Country Status (24)

Country Link
EP (1) EP0668270A3 (en)
JP (1) JPH07278117A (en)
KR (1) KR950032135A (en)
CN (1) CN1111241A (en)
AP (1) AP581A (en)
AU (1) AU1224595A (en)
BR (1) BR9500584A (en)
CA (1) CA2142647A1 (en)
CO (1) CO4410279A1 (en)
CZ (1) CZ39295A3 (en)
FI (1) FI950710A (en)
FR (1) FR2716192B1 (en)
HU (1) HUT71916A (en)
IL (1) IL112631A0 (en)
MA (1) MA23455A1 (en)
NZ (1) NZ270499A (en)
PE (1) PE296A1 (en)
PL (1) PL307295A1 (en)
RU (1) RU95102145A (en)
SI (1) SI9500053A (en)
SK (1) SK21595A3 (en)
TR (1) TR28502A (en)
YU (1) YU9995A (en)
ZA (1) ZA951196B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2049472B1 (en) 2006-06-23 2015-01-21 AbbVie Bahamas Ltd. Cyclopropyl amine derivatives as histamin h3 receptor modulators
US9108948B2 (en) 2006-06-23 2015-08-18 Abbvie Inc. Cyclopropyl amine derivatives
US9186353B2 (en) 2009-04-27 2015-11-17 Abbvie Inc. Treatment of osteoarthritis pain
US8759535B2 (en) 2010-02-18 2014-06-24 High Point Pharmaceuticals, Llc Substituted fused imidazole derivatives, pharmaceutical compositions, and methods of use thereof
CN102762101B (en) 2010-02-18 2014-09-17 高点制药有限责任公司 Substituted fused imidazole derivatives, pharmaceutical compositions, and methods of use thereof
US8853390B2 (en) 2010-09-16 2014-10-07 Abbvie Inc. Processes for preparing 1,2-substituted cyclopropyl derivatives
HUE055262T2 (en) 2014-08-11 2021-11-29 Angion Biomedica Corp Cytochrome p450 inhibitors and uses thereof
WO2016089648A1 (en) 2014-12-01 2016-06-09 Vtv Therapeutics Llc Bach 1 inhibitors in combination with nrf2 activators and pharmaceutical compositions thereof
AU2015374231B2 (en) 2014-12-31 2020-07-23 Angion Biomedica Corp. Methods and agents for treating disease
CN105859598B (en) * 2016-04-19 2017-07-04 青岛科技大学 A kind of preparation method of polysubstituted two sulphur aryl imine derivative

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5036157A (en) * 1986-03-11 1991-07-30 Burroughs Wellcome Co. Aryl derivatives
FR2685328B1 (en) * 1991-12-20 1995-12-01 Rhone Poulenc Agrochimie DERIVATIVES OF 2-IMIDAZOLINE-5-ONES AND 2-IMIDAZOLINE-5-THIONES FUNGICIDES.
FR2693192B1 (en) * 1992-07-02 1994-08-12 Rhone Poulenc Agrochimie Derivatives of 2-imidazoline-5-ones and 2-imidazoline-5-thiones fungicides.
EP1008589A1 (en) * 1992-05-22 2000-06-14 E.I. Du Pont De Nemours & Company Incorporated Fungicidal imidazolinones

Also Published As

Publication number Publication date
HU9500466D0 (en) 1995-04-28
NZ270499A (en) 1996-09-25
BR9500584A (en) 1995-10-24
KR950032135A (en) 1995-12-20
FI950710A0 (en) 1995-02-16
SK21595A3 (en) 1995-09-13
PL307295A1 (en) 1995-08-21
MA23455A1 (en) 1995-10-01
CZ39295A3 (en) 1995-10-18
CN1111241A (en) 1995-11-08
CO4410279A1 (en) 1997-01-09
ZA951196B (en) 1996-07-16
FI950710A (en) 1995-08-18
EP0668270A2 (en) 1995-08-23
HUT71916A (en) 1996-02-28
AP581A (en) 1997-03-27
JPH07278117A (en) 1995-10-24
IL112631A0 (en) 1995-05-26
AU1224595A (en) 1995-08-24
RU95102145A (en) 1996-11-20
YU9995A (en) 1998-07-10
EP0668270A3 (en) 1995-10-11
CA2142647A1 (en) 1995-08-18
AP9500722A0 (en) 1995-04-30
TR28502A (en) 1996-09-02
FR2716192A1 (en) 1995-08-18
FR2716192B1 (en) 1996-04-12
SI9500053A (en) 1995-08-31

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