PE20120348A1 - Combinacion que comprende cabazitaxel y capecitabina - Google Patents

Combinacion que comprende cabazitaxel y capecitabina

Info

Publication number
PE20120348A1
PE20120348A1 PE2011001906A PE2011001906A PE20120348A1 PE 20120348 A1 PE20120348 A1 PE 20120348A1 PE 2011001906 A PE2011001906 A PE 2011001906A PE 2011001906 A PE2011001906 A PE 2011001906A PE 20120348 A1 PE20120348 A1 PE 20120348A1
Authority
PE
Peru
Prior art keywords
capecitabin
cabazitaxel
combination including
solvate
including cabazitaxel
Prior art date
Application number
PE2011001906A
Other languages
English (en)
Inventor
Emmanuelle Magherini
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of PE20120348A1 publication Critical patent/PE20120348A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7068Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

REFERIDA A UNA COMBINACION FARMACEUTICA QUE COMPRENDE CABAZITAXEL Y CAPECITABINA, LOS CUALES PUEDEN ESTAR EN SU FORMA BASE, SAL DE ACIDO, HIDRATO O SOLVATO. DE PREFERENCIA, EL CABAZITAXEL SE ENCUENTRA BAJO LA FORMA DE SOLVATO ACETONICO Y CONTIENE ENTRE 5% Y 8% EN PESO DE ACETONA. DICHA COMBINACION TIENE ACTIVIDAD ANTITUMORAL Y ES UTIL EN PACIENTES CON CANCER DE MAMA METASTASICO
PE2011001906A 2009-05-06 2010-05-06 Combinacion que comprende cabazitaxel y capecitabina PE20120348A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0902189A FR2945211A1 (fr) 2009-05-06 2009-05-06 Combinaison antitumorale comprenant la cabazitaxel et la capecitabine
FR0902264A FR2945212B1 (fr) 2009-05-06 2009-05-11 Combinaison antitumorale comprenant le cabazitaxel et la capecitabine

Publications (1)

Publication Number Publication Date
PE20120348A1 true PE20120348A1 (es) 2012-04-24

Family

ID=41168737

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2011001906A PE20120348A1 (es) 2009-05-06 2010-05-06 Combinacion que comprende cabazitaxel y capecitabina

Country Status (25)

Country Link
US (1) US20120115806A1 (es)
EP (1) EP2427187A1 (es)
JP (1) JP2012526089A (es)
KR (1) KR20120008069A (es)
CN (1) CN102458392A (es)
AU (1) AU2010244253A1 (es)
BR (1) BRPI1011827A2 (es)
CA (1) CA2761079A1 (es)
CL (1) CL2011002774A1 (es)
CO (1) CO6390103A2 (es)
CR (1) CR20110586A (es)
DO (1) DOP2011000336A (es)
EA (1) EA201171360A1 (es)
EC (1) ECSP11011435A (es)
FR (2) FR2945211A1 (es)
IL (1) IL216063A0 (es)
MA (1) MA33343B1 (es)
MX (1) MX2011011765A (es)
NI (1) NI201100192A (es)
NZ (1) NZ596226A (es)
PE (1) PE20120348A1 (es)
SG (1) SG175894A1 (es)
TN (1) TN2011000542A1 (es)
WO (1) WO2010128258A1 (es)
ZA (1) ZA201108109B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA024186B1 (ru) 2009-10-29 2016-08-31 Авентис Фарма С.А. Применение кабазитаксела в комбинации с преднизоном или преднизолоном для лечения рака простаты
CN102068407B (zh) * 2010-12-27 2011-11-23 江苏奥赛康药业股份有限公司 一种cabazitaxel注射液及其制备方法
EP2620148A1 (en) 2012-01-27 2013-07-31 Aventis Pharma S.A. Antitumoral combination comprising cabazitaxel and cisplatin
HUE046232T2 (hu) 2011-02-25 2020-02-28 Sanofi Mature Ip Kabazitaxelt és ciszplatint tartalmazó tumorellenes kombináció
EP2491925A1 (en) 2011-02-25 2012-08-29 Aventis Pharma S.A. Antitumoral combination comprising cabazitaxel and cisplatin
BR212016030926U2 (pt) * 2014-06-30 2018-05-29 Tarveda Therapeutics Inc conjugados de alvo e partículas e formulações dos mesmos
CN108473538B (zh) 2015-10-28 2022-01-28 塔弗达治疗有限公司 Sstr靶向缀合物及其颗粒和制剂

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU671491B2 (en) 1992-12-18 1996-08-29 F. Hoffmann-La Roche Ag N-oxycarbonyl substituted 5'-deoxy-5-fluorcytidines
MA23823A1 (fr) 1995-03-27 1996-10-01 Aventis Pharma Sa Nouveaux taxoides, leur preparation et les compositions qui les contiennent
FR2859996B1 (fr) * 2003-09-19 2006-02-03 Aventis Pharma Sa Solvat acetonique du dimethoxy docetaxel et son procede de preparation

Also Published As

Publication number Publication date
CL2011002774A1 (es) 2012-04-20
FR2945212A1 (fr) 2010-11-12
JP2012526089A (ja) 2012-10-25
MA33343B1 (fr) 2012-06-01
US20120115806A1 (en) 2012-05-10
NI201100192A (es) 2012-01-23
CR20110586A (es) 2011-12-13
TN2011000542A1 (fr) 2013-05-24
DOP2011000336A (es) 2011-12-15
CO6390103A2 (es) 2012-02-29
CA2761079A1 (fr) 2010-11-11
IL216063A0 (en) 2012-01-31
EP2427187A1 (fr) 2012-03-14
MX2011011765A (es) 2012-06-01
KR20120008069A (ko) 2012-01-25
EA201171360A1 (ru) 2012-05-30
WO2010128258A1 (fr) 2010-11-11
FR2945211A1 (fr) 2010-11-12
NZ596226A (en) 2014-01-31
FR2945212B1 (fr) 2011-07-01
AU2010244253A1 (en) 2011-11-24
ZA201108109B (en) 2013-01-30
BRPI1011827A2 (pt) 2016-03-22
ECSP11011435A (es) 2011-12-30
SG175894A1 (en) 2011-12-29
CN102458392A (zh) 2012-05-16

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