PE20091560A1 - ORAL DISINTEGRATION TABLET - Google Patents
ORAL DISINTEGRATION TABLETInfo
- Publication number
- PE20091560A1 PE20091560A1 PE2009000311A PE2009000311A PE20091560A1 PE 20091560 A1 PE20091560 A1 PE 20091560A1 PE 2009000311 A PE2009000311 A PE 2009000311A PE 2009000311 A PE2009000311 A PE 2009000311A PE 20091560 A1 PE20091560 A1 PE 20091560A1
- Authority
- PE
- Peru
- Prior art keywords
- found
- weight
- parts
- dispersion
- disintegration tablet
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Epidemiology (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
SE REFIERE A UNA COMPOSICION FARMACEUTICA EN FORMA DE COMPRIMIDO DESINTEGRANTE ORAL, QUE COMPRENDE: A) CILOSTAZOL Y SACARIDOS TALES COMO MANITOL, XILITOL, ENTRE OTROS EN FORMA DE PARTICULAS GRANULADAS QUE SE PREPARAN POR DISPERSION UNIFORME DE UNA SUSTANCIA INORGANICA Y UN AGENTE DESINTEGRANTE, DONDE (a) LOS SACARIDOS SE ENCUENTRA EN 40-90 PARTES EN PESO, (b) LA SUSTANCIA INORGANICA SE ENCUENTRA EN 1-30 PARTES EN PESO Y (c) EL AGENTE DESINTEGRANTES SE ENCUENTRA EN 5-40 PARTES EN PESO; B) UN DESLIZANTE TAL COMO DIOXIDO DE SILICIO HIDRATADO, ACIDO SILICICO ANHIDRO LIVIANO Y PESADO, QUE SE ENCUENTRA EN UNA CANTIDAD DE 0.2% A 2% (p/p); C) UN EXCIPIENTE ORGANICO TALES COMO ALMIDON DE MAIZ, CELULOSA CRISTALINA, ENTRE OTROS; D) UNO O MAS ADITIVOS OPCIONALES TALES COMO LUBRICANTES, EDULCORANTES, AROMATIZANTES, ENTRE OTROS. DICHO COMPRIMIDO ES UTIL PARA PACIENTES DE EDAD AVANZADA Y PACIENTES QUE SUFREN DE DISFAGIAIT REFERS TO A PHARMACEUTICAL COMPOSITION IN THE FORM OF AN ORAL DISINTEGRANT TABLET, WHICH INCLUDES: A) CILOSTAZOL AND SACCHARIDS SUCH AS MANNITOL, XYLITOL, AMONG OTHERS IN THE FORM OF GRANULATED PARTICLES THAT ARE PREPARED BY A UNIQUE DISPERSION, A UNDEFINANT DISPERSION AND INTO A SUBSTANT DISPERSION. (a) THE SACCHARDS IS FOUND IN 40-90 PARTS BY WEIGHT, (b) THE INORGANIC SUBSTANCE IS FOUND IN 1-30 PARTS BY WEIGHT AND (c) THE DISINTEGRANT AGENT IS FOUND IN 5-40 PARTS BY WEIGHT; B) A SLIPPER SUCH AS HYDRAATED SILICON DIOXIDE, LIGHT AND HEAVY ANHYDROUS SILICONE ACID, WHICH IS IN A QUANTITY OF 0.2% TO 2% (p / p); C) AN ORGANIC EXCIPIENT SUCH AS CORN STARCH, CRYSTALINE CELLULOSE, AMONG OTHERS; D) ONE OR MORE OPTIONAL ADDITIVES SUCH AS LUBRICANTS, SWEETENERS, AROMATIZERS, AMONG OTHERS. SAID COMPRESSED IS USEFUL FOR OLDER PATIENTS AND PATIENTS SUFFERING FROM DYSPHAGIA
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2008050460 | 2008-02-29 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20091560A1 true PE20091560A1 (en) | 2009-10-30 |
Family
ID=40718911
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2009000311A PE20091560A1 (en) | 2008-02-29 | 2009-02-27 | ORAL DISINTEGRATION TABLET |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP2262487A2 (en) |
JP (1) | JP2011513194A (en) |
AR (1) | AR070530A1 (en) |
CL (1) | CL2009000452A1 (en) |
PE (1) | PE20091560A1 (en) |
TW (1) | TW200936184A (en) |
WO (1) | WO2009107864A2 (en) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8779146B2 (en) | 2010-04-28 | 2014-07-15 | Nuformix Limited | Cilostazol cocrystals and compositions |
ES2422657B1 (en) * | 2012-02-10 | 2014-06-11 | Laboratorios Normon S.A. | Cilostazol solid pharmaceutical composition |
US9988542B2 (en) | 2012-07-20 | 2018-06-05 | Otsuka Pharmaceutical Co., Ltd. | Tablet having dry-ink film on surface thereof, and ink for inkjet printer |
JP5713421B1 (en) | 2013-07-19 | 2015-05-07 | 株式会社三和化学研究所 | Orally disintegrating tablets |
US9974738B2 (en) | 2013-09-27 | 2018-05-22 | Daicel Corporation | Disintegrating particle composition produced by two-stage wet granulation process, and intraorally disintegrating tablet containing same composition |
US10231914B2 (en) * | 2015-06-02 | 2019-03-19 | Lynette Batton | Effervescent tablet for elimination of red wine discoloration, offensive odour of mouth and cleaning the palate |
EP3409294A1 (en) | 2017-06-01 | 2018-12-05 | Przedsiebiorstwo Farmaceutyczne Lek-Am Sp Z O. O. | Tablets containing cilostazol of specific particle size distribution |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6548490B1 (en) * | 1997-10-28 | 2003-04-15 | Vivus, Inc. | Transmucosal administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction |
AU2001248751A1 (en) * | 2000-04-12 | 2001-10-23 | Banyu Pharmaceutical Co. Ltd. | Compositions disintegrating in oral cavity and preparations disintegrating in oral cavity |
JP4637338B2 (en) * | 2000-09-22 | 2011-02-23 | 大塚製薬株式会社 | Cilostazol dry coated tablets |
JP4551627B2 (en) * | 2003-02-28 | 2010-09-29 | 東和薬品株式会社 | Method for producing orally disintegrating tablets |
JP3841804B2 (en) * | 2003-10-15 | 2006-11-08 | 富士化学工業株式会社 | Composition for intraorally rapidly disintegrating tablets |
KR101159617B1 (en) * | 2003-10-15 | 2012-06-27 | 후지카가쿠고교가부시키가이샤 | Tablet quickly disintegrating in oral cavity |
TWI383809B (en) * | 2005-06-29 | 2013-02-01 | Otsuka Pharma Co Ltd | Orally disintegrating powder comprising cilostazol |
JP5074190B2 (en) * | 2005-09-02 | 2012-11-14 | 富士化学工業株式会社 | Orally rapidly disintegrating tablets |
-
2009
- 2009-02-26 JP JP2010504975A patent/JP2011513194A/en active Pending
- 2009-02-26 EP EP09714454A patent/EP2262487A2/en not_active Withdrawn
- 2009-02-26 WO PCT/JP2009/054115 patent/WO2009107864A2/en active Application Filing
- 2009-02-27 PE PE2009000311A patent/PE20091560A1/en not_active Application Discontinuation
- 2009-02-27 TW TW098106341A patent/TW200936184A/en unknown
- 2009-02-27 CL CL2009000452A patent/CL2009000452A1/en unknown
- 2009-02-27 AR ARP090100682A patent/AR070530A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
TW200936184A (en) | 2009-09-01 |
JP2011513194A (en) | 2011-04-28 |
WO2009107864A2 (en) | 2009-09-03 |
AR070530A1 (en) | 2010-04-14 |
CL2009000452A1 (en) | 2010-03-26 |
EP2262487A2 (en) | 2010-12-22 |
WO2009107864A3 (en) | 2009-12-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application declared void or lapsed |