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Application filed by Hoffmann La RochefiledCriticalHoffmann La Roche
Publication of PA8535701A1publicationCriticalpatent/PA8535701A1/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A COMPUESTOS QUIMICOS DE FORMULA (I) TANTO COMO A SALES FARMACEUTICAMENTE UTILIZABLES, SOLVATOS Y ESTERES DE LOS MISMOS, EN DONDE R1 A R4 Y n POSEEN EL SIGNIFICADO DADO EN LA REIVINDICACION 1. PUEDEN SER USADOS EN FORMA DE PREPARACIONES FARMACEUTICAS PARA EL TRATAMIENTO O PREVENCION DE TRASTORNOS DEL SISTEMA NERVIOSO CENTRAL, TRASTORNOS CARDIOVASCULARES, TRASTORNOS GASTROINTESTINALES, DIABETES, OBESIDAD Y APNES DURANTE EL SUEÑO.THE PRESENT INVENTION REFERS TO CHEMICAL COMPOUNDS OF FORMULA (I) BOTH AS AS TO PHARMACEUTICALLY USED, SOLVATOS AND STERES SALTS OF THE SAME, WHERE R1 TO R4 AND N HAVE THE MEANING GIVEN IN THE CLAIM 1. CAN BE PREPARED IN USE PHARMACEUTICS FOR THE TREATMENT OR PREVENTION OF DISORDERS OF THE CENTRAL NERVOUS SYSTEM, CARDIOVASCULAR DISORDERS, GASTROINTESTINAL DISORDERS, DIABETES, OBESITY AND APNES DURING THE SLEEP.
PA8535701A2000-12-272001-12-21
DERIVATIVES OF INDOL
PA8535701A1
(en)
A COMPOUND DERIVED FROM PIRAZINOINDOL, USE OF THE SAME, A PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND A METHOD FOR THE MANUFACTURE OF SUCH COMPOSITION