PA8501901A1 - FUSIONATED PIRROLCARBOXAMIDS; A NEW CLASS CLASS OF GABA CEREBRAL RECEPTORS. - Google Patents
FUSIONATED PIRROLCARBOXAMIDS; A NEW CLASS CLASS OF GABA CEREBRAL RECEPTORS.Info
- Publication number
- PA8501901A1 PA8501901A1 PA8501901A PA8501901A PA8501901A1 PA 8501901 A1 PA8501901 A1 PA 8501901A1 PA 8501901 A PA8501901 A PA 8501901A PA 8501901 A PA8501901 A PA 8501901A PA 8501901 A1 PA8501901 A1 PA 8501901A1
- Authority
- PA
- Panama
- Prior art keywords
- class
- compounds
- agonists
- cerebral
- pirrolcarboxamids
- Prior art date
Links
Abstract
SE TRATA DE COMPUESTOS DE PIRROLCARBOXAMIDA SUSTITUIDOS. ESTOS COMPUESTOS SON AGONISTAS, ANTAGONISTAS O AGONISTAS INVERSOS ALTAMENTE SELECTIVOS DE LOS RECEPTORES CEREBRALES GABAa O PRODROGAS DE LOS AGONISTAS, ANTAGONISTAS O AGONISTAS INVERSOS DE LOS RECEPTORES CEREBRALES GABAa. POR LO TANTO, SON UTILES EN EL DIAGNOSTICO Y TRATAMIENTO DE ANSIEDAD, DEPRESION, DEMENCIA CAUSADA POR LA ENFERMEDAD DE ALZHEIMER, TRASTORNOS DEL SUEÑO Y CONVULSIVOS, SOBREDOSIS CON BENZODIAZEPINAS Y PARA MEJORAR LA MEMORIA. TAMBIEN EXISTEN COMPUESTOS FARMACEUTICOS, INCLUIDOS COMPUESTOS FARMACEUTICOS ENVASADOS. LOS COMPUESTOS DEL INVENTO TAMBIEN SON UTILES COMO PRUEBAS PARA LA LOCALIZACION DE RECEPTORES GABAa EN MUESTRAS DE TEJIDOS.IT IS ABOUT REPLACED PIRROLCARBOXAMIDE COMPOUNDS. THESE COMPOUNDS ARE AGONISTS, ANTAGONISTS OR HIGHLY SELECTIVE INVESTED AGONISTS OF THE GABAa CEREBRAL RECEIVERS OR PRODROGES OF THE AGONISTS, ANTAGONISTS OR INVESTED AGONISTS OF THE GABAa CEREBRAL RECEIVERS. THEREFORE, THEY ARE USEFUL IN THE DIAGNOSIS AND TREATMENT OF ANXIETY, DEPRESSION, DEMENTIA CAUSED BY ALZHEIMER'S DISEASE, SLEEP AND CONVULSIVE DISORDERS, OVERDOSE WITH BENZODIAZEPINAS AND TO IMPROVE MEMORY. THERE ARE ALSO PHARMACEUTICAL COMPOUNDS, INCLUDING PACKAGED PHARMACEUTICAL COMPOUNDS. THE COMPOUNDS OF THE INVENTION ARE ALSO USEFUL AS TESTS FOR THE LOCATION OF GABAa RECEPTORS IN FABRIC SAMPLES.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38731199A | 1999-08-31 | 1999-08-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PA8501901A1 true PA8501901A1 (en) | 2002-12-11 |
Family
ID=27805344
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PA8501901A PA8501901A1 (en) | 1999-08-31 | 2000-08-31 | FUSIONATED PIRROLCARBOXAMIDS; A NEW CLASS CLASS OF GABA CEREBRAL RECEPTORS. |
Country Status (10)
| Country | Link |
|---|---|
| AR (1) | AR040397A1 (en) |
| CO (1) | CO5180633A1 (en) |
| EC (1) | ECSP003641A (en) |
| GT (1) | GT200000146A (en) |
| PA (1) | PA8501901A1 (en) |
| PE (1) | PE20010533A1 (en) |
| SV (1) | SV2002000161A (en) |
| TN (1) | TNSN00178A1 (en) |
| UY (1) | UY26322A1 (en) |
| ZA (1) | ZA200201649B (en) |
-
2000
- 2000-08-30 TN TNTNSN00178A patent/TNSN00178A1/en unknown
- 2000-08-31 CO CO00065554A patent/CO5180633A1/en unknown
- 2000-08-31 EC ECSP003641 patent/ECSP003641A/en unknown
- 2000-08-31 AR ARP000104564 patent/AR040397A1/en not_active Application Discontinuation
- 2000-08-31 PE PE2000000891A patent/PE20010533A1/en not_active Application Discontinuation
- 2000-08-31 UY UY26322A patent/UY26322A1/en not_active Application Discontinuation
- 2000-08-31 GT GT200000146A patent/GT200000146A/en unknown
- 2000-08-31 PA PA8501901A patent/PA8501901A1/en unknown
- 2000-08-31 SV SV2000000161A patent/SV2002000161A/en unknown
-
2002
- 2002-02-27 ZA ZA200201649A patent/ZA200201649B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| UY26322A1 (en) | 2001-06-29 |
| SV2002000161A (en) | 2002-09-04 |
| CO5180633A1 (en) | 2002-07-30 |
| ECSP003641A (en) | 2002-03-25 |
| PE20010533A1 (en) | 2001-05-01 |
| ZA200201649B (en) | 2003-05-28 |
| AR040397A1 (en) | 2005-04-06 |
| GT200000146A (en) | 2002-02-22 |
| TNSN00178A1 (en) | 2002-05-30 |
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