NO982709L - Process for Preparation of S- (R, R *) | -3-Methyl-2 (3-oxo-3H-benzoic acid) -thiazol-2-yl) pentaenoic acid and S- (R, R *) | , L-2- {2- £ 2- (1-carboxy-2-methylbutylcarbamoyl) phenyldisulfonyl | benzoylamino-3-metylpentaensyre - Google Patents
Process for Preparation of S- (R, R *) | -3-Methyl-2 (3-oxo-3H-benzoic acid) -thiazol-2-yl) pentaenoic acid and S- (R, R *) | , L-2- {2- £ 2- (1-carboxy-2-methylbutylcarbamoyl) phenyldisulfonyl | benzoylamino-3-metylpentaensyreInfo
- Publication number
- NO982709L NO982709L NO982709A NO982709A NO982709L NO 982709 L NO982709 L NO 982709L NO 982709 A NO982709 A NO 982709A NO 982709 A NO982709 A NO 982709A NO 982709 L NO982709 L NO 982709L
- Authority
- NO
- Norway
- Prior art keywords
- phenyldisulfonyl
- methylbutylcarbamoyl
- benzoylamino
- oxo
- carboxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
- C07C319/22—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of hydropolysulfides or polysulfides
- C07C319/24—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of hydropolysulfides or polysulfides by reactions involving the formation of sulfur-to-sulfur bonds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Foreliggende oppfinnelse tilveiebringer en forbedret syntese av [S-(R*,R*)]-3-metyl-2-(3-okso-3H-benzo[d]isotiazol-2-yl)pentansyreog [S-(R*,R*)],L-2-{2-[2-(1-karboksy-2-metylbutylkarbamoyl)fenyldisulfonyl]- benzoylamino}-3-metylpentansyre.The present invention provides an improved synthesis of [S- (R *, R *)] - 3-methyl-2- (3-oxo-3H-benzo [d] isothiazol-2-yl) pentanoic acid and [S- (R *, R *)], L-2- {2- [2- (1-carboxy-2-methylbutylcarbamoyl) phenyldisulfonyl] benzoylamino} -3-methylpentanoic acid.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US874595P | 1995-12-15 | 1995-12-15 | |
PCT/US1996/018929 WO1997022598A1 (en) | 1995-12-15 | 1996-11-27 | Method of making (s-(r*,r*))-3-methyl-2-(3-oxo-3h-benzo(d)isothiazol-2-yl)pentanoic acid and (s-(r*,r*)), l-2-(2-(2-(1-carboxy-2-methylbutylcarbamoyl)phenyldisulfonyl)benzoyl-amino)-3-methylpentanoic acid |
Publications (2)
Publication Number | Publication Date |
---|---|
NO982709D0 NO982709D0 (en) | 1998-06-12 |
NO982709L true NO982709L (en) | 1998-06-12 |
Family
ID=21733413
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO982709A NO982709L (en) | 1995-12-15 | 1998-06-12 | Process for Preparation of S- (R, R *) | -3-Methyl-2 (3-oxo-3H-benzoic acid) -thiazol-2-yl) pentaenoic acid and S- (R, R *) | , L-2- {2- £ 2- (1-carboxy-2-methylbutylcarbamoyl) phenyldisulfonyl | benzoylamino-3-metylpentaensyre |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP0874835A1 (en) |
JP (1) | JP2000505067A (en) |
KR (1) | KR20000064403A (en) |
CN (1) | CN1208407A (en) |
AU (1) | AU1083597A (en) |
BG (1) | BG102470A (en) |
BR (1) | BR9612020A (en) |
CA (1) | CA2233553A1 (en) |
CZ (1) | CZ182498A3 (en) |
HU (1) | HUP9902043A3 (en) |
IL (1) | IL123903A0 (en) |
NO (1) | NO982709L (en) |
NZ (1) | NZ323803A (en) |
PL (1) | PL327135A1 (en) |
SK (1) | SK81798A3 (en) |
WO (1) | WO1997022598A1 (en) |
ZA (1) | ZA9610479B (en) |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9304903D0 (en) * | 1993-03-10 | 1993-04-28 | Zeneca Ltd | Compounds,preparation and use |
US5734081A (en) * | 1994-08-05 | 1998-03-31 | Warner-Lambert Company | Arylthio compounds |
US5463122A (en) * | 1994-08-05 | 1995-10-31 | Warner-Lambert Company | Arylthio compounds |
-
1996
- 1996-11-27 PL PL96327135A patent/PL327135A1/en unknown
- 1996-11-27 JP JP9522815A patent/JP2000505067A/en active Pending
- 1996-11-27 CA CA002233553A patent/CA2233553A1/en not_active Abandoned
- 1996-11-27 EP EP96940880A patent/EP0874835A1/en not_active Withdrawn
- 1996-11-27 IL IL12390396A patent/IL123903A0/en unknown
- 1996-11-27 NZ NZ323803A patent/NZ323803A/en unknown
- 1996-11-27 AU AU10835/97A patent/AU1083597A/en not_active Abandoned
- 1996-11-27 BR BR9612020A patent/BR9612020A/en not_active Application Discontinuation
- 1996-11-27 WO PCT/US1996/018929 patent/WO1997022598A1/en not_active Application Discontinuation
- 1996-11-27 SK SK817-98A patent/SK81798A3/en unknown
- 1996-11-27 CZ CZ981824A patent/CZ182498A3/en unknown
- 1996-11-27 CN CN96199009A patent/CN1208407A/en active Pending
- 1996-11-27 HU HU9902043A patent/HUP9902043A3/en unknown
- 1996-11-27 KR KR1019980704461A patent/KR20000064403A/en not_active Application Discontinuation
- 1996-12-12 ZA ZA9610479A patent/ZA9610479B/en unknown
-
1998
- 1998-05-20 BG BG102470A patent/BG102470A/en unknown
- 1998-06-12 NO NO982709A patent/NO982709L/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
NO982709D0 (en) | 1998-06-12 |
JP2000505067A (en) | 2000-04-25 |
IL123903A0 (en) | 1998-10-30 |
HUP9902043A2 (en) | 1999-11-29 |
SK81798A3 (en) | 1998-11-04 |
BG102470A (en) | 1999-08-31 |
KR20000064403A (en) | 2000-11-06 |
HUP9902043A3 (en) | 2000-03-28 |
AU1083597A (en) | 1997-07-14 |
CA2233553A1 (en) | 1997-06-26 |
PL327135A1 (en) | 1998-11-23 |
NZ323803A (en) | 1999-02-25 |
CZ182498A3 (en) | 1998-09-16 |
CN1208407A (en) | 1999-02-17 |
EP0874835A1 (en) | 1998-11-04 |
WO1997022598A1 (en) | 1997-06-26 |
ZA9610479B (en) | 1998-06-09 |
BR9612020A (en) | 1999-06-29 |
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Legal Events
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FC2A | Withdrawal, rejection or dismissal of laid open patent application |