NO944487D0 - 8-klor-11[1-[(5-metyl-3-pyridyl)metylÅ-4-piperidylidenÅ-6,11-dihydro-5H-benzo[5,6Åsyklohepta-[1,2-bÅpyridinfumarat - Google Patents

8-klor-11[1-[(5-metyl-3-pyridyl)metylÅ-4-piperidylidenÅ-6,11-dihydro-5H-benzo[5,6Åsyklohepta-[1,2-bÅpyridinfumarat

Info

Publication number
NO944487D0
NO944487D0 NO944487A NO944487A NO944487D0 NO 944487 D0 NO944487 D0 NO 944487D0 NO 944487 A NO944487 A NO 944487A NO 944487 A NO944487 A NO 944487A NO 944487 D0 NO944487 D0 NO 944487D0
Authority
NO
Norway
Prior art keywords
piperidylidenå
metylå
båpyridinfumarat
benzo
pyridyl
Prior art date
Application number
NO944487A
Other languages
English (en)
Other versions
NO944487L (no
NO305436B1 (no
Inventor
Elena Carceller
Nuria Recasens
Carmen Almansa
Javier Bartroli
Manel Merlos
Marta Giral
Julian Garcia-Rafanell
Javier Forn
Original Assignee
Uriach & Cia Sa J
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Uriach & Cia Sa J filed Critical Uriach & Cia Sa J
Publication of NO944487D0 publication Critical patent/NO944487D0/no
Publication of NO944487L publication Critical patent/NO944487L/no
Publication of NO305436B1 publication Critical patent/NO305436B1/no

Links

NO944487A 1993-11-24 1994-11-23 8-klor-11-[1-[(5-metyl-3-pyridyl)metyl]-4-piperidyliden]-6,11-dihydro-5H-benzo[5,6]syklohepta[1,2-b]pyridin-fumarat, fremgangsmÕte for fremstilling derav, farmas°ytisk preparat som omfatter det, samt anvendelse av forbindelsen for fremstilling a NO305436B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES09302460A ES2087818B1 (es) 1993-11-24 1993-11-24 8-cloro-11-(1-((5-metil-3-piridil)metil)-4-piperidiliden)-6,11-dihidro-5h-benzo-(5,6)cicloheptal(1,2-b)piridina, fumarato.

Publications (3)

Publication Number Publication Date
NO944487D0 true NO944487D0 (no) 1994-11-23
NO944487L NO944487L (no) 1995-05-26
NO305436B1 NO305436B1 (no) 1999-05-31

Family

ID=8283716

Family Applications (2)

Application Number Title Priority Date Filing Date
NO944487A NO305436B1 (no) 1993-11-24 1994-11-23 8-klor-11-[1-[(5-metyl-3-pyridyl)metyl]-4-piperidyliden]-6,11-dihydro-5H-benzo[5,6]syklohepta[1,2-b]pyridin-fumarat, fremgangsmÕte for fremstilling derav, farmas°ytisk preparat som omfatter det, samt anvendelse av forbindelsen for fremstilling a
NO2014001C NO2014001I2 (no) 1993-11-24 2014-01-23 Rupatadin fumarat

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO2014001C NO2014001I2 (no) 1993-11-24 2014-01-23 Rupatadin fumarat

Country Status (2)

Country Link
ES (1) ES2087818B1 (no)
NO (2) NO305436B1 (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2120899B1 (es) * 1996-10-07 1999-06-16 Uriach & Cia Sa J Procedimiento para la preparacion de la 8-cloro-6, 11-dihidro-11-(1-(5-metil-3-piridinil)metil)-4-piperidinilideno)-5h-benzo(5,6) ciclohepta (1,2-b)piridina.
ES2311426B1 (es) * 2005-04-27 2009-12-22 Cadila Pharmaceuticals Limited Un procedimiento para la preparacion de rupatadina y sus sales.
CN101531654B (zh) * 2009-04-13 2013-07-17 浙江赐富医药有限公司 一种卢帕他定的制备方法
WO2012001120A1 (en) 2010-06-30 2012-01-05 J. Uriach Y Compañía, S.A. Rupatadine salt as an antihistaminic agent
CA2798028A1 (en) 2010-06-30 2012-01-05 J. Uriach Y Compania S.A. Liquid formulations of rupatadine fumarate
CN102807562A (zh) * 2012-07-31 2012-12-05 东莞达信生物技术有限公司 一种卢帕他定及其盐的制备方法
CN103804357B (zh) * 2014-01-02 2016-03-23 珠海金鸿药业股份有限公司 一种富马酸卢帕他定化合物,其合成方法及其药物组合物
CN109734702B (zh) * 2019-03-01 2020-07-03 南京工业大学 一种采用微通道反应装置制备富马酸卢帕他定的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4826853A (en) * 1986-10-31 1989-05-02 Schering Corporation 6,11-Dihydro-11-(N-substituted-4-piperidylidene)-5H-benzo(5,6)cyclohepta(1,2-B)pyridines and compositions and methods of use
US5089496A (en) * 1986-10-31 1992-02-18 Schering Corporation Benzo[5,6]cycloheptapyridine compounds, compositions and method of treating allergies
IL98572A (en) * 1990-06-22 1995-07-31 Schering Corp Bite-benzo or benzopyrido compounds Cyclohepta piperidine, piperidylidene and piperazine, preparations and methods of use.
ES2042421B1 (es) * 1992-05-22 1994-08-01 Uriach & Cia Sa J Procedimiento para la obtencion de la 8-cloro-11-*1-*(5-metil-3-piridil)metil*-4-piperidiliden*-6,11-dihidro-5h-benzo*5,6*ciclohepta*1,2-b*piridina.

Also Published As

Publication number Publication date
NO944487L (no) 1995-05-26
ES2087818A1 (es) 1996-07-16
NO305436B1 (no) 1999-05-31
NO2014001I1 (no) 2014-06-02
ES2087818B1 (es) 1997-03-16
NO2014001I2 (no) 2015-08-24

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Legal Events

Date Code Title Description
CHAD Change of the owner's name or address (par. 44 patent law, par. patentforskriften)

Owner name: J URIACH Y COMPANIA SA, ES

MK1K Patent expired
SPCG Granted supplementary protection certificate

Free format text: PRODUCT NAME: RUPAFIN, 10 MG TABLETTER; REG.NO/DATE: 13-9499 2013.10.21; FIRST REG.NO/DATE: 16630 2001.07.04

Spc suppl protection certif: 2014001

Filing date: 20140123

Extension date: 20160704