NO863944D0 - L-DOPA DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL MIXTURE CONTAINING THESE DERIVATIVES. - Google Patents
L-DOPA DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL MIXTURE CONTAINING THESE DERIVATIVES.Info
- Publication number
- NO863944D0 NO863944D0 NO863944A NO863944A NO863944D0 NO 863944 D0 NO863944 D0 NO 863944D0 NO 863944 A NO863944 A NO 863944A NO 863944 A NO863944 A NO 863944A NO 863944 D0 NO863944 D0 NO 863944D0
- Authority
- NO
- Norway
- Prior art keywords
- derivatives
- procedure
- preparation
- mixture containing
- dopa
- Prior art date
Links
- WTDRDQBEARUVNC-LURJTMIESA-N L-DOPA Chemical class OC(=O)[C@@H](N)CC1=CC=C(O)C(O)=C1 WTDRDQBEARUVNC-LURJTMIESA-N 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LU85757A LU85757A1 (en) | 1985-02-04 | 1985-02-04 | NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS |
PCT/BE1986/000002 WO1986004579A1 (en) | 1985-02-04 | 1986-01-27 | L-dopa derivatives, preparation thereof and pharmaceutical compositions containing them |
Publications (2)
Publication Number | Publication Date |
---|---|
NO863944D0 true NO863944D0 (en) | 1986-10-03 |
NO863944L NO863944L (en) | 1986-12-01 |
Family
ID=19730402
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO863944A NO863944L (en) | 1985-02-04 | 1986-10-03 | L-DOPA DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL MIXTURE CONTAINING THESE DERIVATIVES. |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP0250403A1 (en) |
JP (1) | JPS63501498A (en) |
DK (1) | DK437586D0 (en) |
FI (1) | FI871270A0 (en) |
LU (1) | LU85757A1 (en) |
NO (1) | NO863944L (en) |
WO (1) | WO1986004579A1 (en) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19631189A1 (en) * | 1996-08-02 | 1998-02-05 | Max Delbrueck Centrum | Novel cationic amphiphiles for liposomal gene transfer |
US7323585B2 (en) | 2004-06-04 | 2008-01-29 | Xenoport, Inc. | Levodopa prodrugs, and compositions and uses thereof |
MX339690B (en) * | 2004-06-04 | 2016-06-06 | Xenoport Inc | Levodopa prodrugs, and compositions and uses thereof. |
US7563821B2 (en) | 2005-12-05 | 2009-07-21 | Xenoport, Inc. | Levodopa prodrug mesylate, compositions thereof, and uses thereof |
JP2011502953A (en) | 2006-12-21 | 2011-01-27 | ゼノポート,インコーポレーテッド | Prodrugs, compositions and methods of use of dimethyl substituted levodopa diesters |
TW200843731A (en) * | 2006-12-21 | 2008-11-16 | Xenoport Inc | Catechol protected levodopa diester prodrugs, compositions, and methods of use |
US9290445B2 (en) | 2008-10-20 | 2016-03-22 | Xenoport, Inc. | Methods of synthesizing a levodopa ester prodrug |
US8399513B2 (en) | 2008-10-20 | 2013-03-19 | Xenoport, Inc. | Levodopa prodrug mesylate hydrate |
GB0904300D0 (en) * | 2009-03-12 | 2009-04-22 | Amarin Neuroscience Ltd | Essential fatty acid compounds |
JP2013520521A (en) | 2009-11-09 | 2013-06-06 | ゼノポート,インコーポレーテッド | Pharmaceutical composition and oral dosage form of levodopa prodrug and method of use |
JP2013043885A (en) * | 2011-08-26 | 2013-03-04 | Kansai Bunri Sogo Gakuen | Dehydroamino acid-containing glycerol derivative |
EP3277660B1 (en) * | 2015-03-30 | 2019-10-16 | Berlirem GmbH | Water-soluble l-dopa esters |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE7605911L (en) * | 1975-06-11 | 1976-12-12 | Merck & Co Inc | IMPROVED PROCEDURE FOR MAKING ESTRARS OF ALFA-METHYL-3,4-DIHYDROXYPHENYLALANINE |
FR2365341A1 (en) * | 1976-09-28 | 1978-04-21 | Synthelabo | L- (PHENYL-3 AMINO-2 PROPIONYLOXY) -2 ACETIC DERIVATIVES |
GR72800B (en) * | 1979-12-17 | 1983-12-05 | Merck & Co Inc | |
US4360533A (en) * | 1981-12-14 | 1982-11-23 | Merck & Co., Inc. | Glyceryl ester of 1-methyl-2-(3,4-dihydroxyphenyl)alanine |
-
1985
- 1985-02-04 LU LU85757A patent/LU85757A1/en unknown
-
1986
- 1986-01-27 JP JP61500751A patent/JPS63501498A/en active Pending
- 1986-01-27 EP EP86900721A patent/EP0250403A1/en not_active Withdrawn
- 1986-01-27 WO PCT/BE1986/000002 patent/WO1986004579A1/en not_active Application Discontinuation
- 1986-09-12 DK DK437586A patent/DK437586D0/en not_active Application Discontinuation
- 1986-10-03 NO NO863944A patent/NO863944L/en unknown
-
1987
- 1987-03-23 FI FI871270A patent/FI871270A0/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
WO1986004579A1 (en) | 1986-08-14 |
EP0250403A1 (en) | 1988-01-07 |
LU85757A1 (en) | 1986-09-02 |
JPS63501498A (en) | 1988-06-09 |
NO863944L (en) | 1986-12-01 |
FI871270A (en) | 1987-03-23 |
DK437586A (en) | 1986-09-12 |
DK437586D0 (en) | 1986-09-12 |
FI871270A0 (en) | 1987-03-23 |
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