LU85757A1 - NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS - Google Patents

NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS Download PDF

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Publication number
LU85757A1
LU85757A1 LU85757A LU85757A LU85757A1 LU 85757 A1 LU85757 A1 LU 85757A1 LU 85757 A LU85757 A LU 85757A LU 85757 A LU85757 A LU 85757A LU 85757 A1 LU85757 A1 LU 85757A1
Authority
LU
Luxembourg
Prior art keywords
novel
compounds
preparation
methods
pharmaceutical compositions
Prior art date
Application number
LU85757A
Other languages
French (fr)
Inventor
Pierre Dumont
Original Assignee
Univ Catholique Louvain
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Catholique Louvain filed Critical Univ Catholique Louvain
Priority to LU85757A priority Critical patent/LU85757A1/en
Priority to PCT/BE1986/000002 priority patent/WO1986004579A1/en
Priority to EP86900721A priority patent/EP0250403A1/en
Priority to JP61500751A priority patent/JPS63501498A/en
Publication of LU85757A1 publication Critical patent/LU85757A1/en
Priority to DK437586A priority patent/DK437586A/en
Priority to NO863944A priority patent/NO863944L/en
Priority to FI871270A priority patent/FI871270A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
LU85757A 1985-02-04 1985-02-04 NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS LU85757A1 (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
LU85757A LU85757A1 (en) 1985-02-04 1985-02-04 NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS
PCT/BE1986/000002 WO1986004579A1 (en) 1985-02-04 1986-01-27 L-dopa derivatives, preparation thereof and pharmaceutical compositions containing them
EP86900721A EP0250403A1 (en) 1985-02-04 1986-01-27 L-dopa derivatives, preparation thereof and pharmaceutical compositions containing them
JP61500751A JPS63501498A (en) 1985-02-04 1986-01-27 Novel derivative of L-dopa, its production method and pharmaceutical composition containing it
DK437586A DK437586A (en) 1985-02-04 1986-09-12 NEW L-DOPA DERIVATIVES, PROCEDURES FOR PREPARING THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH RELATIONSHIPS
NO863944A NO863944L (en) 1985-02-04 1986-10-03 L-DOPA DERIVATIVES, THE PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL MIXTURE CONTAINING THESE DERIVATIVES.
FI871270A FI871270A (en) 1985-02-04 1987-03-23 L-DOPA DERIVATIVES, FOERFARANDE FOER FRAMSTAELLNING AV DEM OCH PHARMACEUTICAL SAMMANSAETTNINGAR SOM INNEHAOLLER DEM.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
LU85757A LU85757A1 (en) 1985-02-04 1985-02-04 NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS

Publications (1)

Publication Number Publication Date
LU85757A1 true LU85757A1 (en) 1986-09-02

Family

ID=19730402

Family Applications (1)

Application Number Title Priority Date Filing Date
LU85757A LU85757A1 (en) 1985-02-04 1985-02-04 NOVEL L-DOPA DERIVATIVES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS RELATING TO SUCH COMPOUNDS

Country Status (7)

Country Link
EP (1) EP0250403A1 (en)
JP (1) JPS63501498A (en)
DK (1) DK437586A (en)
FI (1) FI871270A (en)
LU (1) LU85757A1 (en)
NO (1) NO863944L (en)
WO (1) WO1986004579A1 (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19631189A1 (en) * 1996-08-02 1998-02-05 Max Delbrueck Centrum Novel cationic amphiphiles for liposomal gene transfer
ZA200610042B (en) 2004-06-04 2008-06-25 Xenoport Inc Levodopa prodrugs, and compositions and uses thereof
WO2005121070A1 (en) 2004-06-04 2005-12-22 Xenoport, Inc. Levodopa prodrugs, and compositions and uses thereof
WO2007067495A2 (en) 2005-12-05 2007-06-14 Xenoport, Inc. Levodopa prodrug mesylate, compositions thereof, and uses thereof
WO2008076458A1 (en) 2006-12-21 2008-06-26 Xenoport, Inc. Levodopa dimethyl-substituted diester prodrugs, compositions, and methods of use
US7829592B2 (en) 2006-12-21 2010-11-09 Xenoport, Inc. Catechol protected levodopa diester prodrugs, compositions, and methods of use
CN102186804A (en) 2008-10-20 2011-09-14 克塞诺波特公司 Methods of synthesizing a levodopa ester prodrug
US8399513B2 (en) 2008-10-20 2013-03-19 Xenoport, Inc. Levodopa prodrug mesylate hydrate
GB0904300D0 (en) * 2009-03-12 2009-04-22 Amarin Neuroscience Ltd Essential fatty acid compounds
ES2565644T3 (en) 2009-11-09 2016-04-06 Xenoport, Inc. Pharmaceutical compositions and oral dosage forms of a levodopa pre-medication and methods of use
JP2013043885A (en) * 2011-08-26 2013-03-04 Kansai Bunri Sogo Gakuen Dehydroamino acid-containing glycerol derivative
AU2016239274A1 (en) * 2015-03-30 2017-11-02 Berlirem Gmbh Water-soluble L-DOPA esters
EP3852722A4 (en) * 2018-10-08 2022-08-03 Cellix Bio Private Limited Compositions and methods for the treatment of parkinson's disease

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7605911L (en) * 1975-06-11 1976-12-12 Merck & Co Inc IMPROVED PROCEDURE FOR MAKING ESTRARS OF ALFA-METHYL-3,4-DIHYDROXYPHENYLALANINE
FR2365341A1 (en) * 1976-09-28 1978-04-21 Synthelabo L- (PHENYL-3 AMINO-2 PROPIONYLOXY) -2 ACETIC DERIVATIVES
GR72800B (en) * 1979-12-17 1983-12-05 Merck & Co Inc
US4360533A (en) * 1981-12-14 1982-11-23 Merck & Co., Inc. Glyceryl ester of 1-methyl-2-(3,4-dihydroxyphenyl)alanine

Also Published As

Publication number Publication date
WO1986004579A1 (en) 1986-08-14
DK437586D0 (en) 1986-09-12
FI871270A0 (en) 1987-03-23
JPS63501498A (en) 1988-06-09
FI871270A (en) 1987-03-23
NO863944D0 (en) 1986-10-03
NO863944L (en) 1986-12-01
EP0250403A1 (en) 1988-01-07
DK437586A (en) 1986-09-12

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