NO325958B1 - Enantiomert rent opioid diarylmetylpiperazin samt anvendelse derav - Google Patents
Enantiomert rent opioid diarylmetylpiperazin samt anvendelse derav Download PDFInfo
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- NO325958B1 NO325958B1 NO20041729A NO20041729A NO325958B1 NO 325958 B1 NO325958 B1 NO 325958B1 NO 20041729 A NO20041729 A NO 20041729A NO 20041729 A NO20041729 A NO 20041729A NO 325958 B1 NO325958 B1 NO 325958B1
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- compound
- allyl
- piperazinyl
- thienyl
- phenol
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Psychiatry (AREA)
- Dermatology (AREA)
- Hospice & Palliative Care (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Transplantation (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Otolaryngology (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Investigating Or Analysing Biological Materials (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US32471201P | 2001-09-25 | 2001-09-25 | |
| PCT/US2002/030398 WO2003026660A1 (en) | 2001-09-25 | 2002-09-25 | An enantiomerically pure diarylmethylpiperazine and methods of using same |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20041729L NO20041729L (no) | 2004-06-25 |
| NO325958B1 true NO325958B1 (no) | 2008-08-25 |
Family
ID=23264757
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20041729A NO325958B1 (no) | 2001-09-25 | 2004-04-23 | Enantiomert rent opioid diarylmetylpiperazin samt anvendelse derav |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US6924288B2 (pt) |
| EP (1) | EP1438051A4 (pt) |
| JP (1) | JP2005505575A (pt) |
| KR (1) | KR20040041171A (pt) |
| CN (1) | CN1558765B (pt) |
| AU (1) | AU2002341832B2 (pt) |
| BR (1) | BR0212742A (pt) |
| CA (1) | CA2459577C (pt) |
| IL (2) | IL160794A0 (pt) |
| MX (1) | MXPA04002813A (pt) |
| NO (1) | NO325958B1 (pt) |
| NZ (1) | NZ531875A (pt) |
| PL (1) | PL370346A1 (pt) |
| RU (1) | RU2309153C2 (pt) |
| WO (1) | WO2003026660A1 (pt) |
| ZA (1) | ZA200402325B (pt) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7189725B2 (en) * | 2001-09-25 | 2007-03-13 | Mount Cook Biosciences, Inc. | Enantiomerically pure opioid diarylmethylpiperazine as a cardioprotection agent |
| US7314880B2 (en) * | 2003-01-02 | 2008-01-01 | Mount Cook Biosciences, Inc. | Cardioprotective delta opioid receptor agonists and methods of using same |
| JP2008546638A (ja) * | 2005-04-14 | 2008-12-25 | マウント クック バイオサイエンシズ，インコーポレイテッド | 新規なオピオイド化合物の組成物およびその使用方法 |
| US20070197786A1 (en) * | 2005-07-22 | 2007-08-23 | Kwen-Jen Chang | Enantiomerically pure opioid diarylmethylpiperazine |
| KR101319390B1 (ko) * | 2007-04-25 | 2013-10-17 | 엘지전자 주식회사 | 대중 교통 정보를 제공하고 이를 이용하는 방법 및 장치 |
| CN105646332B (zh) * | 2014-11-09 | 2018-05-25 | 复旦大学 | 氨基甲基哌啶类衍生物及其制备方法和药物用途 |
| US11246865B2 (en) | 2017-04-30 | 2022-02-15 | Versi Group, Llc | Opioid for use to reduce and/or treat drug addiction |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5985880A (en) * | 1996-06-05 | 1999-11-16 | Delta Pharmaceuticals | Compositions and methods for reducing respiratory depression and attendant side effects of mu opioid compounds |
| US5807858A (en) * | 1996-06-05 | 1998-09-15 | Delta Pharmaceutical, Inc. | Compositions and methods for reducing respiratory depression |
| GB9202238D0 (en) * | 1992-02-03 | 1992-03-18 | Wellcome Found | Compounds |
| US20020052007A1 (en) | 1992-02-03 | 2002-05-02 | Chang Kwen Jen | Diarylmethylbenzylpiperazines and corresponding halobenzyl derivatives |
-
2002
- 2002-09-25 NZ NZ531875A patent/NZ531875A/en not_active IP Right Cessation
- 2002-09-25 US US10/254,609 patent/US6924288B2/en not_active Expired - Lifetime
- 2002-09-25 RU RU2004107850/15A patent/RU2309153C2/ru not_active IP Right Cessation
- 2002-09-25 AU AU2002341832A patent/AU2002341832B2/en not_active Ceased
- 2002-09-25 CN CN028187806A patent/CN1558765B/zh not_active Expired - Fee Related
- 2002-09-25 MX MXPA04002813A patent/MXPA04002813A/es active IP Right Grant
- 2002-09-25 KR KR10-2004-7004162A patent/KR20040041171A/ko not_active Application Discontinuation
- 2002-09-25 BR BR0212742-3A patent/BR0212742A/pt not_active IP Right Cessation
- 2002-09-25 IL IL16079402A patent/IL160794A0/xx unknown
- 2002-09-25 EP EP02775985A patent/EP1438051A4/en not_active Withdrawn
- 2002-09-25 JP JP2003530295A patent/JP2005505575A/ja active Pending
- 2002-09-25 WO PCT/US2002/030398 patent/WO2003026660A1/en active Application Filing
- 2002-09-25 CA CA2459577A patent/CA2459577C/en not_active Expired - Fee Related
- 2002-09-25 PL PL02370346A patent/PL370346A1/xx unknown
-
2004
- 2004-03-09 IL IL160794A patent/IL160794A/en not_active IP Right Cessation
- 2004-03-24 ZA ZA200402325A patent/ZA200402325B/en unknown
- 2004-04-23 NO NO20041729A patent/NO325958B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| PL370346A1 (en) | 2005-05-16 |
| KR20040041171A (ko) | 2004-05-14 |
| MXPA04002813A (es) | 2005-06-06 |
| CA2459577C (en) | 2012-01-24 |
| WO2003026660A1 (en) | 2003-04-03 |
| CA2459577A1 (en) | 2003-04-03 |
| RU2004107850A (ru) | 2005-04-20 |
| RU2309153C2 (ru) | 2007-10-27 |
| JP2005505575A (ja) | 2005-02-24 |
| BR0212742A (pt) | 2004-10-05 |
| NO20041729L (no) | 2004-06-25 |
| EP1438051A4 (en) | 2005-01-05 |
| EP1438051A1 (en) | 2004-07-21 |
| NZ531875A (en) | 2006-10-27 |
| IL160794A0 (en) | 2004-08-31 |
| IL160794A (en) | 2012-08-30 |
| ZA200402325B (en) | 2005-01-13 |
| US6924288B2 (en) | 2005-08-02 |
| CN1558765A (zh) | 2004-12-29 |
| CN1558765B (zh) | 2012-01-04 |
| US20030114462A1 (en) | 2003-06-19 |
| AU2002341832B2 (en) | 2008-10-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |