NO20044881L - Acyl-3-carboxyphenylurea derivatives, preparation method and use thereof - Google Patents
Acyl-3-carboxyphenylurea derivatives, preparation method and use thereofInfo
- Publication number
- NO20044881L NO20044881L NO20044881A NO20044881A NO20044881L NO 20044881 L NO20044881 L NO 20044881L NO 20044881 A NO20044881 A NO 20044881A NO 20044881 A NO20044881 A NO 20044881A NO 20044881 L NO20044881 L NO 20044881L
- Authority
- NO
- Norway
- Prior art keywords
- acyl
- preparation
- derivatives
- well
- acceptable salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/46—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylureas
- C07C275/48—Y being a hydrogen or a carbon atom
- C07C275/54—Y being a carbon atom of a six-membered aromatic ring, e.g. benzoylureas
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Hematology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Oppfinnelsen vedrører acyl-3-karboksyfenyl-ureaderivater så vel som deres fysiologisk akseptable salter og fysiologisk funksjonelle derivater. Oppfinnelsen vedrører forbindelsen med formel (I), hvor restene har den angitte betydningen, så vel som deres fysiologisk akseptable salter og fremgangsmåte for deres fremstilling. Forbindelsene egner seg for eksempel som anti-diabetika.The invention relates to acyl-3-carboxyphenyl urea derivatives as well as their physiologically acceptable salts and physiologically functional derivatives. The invention relates to the compound of formula (I), wherein the residues have the indicated meaning, as well as their physiologically acceptable salts and process for their preparation. The compounds are suitable, for example, as anti-diabetics.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10215908A DE10215908B4 (en) | 2002-04-11 | 2002-04-11 | Acyl-3-carboxyphenyl-urea derivatives and their use as medicaments |
PCT/EP2003/003254 WO2003084923A1 (en) | 2002-04-11 | 2003-03-28 | Acyl-3-carboxyphenylurea derivatives, method for production and use thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20044881L true NO20044881L (en) | 2005-01-07 |
Family
ID=28684936
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20044881A NO20044881L (en) | 2002-04-11 | 2004-11-09 | Acyl-3-carboxyphenylurea derivatives, preparation method and use thereof |
Country Status (24)
Country | Link |
---|---|
EP (1) | EP1497263B1 (en) |
JP (1) | JP4328212B2 (en) |
KR (1) | KR20040097332A (en) |
CN (1) | CN1263734C (en) |
AR (1) | AR039402A1 (en) |
AT (1) | ATE404532T1 (en) |
AU (1) | AU2003232192A1 (en) |
BR (1) | BR0309130A (en) |
CA (1) | CA2481819A1 (en) |
DE (2) | DE10215908B4 (en) |
HK (1) | HK1075650A1 (en) |
HR (1) | HRP20040931A2 (en) |
HU (1) | HUP0500203A2 (en) |
IL (1) | IL164248A0 (en) |
MA (1) | MA27195A1 (en) |
MX (1) | MXPA04009239A (en) |
NO (1) | NO20044881L (en) |
NZ (1) | NZ535833A (en) |
PL (1) | PL371317A1 (en) |
RS (1) | RS88704A (en) |
RU (1) | RU2004133046A (en) |
TW (1) | TW200401765A (en) |
WO (1) | WO2003084923A1 (en) |
ZA (1) | ZA200407361B (en) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10215907A1 (en) * | 2002-04-11 | 2003-11-06 | Aventis Pharma Gmbh | Acyl-4-carboxyphenyl-urea derivatives, processes for their preparation and their use |
DE10306502B4 (en) * | 2003-02-17 | 2005-03-17 | Aventis Pharma Deutschland Gmbh | Substituted 3- (benzoylureido) thiophene derivatives and medicaments containing them |
DE10308352A1 (en) | 2003-02-27 | 2004-09-09 | Aventis Pharma Deutschland Gmbh | Branched side chain arylcycloalkyl derivatives, process for their preparation and their use as medicaments |
DE10308355A1 (en) | 2003-02-27 | 2004-12-23 | Aventis Pharma Deutschland Gmbh | Aryl-cycloalkyl-substituted alkanoic acid derivatives, process for their preparation and their use as medicaments |
DE10308353A1 (en) | 2003-02-27 | 2004-12-02 | Aventis Pharma Deutschland Gmbh | Diarylcycloalkyl derivatives, processes for their preparation and their use as medicines |
DE10308351A1 (en) | 2003-02-27 | 2004-11-25 | Aventis Pharma Deutschland Gmbh | 1,3-substituted cycloalkyl derivatives having acidic, usually heterocyclic groups, processes for their preparation and their use as medicaments |
US7148246B2 (en) | 2003-02-27 | 2006-12-12 | Sanofi-Aventis Deutschland Gmbh | Cycloalkyl derivatives having bioisosteric carboxylic acid groups, processes for their preparation and their use as pharmaceuticals |
US7241787B2 (en) | 2004-01-25 | 2007-07-10 | Sanofi-Aventis Deutschland Gmbh | Substituted N-cycloexylimidazolinones, process for their preparation and their use as medicaments |
EP1586573B1 (en) | 2004-04-01 | 2007-02-07 | Sanofi-Aventis Deutschland GmbH | Oxadiazolones, processes for their preparation and their use as pharmaceuticals |
DE102005026762A1 (en) | 2005-06-09 | 2006-12-21 | Sanofi-Aventis Deutschland Gmbh | Azolopyridin-2-one derivatives as inhibitors of lipases and phospholipases |
PE20110235A1 (en) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | PHARMACEUTICAL COMBINATIONS INCLUDING LINAGLIPTIN AND METMORPHINE |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS62111961A (en) * | 1985-09-30 | 1987-05-22 | ユニオン・カ−バイド・コ−ポレ−シヨン | Insecticidal 1-(4-aryloxyphenyl)-3-benzoyl urea compound andits production |
GB9313268D0 (en) * | 1993-06-28 | 1993-08-11 | Zeneca Ltd | Chemical compounds |
ATE205477T1 (en) * | 1995-06-06 | 2001-09-15 | Pfizer | SUBSTITUTED N-(INDOLE-2-CARBONYL)-AMIDES AND DERIVATIVES AS GLYCOGEN PHOSPHORYLASE INHIBITORS |
AU3772800A (en) * | 1999-03-24 | 2000-10-09 | Sepracor, Inc. | Diaryl thioethers, compositions and uses thereof |
US20010053791A1 (en) * | 2000-03-16 | 2001-12-20 | Babcock Walter C. | Glycogen phosphorylase inhibitor |
YU91002A (en) * | 2000-06-09 | 2006-05-25 | Aventis Pharma Deutschland | Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament |
GB0021831D0 (en) * | 2000-09-06 | 2000-10-18 | Astrazeneca Ab | Chemical compounds |
PE20021091A1 (en) * | 2001-05-25 | 2003-02-04 | Aventis Pharma Gmbh | DERIVATIVES OF PHENYLUREA SUBSTITUTED WITH CARBONAMIDE AND PROCEDURE FOR THEIR PREPARATION |
-
2002
- 2002-04-11 DE DE10215908A patent/DE10215908B4/en not_active Expired - Fee Related
-
2003
- 2003-03-28 CN CNB038082241A patent/CN1263734C/en not_active Expired - Fee Related
- 2003-03-28 CA CA002481819A patent/CA2481819A1/en not_active Abandoned
- 2003-03-28 JP JP2003582122A patent/JP4328212B2/en not_active Expired - Fee Related
- 2003-03-28 EP EP03745772A patent/EP1497263B1/en not_active Expired - Lifetime
- 2003-03-28 AT AT03745772T patent/ATE404532T1/en not_active IP Right Cessation
- 2003-03-28 DE DE50310320T patent/DE50310320D1/en not_active Expired - Lifetime
- 2003-03-28 AU AU2003232192A patent/AU2003232192A1/en not_active Abandoned
- 2003-03-28 PL PL03371317A patent/PL371317A1/en not_active Application Discontinuation
- 2003-03-28 NZ NZ535833A patent/NZ535833A/en unknown
- 2003-03-28 MX MXPA04009239A patent/MXPA04009239A/en active IP Right Grant
- 2003-03-28 IL IL16424803A patent/IL164248A0/en unknown
- 2003-03-28 KR KR10-2004-7016149A patent/KR20040097332A/en not_active Application Discontinuation
- 2003-03-28 WO PCT/EP2003/003254 patent/WO2003084923A1/en active IP Right Grant
- 2003-03-28 BR BR0309130-9A patent/BR0309130A/en not_active IP Right Cessation
- 2003-03-28 RS YUP-887/04A patent/RS88704A/en unknown
- 2003-03-28 HU HU0500203A patent/HUP0500203A2/en unknown
- 2003-03-28 RU RU2004133046/04A patent/RU2004133046A/en not_active Application Discontinuation
- 2003-04-09 TW TW092108055A patent/TW200401765A/en unknown
- 2003-04-09 AR ARP030101246A patent/AR039402A1/en unknown
-
2004
- 2004-09-14 ZA ZA200407361A patent/ZA200407361B/en unknown
- 2004-10-07 HR HR20040931A patent/HRP20040931A2/en not_active Application Discontinuation
- 2004-10-08 MA MA27903A patent/MA27195A1/en unknown
- 2004-11-09 NO NO20044881A patent/NO20044881L/en unknown
-
2005
- 2005-09-05 HK HK05107763A patent/HK1075650A1/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
AR039402A1 (en) | 2005-02-16 |
EP1497263A1 (en) | 2005-01-19 |
JP2005522481A (en) | 2005-07-28 |
JP4328212B2 (en) | 2009-09-09 |
RU2004133046A (en) | 2005-04-20 |
TW200401765A (en) | 2004-02-01 |
HK1075650A1 (en) | 2005-12-23 |
DE10215908A1 (en) | 2003-11-06 |
MA27195A1 (en) | 2005-01-03 |
CA2481819A1 (en) | 2003-10-16 |
HUP0500203A2 (en) | 2005-06-28 |
ZA200407361B (en) | 2006-02-22 |
WO2003084923A1 (en) | 2003-10-16 |
EP1497263B1 (en) | 2008-08-13 |
IL164248A0 (en) | 2005-12-18 |
CN1263734C (en) | 2006-07-12 |
KR20040097332A (en) | 2004-11-17 |
HRP20040931A2 (en) | 2005-02-28 |
RS88704A (en) | 2007-02-05 |
PL371317A1 (en) | 2005-06-13 |
ATE404532T1 (en) | 2008-08-15 |
CN1646486A (en) | 2005-07-27 |
BR0309130A (en) | 2005-02-01 |
MXPA04009239A (en) | 2005-01-25 |
DE10215908B4 (en) | 2005-08-18 |
DE50310320D1 (en) | 2008-09-25 |
NZ535833A (en) | 2006-03-31 |
AU2003232192A1 (en) | 2003-10-20 |
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