NO20026167D0 - Condensed cyclic compounds as modulators of nuclear hormone receptor function - Google Patents

Condensed cyclic compounds as modulators of nuclear hormone receptor function

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Publication number
NO20026167D0
NO20026167D0 NO20026167A NO20026167A NO20026167D0 NO 20026167 D0 NO20026167 D0 NO 20026167D0 NO 20026167 A NO20026167 A NO 20026167A NO 20026167 A NO20026167 A NO 20026167A NO 20026167 D0 NO20026167 D0 NO 20026167D0
Authority
NO
Norway
Prior art keywords
hormone receptor
modulators
nuclear hormone
cyclic compounds
receptor function
Prior art date
Application number
NO20026167A
Other languages
Norwegian (no)
Other versions
NO20026167L (en
Inventor
Mark Ernest Salvati
James Aaron Balog
Weifang Shan
Soren Giese
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20026167D0 publication Critical patent/NO20026167D0/en
Publication of NO20026167L publication Critical patent/NO20026167L/en

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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Abstract

Fused cyclic compounds, methods of using such compounds in the treatment of nuclear hormone receptor-associated conditions such as cancer and immune disorders, and pharmaceutical compositions containing such compounds.</SDOAB >
NO20026167A 2000-06-28 2002-12-20 Condensed cyclic compounds as modulators of nuclear hormone receptor function NO20026167L (en)

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US7405234B2 (en) 2002-05-17 2008-07-29 Bristol-Myers Squibb Company Bicyclic modulators of androgen receptor function
BR0313405A (en) 2002-08-12 2005-07-12 Takeda Pharmaceutical Compounds, methods for preparing a compound and for preventing and / or treating cancer, prodrug, drug, androgen receptor modulator, agent for preventing and / or treating male hypogonadism or climatic disorder, osteoporosis and cancer, and use of a compound.
US7199125B2 (en) 2003-10-02 2007-04-03 Bristol-Myers Squibb Company Spiro-cyclic compounds useful as anti-inflammatory agents
US7820702B2 (en) 2004-02-04 2010-10-26 Bristol-Myers Squibb Company Sulfonylpyrrolidine modulators of androgen receptor function and method
US7417040B2 (en) 2004-03-01 2008-08-26 Bristol-Myers Squibb Company Fused tricyclic compounds as inhibitors of 17β-hydroxysteroid dehydrogenase 3
US7625923B2 (en) * 2004-03-04 2009-12-01 Bristol-Myers Squibb Company Bicyclic modulators of androgen receptor function
US7696241B2 (en) 2004-03-04 2010-04-13 Bristol-Myers Squibb Company Bicyclic compounds as modulators of androgen receptor function and method
US8546451B2 (en) 2005-11-28 2013-10-01 Gtx, Inc. Estrogen receptor ligands and methods of use thereof
US9409856B2 (en) 2005-11-28 2016-08-09 Gtx, Inc. Estrogen receptor ligands and methods of use thereof
EP1991549B1 (en) * 2006-02-10 2012-01-11 Janssen Pharmaceutica N.V. Bicyclic imidazole or thiadiazole heterocycles useful as selective androgen receptor modulators
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EP2334683B1 (en) 2008-08-29 2017-03-22 MSD Italia S.r.l. Saturated bicyclic heterocyclic derivatives as smo antagonists
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WO2002000653A2 (en) 2002-01-03
HUP0303165A2 (en) 2003-12-29
BR0111869A (en) 2003-09-23
WO2002000653A3 (en) 2002-07-25
NZ523802A (en) 2005-11-25
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HUP0303165A3 (en) 2006-05-29
CA2413683A1 (en) 2002-01-03

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