NO20026167D0 - Condensed cyclic compounds as modulators of nuclear hormone receptor function - Google Patents
Condensed cyclic compounds as modulators of nuclear hormone receptor functionInfo
- Publication number
- NO20026167D0 NO20026167D0 NO20026167A NO20026167A NO20026167D0 NO 20026167 D0 NO20026167 D0 NO 20026167D0 NO 20026167 A NO20026167 A NO 20026167A NO 20026167 A NO20026167 A NO 20026167A NO 20026167 D0 NO20026167 D0 NO 20026167D0
- Authority
- NO
- Norway
- Prior art keywords
- hormone receptor
- modulators
- nuclear hormone
- cyclic compounds
- receptor function
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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- A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
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- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
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- C07D207/12—Oxygen or sulfur atoms
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Abstract
Fused cyclic compounds, methods of using such compounds in the treatment of nuclear hormone receptor-associated conditions such as cancer and immune disorders, and pharmaceutical compositions containing such compounds.</SDOAB >
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US21439200P | 2000-06-28 | 2000-06-28 | |
US28461701P | 2001-04-18 | 2001-04-18 | |
US28443801P | 2001-04-18 | 2001-04-18 | |
PCT/US2001/019663 WO2002000653A2 (en) | 2000-06-28 | 2001-06-20 | Fused cyclic compounds as modulators of nuclear hormone receptor function |
Publications (2)
Publication Number | Publication Date |
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NO20026167D0 true NO20026167D0 (en) | 2002-12-20 |
NO20026167L NO20026167L (en) | 2002-12-20 |
Family
ID=27485945
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20026167A NO20026167L (en) | 2000-06-28 | 2002-12-20 | Condensed cyclic compounds as modulators of nuclear hormone receptor function |
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EP (1) | EP1299385A2 (en) |
JP (1) | JP2004515462A (en) |
AU (1) | AU2002215609A1 (en) |
BR (1) | BR0111869A (en) |
CA (1) | CA2413683A1 (en) |
HU (1) | HUP0303165A3 (en) |
MX (1) | MXPA02012563A (en) |
NO (1) | NO20026167L (en) |
NZ (1) | NZ523802A (en) |
WO (1) | WO2002000653A2 (en) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2000264876A (en) * | 1998-09-10 | 2000-09-26 | Sumitomo Chem Co Ltd | Condensed heterocyclic ring compound |
AU2001288213B2 (en) * | 2000-06-28 | 2005-04-14 | Bristol-Myers Squibb Company | Selective androgen receptor modulators and methods for their identification, design and use |
US20030114420A1 (en) * | 2000-06-28 | 2003-06-19 | Salvati Mark E. | Fused cyclic modulators of nuclear hormone receptor function |
IL149357A0 (en) * | 2000-09-07 | 2002-11-10 | Bayer Ag | Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents |
DE10162375A1 (en) * | 2001-12-19 | 2003-07-10 | Bayer Ag | Bicyclic N-aryl amides |
ES2310622T3 (en) * | 2001-12-19 | 2009-01-16 | Bristol-Myers Squibb Company | CONDENSED HETEROCICLICAL COMPOUNDS AND ANALOGS OF THE SAME, MODULATORS OF THE FUNCTION OF NUCLEAR HORMONE RECEPTORS. |
CA2479722A1 (en) * | 2002-03-18 | 2003-10-02 | Pharmacia Corporation | Combination of an aldosterone receptor antagonist and a fibric acid derivative |
US7405234B2 (en) | 2002-05-17 | 2008-07-29 | Bristol-Myers Squibb Company | Bicyclic modulators of androgen receptor function |
CA2495383A1 (en) | 2002-08-12 | 2004-02-26 | Takeda Pharmaceutical Company Limited | Fused benzene derivative and use |
US7199125B2 (en) | 2003-10-02 | 2007-04-03 | Bristol-Myers Squibb Company | Spiro-cyclic compounds useful as anti-inflammatory agents |
US7820702B2 (en) | 2004-02-04 | 2010-10-26 | Bristol-Myers Squibb Company | Sulfonylpyrrolidine modulators of androgen receptor function and method |
US7417040B2 (en) | 2004-03-01 | 2008-08-26 | Bristol-Myers Squibb Company | Fused tricyclic compounds as inhibitors of 17β-hydroxysteroid dehydrogenase 3 |
US7625923B2 (en) * | 2004-03-04 | 2009-12-01 | Bristol-Myers Squibb Company | Bicyclic modulators of androgen receptor function |
US7696241B2 (en) | 2004-03-04 | 2010-04-13 | Bristol-Myers Squibb Company | Bicyclic compounds as modulators of androgen receptor function and method |
US8546451B2 (en) | 2005-11-28 | 2013-10-01 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
US9409856B2 (en) | 2005-11-28 | 2016-08-09 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
CN101415710B (en) * | 2006-02-10 | 2013-08-21 | 詹森药业有限公司 | Bicyclic imidazole or thiadiazole heterocycles useful as selective androgen receptor modulators |
EP2039695A4 (en) | 2006-07-11 | 2010-09-15 | Takeda Pharmaceutical | Bicyclic heterocyclic compound and use thereof |
EP2334683B1 (en) | 2008-08-29 | 2017-03-22 | MSD Italia S.r.l. | Saturated bicyclic heterocyclic derivatives as smo antagonists |
US9624161B2 (en) | 2009-02-23 | 2017-04-18 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
US9427418B2 (en) | 2009-02-23 | 2016-08-30 | Gtx, Inc. | Estrogen receptor ligands and methods of use thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69531998T2 (en) * | 1994-12-22 | 2004-07-22 | Ligand Pharmaceuticals, Inc., San Diego | STEROID RECEPTOR MODULATOR COMPOUNDS AND METHODS |
DK0918774T3 (en) * | 1996-06-27 | 2002-05-21 | Ligand Pharm Inc | Androgen receptor modulator compounds and methods |
AU2001288213B2 (en) * | 2000-06-28 | 2005-04-14 | Bristol-Myers Squibb Company | Selective androgen receptor modulators and methods for their identification, design and use |
-
2001
- 2001-06-20 BR BR0111869-2A patent/BR0111869A/en not_active IP Right Cessation
- 2001-06-20 CA CA002413683A patent/CA2413683A1/en not_active Abandoned
- 2001-06-20 MX MXPA02012563A patent/MXPA02012563A/en unknown
- 2001-06-20 HU HU0303165A patent/HUP0303165A3/en unknown
- 2001-06-20 WO PCT/US2001/019663 patent/WO2002000653A2/en active IP Right Grant
- 2001-06-20 EP EP01984054A patent/EP1299385A2/en not_active Withdrawn
- 2001-06-20 AU AU2002215609A patent/AU2002215609A1/en not_active Abandoned
- 2001-06-20 NZ NZ523802A patent/NZ523802A/en unknown
- 2001-06-20 JP JP2002505777A patent/JP2004515462A/en active Pending
-
2002
- 2002-12-20 NO NO20026167A patent/NO20026167L/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
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MXPA02012563A (en) | 2003-05-14 |
EP1299385A2 (en) | 2003-04-09 |
JP2004515462A (en) | 2004-05-27 |
WO2002000653A3 (en) | 2002-07-25 |
CA2413683A1 (en) | 2002-01-03 |
NZ523802A (en) | 2005-11-25 |
AU2002215609A1 (en) | 2002-01-08 |
HUP0303165A3 (en) | 2006-05-29 |
BR0111869A (en) | 2003-09-23 |
HUP0303165A2 (en) | 2003-12-29 |
NO20026167L (en) | 2002-12-20 |
WO2002000653A2 (en) | 2002-01-03 |
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