NO20023107D0 - Carboxamide-diazepine derivatives, method of preparation, use as medicines, pharmaceutical preparations and uses thereof - Google Patents
Carboxamide-diazepine derivatives, method of preparation, use as medicines, pharmaceutical preparations and uses thereofInfo
- Publication number
- NO20023107D0 NO20023107D0 NO20023107A NO20023107A NO20023107D0 NO 20023107 D0 NO20023107 D0 NO 20023107D0 NO 20023107 A NO20023107 A NO 20023107A NO 20023107 A NO20023107 A NO 20023107A NO 20023107 D0 NO20023107 D0 NO 20023107D0
- Authority
- NO
- Norway
- Prior art keywords
- medicines
- carboxamide
- preparation
- pharmaceutical preparations
- products
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Cardiology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
The invention concerns products of formula (I) wherein: R1 represents in particular -C(O) -R5, -SO2 -R5 or -C(O) -NR6R5, R2 and R7 are such that either R7 represents a hydrogen atom and R2 is such that the group (a) represents the radical of a natural or non-natural amino acid, or R2 and R7 form together a cycle with the nitrogen and carbon atom whereto they are bound, R3 represents in particular the radical -CH=N2 or -CH2-L-R4, R4 represents in particular a linear or branched alkyl radical, and their additive salts with mineral or organic acids or with mineral or organic bases of said products of formula (I). The invention also concerns the method for preparing said products and their use as medicines.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9916567A FR2802927B1 (en) | 1999-12-28 | 1999-12-28 | NOVEL DIAZEPINE CARBOXAMIDE DERIVATIVES, THEIR PREPARATION PROCESS, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND THEIR NEW USE |
PCT/FR2000/003622 WO2001047930A1 (en) | 1999-12-28 | 2000-12-21 | Carboxamide diazepin derivatives, preparation method, use as medicines, pharmaceutical compositions and use thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20023107D0 true NO20023107D0 (en) | 2002-06-27 |
NO20023107L NO20023107L (en) | 2002-08-27 |
Family
ID=9553901
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20023107A NO20023107L (en) | 1999-12-28 | 2002-06-27 | Carboxamide-diazepine derivatives, method of preparation, use as medicines, pharmaceutical preparations and uses thereof |
Country Status (26)
Country | Link |
---|---|
EP (1) | EP1246824B1 (en) |
JP (1) | JP2003519152A (en) |
KR (1) | KR20020062772A (en) |
AT (1) | ATE268775T1 (en) |
AU (1) | AU780522B2 (en) |
BR (1) | BR0016845A (en) |
CA (1) | CA2395275A1 (en) |
DE (1) | DE60011473T2 (en) |
DK (1) | DK1246824T3 (en) |
EA (1) | EA005288B1 (en) |
EE (1) | EE200200362A (en) |
ES (1) | ES2218275T3 (en) |
FR (1) | FR2802927B1 (en) |
HR (1) | HRP20020558A2 (en) |
HU (1) | HUP0203921A3 (en) |
IL (1) | IL150419A0 (en) |
MX (1) | MXPA02006413A (en) |
NO (1) | NO20023107L (en) |
NZ (1) | NZ519884A (en) |
PL (1) | PL355950A1 (en) |
PT (1) | PT1246824E (en) |
SI (1) | SI1246824T1 (en) |
SK (1) | SK9092002A3 (en) |
WO (1) | WO2001047930A1 (en) |
YU (1) | YU47502A (en) |
ZA (1) | ZA200205221B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20220115062A (en) | 2021-02-09 | 2022-08-17 | (주)오스티오뉴로젠 | Pharmaceutical Composition For Treating and Preventing Osteoporosis Comprising Compounds of Chromone Scaffold |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6204261B1 (en) * | 1995-12-20 | 2001-03-20 | Vertex Pharmaceuticals Incorporated | Inhibitors of interleukin-1β Converting enzyme inhibitors |
US5552400A (en) * | 1994-06-08 | 1996-09-03 | Sterling Winthrop Inc. | Fused-bicyclic lactams as interleukin-1β converting enzyme inhibitors |
US5847135A (en) * | 1994-06-17 | 1998-12-08 | Vertex Pharmaceuticals, Incorporated | Inhibitors of interleukin-1β converting enzyme |
-
1999
- 1999-12-28 FR FR9916567A patent/FR2802927B1/en not_active Expired - Fee Related
-
2000
- 2000-12-21 DE DE60011473T patent/DE60011473T2/en not_active Expired - Fee Related
- 2000-12-21 SK SK909-2002A patent/SK9092002A3/en unknown
- 2000-12-21 WO PCT/FR2000/003622 patent/WO2001047930A1/en not_active Application Discontinuation
- 2000-12-21 EA EA200200721A patent/EA005288B1/en not_active IP Right Cessation
- 2000-12-21 IL IL15041900A patent/IL150419A0/en unknown
- 2000-12-21 PT PT00990087T patent/PT1246824E/en unknown
- 2000-12-21 AT AT00990087T patent/ATE268775T1/en not_active IP Right Cessation
- 2000-12-21 PL PL00355950A patent/PL355950A1/en not_active Application Discontinuation
- 2000-12-21 DK DK00990087T patent/DK1246824T3/en active
- 2000-12-21 ES ES00990087T patent/ES2218275T3/en not_active Expired - Lifetime
- 2000-12-21 AU AU26888/01A patent/AU780522B2/en not_active Ceased
- 2000-12-21 BR BR0016845-9A patent/BR0016845A/en not_active IP Right Cessation
- 2000-12-21 CA CA002395275A patent/CA2395275A1/en not_active Abandoned
- 2000-12-21 YU YU47502A patent/YU47502A/en unknown
- 2000-12-21 EE EEP200200362A patent/EE200200362A/en unknown
- 2000-12-21 NZ NZ519884A patent/NZ519884A/en unknown
- 2000-12-21 MX MXPA02006413A patent/MXPA02006413A/en active IP Right Grant
- 2000-12-21 KR KR1020027008366A patent/KR20020062772A/en not_active Application Discontinuation
- 2000-12-21 SI SI200030455T patent/SI1246824T1/en unknown
- 2000-12-21 EP EP00990087A patent/EP1246824B1/en not_active Expired - Lifetime
- 2000-12-21 HU HU0203921A patent/HUP0203921A3/en unknown
- 2000-12-21 JP JP2001549400A patent/JP2003519152A/en not_active Abandoned
-
2002
- 2002-06-27 HR HR20020558A patent/HRP20020558A2/en not_active Application Discontinuation
- 2002-06-27 NO NO20023107A patent/NO20023107L/en not_active Application Discontinuation
- 2002-06-28 ZA ZA200205221A patent/ZA200205221B/en unknown
Also Published As
Publication number | Publication date |
---|---|
HUP0203921A3 (en) | 2005-01-28 |
KR20020062772A (en) | 2002-07-29 |
DK1246824T3 (en) | 2004-10-18 |
HUP0203921A2 (en) | 2003-03-28 |
PL355950A1 (en) | 2004-05-31 |
FR2802927A1 (en) | 2001-06-29 |
NO20023107L (en) | 2002-08-27 |
AU2688801A (en) | 2001-07-09 |
ES2218275T3 (en) | 2004-11-16 |
SK9092002A3 (en) | 2003-04-01 |
ZA200205221B (en) | 2003-09-04 |
JP2003519152A (en) | 2003-06-17 |
IL150419A0 (en) | 2002-12-01 |
DE60011473T2 (en) | 2005-06-30 |
BR0016845A (en) | 2002-10-15 |
CA2395275A1 (en) | 2001-07-05 |
FR2802927B1 (en) | 2002-03-01 |
SI1246824T1 (en) | 2004-10-31 |
ATE268775T1 (en) | 2004-06-15 |
AU780522B2 (en) | 2005-03-24 |
DE60011473D1 (en) | 2004-07-15 |
EA005288B1 (en) | 2004-12-30 |
NZ519884A (en) | 2005-03-24 |
EP1246824A1 (en) | 2002-10-09 |
PT1246824E (en) | 2004-10-29 |
EP1246824B1 (en) | 2004-06-09 |
MXPA02006413A (en) | 2002-11-29 |
YU47502A (en) | 2005-03-15 |
WO2001047930A1 (en) | 2001-07-05 |
EE200200362A (en) | 2003-08-15 |
HRP20020558A2 (en) | 2004-02-29 |
EA200200721A1 (en) | 2002-12-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |