NO20020192L - Pseudomycin prodrug - Google Patents

Pseudomycin prodrug

Info

Publication number
NO20020192L
NO20020192L NO20020192A NO20020192A NO20020192L NO 20020192 L NO20020192 L NO 20020192L NO 20020192 A NO20020192 A NO 20020192A NO 20020192 A NO20020192 A NO 20020192A NO 20020192 L NO20020192 L NO 20020192L
Authority
NO
Norway
Prior art keywords
prodrug
pseudomycin
pseudomycin prodrug
acyloxyalkylcarbamate
bond
Prior art date
Application number
NO20020192A
Other languages
Norwegian (no)
Other versions
NO20020192D0 (en
Inventor
Shu-Hui Chen
Michael John Rodriguez
Xicheng Sun
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of NO20020192D0 publication Critical patent/NO20020192D0/en
Publication of NO20020192L publication Critical patent/NO20020192L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)

Abstract

Et pseudomycin prodrug representert ved struktur (A) hvor RI er en acyloksyalkylkarbamat binding er beskrevet. Prodruget viser antifungal aktivitet med færre uheldige bivirkninger.A pseudomycin prodrug represented by structure (A) wherein R 1 is an acyloxyalkylcarbamate bond is disclosed. The prodrug shows antifungal activity with fewer adverse side effects.

NO20020192A 1999-07-15 2002-01-14 Pseudomycin prodrug NO20020192L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14384099P 1999-07-15 1999-07-15
PCT/US2000/015016 WO2001005813A1 (en) 1999-07-15 2000-06-08 Pseudomycin prodrugs

Publications (2)

Publication Number Publication Date
NO20020192D0 NO20020192D0 (en) 2002-01-14
NO20020192L true NO20020192L (en) 2002-03-14

Family

ID=22505903

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20020192A NO20020192L (en) 1999-07-15 2002-01-14 Pseudomycin prodrug

Country Status (11)

Country Link
EP (1) EP1198470A1 (en)
JP (1) JP2003505396A (en)
CN (1) CN1373770A (en)
AU (1) AU5310500A (en)
BR (1) BR0013153A (en)
CA (1) CA2379058A1 (en)
EA (1) EA200200161A1 (en)
HU (1) HUP0202223A3 (en)
MX (1) MXPA02000315A (en)
NO (1) NO20020192L (en)
WO (1) WO2001005813A1 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8048917B2 (en) 2005-04-06 2011-11-01 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US6818787B2 (en) 2001-06-11 2004-11-16 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US7186855B2 (en) 2001-06-11 2007-03-06 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
AU2004267100B2 (en) 2003-08-20 2010-10-07 Xenoport, Inc. Acyloxyalkyl carbamate prodrugs, methods of synthesis and use
CN101486668B (en) * 2003-12-30 2014-07-02 什诺波特有限公司 Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
ES2405329T3 (en) 2003-12-30 2013-05-30 Xenoport, Inc. Synthesis of acyloxyalkyl carbonate prodrugs and intermediates thereof
JP4938771B2 (en) 2005-06-20 2012-05-23 ゼノポート，インコーポレーテッド Acyloxyalkyl carbamate prodrugs of tranexamic acid, methods of synthesis, and uses
TW200820963A (en) 2006-07-28 2008-05-16 Xenoport Inc Acyloxyalkyl carbamate prodrugs of α-amino acids, methods of synthesis and use
WO2010017498A1 (en) * 2008-08-07 2010-02-11 Xenoport, Inc. Methods of synthesizing n-hydroxysuccinimidyl carbonates

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5576298A (en) * 1992-11-30 1996-11-19 Research And Development Institute, Inc. At Montana State University Peptides from pseudomonas syringae possessing broad-spectrum antibiotic activity

Also Published As

Publication number Publication date
WO2001005813A1 (en) 2001-01-25
EA200200161A1 (en) 2002-06-27
JP2003505396A (en) 2003-02-12
HUP0202223A2 (en) 2002-10-28
CA2379058A1 (en) 2001-01-25
HUP0202223A3 (en) 2002-11-28
CN1373770A (en) 2002-10-09
BR0013153A (en) 2002-04-02
EP1198470A1 (en) 2002-04-24
AU5310500A (en) 2001-02-05
MXPA02000315A (en) 2002-06-21
NO20020192D0 (en) 2002-01-14

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application