NO172495C - PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE, NON-Saturated AMINO ACID COMPOUNDS - Google Patents

PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE, NON-Saturated AMINO ACID COMPOUNDS

Info

Publication number
NO172495C
NO172495C NO88883444A NO883444A NO172495C NO 172495 C NO172495 C NO 172495C NO 88883444 A NO88883444 A NO 88883444A NO 883444 A NO883444 A NO 883444A NO 172495 C NO172495 C NO 172495C
Authority
NO
Norway
Prior art keywords
procedure
preparation
amino acid
acid compounds
therapeutic active
Prior art date
Application number
NO88883444A
Other languages
Norwegian (no)
Other versions
NO172495B (en
NO883444L (en
NO883444D0 (en
Inventor
Hans Allgeier
Christof Angst
Guido Bold
Rudolf Duthaler
Roland Heckendorn
Antonio Togni
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of NO883444D0 publication Critical patent/NO883444D0/en
Publication of NO883444L publication Critical patent/NO883444L/en
Publication of NO172495B publication Critical patent/NO172495B/en
Publication of NO172495C publication Critical patent/NO172495C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/16Esters of thiophosphoric acids or thiophosphorous acids
    • C07F9/165Esters of thiophosphoric acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/48Phosphonous acids R—P(OH)2; Thiophosphonous acids including RHP(=O)(OH); Derivatives thereof
    • C07F9/4808Phosphonous acids R—P(OH)2; Thiophosphonous acids including RHP(=O)(OH); Derivatives thereof the acid moiety containing a substituent or structure which is considered as characteristic
    • C07F9/4825Acyclic unsaturated acids or derivatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/30Phosphinic acids R2P(=O)(OH); Thiophosphinic acids, i.e. R2P(=X)(XH) (X = S, Se)
    • C07F9/302Acyclic unsaturated acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se)
    • C07F9/3804Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se) not used, see subgroups
    • C07F9/3826Acyclic unsaturated acids
NO88883444A 1987-08-04 1988-08-03 PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE, NON-Saturated AMINO ACID COMPOUNDS NO172495C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH298687 1987-08-04

Publications (4)

Publication Number Publication Date
NO883444D0 NO883444D0 (en) 1988-08-03
NO883444L NO883444L (en) 1989-02-06
NO172495B NO172495B (en) 1993-04-19
NO172495C true NO172495C (en) 1993-07-28

Family

ID=4246086

Family Applications (1)

Application Number Title Priority Date Filing Date
NO88883444A NO172495C (en) 1987-08-04 1988-08-03 PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE, NON-Saturated AMINO ACID COMPOUNDS

Country Status (16)

Country Link
EP (1) EP0302826A3 (en)
JP (2) JP2714018B2 (en)
KR (1) KR970011164B1 (en)
AU (1) AU605340B2 (en)
CA (1) CA1328113C (en)
DD (1) DD282016A5 (en)
DK (1) DK434788A (en)
FI (1) FI94415C (en)
HU (1) HU202242B (en)
IL (1) IL87246A (en)
NO (1) NO172495C (en)
NZ (1) NZ225649A (en)
PH (1) PH27591A (en)
PT (1) PT88170B (en)
YU (1) YU150188A (en)
ZA (1) ZA885653B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5175344A (en) * 1986-02-13 1992-12-29 Ciba-Geigy Corporation Unsaturated amino acids
ES2060122T3 (en) * 1989-04-07 1994-11-16 Ciba Geigy Ag UNSATURATED DERIVATIVES OF AMINODICARBOXILIC ACIDS.
US5488140A (en) * 1989-09-26 1996-01-30 Ciba-Geigy Corporation 4-substituted 2-aminoalk-3-enoic
ATE124700T1 (en) * 1989-09-26 1995-07-15 Ciba Geigy Ag PHOSPHONIC ACID, METHOD FOR PRODUCTION AND USE AS A MEDICINAL ACTIVE INGREDIENT.
US5294734A (en) * 1989-09-26 1994-03-15 Ciba-Geigy Corp. 4-substituted 2-aminoalk-3-enoic acids
US7414086B2 (en) 2005-05-13 2008-08-19 Shin-Etsu Chemical Co., Ltd. Room temperature-curable organopolysiloxane compositions
US20090170813A1 (en) * 2005-10-18 2009-07-02 Francine Acher Hypophosphorous Acid Derivatives and their Therapeutical Applications
JP4952952B2 (en) 2008-09-12 2012-06-13 信越化学工業株式会社 Method for producing room temperature curable organopolysiloxane composition
EP3427729A1 (en) 2017-07-13 2019-01-16 Paris Sciences et Lettres - Quartier Latin Probenecid for use in treating epileptic diseases, disorders or conditions

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2038690T3 (en) * 1986-02-13 1993-08-01 Ciba-Geigy Ag UNSATURATED AMINO ACIDS.

Also Published As

Publication number Publication date
PT88170A (en) 1989-06-30
IL87246A0 (en) 1989-03-31
JPH1053597A (en) 1998-02-24
AU605340B2 (en) 1991-01-10
KR970011164B1 (en) 1997-07-08
EP0302826A2 (en) 1989-02-08
FI94415C (en) 1995-09-11
AU2038988A (en) 1989-03-02
NO172495B (en) 1993-04-19
FI883589A0 (en) 1988-08-01
FI94415B (en) 1995-05-31
NZ225649A (en) 1991-05-28
HU202242B (en) 1991-02-28
JPH0248586A (en) 1990-02-19
CA1328113C (en) 1994-03-29
NO883444L (en) 1989-02-06
JP2714018B2 (en) 1998-02-16
PH27591A (en) 1993-08-31
NO883444D0 (en) 1988-08-03
IL87246A (en) 1996-07-23
YU150188A (en) 1990-04-30
PT88170B (en) 1995-03-01
KR890003786A (en) 1989-04-18
ZA885653B (en) 1989-04-26
HUT47947A (en) 1989-04-28
EP0302826A3 (en) 1991-04-03
DK434788D0 (en) 1988-08-03
DD282016A5 (en) 1990-08-29
DK434788A (en) 1989-02-05
FI883589A (en) 1989-02-05

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