NO161917C - ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE DERIVATIVES OF TIENO AND FURO (2,3-C) PYROLES. - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE DERIVATIVES OF TIENO AND FURO (2,3-C) PYROLES.

Info

Publication number
NO161917C
NO161917C NO854051A NO854051A NO161917C NO 161917 C NO161917 C NO 161917C NO 854051 A NO854051 A NO 854051A NO 854051 A NO854051 A NO 854051A NO 161917 C NO161917 C NO 161917C
Authority
NO
Norway
Prior art keywords
tieno
pyroles
furo
preparation
active derivatives
Prior art date
Application number
NO854051A
Other languages
Norwegian (no)
Other versions
NO854051L (en
NO161917B (en
Inventor
Didier Festal
Denis Descours
Jean-Claude Depin
Yvette Quentin
Original Assignee
Lipha
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lipha filed Critical Lipha
Publication of NO854051L publication Critical patent/NO854051L/en
Publication of NO161917B publication Critical patent/NO161917B/en
Publication of NO161917C publication Critical patent/NO161917C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO854051A 1984-10-12 1985-10-11 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE DERIVATIVES OF TIENO AND FURO (2,3-C) PYROLES. NO161917C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8415658A FR2571723B1 (en) 1984-10-12 1984-10-12 THIENO AND FURO- (2,3-C) PYRROLES DERIVATIVES, METHODS OF PREPARATION AND MEDICAMENTS CONTAINING THEM

Publications (3)

Publication Number Publication Date
NO854051L NO854051L (en) 1986-04-14
NO161917B NO161917B (en) 1989-07-03
NO161917C true NO161917C (en) 1989-10-11

Family

ID=9308598

Family Applications (1)

Application Number Title Priority Date Filing Date
NO854051A NO161917C (en) 1984-10-12 1985-10-11 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE DERIVATIVES OF TIENO AND FURO (2,3-C) PYROLES.

Country Status (19)

Country Link
EP (1) EP0180500A1 (en)
JP (1) JPS6197286A (en)
AU (1) AU593776B2 (en)
CA (1) CA1250847A (en)
CS (1) CS265211B2 (en)
DD (1) DD237662A5 (en)
DK (1) DK465685A (en)
ES (1) ES8605524A1 (en)
FR (1) FR2571723B1 (en)
HU (1) HU193827B (en)
IL (1) IL76619A (en)
IN (1) IN169684B (en)
MA (1) MA20543A1 (en)
NO (1) NO161917C (en)
OA (1) OA08119A (en)
PT (1) PT81282B (en)
SU (1) SU1329621A3 (en)
YU (1) YU162485A (en)
ZA (1) ZA857809B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60255756A (en) * 1984-06-01 1985-12-17 Ikeda Mohandou:Kk Aminoalkylphenoxy derivative
FR2733750B1 (en) * 1995-05-03 1997-06-13 Synthelabo DERIVATIVES OF GAMMA-OXO-ALPHA- (PHENYLMETHYL) -5,6- DIHYDRO-4H-THIENO (3,4-C) PYRROLE-5-BUTANOIQUE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
ATE325125T1 (en) 2002-09-06 2006-06-15 Janssen Pharmaceutica Nv THIENOPYRROLYL AND FURANOPYRROLYL COMPOUNDS AND THEIR USE AS HISTAMINE H4 RECEPTOR LIGANDS
CN101186612B (en) * 2006-11-15 2012-10-03 天津和美生物技术有限公司 Pyrroline derivative capable of inhibiting cell to release tumor necrotic factor and its preparation and application
EP4196793A1 (en) 2020-08-11 2023-06-21 Université de Strasbourg H2 blockers targeting liver macrophages for the prevention and treatment of liver disease and cancer

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1565966A (en) * 1976-08-04 1980-04-23 Allen & Hanburys Ltd Aminoalkyl furan derivatives
GB1601459A (en) * 1977-05-17 1981-10-28 Allen & Hanburys Ltd Aminoalkyl thiophene derivatives
US4390701A (en) * 1981-05-18 1983-06-28 Bristol-Myers Company 1-Amino-2-[3-(3-piperidinomethylphenoxy)propylamino]cyclobutene-3,4-dione
US4520025A (en) * 1982-07-21 1985-05-28 William H. Rorer, Inc. Bicyclic nitrogen heterocyclic ethers and thioethers, and their pharmaceutical uses

Also Published As

Publication number Publication date
ES547789A0 (en) 1986-03-16
JPS6197286A (en) 1986-05-15
OA08119A (en) 1987-03-31
AU4852885A (en) 1986-04-17
MA20543A1 (en) 1986-07-01
NO854051L (en) 1986-04-14
ZA857809B (en) 1986-05-28
ES8605524A1 (en) 1986-03-16
IL76619A (en) 1990-07-12
CA1250847A (en) 1989-03-07
DK465685A (en) 1986-04-13
CS265211B2 (en) 1989-10-13
FR2571723A1 (en) 1986-04-18
PT81282A (en) 1985-11-01
YU162485A (en) 1987-12-31
FR2571723B1 (en) 1988-08-26
IN169684B (en) 1991-12-07
DK465685D0 (en) 1985-10-11
AU593776B2 (en) 1990-02-22
DD237662A5 (en) 1986-07-23
CS714485A2 (en) 1988-08-16
PT81282B (en) 1988-02-17
HUT40133A (en) 1986-11-28
IL76619A0 (en) 1986-02-28
SU1329621A3 (en) 1987-08-07
NO161917B (en) 1989-07-03
HU193827B (en) 1987-12-28
EP0180500A1 (en) 1986-05-07

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