NO137233C - ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ALFA, ALFA-DIARYLIMIDAZOLE-2-METHANOLS AND ACID ADDITIONAL SALTS THEREOF - Google Patents

ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ALFA, ALFA-DIARYLIMIDAZOLE-2-METHANOLS AND ACID ADDITIONAL SALTS THEREOF

Info

Publication number
NO137233C
NO137233C NO442/73A NO44273A NO137233C NO 137233 C NO137233 C NO 137233C NO 442/73 A NO442/73 A NO 442/73A NO 44273 A NO44273 A NO 44273A NO 137233 C NO137233 C NO 137233C
Authority
NO
Norway
Prior art keywords
alfa
diarylimidazole
methanols
preparation
therapeutic active
Prior art date
Application number
NO442/73A
Other languages
Norwegian (no)
Other versions
NO137233B (en
Inventor
Cornelis Van Der Stelt
Petrus Simon Hofman
Original Assignee
Gist Brocades Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gist Brocades Nv filed Critical Gist Brocades Nv
Publication of NO137233B publication Critical patent/NO137233B/en
Publication of NO137233C publication Critical patent/NO137233C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
NO442/73A 1972-02-04 1973-02-02 ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ALFA, ALFA-DIARYLIMIDAZOLE-2-METHANOLS AND ACID ADDITIONAL SALTS THEREOF NO137233C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB541872 1972-02-04
GB541872A GB1363382A (en) 1972-02-04 1972-09-05 Alpha.alpha-diarylimidazole-2-methanols

Publications (2)

Publication Number Publication Date
NO137233B NO137233B (en) 1977-10-17
NO137233C true NO137233C (en) 1978-01-25

Family

ID=26239878

Family Applications (1)

Application Number Title Priority Date Filing Date
NO442/73A NO137233C (en) 1972-02-04 1973-02-02 ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ALFA, ALFA-DIARYLIMIDAZOLE-2-METHANOLS AND ACID ADDITIONAL SALTS THEREOF

Country Status (16)

Country Link
AT (1) AT322545B (en)
AU (1) AU467008B2 (en)
BE (1) BE794940A (en)
CA (1) CA979899A (en)
CH (1) CH594630A5 (en)
CS (1) CS187368B2 (en)
DE (1) DE2305212A1 (en)
ES (1) ES411222A1 (en)
FI (1) FI57936C (en)
FR (1) FR2173984B1 (en)
GB (1) GB1363382A (en)
HU (1) HU166406B (en)
IL (1) IL41448A (en)
LU (1) LU66953A1 (en)
NL (1) NL7301494A (en)
NO (1) NO137233C (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19951701A1 (en) * 1999-10-27 2001-05-03 Aventis Pharma Gmbh Use of 2-imidazolyl-substituted carbinols for the manufacture of a medicament for the treatment or prophylaxis of diseases caused by ischemic conditions
JP2010522168A (en) * 2007-03-23 2010-07-01 メルク・シャープ・エンド・ドーム・コーポレイション Mineralocorticoid receptor modulators

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2899441A (en) * 1959-08-11 Chjchjoh

Also Published As

Publication number Publication date
IL41448A0 (en) 1973-04-30
NO137233B (en) 1977-10-17
HU166406B (en) 1975-03-28
IL41448A (en) 1977-07-31
FR2173984A1 (en) 1973-10-12
FI57936B (en) 1980-07-31
CA979899A (en) 1975-12-16
NL7301494A (en) 1973-08-07
AU5177473A (en) 1974-08-08
CH594630A5 (en) 1978-01-13
GB1363382A (en) 1974-08-14
FR2173984B1 (en) 1976-08-13
AU467008B2 (en) 1975-11-13
FI57936C (en) 1980-11-10
ES411222A1 (en) 1975-12-01
BE794940A (en) 1973-08-02
CS187368B2 (en) 1979-01-31
LU66953A1 (en) 1973-04-19
DE2305212A1 (en) 1973-08-16
AT322545B (en) 1975-05-26

Similar Documents

Publication Publication Date Title
NO140381C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE ARYLPIPERAZINES
NO138807C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE E 3-MARKAPTOTIADIAZOLE OR MARKAPTOTETRAZOLE-CEPHALOSPORINE
NO137321C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 3-OXO-17ALFA-ACYLOXYANDROST-4-EN-17BETA-CARBOXYLIC ACID ESTERS
NO136459C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF ANTIMICROBIALLY ACTIVE PLEUROMUTILINES.
NO138566C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2,1,3-BENZOTIADIAZOLE DERIVATIVES
NO138374C (en) ANALOGICAL PROCEDURES FOR THE PREPARATION OF THERAPEUTIC ACTIVITIES 4-PHENOXYPHENOXYAL CANCARBOXYLIC ACID DERIVATIVES
NO143575C (en) ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PROSTANIC ACID DERIVATIVES
NO136492C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 3- (TRISUBSTITUTED BENZOYL) PROPHIC ACID.
NO140977C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-AMINO-1,4-DIHYDROPYRIDINES
NO138999C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE DIPHENYLYL-ALKANOYLAMINOPYRIDINES
NO137899C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE N (1H-TETRAZOL-5-YL) -KINAL DAMIDES
NO136251C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PYRIDAZINE DERIVATIVES.
SE400551B (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 3-AMINO-5-CARBAMYLBENZOIC ACID DERIVATIVES
NO137858C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE INDANONS
NO139088C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2BETA, 16BETA-DIAMINO-5ALFA-ANDROSTANES
NO139917C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF 1-AMINOMETHYL-2,2-DIARYL-CYCLOPROPANCARBOXAMIDS AND SALTS THEREOF
NO136795C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE INDOLINES
NO138025C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF ANTIMYCOTIC ACTIVE 1-ETHYL-IMIDAZOLES
NO137728C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PYRASI-4-OXYDE DERIVATIVES
NO138598C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 1- (2-DELTA2-IMIDAZOLINYL) -2,2-DIARYLCYCLOPROPANES AND THEIR ACID ADDITIONAL SALTS
NO137233C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ALFA, ALFA-DIARYLIMIDAZOLE-2-METHANOLS AND ACID ADDITIONAL SALTS THEREOF
SE403612B (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF ANTIBACTERIAL ACTIVE HEXAMETHYLENE-BIS-BIGUANIDS
NO137695C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE N-THENYLMETHYL-HETEROCYCLIC COMPOUNDS
NO136410C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF ANTIDIABETIC ACTIVE 3-METHYL-PYRAZOLE-5-CARBOXAMIDES.
NO139173C (en) ANALOGICAL PROCEDURE FOR THE PREPARATION OF ANTIMICROBIALLY ACTIVE 2-KINOXALINE-CARBOXAMIDE-1,4-DIOXIDES