NL165178B - PROCESS FOR PREPARING A THERAPEUTIC PREPARATION USING A 6-FLUOR-16-METHYL STERID OF THE PREGNA SERIES AND METHOD FOR PREPARING A STERID AND FORMED USE THEREFOR. - Google Patents

PROCESS FOR PREPARING A THERAPEUTIC PREPARATION USING A 6-FLUOR-16-METHYL STERID OF THE PREGNA SERIES AND METHOD FOR PREPARING A STERID AND FORMED USE THEREFOR.

Info

Publication number
NL165178B
NL165178B NL7303262.A NL7303262A NL165178B NL 165178 B NL165178 B NL 165178B NL 7303262 A NL7303262 A NL 7303262A NL 165178 B NL165178 B NL 165178B
Authority
NL
Netherlands
Prior art keywords
sterid
preparing
pregna
fluor
methyl
Prior art date
Application number
NL7303262.A
Other languages
Dutch (nl)
Other versions
NL7303262A (en
NL165178C (en
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of NL7303262A publication Critical patent/NL7303262A/xx
Publication of NL165178B publication Critical patent/NL165178B/en
Application granted granted Critical
Publication of NL165178C publication Critical patent/NL165178C/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NL7303262.A 1972-03-09 1973-03-08 PROCESS FOR PREPARING A THERAPEUTIC PREPARATION USING A 6-FLUOR-16-METHYL STERID OF THE PREGNA SERIES AND METHOD FOR PREPARING A STERID AND FORMED USE THEREFOR. NL165178C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23333772A 1972-03-09 1972-03-09
US31697372A 1972-12-20 1972-12-20

Publications (3)

Publication Number Publication Date
NL7303262A NL7303262A (en) 1973-09-11
NL165178B true NL165178B (en) 1980-10-15
NL165178C NL165178C (en) 1981-03-16

Family

ID=26926821

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7303262.A NL165178C (en) 1972-03-09 1973-03-08 PROCESS FOR PREPARING A THERAPEUTIC PREPARATION USING A 6-FLUOR-16-METHYL STERID OF THE PREGNA SERIES AND METHOD FOR PREPARING A STERID AND FORMED USE THEREFOR.

Country Status (13)

Country Link
JP (3) JPS5331156B2 (en)
AR (1) AR197216A1 (en)
AU (1) AU468257B2 (en)
CH (3) CH580117A5 (en)
DE (1) DE2365992C3 (en)
DK (1) DK133382B (en)
ES (1) ES412235A1 (en)
FR (1) FR2181802B1 (en)
GB (1) GB1403962A (en)
HK (1) HK62680A (en)
NL (1) NL165178C (en)
PH (1) PH14703A (en)
SE (1) SE396756B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1430223A (en) * 1973-10-25 1976-03-31 Upjohn Co Anti-inflammatory composition comprising steroids
ZA77943B (en) * 1976-03-19 1977-12-28 Upjohn Co Topical steroid clindamycin preparations
NL187577C (en) * 1978-04-05 1991-11-18 Sibla Srl 3-ACETOXY-9BETA, 11BETA-EPOXY-PREGNA-1,3,5-TRIEN, PROCESS FOR THE PREPARATION THEREOF, AND PROCESS FOR THE PREPARATION OF 6-alpha-halogen-1,4-diene-3-ones.
DE3071122D1 (en) 1979-11-16 1985-10-31 Sterosynt Ltd 6-alpha-fluoro-9-alpha-chloro-prednisolone-17,21 diesters, pharmaceutical compositions containing them and intermediates
JPH0240957Y2 (en) * 1986-08-30 1990-10-31

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB933859A (en) * 1958-09-06 1963-08-14 Syntex S.A.

Also Published As

Publication number Publication date
AR197216A1 (en) 1974-03-22
FR2181802B1 (en) 1976-10-22
DE2365992A1 (en) 1977-05-18
DK133382B (en) 1976-05-10
FR2181802A1 (en) 1973-12-07
DE2365992C3 (en) 1982-05-19
JPS5344464B2 (en) 1978-11-29
PH14703A (en) 1981-11-10
CH580117A5 (en) 1976-09-30
CH580118A5 (en) 1976-09-30
NL7303262A (en) 1973-09-11
HK62680A (en) 1980-11-14
AU5257973A (en) 1974-08-29
JPS5227761A (en) 1977-03-02
JPS4899157A (en) 1973-12-15
CH580116A5 (en) 1976-09-30
ES412235A1 (en) 1976-01-01
JPS5331156B2 (en) 1978-08-31
JPS5227760A (en) 1977-03-02
GB1403962A (en) 1975-08-28
JPS5344465B2 (en) 1978-11-29
DK133382C (en) 1976-10-04
AU468257B2 (en) 1976-01-08
SE396756B (en) 1977-10-03
NL165178C (en) 1981-03-16
DE2365992B2 (en) 1981-08-06

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Legal Events

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V4 Lapsed because of reaching the maximum lifetime of a patent