NL164040B - METHOD FOR PREPARING 3'-DESOXY DERIVATIVES OF AMINOGLYCOSIDE ANTIBIOTICS, AND METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION INCLUDING SUCH A COMPOUND AS AN ACTIVE SUBSTANCE - Google Patents

METHOD FOR PREPARING 3'-DESOXY DERIVATIVES OF AMINOGLYCOSIDE ANTIBIOTICS, AND METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION INCLUDING SUCH A COMPOUND AS AN ACTIVE SUBSTANCE

Info

Publication number
NL164040B
NL164040B NL7316777.A NL7316777A NL164040B NL 164040 B NL164040 B NL 164040B NL 7316777 A NL7316777 A NL 7316777A NL 164040 B NL164040 B NL 164040B
Authority
NL
Netherlands
Prior art keywords
preparing
compound
active substance
pharmaceutical preparation
aminoglycoside antibiotics
Prior art date
Application number
NL7316777.A
Other languages
Dutch (nl)
Other versions
NL7316777A (en
NL164040C (en
Original Assignee
Microbial Chem Res Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Microbial Chem Res Found filed Critical Microbial Chem Res Found
Publication of NL7316777A publication Critical patent/NL7316777A/xx
Publication of NL164040B publication Critical patent/NL164040B/en
Application granted granted Critical
Publication of NL164040C publication Critical patent/NL164040C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/224—Cyclohexane rings substituted by at least two nitrogen atoms with only one saccharide radical directly attached to the cyclohexyl radical, e.g. destomycin, fortimicin, neamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/228—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to adjacent ring-carbon atoms of the cyclohexane rings
    • C07H15/23—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to adjacent ring-carbon atoms of the cyclohexane rings with only two saccharide radicals in the molecule, e.g. ambutyrosin, butyrosin, xylostatin, ribostamycin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
NL7316777.A 1972-12-08 1973-12-07 METHOD FOR PREPARING 3'-DESOXY DERIVATIVES OF AMINOGLYCOSIDE ANTIBIOTICS, AND METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION INCLUDING SUCH A COMPOUND AS AN ACTIVE SUBSTANCE NL164040C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP12243672A JPS57876B2 (en) 1972-12-08 1972-12-08

Publications (3)

Publication Number Publication Date
NL7316777A NL7316777A (en) 1974-06-11
NL164040B true NL164040B (en) 1980-06-16
NL164040C NL164040C (en) 1980-11-17

Family

ID=14835788

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7316777.A NL164040C (en) 1972-12-08 1973-12-07 METHOD FOR PREPARING 3'-DESOXY DERIVATIVES OF AMINOGLYCOSIDE ANTIBIOTICS, AND METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION INCLUDING SUCH A COMPOUND AS AN ACTIVE SUBSTANCE

Country Status (10)

Country Link
JP (1) JPS57876B2 (en)
AR (1) AR201932A1 (en)
AT (1) AT332543B (en)
BE (1) BE808393A (en)
CA (1) CA1016165A (en)
DE (2) DE2361159C3 (en)
ES (1) ES421251A1 (en)
FR (1) FR2209745B1 (en)
GB (1) GB1426910A (en)
NL (1) NL164040C (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5116642A (en) * 1974-08-01 1976-02-10 Meiji Seika Co 3** deokishineamin oyobi sonokanrenkoseibutsushitsuno seizoho
FR2290908A1 (en) * 1974-11-13 1976-06-11 Roussel Uclaf NEW AMINOGLYCOSIDIC DERIVATIVE AND ITS SALTS, THEIR METHOD OF PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2358156A1 (en) * 1976-03-31 1978-02-10 Roussel Uclaf Antibacterial 2-desoxy-streptamine derivs. - prepd. from methyl-4,6-benzylidene-3-ethoxy:carbonylamino 3-desoxy-gluco:pyranoside
JPS5663993A (en) * 1979-10-30 1981-05-30 Microbial Chem Res Found Novel preparation of tobramycin
JPS6140297A (en) * 1984-08-02 1986-02-26 Microbial Chem Res Found 3'-fluoro-3'-deoxykanamycin a
US4661474A (en) * 1984-12-15 1987-04-28 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai 2',3'-dideoxy-2'-fluorokanamycin A and 1-N-(α-hydroxy-ω-aminoalkanoyl) derivatives thereof
JPH0544930Y2 (en) * 1986-01-24 1993-11-16
JPH01157976A (en) * 1987-12-16 1989-06-21 Towa Kasei Kogyo Kk (4s, 5s)-4,5-cyclohexylidenedioxy-2-cyclopenten-1-one, enantiomer and synthetic intermediate thereof and production thereof

Also Published As

Publication number Publication date
NL7316777A (en) 1974-06-11
DE2366288B2 (en) 1981-07-02
ATA1031873A (en) 1976-01-15
DE2366288C3 (en) 1982-03-18
DE2361159C3 (en) 1982-04-29
BE808393A (en) 1974-03-29
DE2361159B2 (en) 1981-07-02
AR201932A1 (en) 1975-04-30
ES421251A1 (en) 1976-04-01
NL164040C (en) 1980-11-17
GB1426910A (en) 1976-03-03
JPS57876B2 (en) 1982-01-08
AT332543B (en) 1976-10-11
FR2209745B1 (en) 1977-09-23
CA1016165A (en) 1977-08-23
FR2209745A1 (en) 1974-07-05
DE2361159A1 (en) 1974-06-20
JPS4980038A (en) 1974-08-02

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Legal Events

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V4 Lapsed because of reaching the maximum lifetime of a patent