NL160273C - PROCESS FOR PREPARING A PREPARATION WITH A HORMONAL ACTIVITY AND A PROCESS FOR PREPARING SUCH 13-ALKYLGONAN-3, 17-BETA DIOL COMPOUNDS. - Google Patents

PROCESS FOR PREPARING A PREPARATION WITH A HORMONAL ACTIVITY AND A PROCESS FOR PREPARING SUCH 13-ALKYLGONAN-3, 17-BETA DIOL COMPOUNDS.

Info

Publication number
NL160273C
NL160273C NL6715790.A NL6715790A NL160273C NL 160273 C NL160273 C NL 160273C NL 6715790 A NL6715790 A NL 6715790A NL 160273 C NL160273 C NL 160273C
Authority
NL
Netherlands
Prior art keywords
preparing
alkylgonan
preparation
diol compounds
hormonal activity
Prior art date
Application number
NL6715790.A
Other languages
Dutch (nl)
Other versions
NL160273B (en
NL6715790A (en
Original Assignee
Searle & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Searle & Co filed Critical Searle & Co
Publication of NL6715790A publication Critical patent/NL6715790A/xx
Publication of NL160273B publication Critical patent/NL160273B/en
Application granted granted Critical
Publication of NL160273C publication Critical patent/NL160273C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/02Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with oxygen atoms attached in positions 3 and 6, e.g. morphine, morphinone
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Knives (AREA)
NL6715790.A 1966-11-22 1967-11-21 PROCESS FOR PREPARING A PREPARATION WITH A HORMONAL ACTIVITY AND A PROCESS FOR PREPARING SUCH 13-ALKYLGONAN-3, 17-BETA DIOL COMPOUNDS. NL160273C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US59609066A 1966-11-22 1966-11-22

Publications (3)

Publication Number Publication Date
NL6715790A NL6715790A (en) 1968-05-24
NL160273B NL160273B (en) 1979-05-15
NL160273C true NL160273C (en) 1979-10-15

Family

ID=24385944

Family Applications (1)

Application Number Title Priority Date Filing Date
NL6715790.A NL160273C (en) 1966-11-22 1967-11-21 PROCESS FOR PREPARING A PREPARATION WITH A HORMONAL ACTIVITY AND A PROCESS FOR PREPARING SUCH 13-ALKYLGONAN-3, 17-BETA DIOL COMPOUNDS.

Country Status (17)

Country Link
US (1) US3465010A (en)
AT (1) AT275749B (en)
BE (1) BE706819A (en)
CH (1) CH509297A (en)
DE (1) DE1618980B2 (en)
DK (1) DK120489B (en)
ES (1) ES347422A1 (en)
FI (1) FI45857C (en)
FR (2) FR1577245A (en)
GB (1) GB1190240A (en)
GR (1) GR37269B (en)
IL (1) IL28982A (en)
MY (1) MY7300398A (en)
NL (1) NL160273C (en)
NO (1) NO126365B (en)
OA (1) OA02672A (en)
SE (1) SE337818B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3723483A (en) * 1970-07-27 1973-03-27 R Coombs 11{62 -methyl-17{60 -propadienyl steroids
FR2377418A1 (en) * 1977-01-13 1978-08-11 Roussel Uclaf NEW 4,9-DIENIC 11B-SUBSTITUTE STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2377419A1 (en) * 1977-01-13 1978-08-11 Roussel Uclaf NEW 11B-SUBSTITUTES 1,3,5 (10) TRIENIC STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS A MEDICINAL PRODUCT
NL7701384A (en) * 1977-02-10 1978-08-14 Akzo Nv PROCESS FOR PREPARING NEW STEROIDS FROM THE OESTRAINE SERIES.
DE4235220A1 (en) * 1992-10-13 1994-06-16 Schering Ag Gestagen effective 19,11ß-bridged 4-estrene
US5710144A (en) * 1993-02-08 1998-01-20 Akzo Nobel N.V. C-11 substituted steroids for treating menopausal complaints
US6037339A (en) * 1993-02-08 2000-03-14 Akzo Nobel N.V. C-11 substituted steroids for treating menopausal complaints
ZA94715B (en) * 1993-02-08 1994-10-24 Akzo Nv Steroids for treating menopausal complaints
IL148116A0 (en) * 1999-09-06 2002-09-12 Akzo Nobel Nv Non-aromatic estrogenic steroids with a hydrocarbon substituent in position 11
CA2416311C (en) * 2000-07-28 2009-04-28 Akzo Nobel N.V. 16alpha-methyl or ethyl substituted estrogens
UA89964C2 (en) 2004-09-08 2010-03-25 Н.В. Органон 15beta-substituted steroids having selective estrogenic activity

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2843609A (en) * 1955-10-11 1958-07-15 Searle & Co 17-alkenyl and alkynyl derivatives of 4-estrene-3, 17-diol
US3176013A (en) * 1963-07-25 1965-03-30 Searle & Co 17alpha-(aliphatic hydrocarbon)-4, 5-epoxy-19-norandrostane-3beta, 17beta-diols and lower alkanoates thereof
US3346602A (en) * 1966-10-12 1967-10-10 Searle & Co 13beta-alkyl-11-alkylgona-1, 3, 5 (10)-trien-17-ones, ethers and esters thereof

Also Published As

Publication number Publication date
US3465010A (en) 1969-09-02
NL160273B (en) 1979-05-15
AT275749B (en) 1969-11-10
MY7300398A (en) 1973-12-31
FR1577245A (en) 1969-08-08
NL6715790A (en) 1968-05-24
FI45857C (en) 1972-10-10
CH509297A (en) 1971-06-30
NO126365B (en) 1973-01-29
DE1618980B2 (en) 1976-07-22
BE706819A (en) 1968-05-21
FR7830M (en) 1970-05-25
GB1190240A (en) 1970-04-29
ES347422A1 (en) 1969-11-01
IL28982A (en) 1971-12-29
GR37269B (en) 1969-05-12
DE1618980A1 (en) 1971-04-29
SE337818B (en) 1971-08-23
FI45857B (en) 1972-06-30
DK120489B (en) 1971-06-07
OA02672A (en) 1970-12-15

Similar Documents

Publication Publication Date Title
NL158488B (en) PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH A CALMING ACTIVITY, THE PREPARED MEDICINAL PRODUCTS THEREFORE OBTAINED AND PROCESS FOR PREPARING SUITABLE ACTIVE SUBSTANCES.
NL160608C (en) PROCEDURE FOR PREPARING A CLEANING AGENT.
NL138818B (en) PROCESS FOR PREPARING A POTASSIUM BICARBONATE AND CITRIC ACID THERAPEUTIC PREPARATION FOR THE POTASSIUM EMPLACING THERAPY, AND FORMED THERAPEUTIC PREPARATION.
NL157632C (en) PROCEDURE FOR PREPARING A COPOLYESTER.
NL143906B (en) PROCESS FOR PREPARING AN ALPHA, BETA-UNSATURATED N-ALKYLOLAMIDE.
NL158797B (en) PROCESS FOR PREPARING MEDICINAL PRODUCTS WITH ANTI-SPASMODIC AND ANTI-ULCER ACTIVITY, PREPARED MEDICINAL PRODUCTS THEREFORE OBTAINED AND PROCEDURE FOR PREPARING SUITABLE ACTIVE SUBSTANCES THEREOF.
NL152240B (en) PROCEDURE FOR PREPARING A PERFLUORVINYL ETHER.
NL159571B (en) PROCESS FOR PREPARING A TOBACCO SKIN.
NL160273C (en) PROCESS FOR PREPARING A PREPARATION WITH A HORMONAL ACTIVITY AND A PROCESS FOR PREPARING SUCH 13-ALKYLGONAN-3, 17-BETA DIOL COMPOUNDS.
NL141758B (en) PROCEDURE FOR PREPARING A PREPARATION WITH HERBICIDE EFFECT, AND FORMED PREPARATION.
NL156136B (en) PROCEDURE FOR PREPARING INFLAMMATORY COMPOUNDS AND MEDICINAL PRODUCTS, AND PREPARED MEDICINAL PRODUCTS SO OBTAINED.
NL148591B (en) PROCESS FOR PREPARING MEDICINAL PRODUCTS AND ARYLOXYACETAMIDES SUITABLE FOR THIS, AND FORMED MEDICINAL PRODUCTS SO OBTAINED.
NL154246B (en) PROCEDURE FOR PREPARING AN ADHESIVE AND MOLDED PRODUCT CONTAINING AN ADHESIVE SO PREPARED.
NL138925B (en) PROCEDURE FOR PREPARING 4-ACETOXYBENZYLIDEEN MALONITRILES AND ANTI-PROTECTION PRODUCTS CONTAINED THEREOF.
NL150099B (en) PROCEDURE FOR PREPARING A PREPARATION WITH LOCAL ANESTHETIC ACTIVITY, PREPARATION FORMED AND PROCEDURE FOR PREPARING A COMPOUND SUITABLE FOR THE PREPARATION OF SUCH PREPARATION.
NL146708B (en) PROCESS FOR PREPARING A SKIN PREPARATION.
NL153918B (en) PROCESS FOR PREPARING A COATING PREPARATION.
NL160835C (en) PROCESS FOR PREPARING A DEHYDRO-EPIANDROSTERONE ESTER AND PROCEDURE FOR PREPARING A MEDICINAL PRODUCT.
NL157804B (en) PROCEDURE FOR PREPARING A STABILIZED GRAINED ANTIBIOTIC PREPARATION.
NL150170B (en) PROCEDURE FOR PREPARING A STANNIOXYDE PREPARATION AND PROCEDURE FOR GALVANIC VETERINATION AND PREPARED MOLDED PRODUCTS ACCORDING TO THIS PROCESS.
NL154116B (en) METHOD OF PREPARING A MEDICINAL PRODUCT WITH ANTI-BACTERIAL ACTION AND THE MEDICINAL PRODUCT PREPARED.
NL143905B (en) PROCESS FOR PREPARING ALKOXYTRIFLUORMETHYLPHENYL ALKYLAMINS AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS AND THE MEDICINAL PRODUCTS THEREFORE OBTAINED.
NL154751B (en) PROCESS FOR PREPARING POLYALKINS, AND FORMED PRODUCTS MANUFACTURED THEREOF.
NL152866B (en) PROCESS FOR PREPARING 1,2-METHYLENE STEROIDS, AND PROCESS FOR PREPARING ANABOLIC ACTIVE PHARMACEUTICAL AND FORMED PHARMACEUTICAL PREPARATIONS.
NL143960B (en) PROCESS FOR THE PREPARATION PROCESS FOR PREPARING TRIOXANCOPOLYMERS.

Legal Events

Date Code Title Description
V1 Lapsed because of non-payment of the annual fee
NL80 Information provided on patent owner name for an already discontinued patent

Owner name: SEARLE