MY198316A - Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors - Google Patents

Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors

Info

Publication number
MY198316A
MY198316A MYPI2020000301A MYPI2020000301A MY198316A MY 198316 A MY198316 A MY 198316A MY PI2020000301 A MYPI2020000301 A MY PI2020000301A MY PI2020000301 A MYPI2020000301 A MY PI2020000301A MY 198316 A MY198316 A MY 198316A
Authority
MY
Malaysia
Prior art keywords
piperidin
azetidine derivatives
jak1
jak1 inhibitors
activity
Prior art date
Application number
MYPI2020000301A
Inventor
Taisheng Huang
Chu-Biao Xue
Anlai Wang
Ling Kong
Hai Fen Ye
Wenqing Yao
Fames D Rodgers
Stacey Shepard
Haisheng Wang
Lixin Shao
Hui-Yin Li
Qun Li
Original Assignee
Incyte Holdings Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incyte Holdings Corp filed Critical Incyte Holdings Corp
Priority to MYPI2020000301A priority Critical patent/MY198316A/en
Publication of MY198316A publication Critical patent/MY198316A/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The present invention provides piperidin-4-yl azetidine derivatives, as well as their compositions and methods of use, that modulate the 5 activity of Janus kinase 1 (JAK1) and are useful in the treatment of diseases related to the activity of JAK1 including, for example, inflammatory disorders, autoimmune disorders, cancer, and other diseases.
MYPI2020000301A 2012-09-07 2012-09-07 Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors MY198316A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
MYPI2020000301A MY198316A (en) 2012-09-07 2012-09-07 Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
MYPI2020000301A MY198316A (en) 2012-09-07 2012-09-07 Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors

Publications (1)

Publication Number Publication Date
MY198316A true MY198316A (en) 2023-08-23

Family

ID=90931770

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI2020000301A MY198316A (en) 2012-09-07 2012-09-07 Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors

Country Status (1)

Country Link
MY (1) MY198316A (en)

Similar Documents

Publication Publication Date Title
PH12015502575B1 (en) Piperidin-4-yl azetidine derivatives as jak1 inhibitors
PH12018502125A1 (en) Bipyrazole derivatives as jak inhibitors
AU2018236800B2 (en) DNA-PK inhibitors
PH12015500963A1 (en) Tricyclic fused thiophene derivatives as jak inhibitors
NZ700928A (en) Dna-pk inhibitors
MY165963A (en) Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as jak inhibitors
MX2013011908A (en) Compositions and therapeutic uses of ikk-related kinase epsilon and tankbinding kinase 1 inhibitors.
MX2015014234A (en) 2-aminopyrido[4,3-d]pyrimidin-5-one derivatives and their use as wee-1 inhibitors.
PH12014501829A1 (en) Bicyclic pyrazinone derivatives
MY198316A (en) Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors
CY1117435T1 (en) Piperidin-4-yl azetidine derivatives as JAK1 inhibitors
UA110108C2 (en) Azetidine derivatives of piperidine-4-yl as JAK1 inhibitors
EA201890558A1 (en) PETERIDIN-4-ILA ASETIDINE DERIVATIVES AS JAK1 INHIBITORS
MY192305A (en) Bipyrazole derivatives as jak inhibitors
UA110978C2 (en) Azetidinylphenyl, pyridyl or pyrazinylcarboxamide derivatives as JAK inhibitors