MY198316A - Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors - Google Patents
Piperidin-4-YL Azetidine Derivatives as JAK1 InhibitorsInfo
- Publication number
- MY198316A MY198316A MYPI2020000301A MYPI2020000301A MY198316A MY 198316 A MY198316 A MY 198316A MY PI2020000301 A MYPI2020000301 A MY PI2020000301A MY PI2020000301 A MYPI2020000301 A MY PI2020000301A MY 198316 A MY198316 A MY 198316A
- Authority
- MY
- Malaysia
- Prior art keywords
- piperidin
- azetidine derivatives
- jak1
- jak1 inhibitors
- activity
- Prior art date
Links
- DDOFLXMWWKLMSZ-UHFFFAOYSA-N 4-(azetidin-1-yl)piperidine Chemical class C1CCN1C1CCNCC1 DDOFLXMWWKLMSZ-UHFFFAOYSA-N 0.000 title abstract 2
- 229940116839 Janus kinase 1 inhibitor Drugs 0.000 title 1
- 102000002295 Janus Kinase 1 Human genes 0.000 abstract 3
- 108010000837 Janus Kinase 1 Proteins 0.000 abstract 3
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 2
- 208000023275 Autoimmune disease Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 208000027866 inflammatory disease Diseases 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
The present invention provides piperidin-4-yl azetidine derivatives, as well as their compositions and methods of use, that modulate the 5 activity of Janus kinase 1 (JAK1) and are useful in the treatment of diseases related to the activity of JAK1 including, for example, inflammatory disorders, autoimmune disorders, cancer, and other diseases.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MYPI2020000301A MY198316A (en) | 2012-09-07 | 2012-09-07 | Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MYPI2020000301A MY198316A (en) | 2012-09-07 | 2012-09-07 | Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
MY198316A true MY198316A (en) | 2023-08-23 |
Family
ID=90931770
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MYPI2020000301A MY198316A (en) | 2012-09-07 | 2012-09-07 | Piperidin-4-YL Azetidine Derivatives as JAK1 Inhibitors |
Country Status (1)
Country | Link |
---|---|
MY (1) | MY198316A (en) |
-
2012
- 2012-09-07 MY MYPI2020000301A patent/MY198316A/en unknown
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