UA110108C2 - Azetidine derivatives of piperidine-4-yl as JAK1 inhibitors - Google Patents

Azetidine derivatives of piperidine-4-yl as JAK1 inhibitors

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Publication number
UA110108C2
UA110108C2 UAA201211696A UAA201211696A UA110108C2 UA 110108 C2 UA110108 C2 UA 110108C2 UA A201211696 A UAA201211696 A UA A201211696A UA A201211696 A UAA201211696 A UA A201211696A UA 110108 C2 UA110108 C2 UA 110108C2
Authority
UA
Ukraine
Prior art keywords
piperidine
azetidine derivatives
jak1
jak1 inhibitors
activity
Prior art date
Application number
UAA201211696A
Other languages
Russian (ru)
Ukrainian (uk)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2011/027665 external-priority patent/WO2011112662A1/en
Application filed filed Critical
Publication of UA110108C2 publication Critical patent/UA110108C2/en

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Abstract

У даному винаході представлені азетидинові похідні піперидин-4-ілу, а також їх композиції і способи їх застосування, які модулюють активність Янус-кінази 1 (JAK1) і є корисними для лікування захворювань, пов'язаних з активністю JAK1, включаючи, наприклад, запальні порушення, аутоімунні порушення, рак і інші захворювання.The present invention provides azetidine derivatives of piperidin-4-yl, as well as their compositions and methods of use, which modulate the activity of Janus kinase 1 (JAK1) and are useful for the treatment of diseases associated with JAK1 activity, including, for example, inflammatory disorders, autoimmune disorders, cancer and other diseases.

UAA201211696A 2010-03-10 2011-09-03 Azetidine derivatives of piperidine-4-yl as JAK1 inhibitors UA110108C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31258810P 2010-03-10 2010-03-10
PCT/US2011/027665 WO2011112662A1 (en) 2010-03-10 2011-03-09 Piperidin-4-yl azetidine derivatives as jak1 inhibitors

Publications (1)

Publication Number Publication Date
UA110108C2 true UA110108C2 (en) 2015-11-25

Family

ID=55171064

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201211696A UA110108C2 (en) 2010-03-10 2011-09-03 Azetidine derivatives of piperidine-4-yl as JAK1 inhibitors

Country Status (2)

Country Link
AR (1) AR114485A2 (en)
UA (1) UA110108C2 (en)

Also Published As

Publication number Publication date
AR114485A2 (en) 2020-09-09

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