UA110108C2 - Azetidine derivatives of piperidine-4-yl as JAK1 inhibitors - Google Patents
Azetidine derivatives of piperidine-4-yl as JAK1 inhibitorsInfo
- Publication number
- UA110108C2 UA110108C2 UAA201211696A UAA201211696A UA110108C2 UA 110108 C2 UA110108 C2 UA 110108C2 UA A201211696 A UAA201211696 A UA A201211696A UA A201211696 A UAA201211696 A UA A201211696A UA 110108 C2 UA110108 C2 UA 110108C2
- Authority
- UA
- Ukraine
- Prior art keywords
- piperidine
- azetidine derivatives
- jak1
- jak1 inhibitors
- activity
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
У даному винаході представлені азетидинові похідні піперидин-4-ілу, а також їх композиції і способи їх застосування, які модулюють активність Янус-кінази 1 (JAK1) і є корисними для лікування захворювань, пов'язаних з активністю JAK1, включаючи, наприклад, запальні порушення, аутоімунні порушення, рак і інші захворювання.The present invention provides azetidine derivatives of piperidin-4-yl, as well as their compositions and methods of use, which modulate the activity of Janus kinase 1 (JAK1) and are useful for the treatment of diseases associated with JAK1 activity, including, for example, inflammatory disorders, autoimmune disorders, cancer and other diseases.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US31258810P | 2010-03-10 | 2010-03-10 | |
PCT/US2011/027665 WO2011112662A1 (en) | 2010-03-10 | 2011-03-09 | Piperidin-4-yl azetidine derivatives as jak1 inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
UA110108C2 true UA110108C2 (en) | 2015-11-25 |
Family
ID=55171064
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA201211696A UA110108C2 (en) | 2010-03-10 | 2011-09-03 | Azetidine derivatives of piperidine-4-yl as JAK1 inhibitors |
Country Status (2)
Country | Link |
---|---|
AR (1) | AR114485A2 (en) |
UA (1) | UA110108C2 (en) |
-
2011
- 2011-09-03 UA UAA201211696A patent/UA110108C2/en unknown
-
2019
- 2019-04-12 AR ARP190100972A patent/AR114485A2/en unknown
Also Published As
Publication number | Publication date |
---|---|
AR114485A2 (en) | 2020-09-09 |
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