MY185481A - Osteoclast inhibitors for pain - Google Patents

Osteoclast inhibitors for pain

Info

Publication number
MY185481A
MY185481A MYPI2016704377A MYPI2016704377A MY185481A MY 185481 A MY185481 A MY 185481A MY PI2016704377 A MYPI2016704377 A MY PI2016704377A MY PI2016704377 A MYPI2016704377 A MY PI2016704377A MY 185481 A MY185481 A MY 185481A
Authority
MY
Malaysia
Prior art keywords
pain
osteoclast inhibitors
osteoclast
inhibitors
methods
Prior art date
Application number
MYPI2016704377A
Other languages
English (en)
Inventor
Herriot Tabuteau
Eric K M Dinkla
Graeme Jones
Original Assignee
Antecip Bioventures Ii Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US14/288,716 external-priority patent/US8835650B1/en
Priority claimed from US14/288,720 external-priority patent/US8865757B1/en
Priority claimed from US14/310,811 external-priority patent/US8822436B1/en
Priority claimed from PCT/US2014/050427 external-priority patent/WO2015060924A1/fr
Priority claimed from US14/457,659 external-priority patent/US20140349974A1/en
Priority claimed from US14/495,732 external-priority patent/US9127069B1/en
Priority claimed from US14/530,556 external-priority patent/US20150051175A1/en
Priority claimed from US14/536,526 external-priority patent/US20150057250A1/en
Priority claimed from US14/604,524 external-priority patent/US9211257B2/en
Priority claimed from US14/608,855 external-priority patent/US9079927B1/en
Priority claimed from US14/625,457 external-priority patent/US9427403B2/en
Priority claimed from US14/639,013 external-priority patent/US9289441B2/en
Application filed by Antecip Bioventures Ii Llc filed Critical Antecip Bioventures Ii Llc
Priority claimed from PCT/US2015/032739 external-priority patent/WO2015184003A1/fr
Publication of MY185481A publication Critical patent/MY185481A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/662Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
    • A61K31/663Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7088Compounds having three or more nucleosides or nucleotides
    • A61K31/713Double-stranded nucleic acids or oligonucleotides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MYPI2016704377A 2014-05-27 2015-05-27 Osteoclast inhibitors for pain MY185481A (en)

Applications Claiming Priority (28)

Application Number Priority Date Filing Date Title
US201414228241A 2014-05-27 2014-05-27
US14/288,716 US8835650B1 (en) 2014-01-30 2014-05-28 Substituted imidazolium compounds for treating disease
US14/288,720 US8865757B1 (en) 2014-05-28 2014-05-28 Therapeutic compositions comprising imidazole and imidazolium compounds
US14/288,713 US8901162B1 (en) 2014-01-30 2014-05-28 Substituted imidazolium compounds for treating disease
US201462012112P 2014-06-13 2014-06-13
US14/310,811 US8822436B1 (en) 2012-05-14 2014-06-20 Compositions for oral administration of zoledronic acid or related compounds for treating disease
US14/336,642 US20140329773A1 (en) 2012-05-14 2014-07-21 Compositions for Oral Administration of Zoledronic Acid or Related Compounds for Treating Disease
US14/446,184 US9006279B1 (en) 2014-01-30 2014-07-29 Substituted imidazolium compounds for treating disease
PCT/US2014/050427 WO2015060924A1 (fr) 2013-10-25 2014-08-08 Compositions pour administration orale d'acide zolédronique ou de composés associés pour le traitement de maladies
US14/457,659 US20140349974A1 (en) 2014-08-12 2014-08-12 Zoledronic acid dosage forms for the treatment of pain
US14/481,097 US8962599B1 (en) 2014-05-27 2014-09-09 Therapeutic compositions comprising imidazole and imidazolium compounds
US201462053619P 2014-09-22 2014-09-22
US14/495,732 US9127069B1 (en) 2014-06-11 2014-09-24 Compositions comprising rank/rankl antagonists and related compounds for treating pain
US14/530,556 US20150051175A1 (en) 2012-05-14 2014-10-31 Co-Administration of Steroids and Zoledronic Acid to Prevent and Treat Pain
US14/536,526 US20150057250A1 (en) 2012-05-14 2014-11-07 Inhibitors of osteoclast activity for treating arthritis
US14/538,709 US9290575B2 (en) 2014-06-11 2014-11-11 Compositions comprising RANK/RANKL antagonists and related compounds for treating pain
US14/540,333 US9216168B1 (en) 2014-05-27 2014-11-13 Therapeutic compositions comprising imidazole and imidazolium compounds
US14/604,524 US9211257B2 (en) 2012-05-14 2015-01-23 Osteoclast inhibitors for knee conditions
US14/605,822 US9216153B2 (en) 2012-05-14 2015-01-26 Osteoclast inhibitors for knee conditions
US14/607,947 US9289384B2 (en) 2012-05-14 2015-01-28 Osteoclast inhibitors for knee conditions
US14/607,985 US9289385B2 (en) 2012-05-14 2015-01-28 Osteoclast inhibitors for knee conditions
US14/608,855 US9079927B1 (en) 2014-05-27 2015-01-29 Substituted imidazolium compounds for treating disease
US14/625,457 US9427403B2 (en) 2012-05-14 2015-02-18 Methods for the safe administration of imidazole or imidazolium compounds
US201562127214P 2015-03-02 2015-03-02
US14/635,857 US9283239B2 (en) 2012-05-14 2015-03-02 Compositions for oral administration of zoledronic acid or related compounds for treating complex regional pain syndrome
US14/639,013 US9289441B2 (en) 2014-08-08 2015-03-04 Osteoclast inhibitors such as zoledronic acid for low back pain treatment
US14/686,551 US9408860B2 (en) 2012-05-14 2015-04-14 Compositions for oral administration of zoledronic acid or related compounds for treating low back pain
PCT/US2015/032739 WO2015184003A1 (fr) 2014-05-27 2015-05-27 Inhibiteurs d'ostéoclastes contre la douleur

Publications (1)

Publication Number Publication Date
MY185481A true MY185481A (en) 2021-05-19

Family

ID=57483086

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI2016704377A MY185481A (en) 2014-05-27 2015-05-27 Osteoclast inhibitors for pain

Country Status (3)

Country Link
AU (3) AU2017213506B2 (fr)
CA (3) CA3194798A1 (fr)
MY (1) MY185481A (fr)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20130303485A1 (en) * 2012-05-14 2013-11-14 Herriot Tabuteau Compositions for Oral Administration of Zoledronic Acid or Related Compounds for Treating Disease

Also Published As

Publication number Publication date
AU2017272199A1 (en) 2017-12-21
AU2019204559B2 (en) 2020-04-16
AU2019204559A1 (en) 2019-07-18
CA3114271A1 (fr) 2015-12-03
CA3194798A1 (fr) 2015-12-03
AU2017272199B2 (en) 2019-03-28
CA2950443A1 (fr) 2015-12-03
AU2017213506B2 (en) 2017-09-07
AU2017213506A1 (en) 2017-08-31
CA3114271C (fr) 2023-06-06

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