MY145168A - Substituted diaza-spiro-[4.5]-decane derivatives and their use as neurokinin antagonists - Google Patents
Substituted diaza-spiro-[4.5]-decane derivatives and their use as neurokinin antagonistsInfo
- Publication number
- MY145168A MY145168A MYPI20051504A MY145168A MY 145168 A MY145168 A MY 145168A MY PI20051504 A MYPI20051504 A MY PI20051504A MY 145168 A MY145168 A MY 145168A
- Authority
- MY
- Malaysia
- Prior art keywords
- antagonistic activity
- combined
- spiro
- theireof
- antagonistic
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
THIS INVENTION CONCERNS SUBSTITUTED DIAZA-SPIRO-[4.5J-DECANE DENVATIVES HAVING NEUROKININ ANTAGONISTIC ACTIVITY, IN PARTICULAR NK₁ ANTAGONISTIC ACTIVITY, A COMBINED NK₁/NK₂, ANTAGONISTIC ACTIVITY. A COMBINED NK₁/NK₃ ANTAGONISTIC ACTIVIY AND A COMBINED NK₁/NK₂/NK₃ ANTAGONISTIC ACTIVITY, THEIR PREPARATION, COMPOSITIONS COMPRISING THEM AND THEIR USE AS A MEDICINE, IN PARTICULAR FOR THE TREATMENT AND/OR PROPHYLAXIS OF SCHIZOPHRENIA, EMESIS. ANXIETY AND DEPRESSION, INITABLE BOWEL SYNDROME (IBS), CIRCADIAN RHYTHM DISTURBANCES, PRE-ECLAMPSIA, NOCICEPTION, PAM. IN PARTICULAR VISCERAL AND NEUROPATHIC PAIN, PANCREATITIS, NEUROGENIC INFLAMMATION, ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD) AND MICTURITION DISORDERS SUCH AS URINARY INCONTINENCE. THE COMPAUNDS ACCORDING TO THE INVENTION CAN BE REPRESENTED BY GENERAL FORMULA (1) AND COMPRISES ALSO THE PHARMACEUTACALLY ACCEPTABLE ACID OR BASE ADDITION SALTS THEIREOF,THE STEREOCHEMICALLY ISOMERIC FORMS THEIREOF, THE N-OXIDE FORM THEREOF AND PRODRUGS THEREOF, WHEREIN ALL SUBSTITUENTS ARE DEFINED AS IN CLAIM 1.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP04050458 | 2004-04-06 |
Publications (1)
Publication Number | Publication Date |
---|---|
MY145168A true MY145168A (en) | 2011-12-30 |
Family
ID=40257300
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MYPI20051504 MY145168A (en) | 2004-04-06 | 2005-04-04 | Substituted diaza-spiro-[4.5]-decane derivatives and their use as neurokinin antagonists |
Country Status (2)
Country | Link |
---|---|
MY (1) | MY145168A (en) |
PA (1) | PA8628301A1 (en) |
-
2005
- 2005-04-01 PA PA8628301A patent/PA8628301A1/en unknown
- 2005-04-04 MY MYPI20051504 patent/MY145168A/en unknown
Also Published As
Publication number | Publication date |
---|---|
PA8628301A1 (en) | 2005-11-25 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
TW200604198A (en) | Substituted diaza-spiro-[4.5]-decane derivatives and their use as neurokinin antagonists | |
MY142090A (en) | Substituted diaza-spiro-[5.5]-undecane derivatives and their use as neurokinin antagonists | |
MY142773A (en) | Substituted 4-alkyl-and-alkanoyl-piperidine derivatives and their use as neurokinin antagonists | |
WO2006094934A8 (en) | Substituted oxa-diaza-spiro-[5.5]-undecanone derivatives and their use as neurokinin antagonists | |
WO2010018109A3 (en) | Substituted aminotetralines | |
WO2010018113A3 (en) | Bi-aryl aminotetralines | |
MX2012004020A (en) | Heterocyclyl pyrazolopyrimidine analogues as jak inhibitors. | |
IL196543A (en) | Pyridazinone derivatives and pharmaceutical compositions comprising them for use in the treatment of disorders | |
NO20082000L (en) | Pyrimidinamide Compounds as PGDS Inhibitors | |
ATE456565T1 (en) | PYRIDINE AND PYRAZINE DERIVATIVES AS MNK KINASE INHIBITORS | |
SG179437A1 (en) | Pyrimidine hydrazide compounds as pgds inhibitors | |
TW200616967A (en) | Novel indazole carboxamides and their use | |
TW200626601A (en) | Novel compounds | |
WO2010142766A3 (en) | Pyrimidine derivatives as zap-70 inhibitors | |
NZ591914A (en) | Naphthylacetic acids | |
MX350862B (en) | Piperidinyl naphthylacetic acids. | |
MX2009013885A (en) | Fused quinoline derivatives useful as gaba modulators. | |
MX2009005507A (en) | Spiro-piperidine derivatives. | |
WO2004056799A3 (en) | Substituted 1-piperidin-4-yl-4-pyrrolidin-3-yl-piperazine derivatives and their use as neurokinin antagonists | |
WO2006011024A3 (en) | New tricyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them | |
EA200701898A1 (en) | DIAZA-SPYRO- [4.4] -NONAN DERIVATIVES AS ANTAGONISTS NEUROKININ (NK1) | |
MX2009006454A (en) | Spiro-piperidine derivatives. | |
MX2009005544A (en) | Indoles. | |
MX2009005541A (en) | Indoles which act as via receptor antagonists. | |
MX2009005504A (en) | Spiro-piperidine derivatives as via receptor antagonists. |