MX9302986A - Medicamento que contiene metrifonato y procedimiento para su preparacion - Google Patents
Medicamento que contiene metrifonato y procedimiento para su preparacionInfo
- Publication number
- MX9302986A MX9302986A MX9302986A MX9302986A MX9302986A MX 9302986 A MX9302986 A MX 9302986A MX 9302986 A MX9302986 A MX 9302986A MX 9302986 A MX9302986 A MX 9302986A MX 9302986 A MX9302986 A MX 9302986A
- Authority
- MX
- Mexico
- Prior art keywords
- pct
- metrifonate
- procedure
- preparation
- medicines containing
- Prior art date
Links
- 229960001952 metrifonate Drugs 0.000 title abstract 3
- NFACJZMKEDPNKN-UHFFFAOYSA-N trichlorfon Chemical compound COP(=O)(OC)C(O)C(Cl)(Cl)Cl NFACJZMKEDPNKN-UHFFFAOYSA-N 0.000 title abstract 3
- 239000003814 drug Substances 0.000 title abstract 2
- 206010048650 Cholinesterase inhibition Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hospice & Palliative Care (AREA)
- Tropical Medicine & Parasitology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Se ha encontrado un medicamento que contienen metrifonato, el cual contienen al metrifonato enantiómero como única substancia activa. El (-)-metrifonato es básicamente mejor inhibidor de la colineresterasa, que el rasemato, con esto se puede disminuir la cantidad de substancia activa y consecuentemente por ejemplo el tamaño de las tabletas.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4217396A DE4217396A1 (de) | 1992-05-26 | 1992-05-26 | Metrifonat enthaltendes Arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9302986A true MX9302986A (es) | 1993-12-01 |
Family
ID=6459760
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9302986A MX9302986A (es) | 1992-05-26 | 1993-05-21 | Medicamento que contiene metrifonato y procedimiento para su preparacion |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US5629300A (es) |
| EP (1) | EP0669826B1 (es) |
| JP (1) | JPH07507280A (es) |
| AT (1) | ATE169819T1 (es) |
| CA (1) | CA2136548A1 (es) |
| DE (2) | DE4217396A1 (es) |
| DK (1) | DK0669826T3 (es) |
| ES (1) | ES2122005T3 (es) |
| MX (1) | MX9302986A (es) |
| WO (1) | WO1993024130A1 (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9807931D0 (en) * | 1998-04-15 | 1998-06-10 | Medical Res Council | Improvements in or relating to protease inhibitors |
| DE19857716A1 (de) * | 1998-12-15 | 2000-06-21 | Bayer Ag | Neue feste Formulierung von Metrifonat |
| US11446241B2 (en) | 2013-07-29 | 2022-09-20 | Attillaps Holdings Inc. | Treatment of ophthalmological conditions with acetylcholinesterase inhibitors |
| WO2015017328A2 (en) | 2013-07-29 | 2015-02-05 | Spallitta Frank Anthony | Organophosphates for treating afflictions of the skin |
| SI3157534T1 (sl) | 2014-06-19 | 2022-08-31 | Attillaps Holdings | Inhibitorji acetilholinesteraze za zdravljenje dermatoloških obolenj |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4950658A (en) * | 1988-12-06 | 1990-08-21 | Board Of Trustees Of Southern Illinois Univ. | Method of medical treatment of Alzheimer's disease |
-
1992
- 1992-05-26 DE DE4217396A patent/DE4217396A1/de not_active Withdrawn
-
1993
- 1993-05-17 DE DE59308900T patent/DE59308900D1/de not_active Expired - Fee Related
- 1993-05-17 DK DK93910008T patent/DK0669826T3/da active
- 1993-05-17 JP JP6500134A patent/JPH07507280A/ja not_active Ceased
- 1993-05-17 AT AT93910008T patent/ATE169819T1/de not_active IP Right Cessation
- 1993-05-17 EP EP93910008A patent/EP0669826B1/de not_active Expired - Lifetime
- 1993-05-17 WO PCT/EP1993/001228 patent/WO1993024130A1/de not_active Ceased
- 1993-05-17 ES ES93910008T patent/ES2122005T3/es not_active Expired - Lifetime
- 1993-05-17 CA CA002136548A patent/CA2136548A1/en not_active Abandoned
- 1993-05-21 MX MX9302986A patent/MX9302986A/es not_active IP Right Cessation
- 1993-12-09 US US08/331,643 patent/US5629300A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| ATE169819T1 (de) | 1998-09-15 |
| DK0669826T3 (da) | 1999-05-25 |
| EP0669826B1 (de) | 1998-08-19 |
| US5629300A (en) | 1997-05-13 |
| DE59308900D1 (de) | 1998-09-24 |
| CA2136548A1 (en) | 1993-12-09 |
| WO1993024130A1 (de) | 1993-12-09 |
| JPH07507280A (ja) | 1995-08-10 |
| ES2122005T3 (es) | 1998-12-16 |
| DE4217396A1 (de) | 1993-12-02 |
| EP0669826A1 (de) | 1995-09-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration | ||
| MM | Annulment or lapse due to non-payment of fees |